GPRC5A (rai3_mouse)

FAMILY

Class C (Glutamate) Orphan receptors Class C Orphans GPRC5A

GENE

Gprc5a (Rai3, Raig1)

ORGANISM

Mouse (Mus musculus)

ALT. NAMES

Retinoic acid-induced protein 3, G-protein coupled receptor family C group 5 member A, Retinoic acid-induced gene 1 protein, RAIG-1

SOURCE

SWISSPROT

SEQUENCE

N-term        
M
T
T
P
T
T
A
P
S
G
10
                   
C
R
S
D
L
D
S
R
Y
H
20
                   
R
L
C
D
L
A
E
G
W
G
30
TM1              
I
A
L
E
T
L
A
A
V
G
40
                   
A
V
A
T
V
A
C
M
F
A
50
        ICL1    
L
V
F
L
I
C
K
V
Q
D
60
  TM2            
S
N
K
R
K
M
L
P
A
Q
70
                   
F
L
F
L
L
G
V
L
G
V
80
                   
F
G
L
T
F
A
F
I
I
K
90
ECL1 TM3      
L
D
G
A
T
G
P
T
R
F
100
                   
F
L
F
G
V
L
F
A
I
C
110
                   
F
S
C
L
L
A
H
A
F
N
120
          ICL2  
L
I
K
L
V
R
G
R
K
P
130
  TM4            
L
S
W
L
V
I
L
S
L
A
140
                   
V
G
F
S
L
V
Q
D
V
I
150
                   
A
I
E
Y
L
V
L
T
M
N
160
ECL2            
R
T
N
V
N
V
F
S
E
L
170
        TM5      
P
A
P
R
R
N
E
D
F
V
180
                   
M
L
L
I
Y
V
L
V
L
M
190
                   
V
L
T
F
F
T
S
F
L
V
200
ICL3            
F
C
G
S
F
S
G
W
K
R
210
TM6              
H
G
F
H
I
C
F
T
S
F
220
                   
L
S
I
A
I
W
V
A
W
I
230
            ECL3
V
L
L
L
I
P
D
I
D
R
240
TM7              
K
W
D
D
T
I
L
S
T
A
250
                   
L
V
A
N
G
W
V
F
L
A
260
                   
F
Y
I
L
P
E
F
R
Q
L
270
      ICL4 H8  
P
R
Q
R
S
P
T
D
Y
P
280
                   
V
E
D
A
F
C
K
P
Q
L
290
C-term        
M
K
Q
S
Y
G
V
E
N
R
300
                   
A
Y
S
Q
E
E
I
T
Q
G
310
                   
L
E
M
G
D
T
L
Y
A
P
320
                   
Y
S
T
H
F
Q
L
Q
N
H
330
                   
Q
K
D
F
S
I
P
R
A
Q
340
                   
A
P
A
S
P
Y
N
D
Y
E
350
           
G
R
K
G
D
S

LINKS

DIAGRAMS

ICL1 I C K V Q D S ICL1ECL1 I K L ECL1ICL2 R G R K P L ICL2ECL2 M N R T N V N V F S E L P A P R ECL2ICL3 F C G S F S G W K R ICL3ECL3 D I D R ECL3N-term M T T P T T A P S G C R S D L D S R Y H R L C D L A E G N-termC-term P Q L M K Q S Y G V E N R A Y S Q E E I T Q G L E M G D T L Y A P Y S T H F Q L Q N H Q K D F S I P R A Q A P A S P Y N D Y E G R K G D S C-term W G I A L E T L A A V G A V A T V A C M F A L V F L N K R K M L P A Q F L F L L G V L G V F G L T F A F I D G A T G P T R F F L F G V L F A I C F S C L L A H A F N L I K L V S W L V I L S L A V G F S L V Q D V I A I E Y L V L T R N E D F V M L L I Y V L V L M V L T F F T S F L V H G F H I C F T S F L S I A I W V A W I V L L L I P K W D D T I L S T A L V A N G W V F L A F Y I L P E F R Q L P R Q S P T E D A D Y P V F C K
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

V T A V A G V A A L T E L A I G W 1 F L F L L G V L G V F G L T F A F I 2 A L L C S F C I A F L V G F L F F R T P 3 I L S L A V G F S L V Q D V I A I E Y L 4 S T F F T L V M L V L V Y I L L M V F D 5 C F T S F L S I A I W V A W I V L L L I 6 A L F V W G N A V L A T S L I T D D W K 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

MUTATIONS

ENDOGENOUS LIGANDS

No endogenous ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available