Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|
| 3404 | 12 | None | 27 | Mouse | Functional | pEC50 | = | 9.6 | 9.6 | 107 | 3 | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| 5283155 | 12 | None | 27 | Mouse | Functional | pEC50 | = | 9.6 | 9.6 | 107 | 3 | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| 5508 | 12 | None | 27 | Mouse | Functional | pEC50 | = | 9.6 | 9.6 | 107 | 3 | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| CHEMBL1526258 | 12 | None | 27 | Mouse | Functional | pEC50 | = | 9.6 | 9.6 | 107 | 3 | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|
| 3404 | 12 | None | 27 | Mouse | Binding | pKd | = | 8.3 | 8.3 | - | 1 | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| 5283155 | 12 | None | 27 | Mouse | Binding | pKd | = | 8.3 | 8.3 | - | 1 | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| 5508 | 12 | None | 27 | Mouse | Binding | pKd | = | 8.3 | 8.3 | - | 1 | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||
| CHEMBL1526258 | 12 | None | 27 | Mouse | Binding | pKd | = | 8.3 | 8.3 | - | 1 | Guide to Pharmacology | 320 | 14 | 2 | 2 | 5.2 | CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O | 21712392 | |||