GPCRdb

Ligands (move mouse cursor over ligand name to see structure)					Receptor	Activity									Chemical information
Sel. page	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	131648253	3039	None	0	Mouse	Functional	pEC50	=	10.7	10.7	-	1	High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83	Guide to Pharmacology		None	None	None		None	27117253
	155817507	3039	None	0	Mouse	Functional	pEC50	=	10.7	10.7	-	1	High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83	Guide to Pharmacology		None	None	None		None	27117253
	9139	3039	None	0	Mouse	Functional	pEC50	=	10.7	10.7	-	1	High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83	Guide to Pharmacology		None	None	None		None	27117253
	131648253	3039	None	0	Mouse	Functional	pEC50	=	7.0	7.0	-	1	Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83	Guide to Pharmacology		None	None	None		None	27117253
	155817507	3039	None	0	Mouse	Functional	pEC50	=	7.0	7.0	-	1	Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83	Guide to Pharmacology		None	None	None		None	27117253
	9139	3039	None	0	Mouse	Functional	pEC50	=	7.0	7.0	-	1	Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83	Guide to Pharmacology		None	None	None		None	27117253
	32051	4151	None	0	Mouse	Functional	pEC50	=	5	5.0	-	1	UnclassifiedUnclassified	Guide to Pharmacology	64	0	0	0	-0.0	[Zn+2]	23335960
	566	4151	None	0	Mouse	Functional	pEC50	=	5	5.0	-	1	UnclassifiedUnclassified	Guide to Pharmacology	64	0	0	0	-0.0	[Zn+2]	23335960

Ligands (move mouse cursor over ligand name to see structure)	Receptor	Activity	Chemical information
	9140	3040	None	0	Mouse		Binding	pKd	=	8.1	8.1	-	1	N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.	Guide to Pharmacology		None	None	None		None	27117253

Ligands (move mouse cursor over ligand name to see structure)

Receptor

Activity

Chemical information

Sel. page

Common
name

GPCRdb
ID

Reference
ligand

Vendors

Species

Assay
Type

Activity
Type

Activity
Relation

Activity
Value

p-value
(-log)

Fold
selectivity

Tested
GPCRs

Assay
Description

Source

Mol
weight

Rot
Bonds

H don

H acc

LogP

Smiles

DOI

9140

3040

None

Mouse

Binding

pKd

8.1

N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.

Guide to Pharmacology

None

27117253

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Main reference

Ligand source activities (1 row/activity)