Ligand source activities (1 row/activity)





Ligands (move mouse cursor over ligand name to see structure) Receptor Activity Chemical information
Sel. page Common
name
GPCRdb
ID
Reference
ligand
Vendors

Species

Assay
Type

Activity
Type
Activity
Relation
Activity
Value
p-value
(-log)
Fold
selectivity
Tested
GPCRs
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI

3700 3408 None 0 Human Functional pEC50 = 10.1 10.1 4 2
UnclassifiedUnclassified
Guide to Pharmacology None None None None 21693646
3697 3402 None 0 Human Functional pEC50 = 10.7 10.7 -2 2
UnclassifiedUnclassified
Guide to Pharmacology None None None None 21693646
3699 3406 None 0 Human Functional pEC50 = 10.7 10.7 -1 2
UnclassifiedUnclassified
Guide to Pharmacology None None None None 21693646
3698 3405 None 0 Human Functional pEC50 = 12.5 12.5 3 2
UnclassifiedUnclassified
Guide to Pharmacology None None None None 21693646




Ligands (move mouse cursor over ligand name to see structure) Receptor Activity Chemical information
Sel. page Common
name
GPCRdb
ID
Reference
ligand
Vendors

Species

Assay
Type
Activity
Type
Activity
Relation
Activity
Value
p-value
(-log)
Fold
selectivity
Tested
GPCRs
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI

3699 3406 None 0 Human Binding pKd = 8.7 8.7 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 21909076