Ligand source activities (1 row/activity)
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|
4383 | 3409 | None | 0 | Human | Functional | pIC50 | = | 8.2 | 8.2 | - | 1 | Guide to Pharmacology | None | None | None | None | 22615920 | |||||
5539 | 3403 | None | 0 | Human | Functional | pIC50 | = | 8.5 | 8.5 | - | 1 | Guide to Pharmacology | None | None | None | None | 22615920 | |||||
5541 | 3407 | None | 0 | Human | Functional | pIC50 | = | 8.8 | 8.8 | - | 1 | Guide to Pharmacology | None | None | None | None | 22615920 | |||||
5540 | 3404 | None | 0 | Human | Functional | pIC50 | = | 9.3 | 9.3 | - | 1 | Guide to Pharmacology | None | None | None | None | 22615920 |
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |