Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|
| 2365 | 603 | None | 0 | Mouse | Functional | pEC50 | = | 4.4 | 4.4 | -3 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| 239 | 603 | None | 0 | Mouse | Functional | pEC50 | = | 4.4 | 4.4 | -3 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| 4755801 | 603 | None | 0 | Mouse | Functional | pEC50 | = | 4.4 | 4.4 | -3 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| CHEMBL297569 | 603 | None | 0 | Mouse | Functional | pEC50 | = | 4.4 | 4.4 | -3 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| DB03107 | 603 | None | 0 | Mouse | Functional | pEC50 | = | 4.4 | 4.4 | -3 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| 2365 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| 2365 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | |||
| 239 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| 239 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | |||
| 4755801 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| 4755801 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | |||
| CHEMBL297569 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| CHEMBL297569 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | |||
| DB03107 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| DB03107 | 603 | None | 0 | Human | Functional | pEC50 | = | 4.8 | 4.8 | -1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | |||
| 2365 | 603 | None | 0 | Rat | Functional | pEC50 | = | 4.9 | 4.9 | 1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| 239 | 603 | None | 0 | Rat | Functional | pEC50 | = | 4.9 | 4.9 | 1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| 4755801 | 603 | None | 0 | Rat | Functional | pEC50 | = | 4.9 | 4.9 | 1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| CHEMBL297569 | 603 | None | 0 | Rat | Functional | pEC50 | = | 4.9 | 4.9 | 1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| DB03107 | 603 | None | 0 | Rat | Functional | pEC50 | = | 4.9 | 4.9 | 1 | 3 | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | |||
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|