Ligand source activities (1 row/activity)
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|
5506 | 2087 | None | 0 | Mouse | Functional | pEC50 | = | 5 | 5.0 | - | 1 | Guide to Pharmacology | 87 | 2 | 1 | 1 | 1.0 | NCCC(C)C | 16878137 | |||
7894 | 2087 | None | 0 | Mouse | Functional | pEC50 | = | 5 | 5.0 | - | 1 | Guide to Pharmacology | 87 | 2 | 1 | 1 | 1.0 | NCCC(C)C | 16878137 | |||
CHEMBL42003 | 2087 | None | 0 | Mouse | Functional | pEC50 | = | 5 | 5.0 | - | 1 | Guide to Pharmacology | 87 | 2 | 1 | 1 | 1.0 | NCCC(C)C | 16878137 |
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |