Ligand source activities (1 row/activity)





Ligands (move mouse cursor over ligand name to see structure) Receptor Activity Chemical information
Sel. page Common
name
GPCRdb
ID
Reference
ligand
Vendors

Species

Assay
Type

Activity
Type
Activity
Relation
Activity
Value
p-value
(-log)
Fold
selectivity
Tested
GPCRs
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI

1001 620 None 48 Mouse Functional pEC50 = 6 6.0 -11 4
UnclassifiedUnclassified
Guide to Pharmacology 121 2 1 1 1.2 NCCc1ccccc1 16878137
2144 620 None 48 Mouse Functional pEC50 = 6 6.0 -11 4
UnclassifiedUnclassified
Guide to Pharmacology 121 2 1 1 1.2 NCCc1ccccc1 16878137
CHEMBL610 620 None 48 Mouse Functional pEC50 = 6 6.0 -11 4
UnclassifiedUnclassified
Guide to Pharmacology 121 2 1 1 1.2 NCCc1ccccc1 16878137
DB04325 620 None 48 Mouse Functional pEC50 = 6 6.0 -11 4
UnclassifiedUnclassified
Guide to Pharmacology 121 2 1 1 1.2 NCCc1ccccc1 16878137




Ligands (move mouse cursor over ligand name to see structure) Receptor Activity Chemical information
Sel. page Common
name
GPCRdb
ID
Reference
ligand
Vendors

Species

Assay
Type
Activity
Type
Activity
Relation
Activity
Value
p-value
(-log)
Fold
selectivity
Tested
GPCRs
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI