MC2 receptor (q7zsx7_takru)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC2 receptor

GENE

MC2R

ORGANISM

Japanese pufferfish (Takifugu rubripes)

ALT. NAMES

Melanocortin 2 receptor

SOURCE

TREMBL

SEQUENCE

N-term        
M
N
A
T
T
V
N
R
S
D
10
            TM1  
C
P
E
V
N
V
P
I
H
V
20
                   
F
F
T
I
G
F
V
S
L
L
30
                   
E
N
L
L
V
I
G
A
I
S
40
    ICL1 TM2  
W
N
R
N
L
H
S
P
M
Y
50
                   
C
F
I
G
S
L
A
A
F
N
60
                   
T
V
A
S
V
T
K
T
W
E
70
                   
N
L
M
I
T
F
A
E
V
G
80
ECL1   TM3    
H
L
R
K
V
G
F
S
E
R
90
                   
K
A
D
D
V
V
D
S
L
L
100
                   
C
M
S
F
L
G
S
I
F
S
110
                   
F
L
A
I
A
V
D
R
Y
I
120
        ICL2    
T
I
F
H
A
L
R
Y
H
N
130
    TM4          
I
M
T
M
Q
R
T
G
A
I
140
                   
L
G
L
I
W
T
T
C
G
V
150
                   
S
A
M
L
M
V
R
F
F
D
160
TM5              
S
N
L
I
M
S
C
F
V
V
170
                   
F
F
I
I
S
L
A
I
I
Y
180
                   
I
L
Y
V
Y
M
F
I
L
A
190
                   
R
V
H
A
R
K
I
A
A
L
200
ICL3            
P
N
G
S
G
K
H
Q
H
Q
210
          TM6    
R
R
W
G
H
G
M
R
G
I
220
                   
L
T
L
T
I
L
F
G
A
F
230
                   
M
V
C
W
A
P
F
F
L
H
240
                   
L
I
F
L
M
A
C
P
M
N
250
TM7              
P
Y
C
E
C
Y
R
S
M
F
260
                   
Q
L
H
L
V
L
L
M
S
H
270
                   
A
L
I
D
P
V
I
Y
A
F
280
  H8              
R
I
P
E
L
R
H
T
F
R
290
                   
R
M
L
P
C
L
N
W
R
W
300
C-term
R

LINKS

DIAGRAMS

ICL1 R N L H ICL1ECL1 H L R K V ECL1ICL2 A L R Y H N I M ICL2ECL2 D ECL2ICL3 A L P N G S G K H Q H Q R R W G H ICL3ECL3 P M ECL3N-term M N A T T V N R S D C P E V N V N-termC-term N W R W R C-term P I H V F F T I G F V S L L E N L L V I G A I S W N S P M Y C F I G S L A A F N T V A S V T K T W E N L M I T F A E V G G F S E R K A D D V V D S L L C M S F L G S I F S F L A I A V D R Y I T I F H T M Q R T G A I L G L I W T T C G V S A M L M V R F F S N L I M S C F V V F F I I S L A I I Y I L Y V Y M F I L A R V H A R K I A G M R G I L T L T I L F G A F M V C W A P F F L H L I F L M A C N P Y C E C Y R S M F Q L H L V L L M S H A L I D P V I Y A F R I P E F R R L L R H T M L P C
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

L N E L L S V F G I T F F V H I P 1 G S L A A F N T V A S V T K T W E N L M 2 A L F S F I S G L F S M C L L S D V V D 3 T G A I L G L I W T T C G V S A M L M V 4 Y L I Y I I A L S I I F F V V F C S M I 5 T I L F G A F M V C W A P F F L H L I F 6 V P D I L A H S M L L V L H L Q F M S 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

MUTATIONS

ENDOGENOUS LIGANDS

No endogenous ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available