Receptor names:
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Structure coverage
Active Inactive Both



A5-HT1A5-HT1B5-HT1D5-HT1E5-HT1F5-HT2A5-HT2B5-HT2C5-HT45-HT5A5-HT65-HT7M1M2M3M4M5A1A2AA2BA3Α1AΑ1BΑ1DΑ2AΑ2BΑ2CΒ1Β2Β3AT1AT2ApelinGPBABB1BB2BB3B1B2CB1CB2ChemerinChemerin 2CCR1CCR2CCR3CCR4CCR5CCR6CCR7CCR8CCR9CCR10CXCR1CXCR2CXCR3CXCR4CXCR5CXCR6CX3CR1XCR1ACKR1ACKR2ACKR3ACKR4CCRL2CCK1CCK2C3aC5a1C5a2D1D2D3D4D5ETAETBGPERFPR1FPR2/ALXFPR3FFA1FFA2FFA3FFA4GPR42GAL1GAL2GAL3GhrelinFSHLHTSHGnRH1GPR18GPR55GPR119H1H2H3H4HCA1HCA2HCA3KisspeptinBLT1BLT2CysLT1CysLT2OXELPA1LPA2LPA3LPA4LPA5LPA6S1P1S1P2S1P3S1P4S1P5MCH1MCH2MC1MC2MC3MC4MC5MT1MT2MotilinNMU1NMU2NPFF1NPFF2NPSNPBW1NPBW2Y1Y2Y4Y5Y6NTS1NTS2ΔΚΜNOPRhodopsinOPN3OPN4OPN5OPN1SWOPN1MWOPN1LWRRHOX1OX25-HTAcetylcholineAdenosineAdrenoceptorsAngiotensinApelinBile acidBombesinBradykininCannabinoidChemerinChemokineCholecystokininComplement peptideDopamineEndothelinEstrogenFormylpeptideFree fatty acidGalaninGhrelinGlycoprotein hormoneGonadotrophin-rel. hormoneGPR18, 55 & 119HistamineHydroxycarboxylic acidKisspeptinLeukotrieneLysophospholipidLysophospholipidMelanin-conc. hormoneMelanocortinMelatoninMotilinNeuromedin UNeuropeptide FF/AFNeuropeptide SNeuropeptide W/BNeuropeptide YNeurotensinOpioidOpsinsOrexinAOxoglutarateP2Y1P2Y2P2Y4P2Y6P2Y11P2Y12P2Y13P2Y14QRFPPAFPKR1PKR2PrRPDP1DP2EP1EP2EP3EP4FPIPTPPAR1PAR2PAR3PAR4RXFP1RXFP2RXFP3RXFP4SST1SST2SST3SST4SST5SuccinateNK1NK2NK3TRH1TA1UTV1AV1BV2OTGPR3GPR4GPR6GPR12GPR15GPR17GPR19GPR20GPR21GPR22GPR25GPR26GPR27GPR31GPR32GPR33GPR34GPR35GPR37GPR37L1GPR39GPR45GPR50GPR52GPR61GPR62GPR63GPR65GPR68GPR75GPR78GPR82GPR83GPR84GPR85GPR87GPR88GPR101GPR132GPR135GPR139GPR141GPR142GPR146GPR148GPR149GPR150GPR151GPR152GPR153GPR160GPR161GPR162GPR171GPR173GPR174GPR176GPR182GPR183LGR4LGR5LGR6MAS1MAS1LMRGPRDMRGPREMRGPRFMRGPRGMRGPRX1MRGPRX2MRGPRX3MRGPRX4P2RY8P2RY10TAAR2TAAR3TAAR5TAAR6TAAR8TAAR9OxoglutarateP2YPeptide P518Platelet-activating factorProkineticinProlactin-rel. peptideProstanoidProteinase-activatedRelaxin family peptideSomatostatinSuccinateTachykininThyrotropin-rel. hormoneTrace amineUrotensinVasopressin & oxytocinClass A orphansB1CTCLRCRF1CRF2GHRHGIPGLP-1GLP-2GlucagonSecretinPTH1PTH2PAC1VPAC1VPAC2B2ADGRA1ADGRA2ADGRA3ADGRB1ADGRB2ADGRB3CELSR1CELSR2CELSR3ADGRD1ADGRD2ADGRE1ADGRE2ADGRE3ADGRE4PADGRE5ADGRF1ADGRF2ADGRF3ADGRF4ADGRF5ADGRG1ADGRG2ADGRG3ADGRG4ADGRG5ADGRG6ADGRG7ADGRL1ADGRL2ADGRL3ADGRL4ADGRV1CalcitoninCorticotropin-rel. factorGlucagon familyParathyroid hormoneVIP & PACAPADGRAADGRBADGRCADGRDADGREADGRFADGRGADGRLADGRVCCaSGPR156GPR158GPR179GPRC5AGPRC5BGPRC5CGPRC5DGPRC6GABAB1GABAB2MGlu1MGlu2MGlu3MGlu4MGlu5MGlu6MGlu7MGlu8TAS1R1TAS1R2TAS1R3FFZD1FZD2FZD3FZD4FZD5FZD6FZD7FZD8FZD9FZD10SMOCalcium-sensingOrphansGABAMetabotropic glutamateTaste 1FrizzledT2TAS2R1TAS2R3TAS2R4TAS2R5TAS2R7TAS2R8TAS2R9TAS2R10TAS2R13TAS2R14TAS2R16TAS2R19TAS2R20TAS2R30TAS2R31TAS2R38TAS2R39TAS2R40TAS2R41TAS2R42TAS2R43TAS2R45TAS2R46TAS2R50TAS2R60ClasslessGPR107GPR137TPRA1GPR143GPR157

Receptor names:
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Receptor-ligand complexes count (from low to high)



A5-HT1A5-HT1B5-HT1D5-HT1E5-HT1F5-HT2A5-HT2B5-HT2C5-HT45-HT5A5-HT65-HT7M1M2M3M4M5A1A2AA2BA3Α1AΑ1BΑ1DΑ2AΑ2BΑ2CΒ1Β2Β3AT1AT2ApelinGPBABB1BB2BB3B1B2CB1CB2ChemerinChemerin 2CCR1CCR2CCR3CCR4CCR5CCR6CCR7CCR8CCR9CCR10CXCR1CXCR2CXCR3CXCR4CXCR5CXCR6CX3CR1XCR1ACKR1ACKR2ACKR3ACKR4CCRL2CCK1CCK2C3aC5a1C5a2D1D2D3D4D5ETAETBGPERFPR1FPR2/ALXFPR3FFA1FFA2FFA3FFA4GPR42GAL1GAL2GAL3GhrelinFSHLHTSHGnRH1GPR18GPR55GPR119H1H2H3H4HCA1HCA2HCA3KisspeptinBLT1BLT2CysLT1CysLT2OXELPA1LPA2LPA3LPA4LPA5LPA6S1P1S1P2S1P3S1P4S1P5MCH1MCH2MC1MC2MC3MC4MC5MT1MT2MotilinNMU1NMU2NPFF1NPFF2NPSNPBW1NPBW2Y1Y2Y4Y5Y6NTS1NTS2ΔΚΜNOPRhodopsinOPN3OPN4OPN5OPN1SWOPN1MWOPN1LWRRHOX1OX25-HTAcetylcholineAdenosineAdrenoceptorsAngiotensinApelinBile acidBombesinBradykininCannabinoidChemerinChemokineCholecystokininComplement peptideDopamineEndothelinEstrogenFormylpeptideFree fatty acidGalaninGhrelinGlycoprotein hormoneGonadotrophin-rel. hormoneGPR18, 55 & 119HistamineHydroxycarboxylic acidKisspeptinLeukotrieneLysophospholipidLysophospholipidMelanin-conc. hormoneMelanocortinMelatoninMotilinNeuromedin UNeuropeptide FF/AFNeuropeptide SNeuropeptide W/BNeuropeptide YNeurotensinOpioidOpsinsOrexinAOxoglutarateP2Y1P2Y2P2Y4P2Y6P2Y11P2Y12P2Y13P2Y14QRFPPAFPKR1PKR2PrRPDP1DP2EP1EP2EP3EP4FPIPTPPAR1PAR2PAR3PAR4RXFP1RXFP2RXFP3RXFP4SST1SST2SST3SST4SST5SuccinateNK1NK2NK3TRH1TA1UTV1AV1BV2OTGPR3GPR4GPR6GPR12GPR15GPR17GPR19GPR20GPR21GPR22GPR25GPR26GPR27GPR31GPR32GPR33GPR34GPR35GPR37GPR37L1GPR39GPR45GPR50GPR52GPR61GPR62GPR63GPR65GPR68GPR75GPR78GPR82GPR83GPR84GPR85GPR87GPR88GPR101GPR132GPR135GPR139GPR141GPR142GPR146GPR148GPR149GPR150GPR151GPR152GPR153GPR160GPR161GPR162GPR171GPR173GPR174GPR176GPR182GPR183LGR4LGR5LGR6MAS1MAS1LMRGPRDMRGPREMRGPRFMRGPRGMRGPRX1MRGPRX2MRGPRX3MRGPRX4P2RY8P2RY10TAAR2TAAR3TAAR5TAAR6TAAR8TAAR9OxoglutarateP2YPeptide P518Platelet-activating factorProkineticinProlactin-rel. peptideProstanoidProteinase-activatedRelaxin family peptideSomatostatinSuccinateTachykininThyrotropin-rel. hormoneTrace amineUrotensinVasopressin & oxytocinClass A orphansB1CTCLRCRF1CRF2GHRHGIPGLP-1GLP-2GlucagonSecretinPTH1PTH2PAC1VPAC1VPAC2B2ADGRA1ADGRA2ADGRA3ADGRB1ADGRB2ADGRB3CELSR1CELSR2CELSR3ADGRD1ADGRD2ADGRE1ADGRE2ADGRE3ADGRE4PADGRE5ADGRF1ADGRF2ADGRF3ADGRF4ADGRF5ADGRG1ADGRG2ADGRG3ADGRG4ADGRG5ADGRG6ADGRG7ADGRL1ADGRL2ADGRL3ADGRL4ADGRV1CalcitoninCorticotropin-rel. factorGlucagon familyParathyroid hormoneVIP & PACAPADGRAADGRBADGRCADGRDADGREADGRFADGRGADGRLADGRVCCaSGPR156GPR158GPR179GPRC5AGPRC5BGPRC5CGPRC5DGPRC6GABAB1GABAB2MGlu1MGlu2MGlu3MGlu4MGlu5MGlu6MGlu7MGlu8TAS1R1TAS1R2TAS1R3FFZD1FZD2FZD3FZD4FZD5FZD6FZD7FZD8FZD9FZD10SMOCalcium-sensingOrphansGABAMetabotropic glutamateTaste 1FrizzledT2TAS2R1TAS2R3TAS2R4TAS2R5TAS2R7TAS2R8TAS2R9TAS2R10TAS2R13TAS2R14TAS2R16TAS2R19TAS2R20TAS2R30TAS2R31TAS2R38TAS2R39TAS2R40TAS2R41TAS2R42TAS2R43TAS2R45TAS2R46TAS2R50TAS2R60ClasslessGPR107GPR137TPRA1GPR143GPR157

Receptor names:
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Structures count (from low to high)



O2OR1A1OR1A2OR1B1OR1C1OR1D2OR1D4OR1D5OR1E1OR1E2OR1E3OR1F1OR1G1OR1I1OR1J1OR1J2OR1J4OR1K1OR1L1OR1L3OR1L4OR1L6OR1L8OR1M1OR1N1OR1N2OR1P1OR1Q1OR1S1OR1S2OR2A1OR2A2OR2A4OR2A5OR2A7OR2A12OR2A14OR2A25OR2AE1OR2AG1OR2AG2OR2AJ1OR2AK2OR2AP1OR2AT4OR2B2OR2B3OR2B6OR2B11OR2C1OR2C3OR2D2OR2D3OR2F1OR2F2OR2G2OR2G3OR2G6OR2H1OR2H2OR2J1OR2J2OR2J3OR2K2OR2L2OR2L3OR2L5OR2L8OR2L13OR2M2OR2M3OR2M4OR2M5OR2M7OR2S2OR2T1OR2T2OR2T3OR2T4OR2T5OR2T6OR2T7OR2T8OR2T10OR2T11OR2T12OR2T27OR2T29OR2T33OR2T34OR2T35OR2V1OR2V2OR2W1OR2W3OR2Y1OR2Z1OR3A1OR3A2OR3A3OR4A5OR4A8OR4A15OR4A16OR4A47OR4B1OR4C3OR4C5OR4C6OR4C11OR4C12OR4C13OR4C15OR4C16OR4C45OR4C46OR4D1OR4D2OR4D5OR4D6OR4D9OR4D10OR4D11OR4E1OR4E2OR4F3OR4F4OR4F5OR4F6OR4F15OR4F17OR4F21OR4K1OR4K2OR4K3OR4K5OR4K13OR4K14OR4K15OR4K17OR4L1OR4M1OR4M2OR4M2BOR4N2OR4N4OR4N4COR4N5OR4P4OR4Q2OR4Q3OR4S1OR4S2OR4X1OR4X2Family 1Family 2Family 3Family 4O2OR5A1OR5A2OR5AC1OR5AC2OR5AK2OR5AL1OR5AN1OR5AP2OR5AR1OR5AS1OR5AU1OR5B2OR5B3OR5B12OR5B17OR5B21OR5C1OR5D13OR5D14OR5D16OR5D18OR5F1OR5G3OR5H1OR5H2OR5H6OR5H8OR5H14OR5H15OR5I1OR5J2OR5K1OR5K2OR5K3OR5K4OR5L1OR5L2OR5M1OR5M3OR5M8OR5M9OR5M10OR5M11OR5P2OR5P3OR5T1OR5T2OR5T3OR5V1OR5W2OR6A2OR6B1OR6B2OR6B3OR6C1OR6C2OR6C3OR6C4OR6C6OR6C65OR6C68OR6C70OR6C74OR6C75OR6C76OR6F1OR6J1OR6K2OR6K3OR6K6OR6M1OR6N1OR6N2OR6P1OR6Q1OR6S1OR6T1OR6V1OR6X1OR6Y1OR7A5OR7A10OR7A17OR7C1OR7C2OR7D2OR7D4OR7E24OR7G1OR7G2OR7G3OR8A1OR8B2OR8B3OR8B4OR8B8OR8B12OR8D1OR8D2OR8D4OR8G1OR8G5OR8H1OR8H2OR8H3OR8I2OR8J1OR8J2OR8J3OR8K1OR8K3OR8K5OR8S1OR8U1OR8U3OR8U8OR8U9OR9A2OR9A4OR9G1OR9G4OR9G9OR9I1OR9K2OR9Q1OR9Q2Family 5Family 6Family 7Family 8Family 9O2OR10A2OR10A3OR10A4OR10A5OR10A6OR10A7OR10AC1OR10AD1OR10AG1OR10C1OR10D3OR10G2OR10G3OR10G4OR10G6OR10G7OR10G8OR10G9OR10H1OR10H2OR10H3OR10H4OR10H5OR10J1OR10J3OR10J4OR10J5OR10K1OR10K2OR10P1OR10Q1OR10R2OR10S1OR10T2OR10V1OR10W1OR10X1OR10Z1OR11A1OR11G2OR11H1OR11H2OR11H4OR11H6OR11H7OR11H12OR11L1OR12D1OR12D2OR12D3OR13A1OR13C2OR13C3OR13C4OR13C5OR13C7OR13C8OR13C9OR13D1OR13F1OR13G1OR13H1OR13J1OR14A2OR14A16OR14C36OR14I1OR14J1OR14K1OR14L1Family 10Family 11Family 12Family 13Family 14O1OR51A2OR51A4OR51A7OR51B2OR51B4OR51B5OR51B6OR51D1OR51E1OR51E2OR51F1OR51F2OR51G1OR51G2OR51H1OR51I1OR51I2OR51J1OR51L1OR51M1OR51Q1OR51S1OR51T1OR51V1OR52A1OR52A5OR52B2OR52B4OR52B6OR52D1OR52E1OR52E2OR52E4OR52E5OR52E6OR52E8OR52H1OR52I1OR52I2OR52J3OR52K1OR52K2OR52L1OR52M1OR52N1OR52N2OR52N4OR52N5OR52P1OR52R1OR52W1OR56A1OR56A3OR56A4OR56A5OR56B1OR56B4Family 51Family 52Family 56



By class By ligand type The number of unique receptors with structures available. The number of unique receptors GPCR-ligand complexes. The number of structures available. The number of unique receptors with structures. The number of unique GPCR-ligand complexes. The number of structures available.


Number of structures, including multiple of same receptor (complex)

Class
(Family)
A (Rhodopsin) B1 (Secretin) B2 (Adhesion) C (Glutamate) D1
(Ste2-like fungal pheromone)
F (Frizzled) O1 (fish-like odorant) O2 (tetrapod specific odorant) T2 (Taste 2) Other GPCRs Total
Receptors 1305 146 34 105 1 34 5 3 17 0 1650
Receptor - ligand complexes 1303 146 34 105 1 34 5 3 17 0 1648
Receptor - G protein complexes 752 121 32 18 1 11 3 3 15 0 956
Active-state receptors* 847 126 32 38 1 13 4 3 15 0 1079


Number of unique receptor complexes

Class
(Family)
A (Rhodopsin) B1 (Secretin) B2 (Adhesion) C (Glutamate) D1
(Ste2-like fungal pheromone)
F (Frizzled) O1 (fish-like odorant) O2 (tetrapod specific odorant) T2 (Taste 2) Other GPCRs Total
Receptors** 182 15 9 13 1 7 3 3 2 0 235
Receptor - ligand complexes 820 96 13 59 1 19 4 3 6 0 1021
Receptor - G protein complexes 165 15 9 5 1 5 3 3 2 0 208
Active-state receptors* 168 15 9 7 1 5 3 3 2 0 213
*Active state is defined as agonist-bound and opened intracellular TM bundle. **Receptor-orthologues are only counted once.

Specific sets of structures can be downloaded from the Structures page.
The latest released structure is from 2024-10-30.