Data showed in this table is continously collected from the Guide to Pharmacology database. Ref

RECEPTOR PHYSIOLOGICAL LIGANDS STRUCTURE pEC50 pKi REFERENCES
Class Receptor family UniProt IUPHAR Gene Species Ligand GtP
Classification
Potency
Ranking
Type Smiles Inchikey Model Exp Min Mid Max Min Mid Max
A (Rhodopsin) 5-Hydroxytryptamine 5HT1A 5-HT1A HTR1A Human 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - 7E2Y 9.1 9.4 9.7 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT1B 5-HT1B HTR1B Human 5-Ht-Moduline None 3 Peptide OC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(C)C)C)NC(=O)[C@H](CC(C)C)N IMIVWAUMTAIVPJ-XUXIUFHCSA-N - -
A (Rhodopsin) 5-Hydroxytryptamine 5HT1B 5-HT1B HTR1B Human 5-Hydroxytryptamine None 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 7.4 8.1 8.1 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT1B 5-HT1B HTR1B Human Tryptamine None 2 Small molecule NCCc1c[nH]c2c1cccc2 APJYDQYYACXCRM-UHFFFAOYSA-N - - 6.3 6.3 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT1B 5-HT1B Htr1b Mouse 5-Hydroxytryptamine None 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 7.4 8.1 8.1 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT1D 5-HT1D HTR1D Human 5-Ht-Moduline None 2 Peptide OC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(C)C)C)NC(=O)[C@H](CC(C)C)N IMIVWAUMTAIVPJ-XUXIUFHCSA-N - - Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT1D 5-HT1D HTR1D Human 5-Hydroxytryptamine None 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - 7E32 8.0 8.5 9.0 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT1E 5-HT1E HTR1E Human 5-Hydroxytryptamine None 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 8.0 8.1 8.2 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT1E 5-HT1E HTR1E Human Tryptamine None 2 Small molecule NCCc1c[nH]c2c1cccc2 APJYDQYYACXCRM-UHFFFAOYSA-N - - 5.6 6.1 6.5 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT1F 5-HT1F HTR1F Human 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 7.7 7.9 8.0 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT1F 5-HT1F Htr1f Rat 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 7.7 7.9 8.0 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT2A 5-HT2A HTR2A Human 5-Hydroxytryptamine None 2 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - 9ARY 6.0 6.3 6.5 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT2A 5-HT2A HTR2A Human Tryptamine None 1 Small molecule NCCc1c[nH]c2c1cccc2 APJYDQYYACXCRM-UHFFFAOYSA-N - - 5.5 7.1 7.1 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT2A 5-HT2A Htr2a Rat 5-Hydroxytryptamine None 2 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 6.0 6.3 6.5 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT2A 5-HT2A Htr2a Rat Tryptamine None 1 Small molecule NCCc1c[nH]c2c1cccc2 APJYDQYYACXCRM-UHFFFAOYSA-N - - 5.5 7.1 7.1 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT2B 5-HT2B HTR2B Human 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 7.9 8.0 8.0 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT2B 5-HT2B Htr2b Rat 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 7.9 8.0 8.0 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT2C 5-HT2C HTR2C Human 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 6.7 7.3 7.9 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT2C 5-HT2C Htr2c Rat 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 6.7 7.3 7.9 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT4R 5-HT4 HTR4 Human 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - 7XTA 6.7 7.5 8.2 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT4R 5-HT4 Htr4 Mouse 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 6.7 7.5 8.2 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT4R 5-HT4 Htr4 Rat 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 6.7 7.5 8.2 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT5A 5-HT5A HTR5A Human 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 6.0 6.6 6.6 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT5A 5-HT5A Htr5a Mouse 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 6.0 6.6 6.6 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT5A 5-HT5A Htr5a Rat 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 6.0 6.6 6.6 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT5B Htr5b Htr5b Mouse 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - -
A (Rhodopsin) 5-Hydroxytryptamine 5HT6R 5-HT6 HTR6 Human 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - 7XTB 6.6 7.3 7.9 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT6R 5-HT6 Htr6 Rat 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 6.6 7.3 7.9 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT7R 5-HT7 HTR7 Human 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 8.7 9.0 9.2 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT7R 5-HT7 Htr7 Mouse 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 8.7 9.0 9.2 Refs
A (Rhodopsin) 5-Hydroxytryptamine 5HT7R 5-HT7 Htr7 Rat 5-Hydroxytryptamine Principal 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 8.7 9.0 9.2 Refs
A (Rhodopsin) Acetylcholine receptors (muscarinic) ACM1 M1 CHRM1 Human Acetylcholine Principal 1 Small molecule CC(=O)OCC[N+](C)(C)C OIPILFWXSMYKGL-UHFFFAOYSA-N - B2M_ACM1_HUMAN_ACETYLCHOLINE_GNA11_HUMAN 4.3 5.0 5.0 Refs
A (Rhodopsin) Acetylcholine receptors (muscarinic) ACM1 M1 Chrm1 Rat Acetylcholine Principal 1 Small molecule CC(=O)OCC[N+](C)(C)C OIPILFWXSMYKGL-UHFFFAOYSA-N - - 4.3 5.0 5.0 Refs
A (Rhodopsin) Acetylcholine receptors (muscarinic) ACM2 M2 CHRM2 Human Acetylcholine Principal 1 Small molecule CC(=O)OCC[N+](C)(C)C OIPILFWXSMYKGL-UHFFFAOYSA-N - 7T90 4.3 6.4 6.4 Refs
A (Rhodopsin) Acetylcholine receptors (muscarinic) ACM2 M2 Chrm2 Rat Acetylcholine Principal 1 Small molecule CC(=O)OCC[N+](C)(C)C OIPILFWXSMYKGL-UHFFFAOYSA-N - - 4.3 6.4 6.4 Refs
A (Rhodopsin) Acetylcholine receptors (muscarinic) ACM3 M3 CHRM3 Human Acetylcholine Principal 1 Small molecule CC(=O)OCC[N+](C)(C)C OIPILFWXSMYKGL-UHFFFAOYSA-N - B2M_ACM3_HUMAN_ACETYLCHOLINE_GNAQ_HUMAN 4.5 5.6 5.6 Refs
A (Rhodopsin) Acetylcholine receptors (muscarinic) ACM3 M3 Chrm3 Rat Acetylcholine Principal 1 Small molecule CC(=O)OCC[N+](C)(C)C OIPILFWXSMYKGL-UHFFFAOYSA-N - - 4.5 5.6 5.6 Refs
A (Rhodopsin) Acetylcholine receptors (muscarinic) ACM4 M4 CHRM4 Human Acetylcholine Principal 1 Small molecule CC(=O)OCC[N+](C)(C)C OIPILFWXSMYKGL-UHFFFAOYSA-N - 7TRS 4.5 5.1 5.6 Refs
A (Rhodopsin) Acetylcholine receptors (muscarinic) ACM5 M5 CHRM5 Human Acetylcholine Principal 1 Small molecule CC(=O)OCC[N+](C)(C)C OIPILFWXSMYKGL-UHFFFAOYSA-N - 9EJZ 6.1 6.1 Refs
A (Rhodopsin) Adenosine AA1R A1 ADORA1 Human Adenosine Principal 1 Small molecule OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N OIRDTQYFTABQOQ-KQYNXXCUSA-N - 6D9H 7.1 7.1 Refs
A (Rhodopsin) Adenosine AA1R A1 Adora1 Rat Adenosine Principal 1 Small molecule OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N OIRDTQYFTABQOQ-KQYNXXCUSA-N - - 7.1 7.1 Refs
A (Rhodopsin) Adenosine AA2AR A2A ADORA2A Human Adenosine Principal 1 Small molecule OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N OIRDTQYFTABQOQ-KQYNXXCUSA-N - 9EEA 6.5 6.5 Refs
A (Rhodopsin) Adenosine AA2BR A2B ADORA2B Human Adenosine Principal 1 Small molecule OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N OIRDTQYFTABQOQ-KQYNXXCUSA-N - 8HDP 5.3 5.3 Refs
A (Rhodopsin) Adenosine AA2BR A2B Adora2b Rat Adenosine Principal 1 Small molecule OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N OIRDTQYFTABQOQ-KQYNXXCUSA-N - - 5.3 5.3 Refs
A (Rhodopsin) Adenosine AA3R A3 ADORA3 Human Adenosine Principal 1 Small molecule OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N OIRDTQYFTABQOQ-KQYNXXCUSA-N - 9EBH 5.2 5.2 Refs
A (Rhodopsin) Adenosine AA3R A3 Adora3 Rat Adenosine Principal 1 Small molecule OC[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N OIRDTQYFTABQOQ-KQYNXXCUSA-N - - 5.2 5.2 Refs
A (Rhodopsin) Adren ADA1A α1A ADRA1A Human (-)-Adrenaline None 1 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - 8THL 9.1 9.1 5.1 5.8 6.5 Refs
A (Rhodopsin) Adren ADA1A α1A ADRA1A Human (-)-Noradrenaline None 2 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - 7YMH 7.7 8.2 8.6 4.8 5.6 6.4 Refs
A (Rhodopsin) Adren ADA1B α1B ADRA1B Human (-)-Adrenaline None 1 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - 9.4 9.4 3.9 5.2 6.5 Refs
A (Rhodopsin) Adren ADA1B α1B ADRA1B Human (-)-Noradrenaline None 2 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - 9.2 9.2 3.8 5.0 6.2 Refs
A (Rhodopsin) Adren ADA1D α1D ADRA1D Human (-)-Adrenaline None 2 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - 7.7 7.7 5.3 6.3 6.3 Refs
A (Rhodopsin) Adren ADA1D α1D ADRA1D Human (-)-Noradrenaline None 1 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - 7.8 7.8 5.5 6.3 6.3 Refs
A (Rhodopsin) Adren ADA1D α1D Adra1d Rat (-)-Adrenaline None 2 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - - 7.7 7.7 5.3 6.3 6.3 Refs
A (Rhodopsin) Adren ADA1D α1D Adra1d Rat (-)-Noradrenaline None 1 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - - 7.8 7.8 5.5 6.3 6.3 Refs
A (Rhodopsin) Adren ADA2A α2A ADRA2A Human (-)-Adrenaline None 1 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - 9CBL 5.5 6.8 8.0 3.7 5.6 7.4 Refs
A (Rhodopsin) Adren ADA2A α2A ADRA2A Human (-)-Noradrenaline None 2 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - 7EJ0 5.3 6.6 7.7 3.6 5.5 7.4 Refs
A (Rhodopsin) Adren ADA2B α2B ADRA2B Human (-)-Adrenaline None 2 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - 6.3 6.9 7.5 3.6 4.4 5.2 Refs
A (Rhodopsin) Adren ADA2B α2B ADRA2B Human (-)-Noradrenaline None 1 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - 6.9 7.4 7.8 3.5 4.8 6.0 Refs
A (Rhodopsin) Adren ADA2C α2C ADRA2C Human (-)-Adrenaline None 1 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - 7.6 7.6 4.9 5.4 5.8 Refs
A (Rhodopsin) Adren ADA2C α2C ADRA2C Human (-)-Noradrenaline None 2 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - 6.0 6.8 7.7 4.5 5.7 6.8 Refs
A (Rhodopsin) Adren ADRB1 β1 ADRB1 Human (-)-Adrenaline None 2 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - 9L84 7.6 7.6 5.2 5.6 6.0 Refs
A (Rhodopsin) Adren ADRB1 β1 ADRB1 Human (-)-Noradrenaline None 1 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - 7BU6 7.9 7.9 5.5 5.8 6.0 Refs
A (Rhodopsin) Adren ADRB1 β1 ADRB1 Human Noradrenaline None 3 Small molecule NCC(c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-UHFFFAOYSA-N - - 6.0 6.0 Refs
A (Rhodopsin) Adren ADRB2 β2 ADRB2 Human (-)-Adrenaline None 1 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - 4LDO 7.9 7.9 6.0 6.1 6.2 Refs
A (Rhodopsin) Adren ADRB2 β2 ADRB2 Human (-)-Noradrenaline None 2 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - 9CHU 6.4 6.4 4.6 5.0 5.4 Refs
A (Rhodopsin) Adren ADRB2 β2 ADRB2 Human Zn2+ None 3 Small molecule - - - - 3.3 4.3 5.3 Refs
A (Rhodopsin) Adren ADRB2 β2 ADRB2 Human Noradrenaline None 3 Small molecule NCC(c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-UHFFFAOYSA-N - - 5.4 5.4 Refs
A (Rhodopsin) Adren ADRB3 β3 ADRB3 Human (&Plusmn;)-Adrenaline None 3 Small molecule CNCC(c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-UHFFFAOYSA-N - B2M_ADRB3_HUMAN_RACEPINEPHRINE_GNAS2_HUMAN 3.9 5.3 5.3 Refs
A (Rhodopsin) Adren ADRB3 β3 ADRB3 Human (-)-Adrenaline None 2 Small molecule CNC[C@@H](c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-VIFPVBQESA-N - 9IJE 6.5 6.5 3.9 4.3 4.7 Refs
A (Rhodopsin) Adren ADRB3 β3 ADRB3 Human (-)-Noradrenaline None 1 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - 7.2 7.2 4.7 4.2 4.2 Refs
A (Rhodopsin) Adren ADRB3 β3 Adrb3 Mouse (&Plusmn;)-Adrenaline None 3 Small molecule CNCC(c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-UHFFFAOYSA-N - - 3.9 5.3 5.3 Refs
A (Rhodopsin) Adren ADRB3 β3 Adrb3 Mouse (-)-Noradrenaline None 1 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - - 7.2 7.2 4.7 4.2 4.2 Refs
A (Rhodopsin) Adren ADRB3 β3 Adrb3 Rat (&Plusmn;)-Adrenaline None 3 Small molecule CNCC(c1ccc(c(c1)O)O)O UCTWMZQNUQWSLP-UHFFFAOYSA-N - - 3.9 5.3 5.3 Refs
A (Rhodopsin) Adren ADRB3 β3 Adrb3 Rat (-)-Noradrenaline None 1 Small molecule NC[C@@H](c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-QMMMGPOBSA-N - - 7.2 7.2 4.7 4.2 4.2 Refs
A (Rhodopsin) Angiotensin AGTR1 AT1 AGTR1 Human Angiotensin A (Human) 1 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)N)C(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)O CHCOFDZSJYMQMX-NOQNJSOHSA-N - 8.2 8.2 8.8 8.8 Refs
A (Rhodopsin) Angiotensin AGTR1 AT1 AGTR1 Human Angiotensin Ii (Human) 3 Peptide CC[C@@H]([C@@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)O)Cc1ccccc1)Cc1nc[nH]c1)NC(=O)[C@@H](NC(=O)[C@H](C(C)C)NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)N)CCCN=C(N)N)Cc1ccc(cc1)O)C CZGUSIXMZVURDU-JZXHSEFVSA-N - 6OS0
A (Rhodopsin) Angiotensin AGTR1 AT1 AGTR1 Human Angiotensin Iii (Human) 3 Peptide NC(=NCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)O)Cc1[nH]cnc1)C(C)C)Cc1ccc(cc1)O)C(C)C)NC(=O)[C@H](CC(=O)O)N)N UCRMCWFIVZYPFA-LGXQCQDRSA-N -
A (Rhodopsin) Angiotensin AGTR1 AT1 AGTR1 Human Angiotensin Iv (Human) 2 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](N)C(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)O QSBGWDDCOJYQGY-KOQODJNWSA-N - 5.9 5.9 Refs
A (Rhodopsin) Angiotensin AGTR2 AT2 AGTR2 Human Angiotensin Ii (Human) 2 Peptide CC[C@@H]([C@@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)O)Cc1ccccc1)Cc1nc[nH]c1)NC(=O)[C@@H](NC(=O)[C@H](C(C)C)NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)N)CCCN=C(N)N)Cc1ccc(cc1)O)C CZGUSIXMZVURDU-JZXHSEFVSA-N - 6JOD
A (Rhodopsin) Angiotensin AGTR2 AT2 AGTR2 Human Angiotensin Iii (Human) 1 Peptide NC(=NCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)O)Cc1[nH]cnc1)C(C)C)Cc1ccc(cc1)O)C(C)C)NC(=O)[C@H](CC(=O)O)N)N UCRMCWFIVZYPFA-LGXQCQDRSA-N - Refs
A (Rhodopsin) Angiotensin AGTR2 AT2 AGTR2 Human Angiotensin-(1-7) (Human) 3 Peptide CC[C@@H]([C@@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)O)Cc1[nH]cnc1)NC(=O)[C@@H](NC(=O)[C@H](C(C)C)NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)N)CCCN=C(N)N)Cc1ccc(cc1)O)C PVHLMTREZMEJCG-GDTLVBQBSA-N - Refs
A (Rhodopsin) Apelin APJ apelin APLNR Human Elabela/Toddler-11 (Human) 2 Peptide CSCC[C@H](NC(=O)[C@@H](N)CS)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCC[C@H]1C(=O)O)C(C)C XXKPNJFJXZBRMX-HDKAIKTRSA-N -
A (Rhodopsin) Apelin APJ apelin APLNR Human Elabela/Toddler-21 (Human) 2 Peptide CSCC[C@H](NC(=O)[C@H](CS)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CS)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H](N)CC(C)C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)N1CCC[C@H]1C(=O)O)C(C)C TXSAAXFWNUKYQL-FMGZCOAKSA-N -
A (Rhodopsin) Apelin APJ apelin APLNR Human Elabela/Toddler-32 (Human) 2 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)O)Cc1ccccc1)C(C)C)CCCN=C(N)N)CO)Cc1nc[nH]c1)CC(C)C)CCSC)CS)CCCN=C(N)N)CCCN=C(N)N)CCC(=O)N)CC(C)C)CS)CC(=O)N)Cc1nc[nH]c1)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(=O)N)N)CCCN=C(N)N)CC(=O)N)CC(C)C)CCSC)CCCN=C(N)N)CCCN=C(N)N)CCCCN)CC(C)C)CCCN=C(N)N AXGBCVTUKUUUPN-PXWSXZDTSA-N - 7W0O
A (Rhodopsin) Apelin APJ apelin APLNR Human [Pyr1]Apelin-13 (Human) 2 Peptide - - - - Refs
A (Rhodopsin) Apelin APJ apelin APLNR Human Apelin Receptor Early Endogenous Ligand (Human) 1 Peptide - - - Refs
A (Rhodopsin) Apelin APJ apelin APLNR Human Apelin Receptor Early Endogenous Ligand (Mouse) 2 Peptide - - -
A (Rhodopsin) Apelin APJ apelin APLNR Human Apelin-13 (Human) 2 Peptide NCCCC[C@@H](C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)O)Cc1ccccc1)CCSC)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(=O)N)N)CCCN=C(N)N)CCCN=C(N)N)CC(C)C)CO XXCCRHIAIBQDPX-PEWBXTNBSA-N - 8XQE Refs
A (Rhodopsin) Apelin APJ apelin APLNR Human Apelin-17 (Human) 2 Protein CSCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](N)CCCCN)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)O SVWSKJCJNAIKNH-MJZUAXFLSA-N - Refs
A (Rhodopsin) Apelin APJ apelin APLNR Human Apelin-36 (Human) 2 Peptide CSCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)CNC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CO)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@@H](N)CC(C)C)C(C)C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)O BVTLGARMSLXAHI-VDEROMQGSA-N - Refs
A (Rhodopsin) Apelin APJ apelin APLNR Human Apelin-36 (Mouse) 2 Peptide CSCC[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)CNC(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](N)CC(C)C)C(C)C)[C@@H](C)O)[C@@H](C)O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)O NRXGOOSANFUBIE-ZINMNJNTSA-N -
A (Rhodopsin) Bile acid GPBAR GPBA GPBAR1 Human Chenodeoxycholic Acid None 3 Small molecule O[C@@H]1CC[C@]2([C@@H](C1)C[C@H]([C@@H]1[C@@H]2CC[C@]2([C@H]1CC[C@@H]2[C@@H](CCC(=O)O)C)C)O)C RUDATBOHQWOJDD-BSWAIDMHSA-N - - 5.4 5.4 Refs
A (Rhodopsin) Bile acid GPBAR GPBA GPBAR1 Human Cholic Acid None 4 Small molecule O[C@@H]1CC[C@]2([C@@H](C1)C[C@H]([C@@H]1[C@@H]2C[C@H](O)[C@]2([C@H]1CC[C@@H]2[C@@H](CCC(=O)O)C)C)O)C BHQCQFFYRZLCQQ-OELDTZBJSA-N - - 5.0 5.0 Refs
A (Rhodopsin) Bile acid GPBAR GPBA GPBAR1 Human Deoxycholic Acid None 2 Small molecule O[C@@H]1CC[C@]2([C@@H](C1)CC[C@@H]1[C@@H]2C[C@H](O)[C@]2([C@H]1CC[C@@H]2[C@@H](CCC(=O)O)C)C)C KXGVEGMKQFWNSR-LLQZFEROSA-N - - 6.2 6.2 Refs
A (Rhodopsin) Bile acid GPBAR GPBA GPBAR1 Human Lithocholic Acid None 1 Small molecule O[C@@H]1CC[C@]2([C@@H](C1)CC[C@@H]1[C@@H]2CC[C@]2([C@H]1CC[C@@H]2[C@@H](CCC(=O)O)C)C)C SMEROWZSTRWXGI-HVATVPOCSA-N - - 7.5 7.5 Refs
A (Rhodopsin) Bombesin GRPR BB2 GRPR Human Grp-(18-27) (Human) 3 Peptide - - -
A (Rhodopsin) Bombesin GRPR BB2 GRPR Human Grp-(18-27) (Mouse) 3 Peptide - - -
A (Rhodopsin) Bombesin GRPR BB2 GRPR Human Gastrin Releasing Peptide(14-27) (Human) (Human) 3 Peptide CSCC[C@H](N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)N[C@H](C(=O)NCC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCSC)C(=O)O)C(C)C MJHJYGACUDLDMG-QEJDUTAOSA-N - Refs
A (Rhodopsin) Bombesin GRPR BB2 GRPR Human Gastrin-Releasing Peptide (Human) 1 Protein - - - 6.3 7.3 8.2 Refs
A (Rhodopsin) Bombesin GRPR BB2 GRPR Human Neuromedin B (Human) 2 Peptide CSCCC(C(=O)N)NC(=O)C(NC(=O)C(Cc1[nH]cnc1)NC(=O)CNC(=O)C(C(O)C)NC(=O)C(NC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C(NC(=O)CN)CC(=O)N)CC(C)C)C)Cc1ccccc1 YPFNACALNKVZNK-UHFFFAOYSA-N - 6.6 6.6 6.6 Refs
A (Rhodopsin) Bombesin GRPR BB2 GRPR Human Neuromedin C (Human) 3 Peptide - - - - Refs
A (Rhodopsin) Bombesin GRPR BB2 Grpr Mouse Neuromedin B (Human) 2 Peptide CSCCC(C(=O)N)NC(=O)C(NC(=O)C(Cc1[nH]cnc1)NC(=O)CNC(=O)C(C(O)C)NC(=O)C(NC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C(NC(=O)CN)CC(=O)N)CC(C)C)C)Cc1ccccc1 YPFNACALNKVZNK-UHFFFAOYSA-N - - 6.6 6.6 6.6 Refs
A (Rhodopsin) Bombesin GRPR BB2 Grpr Rat Neuromedin B (Human) 2 Peptide CSCCC(C(=O)N)NC(=O)C(NC(=O)C(Cc1[nH]cnc1)NC(=O)CNC(=O)C(C(O)C)NC(=O)C(NC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C(NC(=O)CN)CC(=O)N)CC(C)C)C)Cc1ccccc1 YPFNACALNKVZNK-UHFFFAOYSA-N - - 6.6 6.6 6.6 Refs
A (Rhodopsin) Bombesin NMBR BB1 NMBR Human Grp-(18-27) (Human) 2 Peptide - - -
A (Rhodopsin) Bombesin NMBR BB1 NMBR Human Grp-(18-27) (Mouse) 2 Peptide - - -
A (Rhodopsin) Bombesin NMBR BB1 NMBR Human Gastrin Releasing Peptide(14-27) (Human) (Human) 2 Peptide CSCC[C@H](N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](C)C(=O)N[C@H](C(=O)NCC(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCSC)C(=O)O)C(C)C MJHJYGACUDLDMG-QEJDUTAOSA-N - Refs
A (Rhodopsin) Bombesin NMBR BB1 NMBR Human Gastrin-Releasing Peptide (Human) 2 Protein - - -
A (Rhodopsin) Bombesin NMBR BB1 NMBR Human Gastrin-Releasing Peptide (Mouse) 2 Peptide - - -
A (Rhodopsin) Bombesin NMBR BB1 NMBR Human Gastrin-Releasing Peptide (Pig) 2 Peptide - - -
A (Rhodopsin) Bombesin NMBR BB1 NMBR Human Neuromedin B (Human) 1 Peptide CSCCC(C(=O)N)NC(=O)C(NC(=O)C(Cc1[nH]cnc1)NC(=O)CNC(=O)C(C(O)C)NC(=O)C(NC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C(NC(=O)CN)CC(=O)N)CC(C)C)C)Cc1ccccc1 YPFNACALNKVZNK-UHFFFAOYSA-N - 8.1 9.2 10.3 Refs
A (Rhodopsin) Bradykinin BKRB1 B1 BDKRB1 Human Lys-[Hyp3]-Bradykinin (Human) 6 Peptide - - - -
A (Rhodopsin) Bradykinin BKRB1 B1 BDKRB1 Human T-Kinin (Human) 5 Peptide OC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](CC)C)N)CO)CCCN=C(N)N GKCWYHPGFSRBQV-WRBAKOPXSA-N - 5.0 5.1 5.2 Refs
A (Rhodopsin) Bradykinin BKRB1 B1 BDKRB1 Human [Hyp3]Bradykinin (Human) 6 Peptide - - - -
A (Rhodopsin) Bradykinin BKRB1 B1 BDKRB1 Human [Des-Arg10]Kallidin (Human) 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)O)Cc1ccccc1)CO)Cc1ccccc1)CCCN=C(N)N)N AILVBOHFGXNHCC-TZPCGENMSA-N - 7EIB 9.6 9.8 10.0 Refs
A (Rhodopsin) Bradykinin BKRB1 B1 BDKRB1 Human [Des-Arg9]Bradykinin (Human) 2 Peptide OCC(C(=O)N1CCCC1C(=O)NC(C(=O)O)Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)CNC(=O)C1CCCN1C(=O)C1CCCN1C(=O)C(CCCN=C(N)N)N VCEHWDBVPZFHAG-UHFFFAOYSA-N - 5.7 9.2 9.2 Refs
A (Rhodopsin) Bradykinin BKRB1 B1 BDKRB1 Human Bradykinin (Human) 4 Peptide OC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)N QXZGBUJJYSLZLT-FDISYFBBSA-N - 5.1 5.2 5.3 Refs
A (Rhodopsin) Bradykinin BKRB1 B1 BDKRB1 Human Kallidin (Human) 3 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)CO)Cc1ccccc1)CCCN=C(N)N)N FYSKZKQBTVLYEQ-FSLKYBNLSA-N - 7.0 8.0 8.9 Refs
A (Rhodopsin) Bradykinin BKRB1 B1 Bdkrb1 Mouse [Des-Arg9]Bradykinin (Human) 2 Peptide OCC(C(=O)N1CCCC1C(=O)NC(C(=O)O)Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)CNC(=O)C1CCCN1C(=O)C1CCCN1C(=O)C(CCCN=C(N)N)N VCEHWDBVPZFHAG-UHFFFAOYSA-N - - 5.7 9.2 9.2 Refs
A (Rhodopsin) Bradykinin BKRB1 B1 Bdkrb1 Mouse Bradykinin (Human) 4 Peptide OC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)N QXZGBUJJYSLZLT-FDISYFBBSA-N - - 5.1 5.2 5.3 Refs
A (Rhodopsin) Bradykinin BKRB1 B1 Bdkrb1 Rat T-Kinin (Human) 5 Peptide OC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](CC)C)N)CO)CCCN=C(N)N GKCWYHPGFSRBQV-WRBAKOPXSA-N - - 5.0 5.1 5.2 Refs
A (Rhodopsin) Bradykinin BKRB1 B1 Bdkrb1 Rat Bradykinin (Human) 4 Peptide OC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)N QXZGBUJJYSLZLT-FDISYFBBSA-N - - 5.1 5.2 5.3 Refs
A (Rhodopsin) Bradykinin BKRB2 B2 BDKRB2 Human Lys-[Hyp3]-Bradykinin (Human) 3 Peptide - - - -
A (Rhodopsin) Bradykinin BKRB2 B2 BDKRB2 Human T-Kinin (Human) 3 Peptide OC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](CC)C)N)CO)CCCN=C(N)N GKCWYHPGFSRBQV-WRBAKOPXSA-N -
A (Rhodopsin) Bradykinin BKRB2 B2 BDKRB2 Human [Hyp3]Bradykinin (Human) 3 Peptide - - - -
A (Rhodopsin) Bradykinin BKRB2 B2 BDKRB2 Human [Des-Arg10]Kallidin (Human) 3 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)O)Cc1ccccc1)CO)Cc1ccccc1)CCCN=C(N)N)N AILVBOHFGXNHCC-TZPCGENMSA-N - -
A (Rhodopsin) Bradykinin BKRB2 B2 BDKRB2 Human [Des-Arg9]Bradykinin (Human) 2 Peptide OCC(C(=O)N1CCCC1C(=O)NC(C(=O)O)Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)CNC(=O)C1CCCN1C(=O)C1CCCN1C(=O)C(CCCN=C(N)N)N VCEHWDBVPZFHAG-UHFFFAOYSA-N - Refs
A (Rhodopsin) Bradykinin BKRB2 B2 BDKRB2 Human Bradykinin (Human) 1 Peptide OC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)N QXZGBUJJYSLZLT-FDISYFBBSA-N - 7F2O Refs
A (Rhodopsin) Bradykinin BKRB2 B2 BDKRB2 Human Kallidin (Human) 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)CO)Cc1ccccc1)CCCN=C(N)N)N FYSKZKQBTVLYEQ-FSLKYBNLSA-N - 7F6I Refs
A (Rhodopsin) Bradykinin BKRB2 B2 Bdkrb2 Mouse [Des-Arg9]Bradykinin (Human) 2 Peptide OCC(C(=O)N1CCCC1C(=O)NC(C(=O)O)Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)CNC(=O)C1CCCN1C(=O)C1CCCN1C(=O)C(CCCN=C(N)N)N VCEHWDBVPZFHAG-UHFFFAOYSA-N - - Refs
A (Rhodopsin) Bradykinin BKRB2 B2 Bdkrb2 Mouse Bradykinin (Human) 1 Peptide OC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCCN=C(N)N)Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)N QXZGBUJJYSLZLT-FDISYFBBSA-N - - Refs
A (Rhodopsin) Cannabinoid CNR1 CB1 CNR1 Human 2-Arachidonoylglycerol None 1 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)OC(CO)CO RCRCTBLIHCHWDZ-DOFZRALJSA-N - -
A (Rhodopsin) Cannabinoid CNR1 CB1 CNR1 Human Anandamide None 2 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCCO LGEQQWMQCRIYKG-DOFZRALJSA-N - - 6.3 6.7 7.0 Refs
A (Rhodopsin) Cannabinoid CNR1 CB1 Cnr1 Rat 2-Arachidonoylglycerol None 1 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)OC(CO)CO RCRCTBLIHCHWDZ-DOFZRALJSA-N - - 6.3 6.8 7.2 Refs
A (Rhodopsin) Cannabinoid CNR2 CB2 CNR2 Human 2-Arachidonoylglycerol None 1 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)OC(CO)CO RCRCTBLIHCHWDZ-DOFZRALJSA-N - - 5.8 6.3 6.8 Refs
A (Rhodopsin) Cannabinoid CNR2 CB2 CNR2 Human Anandamide None 2 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCCO LGEQQWMQCRIYKG-DOFZRALJSA-N - - 5.7 6.1 6.4 Refs
A (Rhodopsin) Chemerin CML1 chemerin CMKLR1 Human 18r-Hepe 2 Small molecule CC[C@H](/C=C/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)O)O LRWYBGFSVUBWMO-UAAZXLHOSA-N - -
A (Rhodopsin) Chemerin CML1 chemerin CMKLR1 Human Epa 2 Small molecule CC/C=C\C/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)O JAZBEHYOTPTENJ-JLNKQSITSA-N - -
A (Rhodopsin) Chemerin CML1 chemerin CMKLR1 Human Chemerin (Human) 1 Peptide - - - 7.6 8.0 8.5 Refs
A (Rhodopsin) Chemerin CML1 chemerin CMKLR1 Human Resolvin E1 None 2 Small molecule CC[C@H](/C=C/C=C\C[C@H](/C=C/C=C/C=C\[C@H](CCCC(=O)O)O)O)O AOPOCGPBAIARAV-OTBJXLELSA-N - - Refs
A (Rhodopsin) Chemerin CML2 chemerin 2 CMKLR2 Human Chemerin (Human) Principal 1 Peptide - - - - 8.8 9.2 9.6 Refs
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Ccl11 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Ccl14 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Ccl17 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Ccl2 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Ccl5 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Ccl7 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Cxcl11 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Cxcl5 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Cxcl6 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR1 ACKR1 ACKR1 Human Cxcl8 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl11 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl13 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl14 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl17 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl2 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl22 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl3 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl4 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl5 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl7 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR2 ACKR2 ACKR2 Human Ccl8 (Human) Peptide - - - -
A (Rhodopsin) Chemokine ACKR3 ACKR3 ACKR3 Human Cxcl11 (Human) 3 Peptide - - - -
A (Rhodopsin) Chemokine ACKR3 ACKR3 ACKR3 Human Cxcl12Α (Human) 1 Peptide - - - - 7.5 7.7 7.9 Refs
A (Rhodopsin) Chemokine ACKR3 ACKR3 Ackr3 Rat Adrenomedullin (Rat) 2 Peptide - - - - 7.0 7.0 Refs
A (Rhodopsin) Chemokine ACKR4 ACKR4 ACKR4 Human Ccl19 (Human) 1 Peptide - - - - 8.5 8.8 9.1 8.4 8.4 Refs
A (Rhodopsin) Chemokine ACKR4 ACKR4 ACKR4 Human Ccl21 (Human) 2 Peptide - - - - 7.9 8.2 8.5 6.9 6.9 Refs
A (Rhodopsin) Chemokine ACKR4 ACKR4 ACKR4 Human Ccl25 (Human) 3 Peptide - - - - 7.9 8.1 8.3 7.6 7.6 Refs
A (Rhodopsin) Chemokine CCR10 CCR10 CCR10 Human Ccl27 (Human) Peptide - - - Refs
A (Rhodopsin) Chemokine CCR10 CCR10 CCR10 Human Ccl27 (Mouse) Peptide - - -
A (Rhodopsin) Chemokine CCR10 CCR10 CCR10 Human Ccl28 (Human) Peptide - - -
A (Rhodopsin) Chemokine CCR10 CCR10 CCR10 Human Ccl28 (Mouse) Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl13 (Human) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl14 (Human) 6 Peptide - - - 7.4 7.4 Refs
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl15 (Human) 7 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl16 (Human) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl23 (Human) 2 Peptide - - - 8.9 8.9 Refs
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl3 (Human) 1 Peptide - - - - 7.8 9.0 10.2 Refs
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl3 (Mouse) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl3 (Rat) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl4 (Human) 5 Peptide - - - 7.1 7.5 7.8 Refs
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl4 (Mouse) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl4 (Rat) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl5 (Human) 4 Peptide - - - 6.8 7.5 8.2 Refs
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl5 (Mouse) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl7 (Human) 3 Peptide - - - 8.1 8.1 Refs
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl7 (Mouse) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl7 (Rat) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl8 (Human) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR1 CCR1 CCR1 Human Ccl8 (Mouse) 7 Peptide - - -
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl11 (Human) 6 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl11 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl11 (Rat) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl13 (Human) 2 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl16 (Human) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl2 (Human) 1 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl2 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl2 (Rat) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl24 (Human) 7 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl26 (Human) 5 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl7 (Human) 4 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl7 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl7 (Rat) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl8 (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR2 CCR2 CCR2 Human Ccl8 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl11 (Human) 1 Peptide - - - 9.7 9.9 10.0 Refs
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl11 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl11 (Rat) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl13 (Human) 5 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl15 (Human) 5 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl2 (Human) 4 Peptide - - - 7.2 7.5 7.8 Refs
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl2 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl2 (Rat) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl24 (Human) 5 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl24 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl26 (Human) 5 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl28 (Human) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl28 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl5 (Human) 2 Peptide - - - 8.5 8.9 9.3 Refs
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl5 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl7 (Human) 3 Peptide - - - 8.6 8.9 9.2 Refs
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl7 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl7 (Rat) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl8 (Human) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Ccl8 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Cxcl10 (Human) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Cxcl10 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Cxcl10 (Rat) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Cxcl11 (Human) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Cxcl11 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Cxcl9 (Human) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR3 CCR3 CCR3 Human Cxcl9 (Mouse) 5 Peptide - - -
A (Rhodopsin) Chemokine CCR4 CCR4 CCR4 Human Ccl17 (Human) 2 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR4 CCR4 CCR4 Human Ccl22 (Human) 1 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR4 CCR4 CCR4 Human Ccl22 (Mouse) 3 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl11 (Human) 8 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl11 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl11 (Rat) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl13 (Human) 4 Peptide - - - 9.1 9.1 Refs
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl14 (Human) 7 Peptide - - - 7.2 7.2 Refs
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl16 (Human) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl2 (Human) 6 Peptide - - - 7.5 7.5 Refs
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl2 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl2 (Rat) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl3 (Human) 5 Peptide - - - - 8.0 8.5 8.9 Refs
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl3 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl3 (Rat) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl4 (Human) 1 Peptide - - - 9.4 9.5 9.6 Refs
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl4 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl4 (Rat) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl5 (Human) 2 Peptide - - - 9.2 9.5 9.7 Refs
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl5 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl7 (Human) 6 Peptide - - - 7.5 7.5 Refs
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl7 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl7 (Rat) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl8 (Human) 3 Peptide - - - 9.3 9.3 Refs
A (Rhodopsin) Chemokine CCR5 CCR5 CCR5 Human Ccl8 (Mouse) 8 Peptide - - -
A (Rhodopsin) Chemokine CCR6 CCR6 CCR6 Human Ccl20 (Human) 1 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR6 CCR6 CCR6 Human Ccl20 (Mouse) 2 Peptide - - -
A (Rhodopsin) Chemokine CCR6 CCR6 CCR6 Human Ccl20 (Rat) 2 Peptide - - -
A (Rhodopsin) Chemokine CCR6 CCR6 CCR6 Human Beta-Defensin 4a (Human) 2 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR7 CCR7 CCR7 Human Ccl19 (Human) 1 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR7 CCR7 CCR7 Human Ccl21 (Human) 2 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR7 CCR7 Ccr7 Mouse Ccl19 (Mouse) 2 Peptide - - - - Refs
A (Rhodopsin) Chemokine CCR7 CCR7 Ccr7 Mouse Ccl21a (Mouse) 2 Peptide - - - - Refs
A (Rhodopsin) Chemokine CCR7 CCR7 Ccr7 Mouse Ccl21b (Mouse) 2 Peptide - - - - Refs
A (Rhodopsin) Chemokine CCR8 CCR8 CCR8 Human Ccl1 (Human) 1 Peptide - - - Refs
A (Rhodopsin) Chemokine CCR8 CCR8 CCR8 Human Ccl1 (Mouse) 2 Peptide - - -
A (Rhodopsin) Chemokine CCR8 CCR8 CCR8 Human Ccl8 (Human) 2 Peptide - - - -
A (Rhodopsin) Chemokine CCR8 CCR8 Ccr8 Mouse Ccl8 (Mouse) 2 Peptide - - - -
A (Rhodopsin) Chemokine CCR9 CCR9 CCR9 Human Ccl25 (Human) Principal 1 Peptide - - -
A (Rhodopsin) Chemokine CCR9 CCR9 CCR9 Human Ccl25 (Mouse) Principal 1 Peptide - - -
A (Rhodopsin) Chemokine CCRL2 CCRL2 CCRL2 Human Ccl19 (Human) 1 Peptide - - - - Refs
A (Rhodopsin) Chemokine CCRL2 CCRL2 CCRL2 Human Ccl19 (Mouse) 2 Peptide - - - -
A (Rhodopsin) Chemokine CCRL2 CCRL2 CCRL2 Human Chemerin (Human) 2 Peptide - - - -
A (Rhodopsin) Chemokine CX3C1 CX3CR1 CX3CR1 Human Cx3Cl1 (Human) Principal 1 Peptide - - - Refs
A (Rhodopsin) Chemokine CX3C1 CX3CR1 CX3CR1 Human Cx3Cl1 (Mouse) Principal 1 Peptide - - -
A (Rhodopsin) Chemokine CX3C1 CX3CR1 CX3CR1 Human Cx3Cl1 (Rat) Principal 1 Peptide - - -
A (Rhodopsin) Chemokine CXCR1 CXCR1 CXCR1 Human Cxcl6 (Human) 2 Peptide - - - 7.0 7.0 Refs
A (Rhodopsin) Chemokine CXCR1 CXCR1 CXCR1 Human Cxcl8 (Human) 1 Peptide - - - 8.8 9.2 9.5 Refs
A (Rhodopsin) Chemokine CXCR1 CXCR1 CXCR1 Human Cytokine Domain Of Tyrosyl Trna Synthetase (Human) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl1 (Human) 2 Peptide - - - 8.4 9.1 9.7 Refs
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl1 (Mouse) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl1 (Rat) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl2 (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl2 (Mouse) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl2 (Rat) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl3 (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl3 (Mouse) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl3 (Rat) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl5 (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl5 (Mouse) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl5 (Rat) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl6 (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl7 (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR2 CXCR2 CXCR2 Human Cxcl8 (Human) 1 Peptide - - - 8.8 9.2 9.5 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Ccl11 (Human) 4 Peptide - - - 7.2 7.2 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Ccl13 (Human) 4 Peptide - - - 7.2 7.2 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Ccl19 (Human) 8 Peptide - - - 5.9 5.9 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Ccl20 (Human) 5 Peptide - - - 6.8 6.8 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Ccl5 (Human) 7 Peptide - - - 6.4 6.4 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Ccl7 (Human) 6 Peptide - - - 6.6 6.6 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Cxcl10 (Human) 2 Peptide - - - 7.8 8.8 9.8 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Cxcl10 (Mouse) 9 Peptide - - -
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Cxcl10 (Rat) 9 Peptide - - -
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Cxcl11 (Human) 1 Peptide - - - 10.4 10.5 10.5 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Cxcl11 (Mouse) 9 Peptide - - -
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Cxcl12Α (Human) 7 Peptide - - - 6.4 6.4 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Cxcl9 (Human) 3 Peptide - - - 7.3 7.8 8.3 Refs
A (Rhodopsin) Chemokine CXCR3 CXCR3 CXCR3 Human Cxcl9 (Mouse) 9 Peptide - - -
A (Rhodopsin) Chemokine CXCR4 CXCR4 CXCR4 Human Cxcl12 (Mouse) 3 Peptide - - -
A (Rhodopsin) Chemokine CXCR4 CXCR4 CXCR4 Human Cxcl12Α (Human) 1 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR4 CXCR4 CXCR4 Human Cxcl12Β (Human) 2 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR4 CXCR4 CXCR4 Human Cxcl12Δ (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR4 CXCR4 CXCR4 Human Cxcl12Ε (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR4 CXCR4 CXCR4 Human Cxcl12Γ (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR4 CXCR4 CXCR4 Human Cxcl12Φ (Human) 3 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR5 CXCR5 CXCR5 Human Cxcl13 (Human) Principal 1 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR5 CXCR5 CXCR5 Human Cxcl13 (Mouse) Principal 1 Peptide - - -
A (Rhodopsin) Chemokine CXCR6 CXCR6 CXCR6 Human Cxcl16 (Human) Principal 1 Peptide - - - Refs
A (Rhodopsin) Chemokine CXCR6 CXCR6 CXCR6 Human Cxcl16 (Mouse) Principal 1 Peptide - - -
A (Rhodopsin) Chemokine CXCR6 CXCR6 CXCR6 Human Cxcl16 (Rat) Principal 1 Peptide - - -
A (Rhodopsin) Chemokine XCR1 XCR1 XCR1 Human Xcl1 (Human) 1 Peptide - - - 7.3 7.3 Refs
A (Rhodopsin) Chemokine XCR1 XCR1 XCR1 Human Xcl1 (Mouse) 2 Peptide - - -
A (Rhodopsin) Chemokine XCR1 XCR1 XCR1 Human Xcl1 (Rat) 2 Peptide - - -
A (Rhodopsin) Chemokine XCR1 XCR1 XCR1 Human Xcl2 (Human) 1 Peptide - - - 7.3 7.3 Refs
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Cck-33 (Human) 2 Peptide NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N1CCCC1C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N)Cc1ccccc1)CC(=O)O)CCSC)Cc1c[nH]c2c1cccc2)CCSC)c1ccc(cc1)OS(=O)(=O)O)CC(=O)O)CCCNC(=N)N)CC(=O)O)CO)C(CC)C)CCCNC(=N)N)Cc1nc[nH]c1)CO)CC(=O)O)CC(C)C)CC(=O)N)CCC(=O)N)CC(C)C)CC(=O)N)NC(=O)C(C(C)C)NC(=O)C(C(CC)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)CNC(=O)C(NC(=O)C1CCCN1C(=O)C(NC(=O)C(CCCCN)N)C)CO)CCCNC(=N)N)CCSC)CO QFLBZJPOIZFFJQ-UHFFFAOYSA-N - -
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Cck-33 (Mouse) 2 Peptide - - - -
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Cck-33 (Rat) 2 Peptide - - - -
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Cck-39 (Human) 2 Peptide - - - -
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Cck-4 (Human) 2 Peptide CSCCC(C(=O)NC(C(=O)NC(C(=O)N)Cc1ccccc1)CC(=O)O)NC(=O)C(Cc1c[nH]c2c1cccc2)N RGYLYUZOGHTBRF-UHFFFAOYSA-N - -
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Cck-58 (Human) 2 Peptide - - - -
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Cck-8 (Human) 1 Peptide CSCC[C@@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccccc1)CC(=O)O)CCSC)Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)N)Cc1ccc(cc1)OS(=O)(=O)O IZTQOLKUZKXIRV-YRVFCXMDSA-N - 7EZM Refs
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Desulfated Cholecystokinin-8 2 Peptide CSCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)C(=O)[C@H](CC(=O)O)N)Cc1ccc(cc1)O)CCSC)Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NN)CC(=O)O ZBTPHEHKAHBSMT-YRVFCXMDSA-N - -
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Gastrin-17 (Human) 2 Peptide - - - AFM_CCKAR_HUMAN_hashedseq[KCFYMGL3JABRHKFWN6KFBVOQSYZCN0]
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Gastrin-17 (Mouse) 2 Peptide - - - -
A (Rhodopsin) Cholecystokinin CCKAR CCK1 CCKAR Human Gastrin-17 (Rat) 2 Peptide - - - -
A (Rhodopsin) Cholecystokinin CCKAR CCK1 Cckar Rat Cck-8 (Human) 1 Peptide CSCC[C@@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccccc1)CC(=O)O)CCSC)Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)N)Cc1ccc(cc1)OS(=O)(=O)O IZTQOLKUZKXIRV-YRVFCXMDSA-N - - Refs
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Cck-33 (Human) 2 Peptide NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N1CCCC1C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N)Cc1ccccc1)CC(=O)O)CCSC)Cc1c[nH]c2c1cccc2)CCSC)c1ccc(cc1)OS(=O)(=O)O)CC(=O)O)CCCNC(=N)N)CC(=O)O)CO)C(CC)C)CCCNC(=N)N)Cc1nc[nH]c1)CO)CC(=O)O)CC(C)C)CC(=O)N)CCC(=O)N)CC(C)C)CC(=O)N)NC(=O)C(C(C)C)NC(=O)C(C(CC)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)CNC(=O)C(NC(=O)C1CCCN1C(=O)C(NC(=O)C(CCCCN)N)C)CO)CCCNC(=N)N)CCSC)CO QFLBZJPOIZFFJQ-UHFFFAOYSA-N - - Refs
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Cck-33 (Mouse) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Cck-33 (Rat) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Cck-39 (Human) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Cck-4 (Human) 4 Peptide CSCCC(C(=O)NC(C(=O)NC(C(=O)N)Cc1ccccc1)CC(=O)O)NC(=O)C(Cc1c[nH]c2c1cccc2)N RGYLYUZOGHTBRF-UHFFFAOYSA-N - - Refs
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Cck-58 (Human) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Cck-8 (Human) 1 Peptide CSCC[C@@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccccc1)CC(=O)O)CCSC)Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)N)Cc1ccc(cc1)OS(=O)(=O)O IZTQOLKUZKXIRV-YRVFCXMDSA-N - 8IA7 Refs
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Desulfated Cholecystokinin-8 None 3 Peptide CSCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)C(=O)[C@H](CC(=O)O)N)Cc1ccc(cc1)O)CCSC)Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NN)CC(=O)O ZBTPHEHKAHBSMT-YRVFCXMDSA-N - - Refs
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Desulfated Gastrin-14 (Human) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Desulfated Gastrin-17 (Human) 5 Peptide CSCC[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@@H]1CCC(=O)N1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O GKDWRERMBNGKCZ-RNXBIMIWSA-N - 7F8W
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Desulfated Gastrin-34 (Human) 5 Peptide CSCC[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CO)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCC(=O)N1)C(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O DKONFPYEAKZHHO-JCVYGFDXSA-N - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Desulfated Gastrin-71 (Human) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Gastrin-14 (Human) 5 Peptide CSCC[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O SSBRJDBGIVUNDK-QOGDCIHTSA-N - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Gastrin-17 (Human) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Gastrin-17 (Mouse) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Gastrin-17 (Rat) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Gastrin-34 (Human) 5 Peptide - - - -
A (Rhodopsin) Cholecystokinin GASR CCK2 CCKBR Human Gastrin-71 (Human) 5 Peptide - - - -
A (Rhodopsin) Complement peptide C3AR C3a C3AR1 Human C3a (Human) 1 Peptide - - - - 7.3 8.5 9.6 Refs
A (Rhodopsin) Complement peptide C3AR C3a C3AR1 Human C3a (Mouse) 2 Peptide - - - -
A (Rhodopsin) Complement peptide C3AR C3a C3AR1 Human C3a (Rat) 2 Peptide - - - -
A (Rhodopsin) Complement peptide C3AR C3a C3AR1 Human C5a (Human) 2 Peptide - - - -
A (Rhodopsin) Complement peptide C3AR C3a C3AR1 Human C5a (Mouse) 2 Peptide - - - -
A (Rhodopsin) Complement peptide C3AR C3a C3AR1 Human C5a (Rat) 2 Peptide - - - -
A (Rhodopsin) Complement peptide C5AR1 C5a1 C5AR1 Human C3a (Human) 2 Peptide - - -
A (Rhodopsin) Complement peptide C5AR1 C5a1 C5AR1 Human C3a (Mouse) 2 Peptide - - -
A (Rhodopsin) Complement peptide C5AR1 C5a1 C5AR1 Human C3a (Rat) 2 Peptide - - -
A (Rhodopsin) Complement peptide C5AR1 C5a1 C5AR1 Human C5a (Human) 1 Peptide - - - 8.0 8.5 9.0 Refs
A (Rhodopsin) Complement peptide C5AR1 C5a1 C5AR1 Human C5a (Mouse) 2 Peptide - - -
A (Rhodopsin) Complement peptide C5AR1 C5a1 C5AR1 Human C5a (Rat) 2 Peptide - - -
A (Rhodopsin) Complement peptide C5AR1 C5a1 C5AR1 Human C5a Des-Arg (Human) 2 Peptide - - - 8JZZ Refs
A (Rhodopsin) Complement peptide C5AR1 C5a1 C5AR1 Human Ribosomal Protein S19 (Human) 2 Peptide - - - Refs
A (Rhodopsin) Complement peptide C5AR2 C5a2 C5AR2 Human C3a (Human) 2 Peptide - - - -
A (Rhodopsin) Complement peptide C5AR2 C5a2 C5AR2 Human C5a (Human) 1 Peptide - - - - 8.9 8.9 Refs
A (Rhodopsin) Complement peptide C5AR2 C5a2 C5AR2 Human C5a Des-Arg (Human) 2 Peptide - - - - Refs
A (Rhodopsin) Complement peptide C5AR2 C5a2 C5AR2 Human Ribosomal Protein S19 (Human) 2 Peptide - - - - Refs
A (Rhodopsin) Dopamine DRD1 D1 DRD1 Human 5-Hydroxytryptamine None 1 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 5.0 5.0 Refs
A (Rhodopsin) Dopamine DRD1 D1 DRD1 Human Dopamine None 2 Small molecule NCCc1ccc(c(c1)O)O VYFYYTLLBUKUHU-UHFFFAOYSA-N - 9LLJ 4.3 5.0 5.6 Refs
A (Rhodopsin) Dopamine DRD1 D1 DRD1 Human Noradrenaline None 3 Small molecule NCC(c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-UHFFFAOYSA-N - - 4.3 4.3 Refs
A (Rhodopsin) Dopamine DRD2 D2 DRD2 Human Dopamine Principal 1 Small molecule NCCc1ccc(c(c1)O)O VYFYYTLLBUKUHU-UHFFFAOYSA-N - 8TZQ 5.3 5.9 6.4 Refs
A (Rhodopsin) Dopamine DRD2 D2 Drd2 Rat Dopamine Principal 1 Small molecule NCCc1ccc(c(c1)O)O VYFYYTLLBUKUHU-UHFFFAOYSA-N - - 5.3 5.9 6.4 Refs
A (Rhodopsin) Dopamine DRD3 D3 DRD3 Human Dopamine Principal 1 Small molecule NCCc1ccc(c(c1)O)O VYFYYTLLBUKUHU-UHFFFAOYSA-N - B2M_DRD3_HUMAN_DOPAMINE_GNAO_HUMAN 6.4 6.9 7.3 Refs
A (Rhodopsin) Dopamine DRD4 D4 DRD4 Human Dopamine Principal 1 Small molecule NCCc1ccc(c(c1)O)O VYFYYTLLBUKUHU-UHFFFAOYSA-N - B2M_DRD4_HUMAN_DOPAMINE_GNAO_HUMAN 7.4 7.4 Refs
A (Rhodopsin) Dopamine DRD4 D4 Drd4 Rat Dopamine Principal 1 Small molecule NCCc1ccc(c(c1)O)O VYFYYTLLBUKUHU-UHFFFAOYSA-N - - 7.4 7.4 Refs
A (Rhodopsin) Dopamine DRD5 D5 DRD5 Human 5-Hydroxytryptamine None 2 Small molecule NCCc1c[nH]c2c1cc(O)cc2 QZAYGJVTTNCVMB-UHFFFAOYSA-N - - 5.5 5.5 Refs
A (Rhodopsin) Dopamine DRD5 D5 DRD5 Human Dopamine None 1 Small molecule NCCc1ccc(c(c1)O)O VYFYYTLLBUKUHU-UHFFFAOYSA-N - B2M_DRD5_HUMAN_DOPAMINE_GNAS2_HUMAN 6.6 6.6 Refs
A (Rhodopsin) Dopamine DRD5 D5 DRD5 Human Noradrenaline None 3 Small molecule NCC(c1ccc(c(c1)O)O)O SFLSHLFXELFNJZ-UHFFFAOYSA-N - - 4.9 4.9 Refs
A (Rhodopsin) Endothelin EDNRA ETA EDNRA Human Endothelin-1 (Human) 2 Protein NCCCC[C@@H]1NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@@H](NC1=O)CCC(=O)O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccc(cc1)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CSSC[C@@H](C(=O)N[C@H](C(=O)N2)CO)N)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1c[nH]c2c1cccc2)[C@H](CC)C)[C@H](CC)C)CC(=O)O)CC(C)C)Cc1cnc[nH]1)CO ZUBDGKVDJUIMQQ-ZTNLKOGPSA-N - 8HCQ Refs
A (Rhodopsin) Endothelin EDNRA ETA EDNRA Human Endothelin-2 (Human) 1 Peptide NCCCC[C@@H]1NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@@H](NC1=O)CCC(=O)O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccc(cc1)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CSSC[C@@H](C(=O)N[C@H](C(=O)N2)CO)N)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1c[nH]c2c1cccc2)[C@H](CC)C)[C@H](CC)C)CC(=O)O)CC(C)C)Cc1[nH]cnc1)CO)Cc1c[nH]c2c1cccc2 MLFJHYIHIKEBTQ-IYRKOGFYSA-N - Refs
A (Rhodopsin) Endothelin EDNRA ETA EDNRA Human Endothelin-2 (Mouse) 3 Peptide - - -
A (Rhodopsin) Endothelin EDNRA ETA EDNRA Human Endothelin-3 (Human) 3 Peptide - - -
A (Rhodopsin) Endothelin EDNRB ETB EDNRB Human Endothelin-1 (Human) 2 Protein NCCCC[C@@H]1NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCSC)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@@H](NC1=O)CCC(=O)O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccc(cc1)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CSSC[C@@H](C(=O)N[C@H](C(=O)N2)CO)N)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1c[nH]c2c1cccc2)[C@H](CC)C)[C@H](CC)C)CC(=O)O)CC(C)C)Cc1cnc[nH]1)CO ZUBDGKVDJUIMQQ-ZTNLKOGPSA-N - 8HCX
A (Rhodopsin) Endothelin EDNRB ETB EDNRB Human Endothelin-2 (Human) 2 Peptide NCCCC[C@@H]1NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@@H]2CSSC[C@H](NC(=O)[C@@H](NC1=O)CCC(=O)O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccc(cc1)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CSSC[C@@H](C(=O)N[C@H](C(=O)N2)CO)N)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1c[nH]c2c1cccc2)[C@H](CC)C)[C@H](CC)C)CC(=O)O)CC(C)C)Cc1[nH]cnc1)CO)Cc1c[nH]c2c1cccc2 MLFJHYIHIKEBTQ-IYRKOGFYSA-N -
A (Rhodopsin) Endothelin EDNRB ETB EDNRB Human Endothelin-2 (Mouse) 2 Peptide - - -
A (Rhodopsin) Endothelin EDNRB ETB EDNRB Human Endothelin-3 (Human) 1 Peptide - - - 6IGK Refs
A (Rhodopsin) Endothelin EDNRB ETB Ednrb Rat Endothelin-3 (Human) 1 Peptide - - - - Refs
A (Rhodopsin) Estrogen (G protein-coupled) GPER1 GPER GPER1 Human 17Β-Estradiol Principal 1 Small molecule Oc1ccc2c(c1)CC[C@@H]1[C@@H]2CC[C@]2([C@H]1CC[C@@H]2O)C VOXZDWNPVJITMN-ZBRFXRBCSA-N - - 8.2 8.4 8.5 Refs
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Annexin I (Human) 3 Peptide - - -
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Annexin I (Mouse) 3 Peptide - - -
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Annexin I (Rat) 3 Peptide - - -
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Annexin I-(2-26) (Human) 2 Peptide - - - 5.8 6.0 6.1 Refs
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Cathepsin G (Human) 3 Peptide - - -
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Cathepsin G (Mouse) 3 Peptide - - -
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Cathepsin G (Rat) 3 Peptide - - -
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Fmet-Leu-Phe None 1 Peptide CSCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1ccccc1)CC(C)C)NC=O PRQROPMIIGLWRP-BZSNNMDCSA-N - 7EUO 10.1 10.2 10.2 Refs
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Fmet-Leu-Phe-Ile-Ile None 3 Peptide - - - - Refs
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Mitochondrial Peptde Fmmyalf None 3 Peptide - - - - Refs
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Mitochondrial Peptide Fmfadrw None 3 Peptide - - - - Refs
A (Rhodopsin) Formylpeptide FPR1 FPR1 FPR1 Human Spinorphin (Human) 3 Peptide CC(C[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)O)[C@H](O)C)Cc1c[nH]c2c1cccc2)Cc1ccc(cc1)O)C(C)C)C(C)C)N)C BXIFNVGZIMFBQB-DYDSHOKNSA-N - Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human 15-Deoxy-Lxa4 10 Small molecule CCCCCC/C=C/C=C/C=C/C=C/[C@H]([C@H](CCCC(=O)O)O)O SJIRTDBAYKOBAL-COJKCNNISA-N - -
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Ll-37 (Human) 7 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CO)CCC(=O)O)[C@H](O)C)CCCN=C(N)N)C(C)C)CC(C)C)CC(=O)N)CCCN=C(N)N)CC(C)C)Cc1ccccc1)CC(=O)O)CCCCN)[C@H](CC)C)CCCN=C(N)N)CCC(=O)N)C(C)C)[C@H](CC)C)CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@H]([C@H](CC)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](CC(C)C)N)CC(C)C)CC(=O)O)Cc1ccccc1)Cc1ccccc1)CCCN=C(N)N)CCCCN)CO)CCCCN)CCC(=O)O)CCCCN)CCCCN)CCC(=O)O)Cc1ccccc1 POIUWJQBRNEFGX-XAMSXPGMSA-N - 6.0 6.0 Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Ltc4 None 10 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SC[C@@H](C(=O)NCC(=O)O)NC(=O)CC[C@@H](C(=O)O)N GWNVDXQDILPJIG-NXOLIXFESA-N - -
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Ltd4 None 10 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SCC(C(=O)NCC(=O)O)N YEESKJGWJFYOOK-LDDGIIIKSA-N - -
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Lxa4 None 1 Small molecule CCCCC[C@@H](/C=C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)O)O IXAQOQZEOGMIQS-SSQFXEBMSA-N - - 12.0 12.0 Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Prp106-126 (Human) 9 Peptide CSCC[C@H](NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCSC)NC(=O)[C@H](CC(N)=O)NC(=O)[C@@H](NC(=O)[C@@H](N)CCCCN)[C@@H](C)O)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)O)C(C)C)C(C)C XPZWWTIIKSODDO-MBNDGZRNSA-N - 4.6 4.6 Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Annexin I (Human) 10 Peptide - - - Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Annexin I (Mouse) 10 Peptide - - -
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Annexin I (Rat) 10 Peptide - - -
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Annexin I-(2-26) (Human) 8 Peptide - - - - 5.8 6.0 6.1 Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Aspirin Triggered Lipoxin A4 None 10 Small molecule CCCCC[C@H](/C=C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)O)O IXAQOQZEOGMIQS-JEWNPAEBSA-N - -
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Aspirin-Triggered Resolvin D1 None 3 Small molecule CC/C=C\C[C@H](/C=C/C=C\C=C\C=C\[C@H]([C@H](C/C=C\CCC(=O)O)O)O)O OIWTWACQMDFHJG-BJEBZIPWSA-N - - 11.1 11.1 Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Humanin (Human) 4 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)C)CCCNC(=N)N)CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](CC)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCSC)N)C)CCCNC(=N)N)CO)CS)CC(C)C)CC(C)C)CC(C)C)CC(C)C)CO)CCC(=O)O)CC(=O)O)CC(C)C DPEUWKZJZIPZKE-OFANTOPUSA-N - 8.5 8.5 Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Resolvin D1 None 2 Small molecule CC/C=C\C[C@@H](/C=C/C=C\C=C\C=C\[C@@H]([C@H](C/C=C\CCC(=O)O)O)O)O OIWTWACQMDFHJG-LDOXQWQISA-N - - 11.9 11.9 Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX FPR2 Human Serum Amyloid A (Human) 6 Peptide - - - 6.6 6.6 Refs
A (Rhodopsin) Formylpeptide FPR2 FPR2/ALX Fpr2 Mouse Cramp (Mouse) 5 Peptide CC[C@H](C)[C@H](N)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(N)=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(=O)O)C(=O)O)C(C)C)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC QBSFTGGUOCPHDM-GDCSACRRSA-N - - 6.7 6.9 7.0 Refs
A (Rhodopsin) Formylpeptide FPR3 FPR3 FPR3 Human F2l (Human) 2 Peptide - - - 8.0 8.1 8.2 Refs
A (Rhodopsin) Formylpeptide FPR3 FPR3 FPR3 Human F2l (Mouse) 4 Peptide - - -
A (Rhodopsin) Formylpeptide FPR3 FPR3 FPR3 Human Annexin I-(2-26) (Human) 3 Peptide - - - 5.0 6.0 7.0 Refs
A (Rhodopsin) Formylpeptide FPR3 FPR3 FPR3 Human Humanin (Human) 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)C)CCCNC(=N)N)CCCNC(=N)N)NC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](CC)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCSC)N)C)CCCNC(=N)N)CO)CS)CC(C)C)CC(C)C)CC(C)C)CC(C)C)CO)CCC(=O)O)CC(=O)O)CC(C)C DPEUWKZJZIPZKE-OFANTOPUSA-N - 8.9 8.9 Refs
A (Rhodopsin) Free fatty acid FFAR1 FFA1 FFAR1 Human Α-Linolenic Acid None 2 Small molecule CC/C=C\C/C=C\C/C=C\CCCCCCCC(=O)O DTOSIQBPPRVQHS-PDBXOOCHSA-N - - 4.6 5.2 5.7 Refs
A (Rhodopsin) Free fatty acid FFAR1 FFA1 FFAR1 Human Docosahexaenoic Acid None 1 Small molecule CC/C=C\C/C=C\C/C=C\C/C=C\C/C=C\C/C=C\CCC(=O)O MBMBGCFOFBJSGT-KUBAVDMBSA-N - 8EIT 5.4 5.7 6.0 Refs
A (Rhodopsin) Free fatty acid FFAR1 FFA1 FFAR1 Human Myristic Acid None 3 Lipid CCCCCCCCCCCCCC(=O)O TUNFSRHWOTWDNC-UHFFFAOYSA-N - - 4.5 4.8 5.1 Refs
A (Rhodopsin) Free fatty acid FFAR1 FFA1 FFAR1 Human Oleic Acid None 3 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)O ZQPPMHVWECSIRJ-KTKRTIGZSA-N - - 3.9 4.8 5.7 Refs
A (Rhodopsin) Free fatty acid FFAR2 FFA2 FFAR2 Human Trans-2-Methylcrotonic Acid None 3 Small molecule C/C(=C\C)/C(=O)O UIERETOOQGIECD-ONEGZZNKSA-N - - 3.8 3.8 Refs
A (Rhodopsin) Free fatty acid FFAR2 FFA2 FFAR2 Human Acetic Acid None 2 Small molecule CC(=O)O QTBSBXVTEAMEQO-UHFFFAOYSA-N - 8J24 3.1 3.9 4.6 Refs
A (Rhodopsin) Free fatty acid FFAR2 FFA2 FFAR2 Human Butyric Acid None 4 Small molecule CCCC(=O)O FERIUCNNQQJTOY-UHFFFAOYSA-N - 9K1D 2.9 3.8 4.6 Refs
A (Rhodopsin) Free fatty acid FFAR2 FFA2 FFAR2 Human Propanoic Acid None 1 Small molecule CCC(=O)O XBDQKXXYIPTUBI-UHFFFAOYSA-N - - 3.0 4.0 4.9 Refs
A (Rhodopsin) Free fatty acid FFAR3 FFA3 FFAR3 Human Butyric Acid None 2 Small molecule CCCC(=O)O FERIUCNNQQJTOY-UHFFFAOYSA-N - 8J21 3.8 4.4 4.9 Refs
A (Rhodopsin) Free fatty acid FFAR3 FFA3 FFAR3 Human Propanoic Acid None 1 Small molecule CCC(=O)O XBDQKXXYIPTUBI-UHFFFAOYSA-N - - 3.9 4.8 5.7 Refs
A (Rhodopsin) Free fatty acid FFAR4 FFA4 FFAR4 Human Α-Linolenic Acid None 3 Small molecule CC/C=C\C/C=C\C/C=C\CCCCCCCC(=O)O DTOSIQBPPRVQHS-PDBXOOCHSA-N - - 5.1 5.1 Refs
A (Rhodopsin) Free fatty acid FFAR4 FFA4 FFAR4 Human Linoleic Acid None 1 Small molecule CCCCC/C=C\C/C=C\CCCCCCCC(=O)O OYHQOLUKZRVURQ-HZJYTTRNSA-N - 8ID4 5.9 5.9 Refs
A (Rhodopsin) Free fatty acid FFAR4 FFA4 FFAR4 Human Myristic Acid None 2 Lipid CCCCCCCCCCCCCC(=O)O TUNFSRHWOTWDNC-UHFFFAOYSA-N - - 5.2 5.2 Refs
A (Rhodopsin) Free fatty acid FFAR4 FFA4 FFAR4 Human Oleic Acid None 4 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)O ZQPPMHVWECSIRJ-KTKRTIGZSA-N - 8ID6 4.7 4.7 Refs
A (Rhodopsin) Free fatty acid FFAR4 FFA4 Ffar4 Rat Α-Linolenic Acid None 3 Small molecule CC/C=C\C/C=C\C/C=C\CCCCCCCC(=O)O DTOSIQBPPRVQHS-PDBXOOCHSA-N - - 5.1 5.1 Refs
A (Rhodopsin) GPR18, GPR55 and GPR119 GP119 GPR119 GPR119 Human N-Oleoylethanolamide None 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)NCCO BOWVQLFMWHZBEF-KTKRTIGZSA-N - - 5.4 5.9 6.3 Refs
A (Rhodopsin) GPR18, GPR55 and GPR119 GP119 GPR119 GPR119 Human N-Palmitoylethanolamine None 2 Lipid CCCCCCCCCCCCCCCC(=O)NCCO HXYVTAGFYLMHSO-UHFFFAOYSA-N - -
A (Rhodopsin) GPR18, GPR55 and GPR119 GP119 GPR119 GPR119 Human Sea None 2 Lipid CCCCCCCCCCCCCCCCCC(=O)NCCO OTGQIQQTPXJQRG-UHFFFAOYSA-N - -
A (Rhodopsin) GPR18, GPR55 and GPR119 GP119 GPR119 GPR119 Human Anandamide 2 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCCO LGEQQWMQCRIYKG-DOFZRALJSA-N - -
A (Rhodopsin) GPR18, GPR55 and GPR119 GPR18 GPR18 GPR18 Human N-Arachidonoylglycine Principal 1 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCC(=O)O YLEARPUNMCCKMP-DOFZRALJSA-N - - 7.3 7.5 7.7 Refs
A (Rhodopsin) GPR18, GPR55 and GPR119 GPR55 GPR55 GPR55 Human 2-Arachidonoylglycerol None 1 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)OC(CO)CO RCRCTBLIHCHWDZ-DOFZRALJSA-N - - 8.5 8.5 Refs
A (Rhodopsin) GPR18, GPR55 and GPR119 GPR55 GPR55 GPR55 Human 2-Arachidonoylglycerolphosphoinositol None 5 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)OC(COP(=O)(OC1C(O)C(O)C(C(C1O)O)O)[O-])CO OKEQUIXTUXJQNT-DOFZRALJSA-M - - Refs
A (Rhodopsin) GPR18, GPR55 and GPR119 GPR55 GPR55 GPR55 Human N-Palmitoylethanolamine None 2 Lipid CCCCCCCCCCCCCCCC(=O)NCCO HXYVTAGFYLMHSO-UHFFFAOYSA-N - - 8.4 8.4 Refs
A (Rhodopsin) GPR18, GPR55 and GPR119 GPR55 GPR55 GPR55 Human Anandamide None 3 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCCO LGEQQWMQCRIYKG-DOFZRALJSA-N - - 7.7 7.7 Refs
A (Rhodopsin) GPR18, GPR55 and GPR119 GPR55 GPR55 GPR55 Human Lysophosphatidylinositol None 4 Small molecule O[C@@H](COC(=O)C)COP(=O)(O[C@@H]1[C@H](O)[C@H](O)[C@H]([C@@H]([C@H]1O)O)O)O FBDBXJJQMHPGMP-IFUOQLDVSA-N - - 5.5 6.4 7.3 Refs
A (Rhodopsin) Galanin GALR1 GAL1 GALR1 Human Galanin (Human) 2 Protein CC(C)C[C@H](NC(=O)CNC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(C)C)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O CBSXZYWGVAQSHI-RUKUCZSXSA-N - 9.1 9.8 10.5 Refs
A (Rhodopsin) Galanin GALR1 GAL1 GALR1 Human Galanin-Like Peptide (Human) 2 Peptide - - - Refs
A (Rhodopsin) Galanin GALR1 GAL1 GALR1 Human Galanin-Like Peptide (Mouse) 2 Peptide - - -
A (Rhodopsin) Galanin GALR1 GAL1 GALR1 Human Spexin-1 (Human) 2 Peptide - - - -
A (Rhodopsin) Galanin GALR1 GAL1 Galr1 Mouse Galanin (Mouse) 1 Peptide - - - - 9.8 9.8 9.0 9.6 10.1 Refs
A (Rhodopsin) Galanin GALR1 GAL1 Galr1 Rat Galanin (Mouse) 1 Peptide - - - - 9.8 9.8 9.0 9.6 10.1 Refs
A (Rhodopsin) Galanin GALR1 GAL1 Galr1 Rat Galanin-Like Peptide (Rat) 2 Peptide - - - - Refs
A (Rhodopsin) Galanin GALR2 GAL2 GALR2 Human Galanin (Human) 1 Protein CC(C)C[C@H](NC(=O)CNC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(C)C)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O CBSXZYWGVAQSHI-RUKUCZSXSA-N - 7.9 8.5 9.1 8.6 8.9 9.1 Refs
A (Rhodopsin) Galanin GALR2 GAL2 GALR2 Human Galanin-Like Peptide (Human) 4 Peptide - - - Refs
A (Rhodopsin) Galanin GALR2 GAL2 GALR2 Human Galanin-Like Peptide (Mouse) 4 Peptide - - -
A (Rhodopsin) Galanin GALR2 GAL2 GALR2 Human Galanin-Like Peptide (Rat) 4 Peptide - - -
A (Rhodopsin) Galanin GALR2 GAL2 GALR2 Human Spexin-1 (Human) 3 Peptide - - - 6.8 6.8 Refs
A (Rhodopsin) Galanin GALR2 GAL2 Galr2 Mouse Galanin (Mouse) 2 Peptide - - - - 8.3 8.3 8.3 8.8 9.3 Refs
A (Rhodopsin) Galanin GALR2 GAL2 Galr2 Rat Galanin (Mouse) 2 Peptide - - - - 8.3 8.3 8.3 8.8 9.3 Refs
A (Rhodopsin) Galanin GALR3 GAL3 GALR3 Human Galanin (Human) 2 Protein CC(C)C[C@H](NC(=O)CNC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(N)=O)NC(=O)CNC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(C)C)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)O)[C@@H](C)O CBSXZYWGVAQSHI-RUKUCZSXSA-N - 7.2 7.2 Refs
A (Rhodopsin) Galanin GALR3 GAL3 GALR3 Human Galanin (Mouse) 2 Peptide - - - 8.1 8.5 8.8 Refs
A (Rhodopsin) Galanin GALR3 GAL3 GALR3 Human Galanin-Like Peptide (Human) 2 Peptide - - - Refs
A (Rhodopsin) Galanin GALR3 GAL3 GALR3 Human Galanin-Like Peptide (Mouse) 2 Peptide - - -
A (Rhodopsin) Galanin GALR3 GAL3 GALR3 Human Spexin-1 (Human) 1 Peptide - - - 6.2 6.2 Refs
A (Rhodopsin) Galanin GALR3 GAL3 Galr3 Rat Galanin (Mouse) 2 Peptide - - - - 8.1 8.5 8.8 Refs
A (Rhodopsin) Galanin GALR3 GAL3 Galr3 Rat Galanin-Like Peptide (Rat) 2 Peptide - - - - Refs
A (Rhodopsin) Ghrelin GHSR ghrelin GHSR Human [Des-Gln14]Ghrelin (Human) 2 Peptide - - -
A (Rhodopsin) Ghrelin GHSR ghrelin GHSR Human [Des-Gln14]Ghrelin (Mouse) 2 Peptide - - -
A (Rhodopsin) Ghrelin GHSR ghrelin GHSR Human Ghrelin (Human) 1 Peptide - - - - 7.2 8.1 9.5 7.8 8.0 8.1 Refs
A (Rhodopsin) Ghrelin GHSR ghrelin GHSR Human Ghrelin (Mouse) 2 Peptide - - -
A (Rhodopsin) Ghrelin GHSR ghrelin GHSR Human Liver Enriched Antimicrobial Peptide 2 (Human) 2 Peptide - - - AFM_GHSR_HUMAN_hashedseq[GOLYS53WWDIJMUYE6FCJNZ2ZO40] Refs
A (Rhodopsin) Glycoprotein hormone FSHR FSH FSHR Human Fsh (Human) Principal 1 Peptide - - - -
A (Rhodopsin) Glycoprotein hormone FSHR FSH FSHR Human Fsh (Mouse) Principal 1 Peptide - - - -
A (Rhodopsin) Glycoprotein hormone FSHR FSH FSHR Human Fsh (Rat) Principal 1 Peptide - - - -
A (Rhodopsin) Glycoprotein hormone LSHR LH LHCGR Human Lh (Human) 2 Peptide - - - - Refs
A (Rhodopsin) Glycoprotein hormone LSHR LH LHCGR Human Lh (Mouse) 2 Peptide - - - -
A (Rhodopsin) Glycoprotein hormone LSHR LH LHCGR Human Lh (Rat) 2 Peptide - - - -
A (Rhodopsin) Glycoprotein hormone LSHR LH LHCGR Human Hcg (Human) 1 Peptide - - - - Refs
A (Rhodopsin) Glycoprotein hormone TSHR TSH TSHR Human Tsh (Human) Principal 1 Peptide - - - -
A (Rhodopsin) Glycoprotein hormone TSHR TSH TSHR Human Tsh (Mouse) Principal 1 Peptide - - - -
A (Rhodopsin) Glycoprotein hormone TSHR TSH TSHR Human Tsh (Rat) Principal 1 Peptide - - - -
A (Rhodopsin) Gonadotrophin-releasing hormone GNRHR GnRH1 GNRHR Human Gnrh I (Human) 1 Peptide OCC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)N1CCCC1C(=O)NCC(=O)N)CC(C)C)Cc1c[nH]c2c1cccc2)Cc1ccc(cc1)O)NC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C1CCC(=O)N1)Cc1[nH]cnc1 NMJREATYWWNIKX-UHFFFAOYSA-N - - 7.8 7.9 7.9 7.3 6.8 6.8 Refs
A (Rhodopsin) Gonadotrophin-releasing hormone GNRHR GnRH1 GNRHR Human Gnrh Ii (Human) 2 Peptide - - - - Refs
A (Rhodopsin) Gonadotrophin-releasing hormone GNRHR GnRH1 Gnrhr Mouse Gnrh I (Human) 1 Peptide OCC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)N1CCCC1C(=O)NCC(=O)N)CC(C)C)Cc1c[nH]c2c1cccc2)Cc1ccc(cc1)O)NC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C1CCC(=O)N1)Cc1[nH]cnc1 NMJREATYWWNIKX-UHFFFAOYSA-N - - 7.8 7.9 7.9 7.3 6.8 6.8 Refs
A (Rhodopsin) Gonadotrophin-releasing hormone GNRHR GnRH1 Gnrhr Rat Gnrh I (Human) 1 Peptide OCC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)N1CCCC1C(=O)NCC(=O)N)CC(C)C)Cc1c[nH]c2c1cccc2)Cc1ccc(cc1)O)NC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C1CCC(=O)N1)Cc1[nH]cnc1 NMJREATYWWNIKX-UHFFFAOYSA-N - - 7.8 7.9 7.9 7.3 6.8 6.8 Refs
A (Rhodopsin) Histamine HRH1 H1 HRH1 Human Histamine Principal 1 Small molecule NCCc1cnc[nH]1 NTYJJOPFIAHURM-UHFFFAOYSA-N - 7DFL 4.7 5.3 5.9 Refs
A (Rhodopsin) Histamine HRH2 H2 HRH2 Human Histamine Principal 1 Small molecule NCCc1cnc[nH]1 NTYJJOPFIAHURM-UHFFFAOYSA-N - 8YN4
A (Rhodopsin) Histamine HRH2 H2 Hrh2 Rat Histamine Principal 1 Small molecule NCCc1cnc[nH]1 NTYJJOPFIAHURM-UHFFFAOYSA-N - - 3.8 3.8 Refs
A (Rhodopsin) Histamine HRH3 H3 HRH3 Human Histamine Principal 1 Small molecule NCCc1cnc[nH]1 NTYJJOPFIAHURM-UHFFFAOYSA-N - 8YUU 7.2 7.6 7.9 Refs
A (Rhodopsin) Histamine HRH3 H3 Hrh3 Mouse Histamine Principal 1 Small molecule NCCc1cnc[nH]1 NTYJJOPFIAHURM-UHFFFAOYSA-N - - 7.2 7.6 7.9 Refs
A (Rhodopsin) Histamine HRH3 H3 Hrh3 Rat Histamine Principal 1 Small molecule NCCc1cnc[nH]1 NTYJJOPFIAHURM-UHFFFAOYSA-N - - 7.2 7.6 7.9 Refs
A (Rhodopsin) Histamine HRH4 H4 HRH4 Human Ccl16 (Human) 2 Peptide - - - - Refs
A (Rhodopsin) Histamine HRH4 H4 HRH4 Human Histamine None 1 Small molecule NCCc1cnc[nH]1 NTYJJOPFIAHURM-UHFFFAOYSA-N - 9L42 7.8 7.2 7.2 Refs
A (Rhodopsin) Histamine HRH4 H4 Hrh4 Mouse Histamine None 1 Small molecule NCCc1cnc[nH]1 NTYJJOPFIAHURM-UHFFFAOYSA-N - - 7.8 7.2 7.2 Refs
A (Rhodopsin) Histamine HRH4 H4 Hrh4 Rat Histamine None 1 Small molecule NCCc1cnc[nH]1 NTYJJOPFIAHURM-UHFFFAOYSA-N - - 7.8 7.2 7.2 Refs
A (Rhodopsin) Hydroxycarboxylic acid HCAR1 HCA1 HCAR1 Human D-Lactic Acid Principal 1 Small molecule OC(=O)[C@H](O)C JVTAAEKCZFNVCJ-UWTATZPHSA-N - 8Z8A 2.2 2.5 2.8 Refs
A (Rhodopsin) Hydroxycarboxylic acid HCAR1 HCA1 Hcar1 Mouse D-Lactic Acid Principal 1 Small molecule OC(=O)[C@H](O)C JVTAAEKCZFNVCJ-UWTATZPHSA-N - - 2.2 2.5 2.8 Refs
A (Rhodopsin) Hydroxycarboxylic acid HCAR2 HCA2 HCAR2 Human Β-D-Hydroxybutyric Acid None 1 Small molecule C[C@H](CC(=O)O)O WHBMMWSBFZVSSR-GSVOUGTGSA-N - 8J6Q 3.5 3.5 Refs
A (Rhodopsin) Hydroxycarboxylic acid HCAR2 HCA2 HCAR2 Human Butyric Acid None 2 Small molecule CCCC(=O)O FERIUCNNQQJTOY-UHFFFAOYSA-N - - 2.8 2.8
A (Rhodopsin) Hydroxycarboxylic acid HCAR2 HCA2 Hcar2 Mouse Β-D-Hydroxybutyric Acid None 1 Small molecule C[C@H](CC(=O)O)O WHBMMWSBFZVSSR-GSVOUGTGSA-N - - 3.5 3.5 Refs
A (Rhodopsin) Hydroxycarboxylic acid HCAR3 HCA3 HCAR3 Human 3-Hydroxyoctanoic Acid Principal 1 Small molecule CCCCC[C@@H](CC(=O)O)O NDPLAKGOSZHTPH-ZETCQYMHSA-N - 8JEF 5.1 5.1 Refs
A (Rhodopsin) Kisspeptin KISSR kisspeptin KISS1R Human Kisspeptin-10 (Human) 1 Peptide OC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccccc1)CCCN=C(N)N)CC(C)C)Cc1ccccc1)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccc(cc1)O)N)CC(=O)N)CC(=O)N RITKWYDZSSQNJI-INXYWQKQSA-N - 8ZJD 8.6 9.5 10.4 Refs
A (Rhodopsin) Kisspeptin KISSR kisspeptin KISS1R Human Kisspeptin-10 (Mouse) 5 Peptide - - -
A (Rhodopsin) Kisspeptin KISSR kisspeptin KISS1R Human Kisspeptin-13 (Human) 4 Peptide - - - 8.4 8.4 Refs
A (Rhodopsin) Kisspeptin KISSR kisspeptin KISS1R Human Kisspeptin-14 (Human) 3 Peptide - - - 8.8 8.8 Refs
A (Rhodopsin) Kisspeptin KISSR kisspeptin KISS1R Human Kisspeptin-52 (Mouse) 5 Peptide - - -
A (Rhodopsin) Kisspeptin KISSR kisspeptin KISS1R Human Kisspeptin-52 (Rat) 5 Peptide - - -
A (Rhodopsin) Kisspeptin KISSR kisspeptin KISS1R Human Kisspeptin-54 (Human) 2 Peptide - - - 8.8 9.2 9.5 Refs
A (Rhodopsin) Leukotriene CLTR1 CysLT1 CYSLTR1 Human Ltc4 None 2 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SC[C@@H](C(=O)NCC(=O)O)NC(=O)CC[C@@H](C(=O)O)N GWNVDXQDILPJIG-NXOLIXFESA-N - - 7.4 7.6 7.7 7.0 7.6 8.1 Refs
A (Rhodopsin) Leukotriene CLTR1 CysLT1 CYSLTR1 Human Ltd4 None 1 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SCC(C(=O)NCC(=O)O)N YEESKJGWJFYOOK-LDDGIIIKSA-N - - 7.3 8.6 9.4 Refs
A (Rhodopsin) Leukotriene CLTR1 CysLT1 CYSLTR1 Human Lte4 None 3 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SC[C@@H](C(=O)O)N OTZRAYGBFWZKMX-FRFVZSDQSA-N - - 6.4 6.7 7.2 7.1 7.5 7.8 Refs
A (Rhodopsin) Leukotriene CLTR2 CysLT2 CYSLTR2 Human Ltc4 None 1 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SC[C@@H](C(=O)NCC(=O)O)NC(=O)CC[C@@H](C(=O)O)N GWNVDXQDILPJIG-NXOLIXFESA-N - 9UAM 7.0 7.6 8.6 Refs
A (Rhodopsin) Leukotriene CLTR2 CysLT2 CYSLTR2 Human Ltd4 None 2 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SCC(C(=O)NCC(=O)O)N YEESKJGWJFYOOK-LDDGIIIKSA-N - 9IXX 6.8 7.6 8.6 7.3 7.7 8.1 Refs
A (Rhodopsin) Leukotriene CLTR2 CysLT2 CYSLTR2 Human Lte4 None 3 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SC[C@@H](C(=O)O)N OTZRAYGBFWZKMX-FRFVZSDQSA-N - - 5.6 6.3 7.1 6.5 6.5 Refs
A (Rhodopsin) Leukotriene LT4R1 BLT1 LTB4R Human 12r-Hete None 3 Small molecule CCCCC/C=C\C[C@H](/C=C/C=C\C/C=C\CCCC(=O)O)O ZNHVWPKMFKADKW-ZYBDYUKJSA-N - - 7.5 7.5 Refs
A (Rhodopsin) Leukotriene LT4R1 BLT1 LTB4R Human 20-Hydroxy-Ltb4 None 2 Small molecule OCCCCC/C=C\C[C@H](/C=C/C=C/C=C\[C@H](CCCC(=O)O)O)O PTJFJXLGRSTECQ-PSPARDEHSA-N - - 8.1 8.1 Refs
A (Rhodopsin) Leukotriene LT4R1 BLT1 LTB4R Human Ltb4 None 1 Small molecule CCCCC/C=C\C[C@H](/C=C/C=C/C=C\[C@H](CCCC(=O)O)O)O VNYSSYRCGWBHLG-AMOLWHMGSA-N - 7VKT 9.4 9.4
A (Rhodopsin) Leukotriene LT4R2 BLT2 LTB4R2 Human 12-Epi Ltb4 None 2 Small molecule CCCCC/C=C\C[C@@H](/C=C/C=C/C=C\[C@H](CCCC(=O)O)O)O VNYSSYRCGWBHLG-CBBLYLIKSA-N - - 7.5 7.5 Refs
A (Rhodopsin) Leukotriene LT4R2 BLT2 LTB4R2 Human 12-Hydroxyheptadecatrienoic Acid None 1 Small molecule CCCCC[C@@H](/C=C/C=C/C/C=C\CCCC(=O)O)O KUKJHGXXZWHSBG-WBGSEQOASA-N - - 7.7 7.7 Refs
A (Rhodopsin) Leukotriene LT4R2 BLT2 LTB4R2 Human 12r-Hete 4 Small molecule CCCCC/C=C\C[C@H](/C=C/C=C\C/C=C\CCCC(=O)O)O ZNHVWPKMFKADKW-ZYBDYUKJSA-N - -
A (Rhodopsin) Leukotriene LT4R2 BLT2 LTB4R2 Human 12s-Hete None 2 Small molecule CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O ZNHVWPKMFKADKW-LQWMCKPYSA-N - - 7.5 7.5 Refs
A (Rhodopsin) Leukotriene LT4R2 BLT2 LTB4R2 Human 12s-Hpete 4 Small molecule CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)OO ZIOZYRSDNLNNNJ-LQWMCKPYSA-N - -
A (Rhodopsin) Leukotriene LT4R2 BLT2 LTB4R2 Human 15s-Hete None 2 Small molecule CCCCC[C@@H](/C=C/C=C\C/C=C\C/C=C\CCCC(=O)O)O JSFATNQSLKRBCI-VAEKSGALSA-N - - 7.5 7.5 Refs
A (Rhodopsin) Leukotriene LT4R2 BLT2 LTB4R2 Human 20-Hydroxy-Ltb4 4 Small molecule OCCCCC/C=C\C[C@H](/C=C/C=C/C=C\[C@H](CCCC(=O)O)O)O PTJFJXLGRSTECQ-PSPARDEHSA-N - -
A (Rhodopsin) Leukotriene LT4R2 BLT2 LTB4R2 Human Ltb4 None 3 Small molecule CCCCC/C=C\C[C@H](/C=C/C=C/C=C\[C@H](CCCC(=O)O)O)O VNYSSYRCGWBHLG-AMOLWHMGSA-N - - 6.8 6.8 Refs
A (Rhodopsin) Leukotriene OXER1 OXE OXER1 Human 5-Oxo-12-Hete None 7 Small molecule CCCCC/C=C\C[C@@H](/C=C/C=C\C=C\C(=O)CCCC(=O)O)O MLZJFLKEKVDNAZ-XPKTZJOPSA-N - - Refs
A (Rhodopsin) Leukotriene OXER1 OXE OXER1 Human 5-Oxo-15-Hete None 3 Small molecule CCCCC[C@@H](/C=C/C=C\C/C=C\C=C\C(=O)CCCC(=O)O)O RIUDRKHGFDAKPO-WWWYWCMOSA-N - - 7.7 7.7 Refs
A (Rhodopsin) Leukotriene OXER1 OXE OXER1 Human 5-Oxo-20-Hete None 6 Small molecule OCCCCC/C=C\C/C=C\C/C=C\C=C\C(=O)CCCC(=O)O DTSRZRUIWKDHMR-DHYYJNSCSA-N - - 6.5 6.5 Refs
A (Rhodopsin) Leukotriene OXER1 OXE OXER1 Human 5-Oxo-C20:3 None 2 Small molecule CCCCCCCC/C=C\C/C=C\C=C/C(=O)CCCC(=O)O ULMVEQWNDGUUBR-IEQFDQMRSA-N - - 8.0 8.0 Refs
A (Rhodopsin) Leukotriene OXER1 OXE OXER1 Human 5-Oxo-Ete None 1 Small molecule CCCCC/C=C\C/C=C\C/C=C\C=C\C(=O)CCCC(=O)O MEASLHGILYBXFO-XTDASVJISA-N - - 8.3 8.4 8.5 Refs
A (Rhodopsin) Leukotriene OXER1 OXE OXER1 Human 5-Oxo-Ode None 2 Lipid CCCCCCCCC/C=C\C=C\C(=O)CCCC(=O)O YVWMHFYOIJMUMN-HSINTONASA-N - - 8.0 8.0 Refs
A (Rhodopsin) Leukotriene OXER1 OXE OXER1 Human 5s-Hete None 5 Small molecule CCCCC/C=C\C/C=C\C/C=C\C=C\[C@H](CCCC(=O)O)O KGIJOOYOSFUGPC-JGKLHWIESA-N - - 6.5 6.9 7.2 Refs
A (Rhodopsin) Leukotriene OXER1 OXE OXER1 Human 5s-Hpete None 4 Small molecule CCCCC/C=C\C/C=C\C/C=C\C=C\[C@H](CCCC(=O)O)OO JNUUNUQHXIOFDA-JGKLHWIESA-N - - 7.0 7.0 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR1 LPA1 LPAR1 Human Lpa Principal 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - -
A (Rhodopsin) Lysophospholipid (LPA) LPAR1 LPA1 Lpar1 Mouse Lpa Principal 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 7.9 8.1 8.3 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR2 LPA2 LPAR2 Human Lpa None 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 8.0 8.1 8.2 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR2 LPA2 LPAR2 Human Farnesyl Diphosphate None 2 Small molecule C/C(=C/COP(=O)(OP(=O)(O)O)O)/CC/C=C(\CCC=C(C)C)/C VWFJDQUYCIWHTN-FBXUGWQNSA-N - - Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR2 LPA2 LPAR2 Human Farnesyl Monophosphate None 2 Small molecule C/C(=C/CC/C(=C\COP(=O)(O)O)/C)/CCC=C(C)C ALEWCKXBHSDCCT-FBXUGWQNSA-N - Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR2 LPA2 Lpar2 Mouse Lpa None 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 8.0 8.1 8.2 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR3 LPA3 LPAR3 Human Lpa None 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 6.6 6.6 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR3 LPA3 LPAR3 Human Farnesyl Diphosphate None 2 Small molecule C/C(=C/COP(=O)(OP(=O)(O)O)O)/CC/C=C(\CCC=C(C)C)/C VWFJDQUYCIWHTN-FBXUGWQNSA-N - - Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR3 LPA3 LPAR3 Human Farnesyl Monophosphate None 2 Small molecule C/C(=C/CC/C(=C\COP(=O)(O)O)/C)/CCC=C(C)C ALEWCKXBHSDCCT-FBXUGWQNSA-N - Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR3 LPA3 Lpar3 Mouse Lpa None 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 6.6 6.6 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR4 LPA4 LPAR4 Human Lpa None 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR4 LPA4 LPAR4 Human Farnesyl Diphosphate None 2 Small molecule C/C(=C/COP(=O)(OP(=O)(O)O)O)/CC/C=C(\CCC=C(C)C)/C VWFJDQUYCIWHTN-FBXUGWQNSA-N - - Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR4 LPA4 Lpar4 Mouse Lpa None 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR5 LPA5 LPAR5 Human Lpa None 3 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 4.3 6.1 7.9 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR5 LPA5 LPAR5 Human N-Arachidonoylglycine None 4 Small molecule CCCCC/C=C\C/C=C\C/C=C\C/C=C\CCCC(=O)NCC(=O)O YLEARPUNMCCKMP-DOFZRALJSA-N - - 4.3 4.3 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR5 LPA5 LPAR5 Human Farnesyl Diphosphate None 2 Small molecule C/C(=C/COP(=O)(OP(=O)(O)O)O)/CC/C=C(\CCC=C(C)C)/C VWFJDQUYCIWHTN-FBXUGWQNSA-N - - 5.8 6.2 6.5 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR5 LPA5 LPAR5 Human Farnesyl Monophosphate None 1 Small molecule C/C(=C/CC/C(=C\COP(=O)(O)O)/C)/CCC=C(C)C ALEWCKXBHSDCCT-FBXUGWQNSA-N - - 7.3 7.3 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR6 LPA6 LPAR6 Human Lpa Principal 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 6.0 6.0 Refs
A (Rhodopsin) Lysophospholipid (LPA) LPAR6 LPA6 Lpar6 Mouse Lpa Principal 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 6.0 6.0 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR1 S1P1 S1PR1 Human Dihydrosphingosine 1-Phosphate 2 Lipid CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O YHEDRJPUIRMZMP-ZWKOTPCHSA-N -
A (Rhodopsin) Lysophospholipid (S1P) S1PR1 S1P1 S1PR1 Human Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - 7TD3 7.1 8.7 9.5 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR1 S1P1 S1PR1 Human Sphingosylphosphorylcholine 2 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(OCC[N+](C)(C)C)[O-])N)O JLVSPVFPBBFMBE-HXSWCURESA-N - -
A (Rhodopsin) Lysophospholipid (S1P) S1PR2 S1P2 S1PR2 Human Dihydrosphingosine 1-Phosphate 2 Lipid CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O YHEDRJPUIRMZMP-ZWKOTPCHSA-N -
A (Rhodopsin) Lysophospholipid (S1P) S1PR2 S1P2 S1PR2 Human Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - 7T6B 8.1 8.7 8.7 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR2 S1P2 S1PR2 Human Sphingosylphosphorylcholine 2 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(OCC[N+](C)(C)C)[O-])N)O JLVSPVFPBBFMBE-HXSWCURESA-N - -
A (Rhodopsin) Lysophospholipid (S1P) S1PR2 S1P2 S1pr2 Mouse Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 8.1 8.7 8.7 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR3 S1P3 S1PR3 Human Dihydrosphingosine 1-Phosphate 2 Lipid CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O YHEDRJPUIRMZMP-ZWKOTPCHSA-N -
A (Rhodopsin) Lysophospholipid (S1P) S1PR3 S1P3 S1PR3 Human Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - 9WP9 8.4 8.6 8.6 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR3 S1P3 S1PR3 Human Sphingosylphosphorylcholine 2 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(OCC[N+](C)(C)C)[O-])N)O JLVSPVFPBBFMBE-HXSWCURESA-N - -
A (Rhodopsin) Lysophospholipid (S1P) S1PR3 S1P3 S1pr3 Mouse Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 8.4 8.6 8.6 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR4 S1P4 S1PR4 Human Dihydrosphingosine 1-Phosphate None 2 Lipid CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O YHEDRJPUIRMZMP-ZWKOTPCHSA-N - -
A (Rhodopsin) Lysophospholipid (S1P) S1PR4 S1P4 S1PR4 Human Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - 7.2 7.1 7.1 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR4 S1P4 S1PR4 Human Sphingosylphosphorylcholine 2 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(OCC[N+](C)(C)C)[O-])N)O JLVSPVFPBBFMBE-HXSWCURESA-N - -
A (Rhodopsin) Lysophospholipid (S1P) S1PR4 S1P4 S1pr4 Mouse Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 7.2 7.1 7.1 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR5 S1P5 S1PR5 Human Dihydrosphingosine 1-Phosphate 2 Lipid CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O YHEDRJPUIRMZMP-ZWKOTPCHSA-N - -
A (Rhodopsin) Lysophospholipid (S1P) S1PR5 S1P5 S1PR5 Human Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 7.8 7.9 7.9 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR5 S1P5 S1PR5 Human Sphingosylphosphorylcholine 2 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(OCC[N+](C)(C)C)[O-])N)O JLVSPVFPBBFMBE-HXSWCURESA-N - -
A (Rhodopsin) Lysophospholipid (S1P) S1PR5 S1P5 S1pr5 Mouse Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 7.8 7.9 7.9 Refs
A (Rhodopsin) Lysophospholipid (S1P) S1PR5 S1P5 S1pr5 Rat Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 7.8 7.9 7.9 Refs
A (Rhodopsin) Melanin-concentrating hormon MCHR1 MCH1 MCHR1 Human Melanin-Concentrating Hormone (Human) Principal 1 Peptide CSCCC1NC(=O)C(CSSCC(NC(=O)C2CCCN2C(=O)C(CCCNC(=N)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)CNC(=O)C(NC1=O)C(C)C)CCCNC(=N)N)C(C)C)Cc1ccc(cc1)O)C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)C(C)C)CCC(=O)O)Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(CC(=O)O)N)CCSC)CCCNC(=N)N ORRDHOMWDPJSNL-UHFFFAOYSA-N - 8WSS 9.8 9.9 10.0 Refs
A (Rhodopsin) Melanin-concentrating hormon MCHR1 MCH1 Mchr1 Rat Melanin-Concentrating Hormone (Human) Principal 1 Peptide CSCCC1NC(=O)C(CSSCC(NC(=O)C2CCCN2C(=O)C(CCCNC(=N)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)CNC(=O)C(NC1=O)C(C)C)CCCNC(=N)N)C(C)C)Cc1ccc(cc1)O)C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)C(C)C)CCC(=O)O)Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(CC(=O)O)N)CCSC)CCCNC(=N)N ORRDHOMWDPJSNL-UHFFFAOYSA-N - - 9.8 9.9 10.0 Refs
A (Rhodopsin) Melanin-concentrating hormon MCHR2 MCH2 MCHR2 Human Melanin-Concentrating Hormone (Human) Principal 1 Peptide CSCCC1NC(=O)C(CSSCC(NC(=O)C2CCCN2C(=O)C(CCCNC(=N)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)CNC(=O)C(NC1=O)C(C)C)CCCNC(=N)N)C(C)C)Cc1ccc(cc1)O)C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)C(C)C)CCC(=O)O)Cc1c[nH]c2c1cccc2)NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(CC(=O)O)N)CCSC)CCCNC(=N)N ORRDHOMWDPJSNL-UHFFFAOYSA-N - 8WST Refs
A (Rhodopsin) Melanocortin ACTHR MC2 MC2R Human Acth (Human) Principal 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1ccccc1)CCC(=O)O)CC(C)C)Cc1ccccc1)C)CCC(=O)O)C)CO)CCC(=O)O)CC(=O)O)CCC(=O)O)C)CC(=O)N)Cc1ccc(cc1)O)C(C)C)NC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)CNC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)Cc1ccc(cc1)O)CO)CCSC)CCC(=O)O)Cc1nc[nH]c1)Cc1ccccc1)CCCN=C(N)N)CCCCN)CCCCN)CCCCN)CCCN=C(N)N)CCCN=C(N)N IDLFZVILOHSSID-OVLDLUHVSA-N -
A (Rhodopsin) Melanocortin ACTHR MC2 MC2R Human Acth (Mouse) Principal 1 Peptide - - - Refs
A (Rhodopsin) Melanocortin ACTHR MC2 Mc2r Mouse Acth (Mouse) Principal 1 Peptide - - - - Refs
A (Rhodopsin) Melanocortin MC3R MC3 MC3R Human Α-Msh (Human) 1 Peptide - - - 8.0 8.2 8.4 Refs
A (Rhodopsin) Melanocortin MC3R MC3 MC3R Human Β-Msh (Human) 3 Peptide - - -
A (Rhodopsin) Melanocortin MC3R MC3 MC3R Human Β-Msh (Mouse) 3 Peptide - - -
A (Rhodopsin) Melanocortin MC3R MC3 MC3R Human Β-Msh (Rat) 3 Peptide - - -
A (Rhodopsin) Melanocortin MC3R MC3 MC3R Human Γ-Msh (Human) 3 Peptide - - - 8IOC Refs
A (Rhodopsin) Melanocortin MC3R MC3 MC3R Human Acth (Human) 2 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1ccccc1)CCC(=O)O)CC(C)C)Cc1ccccc1)C)CCC(=O)O)C)CO)CCC(=O)O)CC(=O)O)CCC(=O)O)C)CC(=O)N)Cc1ccc(cc1)O)C(C)C)NC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)CNC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)Cc1ccc(cc1)O)CO)CCSC)CCC(=O)O)Cc1nc[nH]c1)Cc1ccccc1)CCCN=C(N)N)CCCCN)CCCCN)CCCCN)CCCN=C(N)N)CCCN=C(N)N IDLFZVILOHSSID-OVLDLUHVSA-N - 7.1 7.1 Refs
A (Rhodopsin) Melanocortin MC3R MC3 MC3R Human Acth (Mouse) 3 Peptide - - -
A (Rhodopsin) Melanocortin MC3R MC3 MC3R Human Agouti-Related Protein (Human) 3 Peptide - - - Refs
A (Rhodopsin) Melanocortin MC3R MC3 Mc3r Mouse Agouti (Mouse) 3 Peptide - - - - Refs
A (Rhodopsin) Melanocortin MC4R MC4 MC4R Human Α-Msh (Human) 1 Peptide - - - 7.4 7.7 8.0 Refs
A (Rhodopsin) Melanocortin MC4R MC4 MC4R Human Β-Msh (Human) 3 Peptide - - -
A (Rhodopsin) Melanocortin MC4R MC4 MC4R Human Β-Msh (Mouse) 3 Peptide - - -
A (Rhodopsin) Melanocortin MC4R MC4 MC4R Human Β-Msh (Rat) 3 Peptide - - -
A (Rhodopsin) Melanocortin MC4R MC4 MC4R Human Γ-Msh (Human) 3 Peptide - - -
A (Rhodopsin) Melanocortin MC4R MC4 MC4R Human Acth (Human) 2 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1ccccc1)CCC(=O)O)CC(C)C)Cc1ccccc1)C)CCC(=O)O)C)CO)CCC(=O)O)CC(=O)O)CCC(=O)O)C)CC(=O)N)Cc1ccc(cc1)O)C(C)C)NC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)CNC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)Cc1ccc(cc1)O)CO)CCSC)CCC(=O)O)Cc1nc[nH]c1)Cc1ccccc1)CCCN=C(N)N)CCCCN)CCCCN)CCCCN)CCCN=C(N)N)CCCN=C(N)N IDLFZVILOHSSID-OVLDLUHVSA-N - 6.2 6.2 Refs
A (Rhodopsin) Melanocortin MC4R MC4 MC4R Human Acth (Mouse) 3 Peptide - - -
A (Rhodopsin) Melanocortin MC4R MC4 MC4R Human Agouti-Related Protein (Human) 3 Peptide - - - Refs
A (Rhodopsin) Melanocortin MC4R MC4 Mc4r Mouse Agouti (Mouse) 3 Peptide - - - - Refs
A (Rhodopsin) Melanocortin MC5R MC5 MC5R Human Α-Msh (Human) 2 Peptide - - - Refs
A (Rhodopsin) Melanocortin MC5R MC5 MC5R Human Β-Msh (Human) 2 Peptide - - -
A (Rhodopsin) Melanocortin MC5R MC5 MC5R Human Β-Msh (Mouse) 2 Peptide - - -
A (Rhodopsin) Melanocortin MC5R MC5 MC5R Human Β-Msh (Rat) 2 Peptide - - -
A (Rhodopsin) Melanocortin MC5R MC5 MC5R Human Γ-Msh (Human) 2 Peptide - - -
A (Rhodopsin) Melanocortin MC5R MC5 MC5R Human Acth (Human) 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1ccccc1)CCC(=O)O)CC(C)C)Cc1ccccc1)C)CCC(=O)O)C)CO)CCC(=O)O)CC(=O)O)CCC(=O)O)C)CC(=O)N)Cc1ccc(cc1)O)C(C)C)NC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)CNC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)Cc1ccc(cc1)O)CO)CCSC)CCC(=O)O)Cc1nc[nH]c1)Cc1ccccc1)CCCN=C(N)N)CCCCN)CCCCN)CCCCN)CCCN=C(N)N)CCCN=C(N)N IDLFZVILOHSSID-OVLDLUHVSA-N - 5.0 5.0 Refs
A (Rhodopsin) Melanocortin MC5R MC5 MC5R Human Acth (Mouse) 2 Peptide - - -
A (Rhodopsin) Melanocortin MC5R MC5 MC5R Human Agouti-Related Protein (Human) 2 Peptide - - - Refs
A (Rhodopsin) Melanocortin MC5R MC5 Mc5r Mouse Agouti (Mouse) 2 Peptide - - - - Refs
A (Rhodopsin) Melanocortin MSHR MC1 MC1R Human Α-Msh (Human) 2 Peptide - - - Refs
A (Rhodopsin) Melanocortin MSHR MC1 MC1R Human Β-Msh (Human) 2 Peptide - - -
A (Rhodopsin) Melanocortin MSHR MC1 MC1R Human Β-Msh (Mouse) 2 Peptide - - -
A (Rhodopsin) Melanocortin MSHR MC1 MC1R Human Β-Msh (Rat) 2 Peptide - - -
A (Rhodopsin) Melanocortin MSHR MC1 MC1R Human Γ-Msh (Human) 2 Peptide - - -
A (Rhodopsin) Melanocortin MSHR MC1 MC1R Human Acth (Human) 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)Cc1ccccc1)CCC(=O)O)CC(C)C)Cc1ccccc1)C)CCC(=O)O)C)CO)CCC(=O)O)CC(=O)O)CCC(=O)O)C)CC(=O)N)Cc1ccc(cc1)O)C(C)C)NC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@H](C(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)CNC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)Cc1ccc(cc1)O)CO)CCSC)CCC(=O)O)Cc1nc[nH]c1)Cc1ccccc1)CCCN=C(N)N)CCCCN)CCCCN)CCCCN)CCCN=C(N)N)CCCN=C(N)N IDLFZVILOHSSID-OVLDLUHVSA-N - 8.6 8.6 Refs
A (Rhodopsin) Melanocortin MSHR MC1 MC1R Human Acth (Mouse) 2 Peptide - - -
A (Rhodopsin) Melanocortin MSHR MC1 Mc1r Mouse Agouti (Mouse) 2 Peptide - - - - Refs
A (Rhodopsin) Melatonin MTR1A MT1 MTNR1A Human Melatonin Principal 1 Small molecule COc1ccc2c(c1)c(CCNC(=O)C)c[nH]2 DRLFMBDRBRZALE-UHFFFAOYSA-N - - 9.1 9.4 9.7 Refs
A (Rhodopsin) Melatonin MTR1B MT2 MTNR1B Human Melatonin Principal 1 Small molecule COc1ccc2c(c1)c(CCNC(=O)C)c[nH]2 DRLFMBDRBRZALE-UHFFFAOYSA-N - - 9.4 9.6 9.8 Refs
A (Rhodopsin) Motilin MTLR motilin MLNR Human Motilin (Human) Principal 1 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)O)CCC(=O)N)CCCCN)CC(=O)N)CCCNC(=N)N)CCC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@H]([C@H](CC)C)NC(=O)[C@@H]1CCCN1C(=O)[C@H](C(C)C)NC(=O)[C@H](Cc1ccccc1)N)Cc1ccccc1)Cc1ccc(cc1)O)CCC(=O)O)CC(C)C)CCC(=O)N)CCCNC(=N)N)CCSC)CCC(=O)N)CCC(=O)O LVRVABPNVHYXRT-BQWXUCBYSA-N - 8IBV 8.4 8.6 8.7 Refs
A (Rhodopsin) Neuromedin U NMUR1 NMU1 NMUR1 Human Neuromedin S-33 (Human) 1 Peptide - - - - 10.2 10.2 Refs
A (Rhodopsin) Neuromedin U NMUR1 NMU1 NMUR1 Human Neuromedin S-36 (Mouse) 3 Peptide - - - -
A (Rhodopsin) Neuromedin U NMUR1 NMU1 NMUR1 Human Neuromedin S-36 (Rat) 3 Peptide - - - -
A (Rhodopsin) Neuromedin U NMUR1 NMU1 NMUR1 Human Neuromedin U-23 (Mouse) 3 Peptide - - - -
A (Rhodopsin) Neuromedin U NMUR1 NMU1 NMUR1 Human Neuromedin U-23 (Rat) 3 Peptide - - - -
A (Rhodopsin) Neuromedin U NMUR1 NMU1 NMUR1 Human Neuromedin U-25 (Human) 2 Protein - - - 8.4 8.9 9.4 9.5 9.5 Refs
A (Rhodopsin) Neuromedin U NMUR2 NMU2 NMUR2 Human Neuromedin S-33 (Human) 1 Peptide - - - 10.0 10.0 Refs
A (Rhodopsin) Neuromedin U NMUR2 NMU2 NMUR2 Human Neuromedin S-36 (Mouse) 3 Peptide - - -
A (Rhodopsin) Neuromedin U NMUR2 NMU2 NMUR2 Human Neuromedin S-36 (Rat) 3 Peptide - - -
A (Rhodopsin) Neuromedin U NMUR2 NMU2 NMUR2 Human Neuromedin U-23 (Rat) 3 Peptide - - -
A (Rhodopsin) Neuromedin U NMUR2 NMU2 NMUR2 Human Neuromedin U-25 (Human) 2 Protein - - - 8.4 8.9 9.4 9.6 9.6 Refs
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Prrp-31 (Human) 3 Peptide - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Qrfp43 (43rfa) (Human) 3 Peptide - - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Rfrp-1 (Human) 3 Peptide - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Rfrp-3 (Human) 1 Peptide - - - 9.2 9.3 9.3 Refs
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Neuropeptide Af (Human) 3 Peptide CC(C)C[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](C)N)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)O YPBGORNZMUQFSF-KWFINLGMSA-N -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Neuropeptide Af (Mouse) 3 Peptide - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Neuropeptide Af (Rat) 3 Peptide - - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Neuropeptide Ff (Human) 2 Peptide - - - 9VIF 8.5 9.2 9.9 Refs
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Neuropeptide Sf (Human) 3 Peptide - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Neuropeptide Sf (Mouse) 3 Peptide - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF1 NPFF1 NPFFR1 Human Neuropeptide Sf (Rat) 3 Peptide - - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF2 NPFF2 NPFFR2 Human Prrp-31 (Human) 3 Peptide - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF2 NPFF2 NPFFR2 Human Qrfp43 (43rfa) (Human) 3 Peptide - - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF2 NPFF2 NPFFR2 Human Rfrp-1 (Human) 3 Peptide - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF2 NPFF2 NPFFR2 Human Rfrp-3 (Human) 2 Peptide - - - 7.8 7.8 Refs
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF2 NPFF2 NPFFR2 Human Neuropeptide Af (Human) 3 Peptide CC(C)C[C@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)CNC(=O)[C@H](C)N)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)O YPBGORNZMUQFSF-KWFINLGMSA-N -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF2 NPFF2 NPFFR2 Human Neuropeptide Af (Mouse) 3 Peptide - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF2 NPFF2 NPFFR2 Human Neuropeptide Af (Rat) 3 Peptide - - - -
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF2 NPFF2 NPFFR2 Human Neuropeptide Ff (Human) 1 Peptide - - - 9M1O 9.7 9.7 Refs
A (Rhodopsin) Neuropeptide FF/neuropeptide AF NPFF2 NPFF2 NPFFR2 Human Neuropeptide Sf (Human) 3 Peptide - - -
A (Rhodopsin) Neuropeptide S NPSR1 NPS NPSR1 Human Neuropeptide S (Human) Principal 1 Protein - - - - 7.3 7.7 8.0 Refs
A (Rhodopsin) Neuropeptide S NPSR1 NPS NPSR1 Human Neuropeptide S (Mouse) Principal 1 Protein - - -
A (Rhodopsin) Neuropeptide S NPSR1 NPS NPSR1 Human Neuropeptide S (Rat) Principal 1 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Des-Br-Neuropeptide B-23 (Human) 4 Peptide - - - Refs
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Des-Br-Neuropeptide B-29 (Human) 3 Peptide - - - Refs
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide B-23 (Human) 5 Peptide - - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide B-23 (Mouse) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide B-23 (Rat) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide B-29 (Human) 3 Peptide - - - - Refs
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide B-29 (Mouse) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide B-29 (Rat) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide W-23 (Human) 2 Peptide - - - Refs
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide W-23 (Mouse) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide W-30 (Human) 1 Peptide - - - Refs
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide W-30 (Mouse) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW1 NPBW1 NPBWR1 Human Neuropeptide W-30 (Rat) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide B-23 (Human) 4 Peptide - - - - Refs
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide B-23 (Mouse) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide B-23 (Rat) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide B-29 (Human) 3 Peptide - - - - Refs
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide B-29 (Mouse) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide B-29 (Rat) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide W-23 (Human) 1 Peptide - - - Refs
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide W-23 (Mouse) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide W-30 (Human) 2 Peptide - - - Refs
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide W-30 (Mouse) 5 Peptide - - -
A (Rhodopsin) Neuropeptide W/neuropeptide B NPBW2 NPBW2 NPBWR2 Human Neuropeptide W-30 (Rat) 5 Peptide - - -
A (Rhodopsin) Neuropeptide Y NPY1R Y1 NPY1R Human Neuropeptide Y (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccc(cc1)O)CCCN=C(N)N)CCC(=O)N)CCCN=C(N)N)[C@H](O)C)[C@H](CC)C)CC(C)C)CC(=O)N)[C@H](CC)C)Cc1ccc(cc1)O)Cc1c[nH]cn1)CCCN=C(N)N)CC(C)C)C)CO)Cc1ccc(cc1)O)Cc1ccc(cc1)O)CCCN=C(N)N)C)CCSC)CC(=O)O)CCC(=O)O)C)C)CC(=O)O)CCC(=O)O)CC(=O)N)CC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(cc1)O)N)CO XKWCTHKJQNUFOQ-HRPSIEBRSA-N - - 10.5 10.5 Refs
A (Rhodopsin) Neuropeptide Y NPY1R Y1 NPY1R Human Pancreatic Polypeptide (Human) 4 Protein - - -
A (Rhodopsin) Neuropeptide Y NPY1R Y1 NPY1R Human Pancreatic Polypeptide (Mouse) 4 Peptide - - -
A (Rhodopsin) Neuropeptide Y NPY1R Y1 NPY1R Human Peptide Yy (Human) 4 Peptide - - -
A (Rhodopsin) Neuropeptide Y NPY1R Y1 NPY1R Human Peptide Yy (Mouse) 2 Protein - - - 10.2 10.2 Refs
A (Rhodopsin) Neuropeptide Y NPY1R Y1 Npy1r Rat Neuropeptide Y (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccc(cc1)O)CCCN=C(N)N)CCC(=O)N)CCCN=C(N)N)[C@H](O)C)[C@H](CC)C)CC(C)C)CC(=O)N)[C@H](CC)C)Cc1ccc(cc1)O)Cc1c[nH]cn1)CCCN=C(N)N)CC(C)C)C)CO)Cc1ccc(cc1)O)Cc1ccc(cc1)O)CCCN=C(N)N)C)CCSC)CC(=O)O)CCC(=O)O)C)C)CC(=O)O)CCC(=O)O)CC(=O)N)CC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(cc1)O)N)CO XKWCTHKJQNUFOQ-HRPSIEBRSA-N - - 10.5 10.5 Refs
A (Rhodopsin) Neuropeptide Y NPY1R Y1 Npy1r Rat Pancreatic Polypeptide (Rat) 3 Peptide - - - - 7.0 7.0 Refs
A (Rhodopsin) Neuropeptide Y NPY1R Y1 Npy1r Rat Peptide Yy (Mouse) 2 Protein - - - - 10.2 10.2 Refs
A (Rhodopsin) Neuropeptide Y NPY2R Y2 NPY2R Human Pyy-(3-36) (Human) 3 Protein - - - 9.2 9.5 9.7 Refs
A (Rhodopsin) Neuropeptide Y NPY2R Y2 NPY2R Human Neuropeptide Y (Human) 4 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccc(cc1)O)CCCN=C(N)N)CCC(=O)N)CCCN=C(N)N)[C@H](O)C)[C@H](CC)C)CC(C)C)CC(=O)N)[C@H](CC)C)Cc1ccc(cc1)O)Cc1c[nH]cn1)CCCN=C(N)N)CC(C)C)C)CO)Cc1ccc(cc1)O)Cc1ccc(cc1)O)CCCN=C(N)N)C)CCSC)CC(=O)O)CCC(=O)O)C)C)CC(=O)O)CCC(=O)O)CC(=O)N)CC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(cc1)O)N)CO XKWCTHKJQNUFOQ-HRPSIEBRSA-N - - 9.3 9.4 9.4 Refs
A (Rhodopsin) Neuropeptide Y NPY2R Y2 NPY2R Human Neuropeptide Y-(3-36) (Human) 5 Peptide - - -
A (Rhodopsin) Neuropeptide Y NPY2R Y2 NPY2R Human Pancreatic Polypeptide (Human) 5 Protein - - -
A (Rhodopsin) Neuropeptide Y NPY2R Y2 NPY2R Human Pancreatic Polypeptide (Mouse) 5 Peptide - - -
A (Rhodopsin) Neuropeptide Y NPY2R Y2 NPY2R Human Pancreatic Polypeptide (Rat) 5 Peptide - - -
A (Rhodopsin) Neuropeptide Y NPY2R Y2 NPY2R Human Peptide Yy (Human) 2 Peptide - - - 9.5 9.7 9.8 Refs
A (Rhodopsin) Neuropeptide Y NPY2R Y2 NPY2R Human Peptide Yy (Mouse) 1 Protein - - - 10.0 10.0 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 NPY4R Human Pyy-(3-36) (Mouse) 6 Peptide - - - 6.2 6.2 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 NPY4R Human Neuropeptide Y (Human) 4 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccc(cc1)O)CCCN=C(N)N)CCC(=O)N)CCCN=C(N)N)[C@H](O)C)[C@H](CC)C)CC(C)C)CC(=O)N)[C@H](CC)C)Cc1ccc(cc1)O)Cc1c[nH]cn1)CCCN=C(N)N)CC(C)C)C)CO)Cc1ccc(cc1)O)Cc1ccc(cc1)O)CCCN=C(N)N)C)CCSC)CC(=O)O)CCC(=O)O)C)C)CC(=O)O)CCC(=O)O)CC(=O)N)CC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(cc1)O)N)CO XKWCTHKJQNUFOQ-HRPSIEBRSA-N - - 6.4 7.2 8.8 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 NPY4R Human Pancreatic Polypeptide (Human) 2 Protein - - - 8.7 9.8 10.9 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 NPY4R Human Pancreatic Polypeptide (Mouse) 7 Peptide - - -
A (Rhodopsin) Neuropeptide Y NPY4R Y4 NPY4R Human Peptide Yy (Human) 3 Peptide - - - 8.8 8.8 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 NPY4R Human Peptide Yy (Mouse) 5 Protein - - - 6.3 7.0 8.5 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 Npy4r Mouse Peptide Yy (Mouse) 5 Protein - - - - 6.3 7.0 8.5 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 Npy4r Rat Pyy-(3-36) (Mouse) 6 Peptide - - - - 6.2 6.2 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 Npy4r Rat Neuropeptide Y (Human) 4 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccc(cc1)O)CCCN=C(N)N)CCC(=O)N)CCCN=C(N)N)[C@H](O)C)[C@H](CC)C)CC(C)C)CC(=O)N)[C@H](CC)C)Cc1ccc(cc1)O)Cc1c[nH]cn1)CCCN=C(N)N)CC(C)C)C)CO)Cc1ccc(cc1)O)Cc1ccc(cc1)O)CCCN=C(N)N)C)CCSC)CC(=O)O)CCC(=O)O)C)C)CC(=O)O)CCC(=O)O)CC(=O)N)CC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(cc1)O)N)CO XKWCTHKJQNUFOQ-HRPSIEBRSA-N - - 6.4 7.2 8.8 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 Npy4r Rat Pancreatic Polypeptide (Rat) 1 Peptide - - - - 10.3 10.6 10.8 Refs
A (Rhodopsin) Neuropeptide Y NPY4R Y4 Npy4r Rat Peptide Yy (Mouse) 5 Protein - - - - 6.3 7.0 8.5 Refs
A (Rhodopsin) Neuropeptide Y NPY5R Y5 NPY5R Human Pyy-(3-36) (Mouse) 3 Peptide - - - - 8.4 8.4 Refs
A (Rhodopsin) Neuropeptide Y NPY5R Y5 NPY5R Human Neuropeptide Y (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccc(cc1)O)CCCN=C(N)N)CCC(=O)N)CCCN=C(N)N)[C@H](O)C)[C@H](CC)C)CC(C)C)CC(=O)N)[C@H](CC)C)Cc1ccc(cc1)O)Cc1c[nH]cn1)CCCN=C(N)N)CC(C)C)C)CO)Cc1ccc(cc1)O)Cc1ccc(cc1)O)CCCN=C(N)N)C)CCSC)CC(=O)O)CCC(=O)O)C)C)CC(=O)O)CCC(=O)O)CC(=O)N)CC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(cc1)O)N)CO XKWCTHKJQNUFOQ-HRPSIEBRSA-N - - 9.3 9.3 Refs
A (Rhodopsin) Neuropeptide Y NPY5R Y5 NPY5R Human Pancreatic Polypeptide (Human) 4 Protein - - - - 8.0 8.0 Refs
A (Rhodopsin) Neuropeptide Y NPY5R Y5 NPY5R Human Pancreatic Polypeptide (Mouse) 6 Peptide - - - -
A (Rhodopsin) Neuropeptide Y NPY5R Y5 NPY5R Human Peptide Yy (Human) 6 Peptide - - - -
A (Rhodopsin) Neuropeptide Y NPY5R Y5 NPY5R Human Peptide Yy (Mouse) 2 Protein - - - - 9.0 9.0 Refs
A (Rhodopsin) Neuropeptide Y NPY5R Y5 Npy5r Rat Pyy-(3-36) (Mouse) 3 Peptide - - - - 8.4 8.4 Refs
A (Rhodopsin) Neuropeptide Y NPY5R Y5 Npy5r Rat Neuropeptide Y (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccc(cc1)O)CCCN=C(N)N)CCC(=O)N)CCCN=C(N)N)[C@H](O)C)[C@H](CC)C)CC(C)C)CC(=O)N)[C@H](CC)C)Cc1ccc(cc1)O)Cc1c[nH]cn1)CCCN=C(N)N)CC(C)C)C)CO)Cc1ccc(cc1)O)Cc1ccc(cc1)O)CCCN=C(N)N)C)CCSC)CC(=O)O)CCC(=O)O)C)C)CC(=O)O)CCC(=O)O)CC(=O)N)CC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(cc1)O)N)CO XKWCTHKJQNUFOQ-HRPSIEBRSA-N - - 9.3 9.3 Refs
A (Rhodopsin) Neuropeptide Y NPY5R Y5 Npy5r Rat Pancreatic Polypeptide (Rat) 5 Peptide - - - - 6.5 6.5 Refs
A (Rhodopsin) Neuropeptide Y NPY5R Y5 Npy5r Rat Peptide Yy (Mouse) 2 Protein - - - - 9.0 9.0 Refs
A (Rhodopsin) Neuropeptide Y Q9ERC0 Y2 Npy2r Rat Neuropeptide Y (Human) 4 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccc(cc1)O)CCCN=C(N)N)CCC(=O)N)CCCN=C(N)N)[C@H](O)C)[C@H](CC)C)CC(C)C)CC(=O)N)[C@H](CC)C)Cc1ccc(cc1)O)Cc1c[nH]cn1)CCCN=C(N)N)CC(C)C)C)CO)Cc1ccc(cc1)O)Cc1ccc(cc1)O)CCCN=C(N)N)C)CCSC)CC(=O)O)CCC(=O)O)C)C)CC(=O)O)CCC(=O)O)CC(=O)N)CC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(cc1)O)N)CO XKWCTHKJQNUFOQ-HRPSIEBRSA-N - - 9.3 9.4 9.4 Refs
A (Rhodopsin) Neuropeptide Y Q9ERC0 Y2 Npy2r Rat Peptide Yy (Mouse) 1 Protein - - - - 10.0 10.0 Refs
A (Rhodopsin) Neurotensin NTR1 NTS1 NTSR1 Human Large Neuromedin N (Human) 3 Peptide - - - - Refs
A (Rhodopsin) Neurotensin NTR1 NTS1 NTSR1 Human Large Neuromedin N (Mouse) 3 Peptide - - - -
A (Rhodopsin) Neurotensin NTR1 NTS1 NTSR1 Human Large Neuromedin N (Rat) 3 Peptide - - - -
A (Rhodopsin) Neurotensin NTR1 NTS1 NTSR1 Human Large Neurotensin (Human) 3 Peptide - - - - Refs
A (Rhodopsin) Neurotensin NTR1 NTS1 NTSR1 Human Neuromedin N (Human) 3 Peptide - - - -
A (Rhodopsin) Neurotensin NTR1 NTS1 NTSR1 Human Neuromedin N (Mouse) 2 Peptide - - - - 8.7 8.7 Refs
A (Rhodopsin) Neurotensin NTR1 NTS1 NTSR1 Human Neurotensin (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(C)C)[C@H](CC)C)Cc1ccc(cc1)O)CCCN=C(N)N)CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCC(=O)N1)CC(C)C)Cc1ccc(cc1)O)CCC(=O)O)CC(=O)N PCJGZPGTCUMMOT-ISULXFBGSA-N - - 8.2 9.1 10.0 Refs
A (Rhodopsin) Neurotensin NTR1 NTS1 Ntsr1 Rat Neuromedin N (Mouse) 2 Peptide - - - - 8.7 8.7 Refs
A (Rhodopsin) Neurotensin NTR1 NTS1 Ntsr1 Rat Neurotensin (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(C)C)[C@H](CC)C)Cc1ccc(cc1)O)CCCN=C(N)N)CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCC(=O)N1)CC(C)C)Cc1ccc(cc1)O)CCC(=O)O)CC(=O)N PCJGZPGTCUMMOT-ISULXFBGSA-N - - 8.2 9.1 10.0 Refs
A (Rhodopsin) Neurotensin NTR2 NTS2 NTSR2 Human Neuromedin N (Human) 2 Peptide - - - -
A (Rhodopsin) Neurotensin NTR2 NTS2 NTSR2 Human Neurotensin (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(C)C)[C@H](CC)C)Cc1ccc(cc1)O)CCCN=C(N)N)CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCC(=O)N1)CC(C)C)Cc1ccc(cc1)O)CCC(=O)O)CC(=O)N PCJGZPGTCUMMOT-ISULXFBGSA-N - - 8.8 8.8 Refs
A (Rhodopsin) Neurotensin NTR2 NTS2 NTSR2 Human Xenin (Human) 2 Peptide NCCCC[C@@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(C)C)[C@H](CC)C)Cc1c[nH]c2c1cccc2)CCCNC(=N)N)CCCCN)Cc1[nH]cnc1)Cc1ccccc1)CO)CC(C)C)NC(=O)[C@H](C(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@H](CCSC)N)CC(C)C)CCCCN)Cc1ccccc1)CCC(=O)O)CCCCN)CO)C)CCCNC(=N)N IDHVLSACPFUBDY-QCDLPZBNSA-N - - Refs
A (Rhodopsin) Neurotensin NTR2 NTS2 Ntsr2 Mouse Neuromedin N (Mouse) 2 Peptide - - - - Refs
A (Rhodopsin) Neurotensin NTR2 NTS2 Ntsr2 Mouse Neurotensin (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(C)C)[C@H](CC)C)Cc1ccc(cc1)O)CCCN=C(N)N)CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCC(=O)N1)CC(C)C)Cc1ccc(cc1)O)CCC(=O)O)CC(=O)N PCJGZPGTCUMMOT-ISULXFBGSA-N - - 8.8 8.8 Refs
A (Rhodopsin) Neurotensin NTR2 NTS2 Ntsr2 Mouse Xenin (Human) 2 Peptide NCCCC[C@@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(C)C)[C@H](CC)C)Cc1c[nH]c2c1cccc2)CCCNC(=N)N)CCCCN)Cc1[nH]cnc1)Cc1ccccc1)CO)CC(C)C)NC(=O)[C@H](C(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@H](CCSC)N)CC(C)C)CCCCN)Cc1ccccc1)CCC(=O)O)CCCCN)CO)C)CCCNC(=N)N IDHVLSACPFUBDY-QCDLPZBNSA-N - - Refs
A (Rhodopsin) Neurotensin NTR2 NTS2 Ntsr2 Rat Neuromedin N (Mouse) 2 Peptide - - - - Refs
A (Rhodopsin) Neurotensin NTR2 NTS2 Ntsr2 Rat Neurotensin (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CC(C)C)[C@H](CC)C)Cc1ccc(cc1)O)CCCN=C(N)N)CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCC(=O)N1)CC(C)C)Cc1ccc(cc1)O)CCC(=O)O)CC(=O)N PCJGZPGTCUMMOT-ISULXFBGSA-N - - 8.8 8.8 Refs
A (Rhodopsin) Opioid OPRD δ OPRD1 Human Α-Neoendorphin (Human) 6 Peptide CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)O KZTDMJBCZSGHOG-XJIZABAQSA-N - Refs
A (Rhodopsin) Opioid OPRD δ OPRD1 Human Β-Endorphin (Human) 2 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O)[C@@H](C)O)C(C)C)[C@@H](C)O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)O)[C@@H](C)CC JMHFFDIMOUKDCZ-NTXHZHDSSA-N - 8.3 8.3 Refs
A (Rhodopsin) Opioid OPRD δ OPRD1 Human Β-Endorphin (Mouse) 6 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O)[C@@H](C)O)C(C)C)[C@@H](C)O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)O)[C@@H](C)CC HQALISCIMNBRAE-XJTHNYJFSA-N -
A (Rhodopsin) Opioid OPRD δ OPRD1 Human Β-Endorphin (Rat) 6 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O)[C@@H](C)O)C(C)C)[C@@H](C)O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)O)C(C)C)[C@@H](C)CC KSZMZNRVPCEDEO-KFHPFRHLSA-N -
A (Rhodopsin) Opioid OPRD δ OPRD1 Human [Leu]Enkephalin (Human) 1 Peptide O=C(CNC(=O)C(Cc1ccc(cc1)O)N)NCC(=O)NC(C(=O)NC(C(=O)O)CC(C)C)Cc1ccccc1 URLZCHNOLZSCCA-UHFFFAOYSA-N - 9XF4 8.4 8.4 Refs
A (Rhodopsin) Opioid OPRD δ OPRD1 Human [Met]Enkephalin (Human) 6 Peptide CSCC[C@@H](C(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N YFGBQHOOROIVKG-FKBYEOEOSA-N - Refs
A (Rhodopsin) Opioid OPRD δ OPRD1 Human Dynorphin A (Human) 4 Protein CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)O JMNJYGMAUMANNW-FIXZTSJVSA-N - - 7.4 7.4 Refs
A (Rhodopsin) Opioid OPRD δ OPRD1 Human Dynorphin A-(1-13) (Human) 3 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)O OVVIBUHLQIYUEU-IWIISZHXSA-N - 7.8 7.8 Refs
A (Rhodopsin) Opioid OPRD δ OPRD1 Human Dynorphin A-(1-8) (Human) 1 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)O WRPLGMBDXVBPEG-VGXZEHLRSA-N - 8.4 8.4 Refs
A (Rhodopsin) Opioid OPRD δ OPRD1 Human Dynorphin B (Human) 3 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)[C@H](O)C)C(C)C)C(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N)CC(C)C)CCCN=C(N)N)CCCN=C(N)N)CCC(=O)N)Cc1ccccc1 AGTSSZRZBSNTGQ-ITZCFHCWSA-N - 7.8 7.8 Refs
A (Rhodopsin) Opioid OPRD δ OPRD1 Human Endomorphin-1 (Human) 5 Peptide Oc1ccc(cc1)C[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccccc1)Cc1c[nH]c2c1cccc2)N ZEXLJFNSKAHNFH-SYKYGTKKSA-N - 6.1 6.1 Refs
A (Rhodopsin) Opioid OPRD δ Oprd1 Mouse Α-Neoendorphin (Human) 6 Peptide CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)O KZTDMJBCZSGHOG-XJIZABAQSA-N - - Refs
A (Rhodopsin) Opioid OPRD δ Oprd1 Mouse [Leu]Enkephalin (Human) 1 Peptide O=C(CNC(=O)C(Cc1ccc(cc1)O)N)NCC(=O)NC(C(=O)NC(C(=O)O)CC(C)C)Cc1ccccc1 URLZCHNOLZSCCA-UHFFFAOYSA-N - - 8.4 8.4 Refs
A (Rhodopsin) Opioid OPRD δ Oprd1 Mouse [Met]Enkephalin (Human) 6 Peptide CSCC[C@@H](C(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N YFGBQHOOROIVKG-FKBYEOEOSA-N - - Refs
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Α-Neoendorphin (Human) 4 Peptide CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)O KZTDMJBCZSGHOG-XJIZABAQSA-N - 8.9 9.5 10.0 Refs
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Β-Endorphin (Human) 7 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O)[C@@H](C)O)C(C)C)[C@@H](C)O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)O)[C@@H](C)CC JMHFFDIMOUKDCZ-NTXHZHDSSA-N - 6.3 7.1 7.9 Refs
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Β-Endorphin (Mouse) 9 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O)[C@@H](C)O)C(C)C)[C@@H](C)O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)O)[C@@H](C)CC HQALISCIMNBRAE-XJTHNYJFSA-N -
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Β-Endorphin (Rat) 9 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O)[C@@H](C)O)C(C)C)[C@@H](C)O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)O)C(C)C)[C@@H](C)CC KSZMZNRVPCEDEO-KFHPFRHLSA-N -
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Β-Neoendorphin (Human) 5 Peptide CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)O RTXIYIQLESPXIV-VLOLPVCOSA-N - 9.1 9.1 Refs
A (Rhodopsin) Opioid OPRK κ OPRK1 Human [Leu]Enkephalin (Human) 8 Peptide O=C(CNC(=O)C(Cc1ccc(cc1)O)N)NCC(=O)NC(C(=O)NC(C(=O)O)CC(C)C)Cc1ccccc1 URLZCHNOLZSCCA-UHFFFAOYSA-N - 6.0 6.0 Refs
A (Rhodopsin) Opioid OPRK κ OPRK1 Human [Met]Enkephalin (Human) 8 Peptide CSCC[C@@H](C(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N YFGBQHOOROIVKG-FKBYEOEOSA-N - 6.0 6.0 Refs
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Big Dynorphin (Human) 9 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)NCC(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)[C@@H](C)O)C(C)C)C(C)C VPZXNPNLCOYTOT-MBGMINRZSA-N -
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Dynorphin A (Human) 1 Protein CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)O JMNJYGMAUMANNW-FIXZTSJVSA-N - - 10.0 10.2 10.3 Refs
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Dynorphin A-(1-13) (Human) 2 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)O OVVIBUHLQIYUEU-IWIISZHXSA-N - 9.3 9.9 9.9 Refs
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Dynorphin A-(1-8) (Human) 6 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)O WRPLGMBDXVBPEG-VGXZEHLRSA-N - 8F7W 8.0 9.0 9.9 Refs
A (Rhodopsin) Opioid OPRK κ OPRK1 Human Dynorphin B (Human) 3 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)[C@H](O)C)C(C)C)C(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N)CC(C)C)CCCN=C(N)N)CCCN=C(N)N)CCC(=O)N)Cc1ccccc1 AGTSSZRZBSNTGQ-ITZCFHCWSA-N - 8.1 9.5 9.5 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Mouse Α-Neoendorphin (Human) 4 Peptide CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)O KZTDMJBCZSGHOG-XJIZABAQSA-N - - 8.9 9.5 10.0 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Mouse Dynorphin A (Human) 1 Protein CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)O JMNJYGMAUMANNW-FIXZTSJVSA-N - - 10.0 10.2 10.3 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Mouse Dynorphin A-(1-8) (Human) 6 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)O WRPLGMBDXVBPEG-VGXZEHLRSA-N - - 8.0 9.0 9.9 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Mouse Dynorphin B (Human) 3 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)[C@H](O)C)C(C)C)C(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N)CC(C)C)CCCN=C(N)N)CCCN=C(N)N)CCC(=O)N)Cc1ccccc1 AGTSSZRZBSNTGQ-ITZCFHCWSA-N - - 8.1 9.5 9.5 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Rat Α-Neoendorphin (Human) 4 Peptide CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)O KZTDMJBCZSGHOG-XJIZABAQSA-N - - 8.9 9.5 10.0 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Rat Β-Neoendorphin (Human) 5 Peptide CC(C)C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)O RTXIYIQLESPXIV-VLOLPVCOSA-N - - 9.1 9.1 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Rat [Leu]Enkephalin (Human) 8 Peptide O=C(CNC(=O)C(Cc1ccc(cc1)O)N)NCC(=O)NC(C(=O)NC(C(=O)O)CC(C)C)Cc1ccccc1 URLZCHNOLZSCCA-UHFFFAOYSA-N - - 6.0 6.0 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Rat [Met]Enkephalin (Human) 8 Peptide CSCC[C@@H](C(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N YFGBQHOOROIVKG-FKBYEOEOSA-N - - 6.0 6.0 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Rat Dynorphin A (Human) 1 Protein CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)O JMNJYGMAUMANNW-FIXZTSJVSA-N - - 10.0 10.2 10.3 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Rat Dynorphin A-(1-13) (Human) 2 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)O OVVIBUHLQIYUEU-IWIISZHXSA-N - - 9.3 9.9 9.9 Refs
A (Rhodopsin) Opioid OPRK κ Oprk1 Rat Dynorphin B (Human) 3 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)[C@H](O)C)C(C)C)C(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N)CC(C)C)CCCN=C(N)N)CCCN=C(N)N)CCC(=O)N)Cc1ccccc1 AGTSSZRZBSNTGQ-ITZCFHCWSA-N - - 8.1 9.5 9.5 Refs
A (Rhodopsin) Opioid OPRM μ OPRM1 Human Β-Endorphin (Human) 6 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O)[C@@H](C)O)C(C)C)[C@@H](C)O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(=O)O)C(=O)O)[C@@H](C)CC JMHFFDIMOUKDCZ-NTXHZHDSSA-N -
A (Rhodopsin) Opioid OPRM μ OPRM1 Human Β-Endorphin (Mouse) 6 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O)[C@@H](C)O)C(C)C)[C@@H](C)O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)O)[C@@H](C)CC HQALISCIMNBRAE-XJTHNYJFSA-N -
A (Rhodopsin) Opioid OPRM μ OPRM1 Human Β-Endorphin (Rat) 6 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)[C@@H](C)O)[C@@H](C)O)C(C)C)[C@@H](C)O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)O)C(C)C)[C@@H](C)CC KSZMZNRVPCEDEO-KFHPFRHLSA-N -
A (Rhodopsin) Opioid OPRM μ OPRM1 Human [Leu]Enkephalin (Human) 5 Peptide O=C(CNC(=O)C(Cc1ccc(cc1)O)N)NCC(=O)NC(C(=O)NC(C(=O)O)CC(C)C)Cc1ccccc1 URLZCHNOLZSCCA-UHFFFAOYSA-N - 8.1 8.1 Refs
A (Rhodopsin) Opioid OPRM μ OPRM1 Human [Met]Enkephalin (Human) 1 Peptide CSCC[C@@H](C(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N YFGBQHOOROIVKG-FKBYEOEOSA-N - 9.2 9.2 Refs
A (Rhodopsin) Opioid OPRM μ OPRM1 Human Dynorphin A (Human) 5 Protein CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCC(N)=O)C(=O)O JMNJYGMAUMANNW-FIXZTSJVSA-N - - 8.1 8.1 Refs
A (Rhodopsin) Opioid OPRM μ OPRM1 Human Dynorphin A-(1-13) (Human) 4 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCCN)C(=O)O OVVIBUHLQIYUEU-IWIISZHXSA-N - 8.3 8.3 Refs
A (Rhodopsin) Opioid OPRM μ OPRM1 Human Dynorphin A-(1-8) (Human) 3 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)O WRPLGMBDXVBPEG-VGXZEHLRSA-N - 8.4 8.4 Refs
A (Rhodopsin) Opioid OPRM μ OPRM1 Human Dynorphin B (Human) 2 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)[C@H](O)C)C(C)C)C(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N)CC(C)C)CCCN=C(N)N)CCCN=C(N)N)CCC(=O)N)Cc1ccccc1 AGTSSZRZBSNTGQ-ITZCFHCWSA-N - 8.5 8.5 Refs
A (Rhodopsin) Opioid OPRM μ OPRM1 Human Endomorphin-1 (Human) 4 Peptide Oc1ccc(cc1)C[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccccc1)Cc1c[nH]c2c1cccc2)N ZEXLJFNSKAHNFH-SYKYGTKKSA-N - 8F7R 8.3 8.3 Refs
A (Rhodopsin) Opioid OPRM μ OPRM1 Human Endomorphin-2 (Human) 6 Peptide Oc1ccc(cc1)C[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccccc1)Cc1ccccc1)N XIJHWXXXIMEHKW-LJWNLINESA-N -
A (Rhodopsin) Opioid OPRM μ Oprm1 Rat [Met]Enkephalin (Human) 1 Peptide CSCC[C@@H](C(=O)O)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccc(cc1)O)N YFGBQHOOROIVKG-FKBYEOEOSA-N - - 9.2 9.2 Refs
A (Rhodopsin) Opioid OPRX NOP OPRL1 Human Nociceptin/Orphanin Fq (Human) Principal 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCC(=O)N)CC(=O)N)C)CC(C)C)CCCCN)CCCNC(=N)N)C)CO)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@H]([C@H](O)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccccc1)N)C)CCCNC(=N)N PULGYDLMFSFVBL-SMFNREODSA-N - 8F7X 8.4 9.1 9.8 9.7 9.4 9.4 Refs
A (Rhodopsin) Opioid OPRX NOP Oprl1 Mouse Nociceptin/Orphanin Fq (Human) Principal 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)CCC(=O)N)CC(=O)N)C)CC(C)C)CCCCN)CCCNC(=N)N)C)CO)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)CNC(=O)[C@H]([C@H](O)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CNC(=O)[C@H](Cc1ccccc1)N)C)CCCNC(=N)N PULGYDLMFSFVBL-SMFNREODSA-N - - 8.4 9.1 9.8 9.7 9.4 9.4 Refs
A (Rhodopsin) Orexin OX1R OX1 HCRTR1 Human Orexin-A (Human) 1 Peptide - - - - 6.5 8.4 10.2 Refs
A (Rhodopsin) Orexin OX1R OX1 HCRTR1 Human Orexin-B (Human) 2 Protein CSCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCCN=C(N)N)CO)CC(C)C)CCC(=O)N)CCCN=C(N)N)CC(C)C)CCC(=O)N)CCCN=C(N)N)CC(C)C)CC(C)C)CCC(=O)N)C)CO)CC(=O)N)Cc1nc[nH]c1)C)C)[C@H](CC)C)CC(C)C)[C@H](O)C)N OHOWSYIKESXDMN-WMQZXSDYSA-N - - 5.8 7.5 9.2 Refs
A (Rhodopsin) Orexin OX1R OX1 HCRTR1 Human Orexin-B (Mouse) 3 Protein - - - -
A (Rhodopsin) Orexin OX2R OX2 HCRTR2 Human Orexin-A (Human) 1 Peptide - - - - 6.5 8.3 10.0 Refs
A (Rhodopsin) Orexin OX2R OX2 HCRTR2 Human Orexin-B (Human) 1 Protein CSCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCCN=C(N)N)CO)CC(C)C)CCC(=O)N)CCCN=C(N)N)CC(C)C)CCC(=O)N)CCCN=C(N)N)CC(C)C)CC(C)C)CCC(=O)N)C)CO)CC(=O)N)Cc1nc[nH]c1)C)C)[C@H](CC)C)CC(C)C)[C@H](O)C)N OHOWSYIKESXDMN-WMQZXSDYSA-N - 7L1U 6.5 8.3 10.0 Refs
A (Rhodopsin) Orexin OX2R OX2 HCRTR2 Human Orexin-B (Mouse) 2 Protein - - - -
A (Rhodopsin) Orphan G37L1 GPR37L1 GPR37L1 Human Prosaptide (Human) Principal 1 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](N)CS)C(C)C)C(C)C)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)O KSDDQEGWVBODMD-OULINLAESA-N - 8.3 8.3 Refs
A (Rhodopsin) Orphan GP139 GPR139 GPR139 Human D-Phenylalanine None 2 Small molecule N[C@@H](C(=O)O)Cc1ccccc1 COLNVLDHVKWLRT-MRVPVSSYSA-N - - 3.5 3.5 3.1 3.1 Refs
A (Rhodopsin) Orphan GP139 GPR139 GPR139 Human D-Tryptophan None 1 Small molecule OC(=O)[C@@H](Cc1c[nH]c2c1cccc2)N QIVBCDIJIAJPQS-SECBINFHSA-N - - 3.7 3.7 3.1 3.1 Refs
A (Rhodopsin) Orphan GP174 GPR174 GPR174 Human Lysophosphatidylserine Principal 1 Lipid CCCCCCCCCCCCCCCCCC(=O)OC[C@H](COP(=O)(OC[C@@H](C(=O)O)N)O)O ZPDQFUYPBVXUKS-YADHBBJMSA-N - 9XXT 7.1 7.1 Refs
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Ccl1 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Ccl11 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Ccl19 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Ccl25 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Ccl26 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Cxcl1 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Cxcl10 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Cxcl11 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Cxcl12Α (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Cxcl13 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Cxcl14 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP182 GPR182 GPR182 Human Cxcl17 (Human) Peptide - - - -
A (Rhodopsin) Orphan GP183 GPR183 GPR183 Human 25-Hydroxycholesterol None 6 Small molecule O[C@H]1CC[C@]2(C(=CC[C@@H]3[C@@H]2CC[C@]2([C@H]3CC[C@@H]2[C@@H](CCCC(O)(C)C)C)C)C1)C INBGSXNNRGWLJU-ZHHJOTBYSA-N - - 6.9 6.9 Refs
A (Rhodopsin) Orphan GP183 GPR183 GPR183 Human 27-Hydroxycholesterol None 8 Small molecule OC[C@@H](CCC[C@H]([C@H]1CC[C@@H]2[C@]1(C)CC[C@H]1[C@H]2CC=C2[C@]1(C)CC[C@@H](C2)O)C)C FYHRJWMENCALJY-YSQMORBQSA-N - - 5.5 5.5 Refs
A (Rhodopsin) Orphan GP183 GPR183 GPR183 Human 7Α,25-Dihydroxycholesterol None 1 Small molecule O[C@H]1CC[C@]2(C(=C[C@H]([C@@H]3[C@@H]2CC[C@]2([C@H]3CC[C@@H]2[C@@H](CCCC(O)(C)C)C)C)O)C1)C BQMSKLCEWBSPPY-IKVTXIKFSA-N - 7TUZ 8.1 9.0 9.9 Refs
A (Rhodopsin) Orphan GP183 GPR183 GPR183 Human 7Α,27-Dihydroxycholesterol None 2 Small molecule OC[C@@H](CCC[C@H]([C@H]1CC[C@@H]2[C@]1(C)CC[C@H]1[C@H]2[C@H](O)C=C2[C@]1(C)CC[C@@H](C2)O)C)C RXMHNAKZMGJANZ-GNENNHQYSA-N - - 8.9 8.9 Refs
A (Rhodopsin) Orphan GP183 GPR183 GPR183 Human 7Α-Hydroxycholesterol None 5 Small molecule CC(CCC[C@H]([C@H]1CC[C@@H]2[C@]1(C)CC[C@H]1[C@H]2[C@H](O)C=C2[C@]1(C)CC[C@@H](C2)O)C)C OYXZMSRRJOYLLO-RVOWOUOISA-N - - 7.1 7.1 Refs
A (Rhodopsin) Orphan GP183 GPR183 GPR183 Human 7Β, 25-Dihydroxycholesterol None 3 Small molecule O[C@H]1CC[C@]2(C(=C[C@@H]([C@@H]3[C@@H]2CC[C@]2([C@H]3CC[C@@H]2[C@@H](CCCC(O)(C)C)C)C)O)C1)C BQMSKLCEWBSPPY-CGSQRZAOSA-N - - 8.7 8.7 Refs
A (Rhodopsin) Orphan GP183 GPR183 GPR183 Human 7Β, 27-Dihydroxycholesterol None 4 Small molecule OC[C@@H](CCC[C@H]([C@H]1CC[C@@H]2[C@]1(C)CC[C@H]1[C@H]2[C@@H](O)C=C2[C@]1(C)CC[C@@H](C2)O)C)C RXMHNAKZMGJANZ-BMOLSTJGSA-N - - 7.3 7.3 Refs
A (Rhodopsin) Orphan GP183 GPR183 GPR183 Human 7Β-Hydroxycholesterol None 7 Small molecule CC(CCC[C@H]([C@H]1CC[C@@H]2[C@]1(C)CC[C@H]1[C@H]2[C@@H](O)C=C2[C@]1(C)CC[C@@H](C2)O)C)C OYXZMSRRJOYLLO-KGZHIOMZSA-N - - 5.8 5.8 Refs
A (Rhodopsin) Orphan GPR12 GPR12 GPR12 Human Sphingosine 1-Phosphate Principal 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 5.5 6.3 7.0 Refs
A (Rhodopsin) Orphan GPR17 GPR17 GPR17 Human Atp None 4 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N ZKHQWZAMYRWXGA-KQYNXXCUSA-N - - 7.4 7.4 Refs
A (Rhodopsin) Orphan GPR17 GPR17 GPR17 Human Ltc4 None 3 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SC[C@@H](C(=O)NCC(=O)O)NC(=O)CC[C@@H](C(=O)O)N GWNVDXQDILPJIG-NXOLIXFESA-N - - 7.8 9.1 9.1 Refs
A (Rhodopsin) Orphan GPR17 GPR17 GPR17 Human Ltd4 None 2 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SCC(C(=O)NCC(=O)O)N YEESKJGWJFYOOK-LDDGIIIKSA-N - - 8.1 9.2 9.2 Refs
A (Rhodopsin) Orphan GPR17 GPR17 GPR17 Human Lte4 None 1 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SC[C@@H](C(=O)O)N OTZRAYGBFWZKMX-FRFVZSDQSA-N - -
A (Rhodopsin) Orphan GPR17 GPR17 GPR17 Human Udp None 4 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O XCCTYIAWTASOJW-XVFCMESISA-N - - 6.0 7.4 8.8 Refs
A (Rhodopsin) Orphan GPR17 GPR17 GPR17 Human Udp-Galactose None 5 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@H]1O)O)O HSCJRCZFDFQWRP-ABVWGUQPSA-N - - 6.0 7.2 7.2 Refs
A (Rhodopsin) Orphan GPR17 GPR17 GPR17 Human Udp-Glucose None 6 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@@H]1O)O)O HSCJRCZFDFQWRP-JZMIEXBBSA-N - - 7.1 7.2 7.3 Refs
A (Rhodopsin) Orphan GPR17 GPR17 Gpr17 Mouse Ltc4 None 3 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SC[C@@H](C(=O)NCC(=O)O)NC(=O)CC[C@@H](C(=O)O)N GWNVDXQDILPJIG-NXOLIXFESA-N - - 7.8 9.1 9.1 Refs
A (Rhodopsin) Orphan GPR17 GPR17 Gpr17 Mouse Ltd4 None 2 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SCC(C(=O)NCC(=O)O)N YEESKJGWJFYOOK-LDDGIIIKSA-N - - 8.1 9.2 9.2 Refs
A (Rhodopsin) Orphan GPR17 GPR17 Gpr17 Mouse Lte4 None 1 Small molecule CCCCC/C=C\C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)SC[C@@H](C(=O)O)N OTZRAYGBFWZKMX-FRFVZSDQSA-N - - 9.5 9.5 Refs
A (Rhodopsin) Orphan GPR17 GPR17 Gpr17 Mouse Udp-Galactose None 5 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@H]1O)O)O HSCJRCZFDFQWRP-ABVWGUQPSA-N - - 6.0 7.2 7.2 Refs
A (Rhodopsin) Orphan GPR17 GPR17 Gpr17 Mouse Udp-Glucose None 6 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@@H]1O)O)O HSCJRCZFDFQWRP-JZMIEXBBSA-N - - 7.1 7.2 7.3 Refs
A (Rhodopsin) Orphan GPR31 GPR31 GPR31 Human 12s-Hete Principal 1 Small molecule CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O ZNHVWPKMFKADKW-LQWMCKPYSA-N - -
A (Rhodopsin) Orphan GPR31 GPR31 Gpr31 Mouse 12s-Hete Principal 1 Small molecule CCCCC/C=C\C[C@@H](/C=C/C=C\C/C=C\CCCC(=O)O)O ZNHVWPKMFKADKW-LQWMCKPYSA-N - - 9.6 9.6 Refs
A (Rhodopsin) Orphan GPR32 GPR32 GPR32 Human Lxa4 None 2 Small molecule CCCCC[C@@H](/C=C/C=C\C=C\C=C\[C@H]([C@H](CCCC(=O)O)O)O)O IXAQOQZEOGMIQS-SSQFXEBMSA-N - - 9.7 9.7 Refs
A (Rhodopsin) Orphan GPR32 GPR32 GPR32 Human Resolvin D1 None 1 Small molecule CC/C=C\C[C@@H](/C=C/C=C\C=C\C=C\[C@@H]([C@H](C/C=C\CCC(=O)O)O)O)O OIWTWACQMDFHJG-LDOXQWQISA-N - - 11.1 11.1 Refs
A (Rhodopsin) Orphan GPR34 GPR34 GPR34 Human Lysophosphatidylserine Principal 1 Lipid CCCCCCCCCCCCCCCCCC(=O)OC[C@H](COP(=O)(OC[C@@H](C(=O)O)N)O)O ZPDQFUYPBVXUKS-YADHBBJMSA-N - 6.6 7.3 7.3 Refs
A (Rhodopsin) Orphan GPR34 GPR34 Gpr34 Mouse Lysophosphatidylserine Principal 1 Lipid CCCCCCCCCCCCCCCCCC(=O)OC[C@H](COP(=O)(OC[C@@H](C(=O)O)N)O)O ZPDQFUYPBVXUKS-YADHBBJMSA-N - - 6.6 7.3 7.3 Refs
A (Rhodopsin) Orphan GPR35 GPR35 GPR35 Human 2-Oleoyl-Lpa None 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OC(COP(=O)(O)O)CO ZOOLJLSXNRZLDH-KTKRTIGZSA-N - - 7.3 7.4 7.5 Refs
A (Rhodopsin) Orphan GPR35 GPR35 GPR35 Human Kynurenic Acid None 2 Small molecule OC(=O)c1cc(=O)c2c([nH]1)cccc2 HCZHHEIFKROPDY-UHFFFAOYSA-N - - 3.9 5.2 5.2 Refs
A (Rhodopsin) Orphan GPR35 GPR35 Gpr35 Mouse Kynurenic Acid None 2 Small molecule OC(=O)c1cc(=O)c2c([nH]1)cccc2 HCZHHEIFKROPDY-UHFFFAOYSA-N - - 3.9 5.2 5.2 Refs
A (Rhodopsin) Orphan GPR37 GPR37 GPR37 Human Prosaptide (Human) Principal 1 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@@H](N)CS)C(C)C)C(C)C)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)C(=O)N[C@@H](CC(C)C)C(=O)O KSDDQEGWVBODMD-OULINLAESA-N - 8.1 8.1 Refs
A (Rhodopsin) Orphan GPR39 GPR39 GPR39 Human Zn2+ None Small molecule - - - - Refs
A (Rhodopsin) Orphan GPR39 GPR39 GPR39 Human Obestatin (Human) Peptide - - -
A (Rhodopsin) Orphan GPR39 GPR39 GPR39 Human Obestatin (Mouse) Peptide - - -
A (Rhodopsin) Orphan GPR3 GPR3 GPR3 Human Sphingosine 1-Phosphate Principal 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 7.1 7.4 7.7 Refs
A (Rhodopsin) Orphan GPR63 GPR63 GPR63 Human Dihydrosphingosine 1-Phosphate None 2 Lipid CCCCCCCCCCCCCCC[C@H]([C@H](COP(=O)(O)O)N)O YHEDRJPUIRMZMP-ZWKOTPCHSA-N - - 6.2 6.2 Refs
A (Rhodopsin) Orphan GPR63 GPR63 GPR63 Human Dioleoylphosphatidic Acid None 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(OC(=O)CCCCCCC/C=C\CCCCCCCC)COP(=O)(O)O MHUWZNTUIIFHAS-CLFAGFIQSA-N - - 6.3 6.3 Refs
A (Rhodopsin) Orphan GPR63 GPR63 GPR63 Human Sphingosine 1-Phosphate None 3 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 6.1 6.2 6.2 Refs
A (Rhodopsin) Orphan GPR6 GPR6 GPR6 Human Sphingosine 1-Phosphate Principal 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - -
A (Rhodopsin) Orphan GPR6 GPR6 Gpr6 Mouse Sphingosine 1-Phosphate Principal 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 7.3 7.5 7.7 Refs
A (Rhodopsin) Orphan GPR75 GPR75 GPR75 Human Ccl5 (Human) Principal 1 Peptide - - - - 9.6 9.6 Refs
A (Rhodopsin) Orphan GPR87 GPR87 GPR87 Human Lpa Principal 1 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 7.4 7.4 Refs
A (Rhodopsin) Orphan LGR4 LGR4 LGR4 Human R-Spondin-1 (Human) 2 Peptide - - - - 10.7 10.7 Refs
A (Rhodopsin) Orphan LGR4 LGR4 LGR4 Human R-Spondin-2 (Human) 1 Peptide - - - - 12.5 12.5 Refs
A (Rhodopsin) Orphan LGR4 LGR4 LGR4 Human R-Spondin-3 (Human) 2 Peptide - - - - 10.7 10.7 Refs
A (Rhodopsin) Orphan LGR4 LGR4 LGR4 Human R-Spondin-4 (Human) 3 Peptide - - - - 10.1 10.1 Refs
A (Rhodopsin) Orphan LGR5 LGR5 LGR5 Human R-Spondin-1 (Human) 2 Peptide - - - - 11.1 11.1 Refs
A (Rhodopsin) Orphan LGR5 LGR5 LGR5 Human R-Spondin-2 (Human) 1 Peptide - - - - 12.0 12.0 Refs
A (Rhodopsin) Orphan LGR5 LGR5 LGR5 Human R-Spondin-3 (Human) 3 Peptide - - - - 11.0 11.0 Refs
A (Rhodopsin) Orphan LGR5 LGR5 LGR5 Human R-Spondin-4 (Human) 4 Peptide - - - - 9.4 9.4 Refs
A (Rhodopsin) Orphan LGR6 LGR6 LGR6 Human R-Spondin-1 (Human) Peptide - - - - Refs
A (Rhodopsin) Orphan LGR6 LGR6 LGR6 Human R-Spondin-2 (Human) Peptide - - - - Refs
A (Rhodopsin) Orphan LGR6 LGR6 LGR6 Human R-Spondin-3 (Human) Peptide - - - - Refs
A (Rhodopsin) Orphan LGR6 LGR6 LGR6 Human R-Spondin-4 (Human) Peptide - - - - Refs
A (Rhodopsin) Orphan MRGRD MRGPRD MRGPRD Human Β-Alanine Principal 1 Small molecule NCCC(=O)O UCMIRNVEIXFBKS-UHFFFAOYSA-N - 7Y14 4.8 4.8 Refs
A (Rhodopsin) Orphan MRGX1 MRGPRX1 MRGPRX1 Human Bovine Adrenal Medulla Peptide 8-22 (Human) Principal 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)O)Cc1ccc(cc1)O)CCCNC(=N)N)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)CNC(=O)[C@H](C(C)C)N)CCCNC(=N)N)CCC(=O)O)CCSC)CC(=O)O)Cc1ccc(cc1)O)CCC(=O)N GOEYECACIBFJGZ-NPAGUKBMSA-N - 8DWC 5.3 6.6 7.8 7.7 7.7 Refs
A (Rhodopsin) Orphan MRGX2 MRGPRX2 MRGPRX2 Human Pamp-20 (Human) Principal 1 Peptide - - - Refs
A (Rhodopsin) Orphan P2Y10 P2RY10 P2RY10 Human Lpa None 2 Small molecule CCCCCCCC/C=C\CCCCCCCC(=O)OCC(COP(=O)(O)O)O WRGQSWVCFNIUNZ-KTKRTIGZSA-N - - 6.9 6.9 Refs
A (Rhodopsin) Orphan P2Y10 P2RY10 P2RY10 Human Sphingosine 1-Phosphate None 1 Lipid CCCCCCCCCCCCC/C=C/[C@H]([C@H](COP(=O)(O)O)N)O DUYSYHSSBDVJSM-KRWOKUGFSA-N - - 7.3 7.3 Refs
A (Rhodopsin) Orphan Q33BM1 GPR35 Gpr35 Rat Kynurenic Acid None 2 Small molecule OC(=O)c1cc(=O)c2c([nH]1)cccc2 HCZHHEIFKROPDY-UHFFFAOYSA-N - - 3.9 5.2 5.2 Refs
A (Rhodopsin) Orphan TAAR2 TAAR2 TAAR2 Human Β-Phenylethylamine Small molecule NCCc1ccccc1 BHHGXPLMPWCGHP-UHFFFAOYSA-N - -
A (Rhodopsin) Orphan TAAR2 TAAR2 TAAR2 Human Tryptamine Small molecule NCCc1c[nH]c2c1cccc2 APJYDQYYACXCRM-UHFFFAOYSA-N - -
A (Rhodopsin) Orphan TAAR3 TAAR3 TAAR3P Human Isoamylamine Principal 1 Small molecule NCCC(C)C BMFVGAAISNGQNM-UHFFFAOYSA-N - -
A (Rhodopsin) Orphan TAAR3 TAAR3 Taar3 Mouse Isoamylamine Principal 1 Small molecule NCCC(C)C BMFVGAAISNGQNM-UHFFFAOYSA-N - - 5.0 5.0 Refs
A (Rhodopsin) Oxoglutarate OXGR1 oxoglutarate OXGR1 Human Α-Ketoglutaric Acid Principal 1 Small molecule OC(=O)CCC(=O)C(=O)O KPGXRSRHYNQIFN-UHFFFAOYSA-N - 8YYW 3.3 3.9 4.5 Refs
A (Rhodopsin) P2Y P2RY1 P2Y1 P2RY1 Human Adp None 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N XTWYTFMLZFPYCI-KQYNXXCUSA-N - 8WJX Refs
A (Rhodopsin) P2Y P2RY1 P2Y1 P2RY1 Human Atp None 1 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N ZKHQWZAMYRWXGA-KQYNXXCUSA-N - - 4.8 4.8 Refs
A (Rhodopsin) P2Y P2RY2 P2Y2 P2RY2 Human Atp None 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N ZKHQWZAMYRWXGA-KQYNXXCUSA-N - 9K0X 6.6 6.9 7.1 Refs
A (Rhodopsin) P2Y P2RY2 P2Y2 P2RY2 Human Utp None 1 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O PGAVKCOVUIYSFO-XVFCMESISA-N - - 8.1 8.1 Refs
A (Rhodopsin) P2Y P2RY4 P2Y4 P2RY4 Human Atp None 1 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N ZKHQWZAMYRWXGA-KQYNXXCUSA-N - - 5.7 6.0 6.3 Refs
A (Rhodopsin) P2Y P2RY4 P2Y4 P2RY4 Human Utp None 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O PGAVKCOVUIYSFO-XVFCMESISA-N - 9K0K 5.6 5.6 Refs
A (Rhodopsin) P2Y P2RY4 P2Y4 P2ry4 Rat Atp None 1 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N ZKHQWZAMYRWXGA-KQYNXXCUSA-N - - 5.7 6.0 6.3 Refs
A (Rhodopsin) P2Y P2RY4 P2Y4 P2ry4 Rat Utp None 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O PGAVKCOVUIYSFO-XVFCMESISA-N - - 5.6 5.6 Refs
A (Rhodopsin) P2Y P2RY6 P2Y6 P2RY6 Human Adp None 3 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N XTWYTFMLZFPYCI-KQYNXXCUSA-N - 4.5 4.5 Refs
A (Rhodopsin) P2Y P2RY6 P2Y6 P2RY6 Human Udp None 1 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O XCCTYIAWTASOJW-XVFCMESISA-N - 6.5 6.5 Refs
A (Rhodopsin) P2Y P2RY6 P2Y6 P2RY6 Human Utp None 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O PGAVKCOVUIYSFO-XVFCMESISA-N - - 5.2 5.2 Refs
A (Rhodopsin) P2Y P2Y11 P2Y11 P2RY11 Human Adp None 3 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N XTWYTFMLZFPYCI-KQYNXXCUSA-N - Refs
A (Rhodopsin) P2Y P2Y11 P2Y11 P2RY11 Human Atp None 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N ZKHQWZAMYRWXGA-KQYNXXCUSA-N - 4.2 4.9 5.6 Refs
A (Rhodopsin) P2Y P2Y11 P2Y11 P2RY11 Human Utp None 1 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O PGAVKCOVUIYSFO-XVFCMESISA-N - - 5.2 5.2 Refs
A (Rhodopsin) P2Y P2Y12 P2Y12 P2RY12 Human Adp None 1 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N XTWYTFMLZFPYCI-KQYNXXCUSA-N - 5.9 5.9 Refs
A (Rhodopsin) P2Y P2Y12 P2Y12 P2RY12 Human Atp 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N ZKHQWZAMYRWXGA-KQYNXXCUSA-N -
A (Rhodopsin) P2Y P2Y13 P2Y13 P2RY13 Human Adp None 1 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N XTWYTFMLZFPYCI-KQYNXXCUSA-N - 24XY Refs
A (Rhodopsin) P2Y P2Y13 P2Y13 P2RY13 Human Atp None 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N ZKHQWZAMYRWXGA-KQYNXXCUSA-N - Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2RY14 Human Udp None 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O XCCTYIAWTASOJW-XVFCMESISA-N - 24XZ 7.1 7.1 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2RY14 Human Udp N-Acetyl-Glucosamine None 4 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@@H]1O)O)NC(=O)C LFTYTUAZOPRMMI-CFRASDGPSA-N -
A (Rhodopsin) P2Y P2Y14 P2Y14 P2RY14 Human Udp-Galactose None 2 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@H]1O)O)O HSCJRCZFDFQWRP-ABVWGUQPSA-N - 7.1 7.1 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2RY14 Human Udp-Glucose None 1 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@@H]1O)O)O HSCJRCZFDFQWRP-JZMIEXBBSA-N - 9J0B 7.6 7.6 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2RY14 Human Udp-Glucuronic Acid None 3 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O[C@H]2O[C@H](C(=O)O)[C@H]([C@@H]([C@H]2O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O HDYANYHVCAPMJV-LXQIFKJMSA-N - 9J0I
A (Rhodopsin) P2Y P2Y14 P2Y14 P2ry14 Mouse Udp N-Acetyl-Glucosamine None 4 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@@H]1O)O)NC(=O)C LFTYTUAZOPRMMI-CFRASDGPSA-N - - 6.8 6.8 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2ry14 Mouse Udp-Galactose None 2 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@H]1O)O)O HSCJRCZFDFQWRP-ABVWGUQPSA-N - - 7.1 7.1 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2ry14 Mouse Udp-Glucose None 1 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@@H]1O)O)O HSCJRCZFDFQWRP-JZMIEXBBSA-N - - 7.6 7.6 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2ry14 Mouse Udp-Glucuronic Acid None 3 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O[C@H]2O[C@H](C(=O)O)[C@H]([C@@H]([C@H]2O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O HDYANYHVCAPMJV-LXQIFKJMSA-N - - 7.0 7.0 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2ry14 Rat Udp None 2 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O XCCTYIAWTASOJW-XVFCMESISA-N - - 7.1 7.1 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2ry14 Rat Udp N-Acetyl-Glucosamine None 4 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@@H]1O)O)NC(=O)C LFTYTUAZOPRMMI-CFRASDGPSA-N - - 6.8 6.8 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2ry14 Rat Udp-Galactose None 2 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@H]1O)O)O HSCJRCZFDFQWRP-ABVWGUQPSA-N - - 7.1 7.1 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2ry14 Rat Udp-Glucose None 1 Small molecule OC[C@H]1O[C@H](OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)[C@@H]([C@H]([C@@H]1O)O)O HSCJRCZFDFQWRP-JZMIEXBBSA-N - - 7.6 7.6 Refs
A (Rhodopsin) P2Y P2Y14 P2Y14 P2ry14 Rat Udp-Glucuronic Acid None 3 Small molecule O[C@@H]1[C@@H](COP(=O)(OP(=O)(O[C@H]2O[C@H](C(=O)O)[C@H]([C@@H]([C@H]2O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O HDYANYHVCAPMJV-LXQIFKJMSA-N - - 7.0 7.0 Refs
A (Rhodopsin) Platelet-activating factor PTAFR PAF PTAFR Human Paf Principal 1 Lipid CCCCCCCCCCCCCCCCOC[C@@H](OC(=O)C)COP(=O)(OCC[N+](C)(C)C)[O-] HVAUUPRFYPCOCA-AREMUKBSSA-N - 8XYD 7.5 7.7 7.9 Refs
A (Rhodopsin) Prokineticin PKR1 PKR1 PROKR1 Human Prokineticin-1 (Human) 3 Peptide - - - Refs
A (Rhodopsin) Prokineticin PKR1 PKR1 PROKR1 Human Prokineticin-1 (Mouse) 4 Peptide - - -
A (Rhodopsin) Prokineticin PKR1 PKR1 PROKR1 Human Prokineticin-1 (Rat) 4 Peptide - - -
A (Rhodopsin) Prokineticin PKR1 PKR1 PROKR1 Human Prokineticin-2 (Human) 1 Peptide - - - Refs
A (Rhodopsin) Prokineticin PKR1 PKR1 PROKR1 Human Prokineticin-2 (Mouse) 4 Peptide - - -
A (Rhodopsin) Prokineticin PKR1 PKR1 PROKR1 Human Prokineticin-2Β (Human) 2 Peptide - - - Refs
A (Rhodopsin) Prokineticin PKR2 PKR2 PROKR2 Human Prokineticin-1 (Human) 2 Peptide - - - Refs
A (Rhodopsin) Prokineticin PKR2 PKR2 PROKR2 Human Prokineticin-1 (Mouse) 4 Peptide - - -
A (Rhodopsin) Prokineticin PKR2 PKR2 PROKR2 Human Prokineticin-1 (Rat) 4 Peptide - - -
A (Rhodopsin) Prokineticin PKR2 PKR2 PROKR2 Human Prokineticin-2 (Human) 1 Peptide - - - Refs
A (Rhodopsin) Prokineticin PKR2 PKR2 PROKR2 Human Prokineticin-2 (Mouse) 4 Peptide - - -
A (Rhodopsin) Prokineticin PKR2 PKR2 PROKR2 Human Prokineticin-2Β (Human) 3 Peptide - - - Refs
A (Rhodopsin) Prolactin-releasing peptide PRLHR PrRP PRLHR Human Pthrp (Human) 4 Peptide - - - -
A (Rhodopsin) Prolactin-releasing peptide PRLHR PrRP PRLHR Human Prrp-20 (Human) 1 Peptide - - - - 9.0 9.3 9.6 Refs
A (Rhodopsin) Prolactin-releasing peptide PRLHR PrRP PRLHR Human Prrp-20 (Rat) 4 Peptide - - - -
A (Rhodopsin) Prolactin-releasing peptide PRLHR PrRP PRLHR Human Prrp-31 (Human) 2 Peptide - - - - 9.0 9.1 9.2 Refs
A (Rhodopsin) Prolactin-releasing peptide PRLHR PrRP PRLHR Human Prrp-31 (Rat) 4 Peptide - - - -
A (Rhodopsin) Prolactin-releasing peptide PRLHR PrRP PRLHR Human Neuropeptide Y (Human) 3 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N)Cc1ccc(cc1)O)CCCN=C(N)N)CCC(=O)N)CCCN=C(N)N)[C@H](O)C)[C@H](CC)C)CC(C)C)CC(=O)N)[C@H](CC)C)Cc1ccc(cc1)O)Cc1c[nH]cn1)CCCN=C(N)N)CC(C)C)C)CO)Cc1ccc(cc1)O)Cc1ccc(cc1)O)CCCN=C(N)N)C)CCSC)CC(=O)O)CCC(=O)O)C)C)CC(=O)O)CCC(=O)O)CC(=O)N)CC(=O)O)NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1ccc(cc1)O)N)CO XKWCTHKJQNUFOQ-HRPSIEBRSA-N - - 5.4 5.4 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 PTGDR2 Human Δ12-Pgj2 None 3 Small molecule CCCCC[C@@H](C/C=C/1\[C@@H](C/C=C\CCCC(=O)O)C=CC1=O)O TUXFWOHFPFBNEJ-GJGHEGAFSA-N - - 7.3 7.3 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 PTGDR2 Human Pgd2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - 9IYB 7.4 7.5 7.5 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 PTGDR2 Human Pgd3 None 2 Small molecule CCC=CC[C@@H](C=C[C@H]1C(=O)C[C@@H]([C@@H]1CC=CCCCC(=O)O)O)O ANOICLBSJIMQTA-MLHJIOFPSA-N - -
A (Rhodopsin) Prostanoid PD2R2 DP2 PTGDR2 Human Pge2 None 5 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 5.5 5.5 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 PTGDR2 Human Pgf2Α None 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 6.2 6.2 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 PTGDR2 Human Pgi2 6 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@H]2[C@@H]1C/C(=C/CCCC(=O)O)/O2)O KAQKFAOMNZTLHT-OZUDYXHBSA-N - -
A (Rhodopsin) Prostanoid PD2R2 DP2 PTGDR2 Human Thromboxane A2 6 Small molecule CCCCC[C@@H](/C=C/[C@H]1O[C@H]2C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O2)O DSNBHJFQCNUKMA-SCKDECHMSA-N - -
A (Rhodopsin) Prostanoid PD2R2 DP2 Ptgdr2 Mouse Δ12-Pgj2 None 3 Small molecule CCCCC[C@@H](C/C=C/1\[C@@H](C/C=C\CCCC(=O)O)C=CC1=O)O TUXFWOHFPFBNEJ-GJGHEGAFSA-N - - 7.3 7.3 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 Ptgdr2 Mouse Pgd2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 7.4 7.5 7.5 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 Ptgdr2 Mouse Pgd3 None 2 Small molecule CCC=CC[C@@H](C=C[C@H]1C(=O)C[C@@H]([C@@H]1CC=CCCCC(=O)O)O)O ANOICLBSJIMQTA-MLHJIOFPSA-N - - 7.4 7.4 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 Ptgdr2 Mouse Pge2 None 5 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 5.5 5.5 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 Ptgdr2 Mouse Pgf2Α None 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 6.2 6.2 Refs
A (Rhodopsin) Prostanoid PD2R2 DP2 Ptgdr2 Rat Pgd2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 7.4 7.5 7.5 Refs
A (Rhodopsin) Prostanoid PD2R DP1 PTGDR Human Δ12-Pgj2 None 1 Small molecule CCCCC[C@@H](C/C=C/1\[C@@H](C/C=C\CCCC(=O)O)C=CC1=O)O TUXFWOHFPFBNEJ-GJGHEGAFSA-N - - 9.0 9.0 Refs
A (Rhodopsin) Prostanoid PD2R DP1 PTGDR Human Pgd2 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - 9E9S 7.8 7.6 7.6 Refs
A (Rhodopsin) Prostanoid PD2R DP1 PTGDR Human Pge1 None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 7.3 7.3 Refs
A (Rhodopsin) Prostanoid PD2R DP1 PTGDR Human Pge2 None 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 6.5 6.8 7.0 Refs
A (Rhodopsin) Prostanoid PD2R DP1 PTGDR Human Pgf2Α None 5 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - 6.1 6.3 6.4 Refs
A (Rhodopsin) Prostanoid PD2R DP1 PTGDR Human Pgi2 6 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@H]2[C@@H]1C/C(=C/CCCC(=O)O)/O2)O KAQKFAOMNZTLHT-OZUDYXHBSA-N - -
A (Rhodopsin) Prostanoid PD2R DP1 PTGDR Human Thromboxane A2 6 Small molecule CCCCC[C@@H](/C=C/[C@H]1O[C@H]2C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O2)O DSNBHJFQCNUKMA-SCKDECHMSA-N - -
A (Rhodopsin) Prostanoid PD2R DP1 Ptgdr Mouse Pgd2 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 7.8 7.6 7.6 Refs
A (Rhodopsin) Prostanoid PD2R DP1 Ptgdr Rat Pgd2 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 7.8 7.6 7.6 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 PTGER1 Human Pgd2 None 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 5.2 5.2 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 PTGER1 Human Pge1 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - 7.0 7.0 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 PTGER1 Human Pge2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - 9M1H 7.3 7.7 7.7 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 PTGER1 Human Pgf2Α None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - 6.2 6.4 6.4 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 PTGER1 Human Pgi2 None 5 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@H]2[C@@H]1C/C(=C/CCCC(=O)O)/O2)O KAQKFAOMNZTLHT-OZUDYXHBSA-N - - 4.8 4.8 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 PTGER1 Human Thromboxane A2 6 Small molecule CCCCC[C@@H](/C=C/[C@H]1O[C@H]2C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O2)O DSNBHJFQCNUKMA-SCKDECHMSA-N -
A (Rhodopsin) Prostanoid PE2R1 EP1 Ptger1 Mouse Pge1 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 7.0 7.0 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 Ptger1 Mouse Pge2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 7.3 7.7 7.7 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 Ptger1 Mouse Pgf2Α None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 6.2 6.4 6.4 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 Ptger1 Rat Pgd2 None 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 5.2 5.2 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 Ptger1 Rat Pge1 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 7.0 7.0 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 Ptger1 Rat Pge2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 7.3 7.7 7.7 Refs
A (Rhodopsin) Prostanoid PE2R1 EP1 Ptger1 Rat Pgf2Α None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 6.2 6.4 6.4 Refs
A (Rhodopsin) Prostanoid PE2R2 EP2 PTGER2 Human Pgd2 None 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 5.3 5.3 Refs
A (Rhodopsin) Prostanoid PE2R2 EP2 PTGER2 Human Pge1 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N -
A (Rhodopsin) Prostanoid PE2R2 EP2 PTGER2 Human Pge2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - 7CX2 7.4 8.2 8.2 Refs
A (Rhodopsin) Prostanoid PE2R2 EP2 PTGER2 Human Pgf2Α None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - 5.2 5.6 5.6 Refs
A (Rhodopsin) Prostanoid PE2R2 EP2 PTGER2 Human Pgi2 5 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@H]2[C@@H]1C/C(=C/CCCC(=O)O)/O2)O KAQKFAOMNZTLHT-OZUDYXHBSA-N -
A (Rhodopsin) Prostanoid PE2R2 EP2 PTGER2 Human Thromboxane A2 5 Small molecule CCCCC[C@@H](/C=C/[C@H]1O[C@H]2C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O2)O DSNBHJFQCNUKMA-SCKDECHMSA-N - -
A (Rhodopsin) Prostanoid PE2R2 EP2 Ptger2 Mouse Pge1 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 8.0 8.0 Refs
A (Rhodopsin) Prostanoid PE2R2 EP2 Ptger2 Mouse Pge2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 7.4 8.2 8.2 Refs
A (Rhodopsin) Prostanoid PE2R2 EP2 Ptger2 Rat Pgd2 None 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 5.3 5.3 Refs
A (Rhodopsin) Prostanoid PE2R2 EP2 Ptger2 Rat Pge1 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 8.0 8.0 Refs
A (Rhodopsin) Prostanoid PE2R2 EP2 Ptger2 Rat Pge2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 7.4 8.2 8.2 Refs
A (Rhodopsin) Prostanoid PE2R2 EP2 Ptger2 Rat Pgf2Α None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 5.2 5.6 5.6 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 PTGER3 Human Pgd2 None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - -
A (Rhodopsin) Prostanoid PE2R3 EP3 PTGER3 Human Pge1 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N -
A (Rhodopsin) Prostanoid PE2R3 EP3 PTGER3 Human Pge2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - 6AK3 9.4 9.4 9.0 9.0 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 PTGER3 Human Pgf2Α None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - 8.4 8.4 6.7 6.7 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 PTGER3 Human Pgi2 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@H]2[C@@H]1C/C(=C/CCCC(=O)O)/O2)O KAQKFAOMNZTLHT-OZUDYXHBSA-N -
A (Rhodopsin) Prostanoid PE2R3 EP3 PTGER3 Human Thromboxane A2 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1O[C@H]2C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O2)O DSNBHJFQCNUKMA-SCKDECHMSA-N -
A (Rhodopsin) Prostanoid PE2R3 EP3 Ptger3 Mouse Pgd2 None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 7.9 7.9 5.9 7.4 8.9 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 Ptger3 Mouse Pge1 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 9.4 9.4 9.0 9.0 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 Ptger3 Mouse Pge2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 9.4 9.4 9.0 9.0 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 Ptger3 Mouse Pgf2Α None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 8.4 8.4 6.7 6.7 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 Ptger3 Rat Pgd2 None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 7.9 7.9 5.9 7.4 8.9 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 Ptger3 Rat Pge1 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 9.4 9.4 9.0 9.0 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 Ptger3 Rat Pge2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 9.4 9.4 9.0 9.0 Refs
A (Rhodopsin) Prostanoid PE2R3 EP3 Ptger3 Rat Pgf2Α None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 8.4 8.4 6.7 6.7 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 PTGER4 Human Pgd2 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 8.8 8.8 8.7 5.9 5.9 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 PTGER4 Human Pge1 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 9.5 9.5 9.2 9.2 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 PTGER4 Human Pge2 None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - 7D7M 6.1 6.1 8.5 9.0 9.0 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 PTGER4 Human Pgf2Α None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 6.1 6.1 9.1 6.2 6.2 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 PTGER4 Human Pgi2 None 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@H]2[C@@H]1C/C(=C/CCCC(=O)O)/O2)O KAQKFAOMNZTLHT-OZUDYXHBSA-N - - 5.1 5.1 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 PTGER4 Human Thromboxane A2 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1O[C@H]2C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O2)O DSNBHJFQCNUKMA-SCKDECHMSA-N - -
A (Rhodopsin) Prostanoid PE2R4 EP4 Ptger4 Mouse Pge1 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 9.5 9.5 9.2 9.2 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 Ptger4 Mouse Pge2 None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 6.1 6.1 8.5 9.0 9.0 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 Ptger4 Rat Pgd2 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 8.8 8.8 8.7 5.9 5.9 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 Ptger4 Rat Pge1 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 9.5 9.5 9.2 9.2 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 Ptger4 Rat Pge2 None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 6.1 6.1 8.5 9.0 9.0 Refs
A (Rhodopsin) Prostanoid PE2R4 EP4 Ptger4 Rat Pgf2Α None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 6.1 6.1 9.1 6.2 6.2 Refs
A (Rhodopsin) Prostanoid PF2R FP PTGFR Human Pgd2 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 7.3 7.3 Refs
A (Rhodopsin) Prostanoid PF2R FP PTGFR Human Pge2 None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 6.4 7.0 7.0 Refs
A (Rhodopsin) Prostanoid PF2R FP PTGFR Human Pgf2Α None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - 8IUK 7.9 8.5 8.5 Refs
A (Rhodopsin) Prostanoid PF2R FP PTGFR Human Pgi2 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@H]2[C@@H]1C/C(=C/CCCC(=O)O)/O2)O KAQKFAOMNZTLHT-OZUDYXHBSA-N -
A (Rhodopsin) Prostanoid PF2R FP PTGFR Human Thromboxane A2 4 Small molecule CCCCC[C@@H](/C=C/[C@H]1O[C@H]2C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O2)O DSNBHJFQCNUKMA-SCKDECHMSA-N -
A (Rhodopsin) Prostanoid PF2R FP Ptgfr Mouse Pgd2 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - - 7.3 7.3 Refs
A (Rhodopsin) Prostanoid PF2R FP Ptgfr Mouse Pge2 None 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 6.4 7.0 7.0 Refs
A (Rhodopsin) Prostanoid PF2R FP Ptgfr Mouse Pgf2Α None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - - 7.9 8.5 8.5 Refs
A (Rhodopsin) Prostanoid PI2R IP PTGIR Human Pgd2 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - -
A (Rhodopsin) Prostanoid PI2R IP PTGIR Human Pge1 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - 6.5 7.5 7.5 Refs
A (Rhodopsin) Prostanoid PI2R IP PTGIR Human Pge2 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - -
A (Rhodopsin) Prostanoid PI2R IP PTGIR Human Pgf2Α 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N -
A (Rhodopsin) Prostanoid PI2R IP PTGIR Human Pgi2 None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@H]2[C@@H]1C/C(=C/CCCC(=O)O)/O2)O KAQKFAOMNZTLHT-OZUDYXHBSA-N - B2M_PI2R_HUMAN_EPOPROSTENOL_GNA12_HUMAN 7.8 7.8 Refs
A (Rhodopsin) Prostanoid PI2R IP PTGIR Human Thromboxane A2 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1O[C@H]2C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O2)O DSNBHJFQCNUKMA-SCKDECHMSA-N - -
A (Rhodopsin) Prostanoid PI2R IP Ptgir Mouse Pge1 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1CCCCCCC(=O)O)O GMVPRGQOIOIIMI-DWKJAMRDSA-N - - 6.5 7.5 7.5 Refs
A (Rhodopsin) Prostanoid TA2R TP TBXA2R Human Pgd2 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1C(=O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O BHMBVRSPMRCCGG-OUTUXVNYSA-N - -
A (Rhodopsin) Prostanoid TA2R TP TBXA2R Human Pge2 None 2 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)CC(=O)[C@@H]1C/C=C\CCCC(=O)O)O XEYBRNLFEZDVAW-ARSRFYASSA-N - - 4.5 4.5 Refs
A (Rhodopsin) Prostanoid TA2R TP TBXA2R Human Pgf2Α None 1 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O)O PXGPLTODNUVGFL-YNNPMVKQSA-N - 5.1 5.1 Refs
A (Rhodopsin) Prostanoid TA2R TP TBXA2R Human Pgh2 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@@H]2OO[C@H]([C@@H]1C/C=C\CCCC(=O)O)C2)O YIBNHAJFJUQSRA-YNNPMVKQSA-N -
A (Rhodopsin) Prostanoid TA2R TP TBXA2R Human Pgi2 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1[C@H](O)C[C@H]2[C@@H]1C/C(=C/CCCC(=O)O)/O2)O KAQKFAOMNZTLHT-OZUDYXHBSA-N -
A (Rhodopsin) Prostanoid TA2R TP TBXA2R Human Thromboxane A2 3 Small molecule CCCCC[C@@H](/C=C/[C@H]1O[C@H]2C[C@@H]([C@@H]1C/C=C\CCCC(=O)O)O2)O DSNBHJFQCNUKMA-SCKDECHMSA-N -
A (Rhodopsin) Proteinase-activated PAR1 PAR1 F2R Human Thrombin (Human) Principal 1 Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR1 PAR1 F2R Human Thrombin (Mouse) Principal 1 Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR1 PAR1 F2R Human Thrombin (Rat) Principal 1 Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR3 PAR3 F2RL2 Human Thrombin (Human) Principal 1 Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR3 PAR3 F2RL2 Human Thrombin (Mouse) Principal 1 Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR3 PAR3 F2RL2 Human Thrombin (Rat) Principal 1 Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR4 PAR4 F2RL3 Human Cathepsin G (Human) Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR4 PAR4 F2RL3 Human Cathepsin G (Mouse) Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR4 PAR4 F2RL3 Human Cathepsin G (Rat) Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR4 PAR4 F2RL3 Human Thrombin (Human) Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR4 PAR4 F2RL3 Human Thrombin (Mouse) Peptide - - - -
A (Rhodopsin) Proteinase-activated PAR4 PAR4 F2RL3 Human Thrombin (Rat) Peptide - - - -
A (Rhodopsin) Proton GP132 GPR132 GPR132 Human 9-Hydroxyoctadecadienoic Acid Principal 1 Small molecule CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O NPDSHTNEKLQQIJ-UINYOVNOSA-N - 8HQN 5.7 5.7 Refs
A (Rhodopsin) QRFP QRFPR QRFP QRFPR Human Qrfp26 (26rfa) (Human) 2 Peptide - - - 8.1 8.1 Refs
A (Rhodopsin) QRFP QRFPR QRFP QRFPR Human Qrfp43 (43rfa) (Human) 3 Peptide - - - - 6.9 7.8 8.6 Refs
A (Rhodopsin) QRFP QRFPR QRFP QRFPR Human Qrfp43 (Rat) 5 Peptide - - - -
A (Rhodopsin) QRFP QRFPR QRFP Qrfpr Mouse Qrfp26 (Mouse) 1 Peptide - - - - 8.2 8.2 Refs
A (Rhodopsin) QRFP QRFPR QRFP Qrfpr Mouse Qrfp43 (Mouse) 4 Peptide - - - - 6.7 7.0 7.2 Refs
A (Rhodopsin) QRFP QRFPR QRFP Qrfpr Rat Qrfp26 (Rat) 5 Peptide - - - - Refs
A (Rhodopsin) Relaxin family peptide Q5Y986 RXFP3 Rxfp3 Rat Relaxin-3 (Rat) 3 Peptide - - - - Refs
A (Rhodopsin) Relaxin family peptide RL3R1 RXFP3 RXFP3 Human Insl5 (Human) 3 Peptide - - - - 7.0 7.0 Refs
A (Rhodopsin) Relaxin family peptide RL3R1 RXFP3 RXFP3 Human Relaxin (Human) 2 Peptide - - - - 7.1 7.8 8.4 Refs
A (Rhodopsin) Relaxin family peptide RL3R1 RXFP3 RXFP3 Human Relaxin-3 (B Chain) (Human) 3 Peptide - - - - Refs
A (Rhodopsin) Relaxin family peptide RL3R1 RXFP3 RXFP3 Human Relaxin-3 (Human) 1 Peptide - - - - 8.3 9.1 9.9 7.8 8.4 8.9 Refs
A (Rhodopsin) Relaxin family peptide RL3R2 RXFP4 RXFP4 Human Insl5 (Human) 3 Peptide - - - - 7.0 7.7 8.9 7.3 8.1 8.8 Refs
A (Rhodopsin) Relaxin family peptide RL3R2 RXFP4 RXFP4 Human Relaxin-3 (B Chain) (Human) 4 Peptide - - - - 7.0 7.0 Refs
A (Rhodopsin) Relaxin family peptide RL3R2 RXFP4 RXFP4 Human Relaxin-3 (Human) 1 Peptide - - - - 8.7 9.2 9.7 8.8 8.9 9.0 Refs
A (Rhodopsin) Relaxin family peptide RL3R2 RXFP4 Rxfp4 Mouse Insl5 (Mouse) 2 Peptide - - - - 7.8 8.6 9.4 8.5 8.7 8.8 Refs
A (Rhodopsin) Relaxin family peptide RXFP1 RXFP1 RXFP1 Human Relaxin (Human) 1 Peptide - - - - 10.4 10.4 9.2 9.7 10.2 Refs
A (Rhodopsin) Relaxin family peptide RXFP1 RXFP1 RXFP1 Human Relaxin-1 (Human) 2 Peptide - - - - 8.8 8.8 Refs
A (Rhodopsin) Relaxin family peptide RXFP1 RXFP1 RXFP1 Human Relaxin-3 (Human) 3 Peptide - - - - 7.5 7.8 8.0 Refs
A (Rhodopsin) Relaxin family peptide RXFP2 RXFP2 RXFP2 Human Insl3 (Human) 2 Peptide - - - - 9.3 9.5 9.7 Refs
A (Rhodopsin) Relaxin family peptide RXFP2 RXFP2 RXFP2 Human Relaxin (Human) 1 Peptide - - - - 9.1 9.1 8.3 8.4 8.5 Refs
A (Rhodopsin) Relaxin family peptide RXFP2 RXFP2 RXFP2 Human Relaxin-1 (Human) 2 Peptide - - - - 8.8 8.8 Refs
A (Rhodopsin) Relaxin family peptide RXFP2 RXFP2 RXFP2 Human Relaxin-3 (Human) 2 Peptide - - - - 7.0 7.0 Refs
A (Rhodopsin) Somatostatin SSR1 SST1 SSTR1 Human Cst-17 (Human) 1 Peptide - - - 9.1 9.4 9.6 Refs
A (Rhodopsin) Somatostatin SSR1 SST1 SSTR1 Human Srif-14 (Human) 2 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - AFM_SSR1_HUMAN_hashedseq[NJ4IM4MWSOW2HEXWNXNOALOKZM0] 8.6 9.1 9.5 Refs
A (Rhodopsin) Somatostatin SSR1 SST1 SSTR1 Human Srif-28 (Human) 3 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - 8.6 9.0 9.4 Refs
A (Rhodopsin) Somatostatin SSR1 SST1 SSTR1 Human Cortistatin-14 (Mouse) 4 Peptide - - -
A (Rhodopsin) Somatostatin SSR1 SST1 Sstr1 Rat Srif-14 (Human) 2 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - - 8.6 9.1 9.5 Refs
A (Rhodopsin) Somatostatin SSR2 SST2 SSTR2 Human Cst-17 (Human) 2 Peptide - - - 8.8 9.1 9.3 Refs
A (Rhodopsin) Somatostatin SSR2 SST2 SSTR2 Human Srif-14 (Human) 1 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - AFM_SSR2_HUMAN_hashedseq[NJ4IM4MWSOW2HEXWNXNOALOKZM0] 9.0 9.1 9.1 8.8 8.8 8.8 Refs
A (Rhodopsin) Somatostatin SSR2 SST2 SSTR2 Human Srif-28 (Human) 2 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - 8.4 8.8 8.8 Refs
A (Rhodopsin) Somatostatin SSR2 SST2 SSTR2 Human Cortistatin-14 (Mouse) 2 Peptide - - -
A (Rhodopsin) Somatostatin SSR2 SST2 Sstr2 Mouse Srif-14 (Human) 1 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - - 9.0 9.1 9.1 8.8 8.8 8.8 Refs
A (Rhodopsin) Somatostatin SSR2 SST2 Sstr2 Mouse Srif-28 (Human) 2 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - - 8.4 8.8 8.8 Refs
A (Rhodopsin) Somatostatin SSR2 SST2 Sstr2 Rat Srif-14 (Human) 1 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - - 9.0 9.1 9.1 8.8 8.8 8.8 Refs
A (Rhodopsin) Somatostatin SSR2 SST2 Sstr2 Rat Srif-28 (Human) 2 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - - 8.4 8.8 8.8 Refs
A (Rhodopsin) Somatostatin SSR3 SST3 SSTR3 Human Cst-17 (Human) 1 Peptide - - - 8.7 9.3 9.9 Refs
A (Rhodopsin) Somatostatin SSR3 SST3 SSTR3 Human Srif-14 (Human) 3 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - AFM_SSR3_HUMAN_hashedseq[NJ4IM4MWSOW2HEXWNXNOALOKZM0] 8.7 8.9 8.9 Refs
A (Rhodopsin) Somatostatin SSR3 SST3 SSTR3 Human Srif-28 (Human) 2 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - 8.1 9.1 9.1 Refs
A (Rhodopsin) Somatostatin SSR3 SST3 SSTR3 Human Cortistatin-14 (Mouse) 4 Peptide - - -
A (Rhodopsin) Somatostatin SSR3 SST3 Sstr3 Mouse Srif-14 (Human) 3 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - - 8.7 8.9 8.9 Refs
A (Rhodopsin) Somatostatin SSR3 SST3 Sstr3 Mouse Srif-28 (Human) 2 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - - 8.1 9.1 9.1 Refs
A (Rhodopsin) Somatostatin SSR3 SST3 Sstr3 Rat Srif-14 (Human) 3 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - - 8.7 8.9 8.9 Refs
A (Rhodopsin) Somatostatin SSR3 SST3 Sstr3 Rat Srif-28 (Human) 2 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - - 8.1 9.1 9.1 Refs
A (Rhodopsin) Somatostatin SSR4 SST4 SSTR4 Human Cst-17 (Human) 1 Peptide - - - 8.5 9.1 9.6 Refs
A (Rhodopsin) Somatostatin SSR4 SST4 SSTR4 Human Srif-14 (Human) 2 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - 8.4 8.9 9.3 Refs
A (Rhodopsin) Somatostatin SSR4 SST4 SSTR4 Human Srif-28 (Human) 3 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - 8.1 8.7 9.2 Refs
A (Rhodopsin) Somatostatin SSR4 SST4 SSTR4 Human Cortistatin-14 (Mouse) 4 Peptide - - -
A (Rhodopsin) Somatostatin SSR4 SST4 Sstr4 Rat Srif-14 (Human) 2 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - - 8.4 8.9 9.3 Refs
A (Rhodopsin) Somatostatin SSR5 SST5 SSTR5 Human Cst-17 (Human) 1 Peptide - - - 8.5 9.4 10.2 Refs
A (Rhodopsin) Somatostatin SSR5 SST5 SSTR5 Human Srif-14 (Human) 4 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - 7.7 8.4 8.4 Refs
A (Rhodopsin) Somatostatin SSR5 SST5 SSTR5 Human Srif-28 (Human) 3 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - 9.8 9.0 9.0 Refs
A (Rhodopsin) Somatostatin SSR5 SST5 SSTR5 Human Cortistatin-14 (Mouse) 2 Peptide - - - 8.7 9.1 9.4 Refs
A (Rhodopsin) Somatostatin SSR5 SST5 Sstr5 Mouse Srif-14 (Human) 4 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - - 7.7 8.4 8.4 Refs
A (Rhodopsin) Somatostatin SSR5 SST5 Sstr5 Mouse Srif-28 (Human) 3 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - - 9.8 9.0 9.0 Refs
A (Rhodopsin) Somatostatin SSR5 SST5 Sstr5 Mouse Cortistatin-14 (Mouse) 2 Peptide - - - - 8.7 9.1 9.4 Refs
A (Rhodopsin) Somatostatin SSR5 SST5 Sstr5 Rat Srif-14 (Human) 4 Peptide NCCCC[C@H]1NC(=O)[C@@H](CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC(=O)[C@H](NC(=O)[C@@H](NC1=O)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)C(=O)O)NC(=O)CNC(=O)[C@@H](N)C VVEJUSYNERNRME-XGFVQVCISA-N - - 7.7 8.4 8.4 Refs
A (Rhodopsin) Somatostatin SSR5 SST5 Sstr5 Rat Srif-28 (Human) 3 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCCCN)CC(=O)N)Cc1ccccc1)Cc1ccccc1)Cc1c[nH]c2c1cccc2)CCCCN)[C@H](O)C)[C@H](O)C)C(=O)O)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)N)C)CC(=O)N)CO)CC(=O)N)C)CCSC)C)CCCNC(=N)N)CCC(=O)O)CCCNC(=N)N GGYTXJNZMFRSLX-DFTNLTQTSA-N - - 9.8 9.0 9.0 Refs
A (Rhodopsin) Succinate SUCR1 succinate SUCNR1 Human Succinic Acid Principal 1 Small molecule OC(=O)CCC(=O)O KDYFGRWQOYBRFD-UHFFFAOYSA-N - 8JPP 3.1 3.9 4.7 Refs
A (Rhodopsin) Tachykinin NK1R NK1 TACR1 Human Hemokinin 1 (Mouse) 4 Peptide - - -
A (Rhodopsin) Tachykinin NK1R NK1 TACR1 Human Neurokinin A (Human) 2 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)C(C)C)Cc1ccccc1)CO)CC(=O)O)[C@H](O)C)NC(=O)[C@H](Cc1[nH]cnc1)N HEAUFJZALFKPBA-JPQUDPSNSA-N - 6.2 7.8 9.3 Refs
A (Rhodopsin) Tachykinin NK1R NK1 TACR1 Human Neurokinin B (Human) 3 Peptide CSCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)C(C)C)Cc1ccccc1)Cc1ccccc1)CC(=O)O)Cc1[nH]cnc1)NC(=O)[C@H](CC(=O)O)N NHXYSAFTNPANFK-HDMCBQFHSA-N - 6.1 6.3 6.4 Refs
A (Rhodopsin) Tachykinin NK1R NK1 TACR1 Human Neuropeptide Γ (Human) 4 Peptide - - - Refs
A (Rhodopsin) Tachykinin NK1R NK1 TACR1 Human Neuropeptide K (Human) 4 Peptide - - - Refs
A (Rhodopsin) Tachykinin NK1R NK1 TACR1 Human Substance P (Human) 1 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)Cc1ccccc1)Cc1ccccc1)CCC(=O)N)CCC(=O)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)N ADNPLDHMAVUMIW-CUZNLEPHSA-N - 7P00 8.5 9.4 10.3 Refs
A (Rhodopsin) Tachykinin NK2R NK2 TACR2 Human Hemokinin 1 (Mouse) 4 Peptide - - -
A (Rhodopsin) Tachykinin NK2R NK2 TACR2 Human Neurokinin A (Human) 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)C(C)C)Cc1ccccc1)CO)CC(=O)O)[C@H](O)C)NC(=O)[C@H](Cc1[nH]cnc1)N HEAUFJZALFKPBA-JPQUDPSNSA-N - 7XWO 8.0 8.6 9.1 Refs
A (Rhodopsin) Tachykinin NK2R NK2 TACR2 Human Neurokinin B (Human) 3 Peptide CSCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)C(C)C)Cc1ccccc1)Cc1ccccc1)CC(=O)O)Cc1[nH]cnc1)NC(=O)[C@H](CC(=O)O)N NHXYSAFTNPANFK-HDMCBQFHSA-N - 5.0 6.4 7.7 Refs
A (Rhodopsin) Tachykinin NK2R NK2 TACR2 Human Neuropeptide Γ (Human) 4 Peptide - - -
A (Rhodopsin) Tachykinin NK2R NK2 TACR2 Human Neuropeptide K (Human) 4 Peptide - - -
A (Rhodopsin) Tachykinin NK2R NK2 TACR2 Human Substance P (Human) 2 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)Cc1ccccc1)Cc1ccccc1)CCC(=O)N)CCC(=O)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)N ADNPLDHMAVUMIW-CUZNLEPHSA-N - - 5.9 6.4 6.9 Refs
A (Rhodopsin) Tachykinin NK3R NK3 TACR3 Human Neurokinin A (Human) 2 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)C(C)C)Cc1ccccc1)CO)CC(=O)O)[C@H](O)C)NC(=O)[C@H](Cc1[nH]cnc1)N HEAUFJZALFKPBA-JPQUDPSNSA-N - 7.4 7.4 5.5 6.1 6.1 Refs
A (Rhodopsin) Tachykinin NK3R NK3 TACR3 Human Neurokinin B (Human) 1 Peptide CSCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)C(C)C)Cc1ccccc1)Cc1ccccc1)CC(=O)O)Cc1[nH]cnc1)NC(=O)[C@H](CC(=O)O)N NHXYSAFTNPANFK-HDMCBQFHSA-N - 8JBG 8.4 8.4 8.6 8.7 8.7 Refs
A (Rhodopsin) Tachykinin NK3R NK3 TACR3 Human Substance P (Human) 3 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)Cc1ccccc1)Cc1ccccc1)CCC(=O)N)CCC(=O)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)N ADNPLDHMAVUMIW-CUZNLEPHSA-N - 8JBH 5.0 5.3 5.3 Refs
A (Rhodopsin) Tachykinin NK3R NK3 Tacr3 Mouse Hemokinin 1 (Mouse) 3 Peptide - - - - 9.2 9.3 9.3 Refs
A (Rhodopsin) Tachykinin NK3R NK3 Tacr3 Mouse Neurokinin A (Human) 2 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)C(C)C)Cc1ccccc1)CO)CC(=O)O)[C@H](O)C)NC(=O)[C@H](Cc1[nH]cnc1)N HEAUFJZALFKPBA-JPQUDPSNSA-N - - 7.4 7.4 5.5 6.1 6.1 Refs
A (Rhodopsin) Tachykinin NK3R NK3 Tacr3 Mouse Neurokinin B (Human) 1 Peptide CSCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)C(C)C)Cc1ccccc1)Cc1ccccc1)CC(=O)O)Cc1[nH]cnc1)NC(=O)[C@H](CC(=O)O)N NHXYSAFTNPANFK-HDMCBQFHSA-N - - 8.4 8.4 8.6 8.7 8.7 Refs
A (Rhodopsin) Tachykinin NK3R NK3 Tacr3 Mouse Substance P (Human) 3 Peptide NCCCC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N)CCSC)CC(C)C)Cc1ccccc1)Cc1ccccc1)CCC(=O)N)CCC(=O)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCN=C(N)N)N ADNPLDHMAVUMIW-CUZNLEPHSA-N - - 5.0 5.3 5.3 Refs
A (Rhodopsin) Thyrotropin-releasing hormone TRFR TRH1 TRHR Human Trh (Human) Principal 1 Peptide O=C1CC[C@H](N1)C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N)Cc1nc[nH]c1 XNSAINXGIQZQOO-SRVKXCTJSA-N - 7WKD 7.4 7.4 Refs
A (Rhodopsin) Thyrotropin-releasing hormone TRHR TRH1 Trhr Rat Trh (Human) Principal 1 Peptide O=C1CC[C@H](N1)C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N)Cc1nc[nH]c1 XNSAINXGIQZQOO-SRVKXCTJSA-N - - 7.4 7.4 Refs
A (Rhodopsin) Trace amine TAAR1 TA1 TAAR1 Human Β-Phenylethylamine None 3 Small molecule NCCc1ccccc1 BHHGXPLMPWCGHP-UHFFFAOYSA-N - 8WCA 6.4 6.5 6.6 Refs
A (Rhodopsin) Trace amine TAAR1 TA1 TAAR1 Human 3-Iodothyronamine None 1 Small molecule NCCc1ccc(cc1)Oc1ccc(c(c1)I)O HCYGDNGLWSZCCA-UHFFFAOYSA-N - -
A (Rhodopsin) Trace amine TAAR1 TA1 TAAR1 Human Dopamine 4 Small molecule NCCc1ccc(c(c1)O)O VYFYYTLLBUKUHU-UHFFFAOYSA-N - -
A (Rhodopsin) Trace amine TAAR1 TA1 TAAR1 Human Octopamine None 4 Small molecule NCC(c1ccc(cc1)O)O QHGUCRYDKWKLMG-UHFFFAOYSA-N - -
A (Rhodopsin) Trace amine TAAR1 TA1 TAAR1 Human Tyramine None 2 Small molecule NCCc1ccc(cc1)O DZGWFCGJZKJUFP-UHFFFAOYSA-N - - 6.9 7.1 7.2 7.2 7.2 Refs
A (Rhodopsin) Trace amine TAAR1 TA1 Taar1 Mouse Β-Phenylethylamine None 3 Small molecule NCCc1ccccc1 BHHGXPLMPWCGHP-UHFFFAOYSA-N - 8WC6 6.4 6.5 6.6 Refs
A (Rhodopsin) Trace amine TAAR1 TA1 Taar1 Mouse 3-Iodothyronamine None 1 Small molecule NCCc1ccc(cc1)Oc1ccc(c(c1)I)O HCYGDNGLWSZCCA-UHFFFAOYSA-N - - 7.5 7.7 7.9 Refs
A (Rhodopsin) Trace amine TAAR1 TA1 Taar1 Mouse Tyramine None 2 Small molecule NCCc1ccc(cc1)O DZGWFCGJZKJUFP-UHFFFAOYSA-N - - 6.9 7.1 7.2 7.2 7.2 Refs
A (Rhodopsin) Trace amine TAAR1 TA1 Taar1 Rat Β-Phenylethylamine None 3 Small molecule NCCc1ccccc1 BHHGXPLMPWCGHP-UHFFFAOYSA-N - - 6.4 6.5 6.6 Refs
A (Rhodopsin) Trace amine TAAR1 TA1 Taar1 Rat 3-Iodothyronamine None 1 Small molecule NCCc1ccc(cc1)Oc1ccc(c(c1)I)O HCYGDNGLWSZCCA-UHFFFAOYSA-N - - 7.5 7.7 7.9 Refs
A (Rhodopsin) Trace amine TAAR1 TA1 Taar1 Rat Tyramine None 2 Small molecule NCCc1ccc(cc1)O DZGWFCGJZKJUFP-UHFFFAOYSA-N - - 6.9 7.1 7.2 7.2 7.2 Refs
A (Rhodopsin) Urotensin UR2R UT UTS2R Human Urotensin Ii-Related Peptide (Human) 4 Peptide NCCCC[C@@H]1NC(=O)[C@@H](NC(=O)[C@H](CC2CCCCC2)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@@H](NC1=O)Cc1ccc(cc1)O)C(=O)N[C@H](C(=O)O)C(C)C)NC(=O)[C@@H](N)C)Cc1c[nH]c2c1cccc2 BKBNRUZZGBUWOM-KOOAXUMWSA-N - Refs
A (Rhodopsin) Urotensin UR2R UT UTS2R Human Urotensin-Ii (Human) 2 Peptide - - - - 8.6 8.6 Refs
A (Rhodopsin) Urotensin UR2R UT Uts2r Mouse Urotensin-Ii (Mouse) 3 Peptide - - - - 8.4 8.5 8.6 Refs
A (Rhodopsin) Urotensin UR2R UT Uts2r Rat Urotensin-Ii (Rat) 1 Peptide - - - - 8.8 8.8 Refs
A (Rhodopsin) Vasopressin and oxytocin OXYR OT OXTR Human Oxytocin (Human) 1 Peptide CC[C@@H]([C@@H]1NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCC(=O)N)CC(=O)N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CC(C)C)C XNOPRXBHLZRZKH-DSZYJQQASA-N - 7RYC 8.2 8.7 8.7 Refs
A (Rhodopsin) Vasopressin and oxytocin OXYR OT OXTR Human Vasopressin (Human) 2 Peptide NC(=O)C[C@@H]1NC(=O)[C@H](CCC(=O)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@H](CSSC[C@H](NC1=O)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CCCN=C(N)N)N KBZOIRJILGZLEJ-LGYYRGKSSA-N - B2M_OXYR_HUMAN_VASOPRESSIN_GNAQ_HUMAN 7.3 8.3 9.3 Refs
A (Rhodopsin) Vasopressin and oxytocin OXYR OT Oxtr Rat Oxytocin (Human) 1 Peptide CC[C@@H]([C@@H]1NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCC(=O)N)CC(=O)N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CC(C)C)C XNOPRXBHLZRZKH-DSZYJQQASA-N - - 8.2 8.7 8.7 Refs
A (Rhodopsin) Vasopressin and oxytocin V1AR V1A AVPR1A Human Oxytocin (Human) 2 Peptide CC[C@@H]([C@@H]1NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCC(=O)N)CC(=O)N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CC(C)C)C XNOPRXBHLZRZKH-DSZYJQQASA-N - - 6.9 6.1 6.1 Refs
A (Rhodopsin) Vasopressin and oxytocin V1AR V1A AVPR1A Human Vasopressin (Human) 1 Peptide NC(=O)C[C@@H]1NC(=O)[C@H](CCC(=O)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@H](CSSC[C@H](NC1=O)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CCCN=C(N)N)N KBZOIRJILGZLEJ-LGYYRGKSSA-N - B2M_V1AR_HUMAN_VASOPRESSIN_GNA11_HUMAN 8.5 8.4 8.4 Refs
A (Rhodopsin) Vasopressin and oxytocin V1AR V1A Avpr1a Rat Oxytocin (Human) 2 Peptide CC[C@@H]([C@@H]1NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCC(=O)N)CC(=O)N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CC(C)C)C XNOPRXBHLZRZKH-DSZYJQQASA-N - - 6.9 6.1 6.1 Refs
A (Rhodopsin) Vasopressin and oxytocin V1AR V1A Avpr1a Rat Vasopressin (Human) 1 Peptide NC(=O)C[C@@H]1NC(=O)[C@H](CCC(=O)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@H](CSSC[C@H](NC1=O)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CCCN=C(N)N)N KBZOIRJILGZLEJ-LGYYRGKSSA-N - - 8.5 8.4 8.4 Refs
A (Rhodopsin) Vasopressin and oxytocin V1BR V1B AVPR1B Human Oxytocin (Human) 2 Peptide CC[C@@H]([C@@H]1NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCC(=O)N)CC(=O)N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CC(C)C)C XNOPRXBHLZRZKH-DSZYJQQASA-N - - 5.7 6.4 7.0 Refs
A (Rhodopsin) Vasopressin and oxytocin V1BR V1B AVPR1B Human Vasopressin (Human) 1 Peptide NC(=O)C[C@@H]1NC(=O)[C@H](CCC(=O)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@H](CSSC[C@H](NC1=O)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CCCN=C(N)N)N KBZOIRJILGZLEJ-LGYYRGKSSA-N - B2M_V1BR_HUMAN_VASOPRESSIN_GNAQ_HUMAN 9.0 9.9 9.9 Refs
A (Rhodopsin) Vasopressin and oxytocin V1BR V1B Avpr1b Rat Vasopressin (Human) 1 Peptide NC(=O)C[C@@H]1NC(=O)[C@H](CCC(=O)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@H](CSSC[C@H](NC1=O)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CCCN=C(N)N)N KBZOIRJILGZLEJ-LGYYRGKSSA-N - - 9.0 9.9 9.9 Refs
A (Rhodopsin) Vasopressin and oxytocin V2R V2 AVPR2 Human Oxytocin (Human) 2 Peptide CC[C@@H]([C@@H]1NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@@H](N)CSSC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](NC1=O)CCC(=O)N)CC(=O)N)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CC(C)C)C XNOPRXBHLZRZKH-DSZYJQQASA-N - - 5.4 6.1 6.8 Refs
A (Rhodopsin) Vasopressin and oxytocin V2R V2 AVPR2 Human Vasopressin (Human) 1 Peptide NC(=O)C[C@@H]1NC(=O)[C@H](CCC(=O)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccc(cc2)O)NC(=O)[C@H](CSSC[C@H](NC1=O)C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)NCC(=O)N)CCCN=C(N)N)N KBZOIRJILGZLEJ-LGYYRGKSSA-N - 7BB6 7.9 8.5 9.1 Refs
B1 (Secretin) Calcitonin CALCR CT CALCR Human Α-Cgrp (Human) 3 Peptide - - - 6.2 7.3 8.4 Refs
B1 (Secretin) Calcitonin CALCR CT CALCR Human Α-Cgrp (Mouse) 6 Peptide - - -
B1 (Secretin) Calcitonin CALCR CT CALCR Human Β-Cgrp (Human) 4 Peptide - - - 7.2 7.2 Refs
B1 (Secretin) Calcitonin CALCR CT CALCR Human Β-Cgrp (Mouse) 6 Peptide - - -
B1 (Secretin) Calcitonin CALCR CT CALCR Human Β-Cgrp (Rat) 6 Peptide - - -
B1 (Secretin) Calcitonin CALCR CT CALCR Human Adrenomedullin (Human) 4 Peptide - - - 6.7 7.2 7.7 Refs
B1 (Secretin) Calcitonin CALCR CT CALCR Human Adrenomedullin 2/Intermedin (Human) 5 Peptide - - - 6.5 6.5 Refs
B1 (Secretin) Calcitonin CALCR CT CALCR Human Amylin (Human) 2 Peptide - - - 8.0 8.6 9.2 Refs
B1 (Secretin) Calcitonin CALCR CT CALCR Human Amylin (Mouse) 6 Peptide - - -
B1 (Secretin) Calcitonin CALCR CT CALCR Human Calcitonin (Human) 1 Peptide NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N1CCC[C@H]1C(=O)N)C)C(C)C)[C@H](CC)C)C)[C@H](O)C)CCC(=O)N)Cc1ccccc1)[C@H](O)C)Cc1nc[nH]c1)Cc1ccccc1)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)CNC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H]1CSSC[C@H](N)C(=O)NCC(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)NC(C(=O)N1)[C@H](O)C)CO)CC(C)C)CC(=O)N)CCSC)CC(C)C)Cc1ccc(cc1)O)CCC(=O)N)CC(=O)O)Cc1ccccc1)CC(=O)N LDVRMNJZLWXJPL-GXQFRRLTSA-N - 7TYH 9.0 10.1 11.2 Refs
B1 (Secretin) Calcitonin CALCR CT CALCR Human Calcitonin (Mouse) 6 Peptide - - -
B1 (Secretin) Corticotropin-releasing factor CRHR1 CRF1 CRHR1 Human Corticotrophin-Releasing Hormone (Human) 2 Peptide - - - AFM_CRHR1_HUMAN_hashedseq[MXKE57KVTIFLBOBIYYEV4DKRYY0] Refs
B1 (Secretin) Corticotropin-releasing factor CRHR1 CRF1 CRHR1 Human Urocortin 1 (Human) 1 Peptide - - - - Refs
B1 (Secretin) Corticotropin-releasing factor CRHR1 CRF1 CRHR1 Human Urocortin 1 (Mouse) 4 Peptide - - - -
B1 (Secretin) Corticotropin-releasing factor CRHR1 CRF1 CRHR1 Human Urocortin 2 (Human) 3 Protein - - - - Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 CRHR2 Human Corticotrophin-Releasing Hormone (Human) 1 Peptide - - - AFM_CRHR2_HUMAN_hashedseq[MXKE57KVTIFLBOBIYYEV4DKRYY0] 7.8 7.8 Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 CRHR2 Human Urocortin 1 (Human) 2 Peptide - - - Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 CRHR2 Human Urocortin 1 (Mouse) 2 Peptide - - - Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 CRHR2 Human Urocortin 2 (Human) 2 Protein - - - Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 CRHR2 Human Urocortin 2 (Rat) 2 Peptide - - -
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 CRHR2 Human Urocortin 3 (Human) 2 Peptide - - - Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 Crhr2 Mouse Corticotrophin-Releasing Hormone (Human) 1 Peptide - - - - 7.8 7.8 Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 Crhr2 Mouse Urocortin 1 (Mouse) 2 Peptide - - - - Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 Crhr2 Mouse Urocortin 2 (Mouse) 2 Peptide - - - - Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 Crhr2 Mouse Urocortin 3 (Mouse) 2 Peptide - - - - Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 Crhr2 Rat Corticotrophin-Releasing Hormone (Human) 1 Peptide - - - - 7.8 7.8 Refs
B1 (Secretin) Corticotropin-releasing factor CRHR2 CRF2 Crhr2 Rat Urocortin 3 (Mouse) 2 Peptide - - - - Refs
B1 (Secretin) Glucagon receptor family GHRHR GHRH GHRHR Human Ghrh (Human) Principal 1 Peptide - - - 7CZ5
B1 (Secretin) Glucagon receptor family GHRHR GHRH GHRHR Human Ghrh (Mouse) Principal 1 Peptide - - -
B1 (Secretin) Glucagon receptor family GHRHR GHRH GHRHR Human Ghrh (Rat) Principal 1 Peptide - - -
B1 (Secretin) Glucagon receptor family GIPR GIP GIPR Human Gastric Inhibitory Polypeptide (Human) Principal 1 Peptide - - - 9.1 9.1 Refs
B1 (Secretin) Glucagon receptor family GIPR GIP GIPR Human Gastric Inhibitory Polypeptide (Mouse) Principal 1 Peptide - - -
B1 (Secretin) Glucagon receptor family GIPR GIP Gipr Rat Gastric Inhibitory Polypeptide (Rat) Principal 1 Peptide - - - - Refs
B1 (Secretin) Glucagon receptor family GLP1R GLP-1 GLP1R Human Glucagon (Human) 2 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)[C@H](O)C)CC(=O)N)CCSC)CC(C)C)Cc1c[nH]c2c1cccc2)CCC(=O)N)C(C)C)Cc1ccccc1)CC(=O)O)CCC(=O)N)C)CCCN=C(N)N)CCCN=C(N)N)CO)CC(=O)O)CC(C)C)Cc1ccc(cc1)O)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)CNC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1nc[nH]c1)N)CO)CCC(=O)N)Cc1ccccc1)CO)CC(=O)O)Cc1ccc(cc1)O)CO MASNOZXLGMXCHN-ZLPAWPGGSA-N - 6.9 7.0 7.0 Refs
B1 (Secretin) Glucagon receptor family GLP1R GLP-1 GLP1R Human Glucagon-Like Peptide 1-(7-36) Amide (Human) 1 Protein - - - 9.2 9.2 Refs
B1 (Secretin) Glucagon receptor family GLP1R GLP-1 GLP1R Human Glucagon-Like Peptide 1-(7-37) (Human) 3 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CCC(N)=O)NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)CNC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1c[nH]cn1)[C@@H](C)O)[C@@H](C)O)C(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)NCC(=O)N[C@@H](CCCN=C(N)N)C(=O)NCC(=O)O)C(C)C GCYXWQUSHADNBF-AAEALURTSA-N - 7DUQ Refs
B1 (Secretin) Glucagon receptor family GLP2R GLP-2 GLP2R Human Glucagon-Like Peptide 2 (Human) 4 Protein CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1c[nH]cn1)[C@@H](C)O)[C@@H](C)CC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)[C@@H](C)CC TWSALRJGPBVBQU-PKQQPRCHSA-N - 7D68 Refs
B1 (Secretin) Glucagon receptor family GLP2R GLP-2 GLP2R Human Glucagon-Like Peptide 2 (Mouse) 4 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1c[nH]cn1)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)[C@@H](C)CC VSJTUHNYLFMYOE-HUADCCRNSA-N -
B1 (Secretin) Glucagon receptor family GLP2R GLP-2 GLP2R Human Glucagon-Like Peptide 2-(3-33) (Human) 4 Protein CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](N)CC(=O)O)[C@@H](C)O)[C@@H](C)CC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)[C@@H](C)CC MYKFSDGCGNRIEA-KXTJMAPWSA-N - Refs
B1 (Secretin) Glucagon receptor family GLP2R GLP-2 GLP2R Human Glucagon-Like Peptide 2-(3-33) (Mouse) 4 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](N)CC(=O)O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)[C@@H](C)CC FGSZUMQGXARWAJ-XVADTHAUSA-N -
B1 (Secretin) Glucagon receptor family GLP2R GLP-2 Glp2r Rat Glucagon-Like Peptide 2 (Rat) 1 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1c[nH]cn1)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)[C@@H](C)CC JPRUMPQGPCFDGW-CWHSZFSPSA-N - - 10.2 10.2 Refs
B1 (Secretin) Glucagon receptor family GLP2R GLP-2 Glp2r Rat Glucagon-Like Peptide 2-(2-33) (Rat) 3 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)N)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)[C@@H](C)CC OQGQYLSDVZWIPO-QSSAVJFTSA-N - - 6.1 6.1 Refs
B1 (Secretin) Glucagon receptor family GLP2R GLP-2 Glp2r Rat Glucagon-Like Peptide 2-(3-33) (Rat) 2 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)CNC(=O)[C@@H](N)CC(=O)O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H](CC(C)C)C(=O)N[C@H](C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CC(=O)O)C(=O)O)[C@@H](C)O)[C@@H](C)CC)[C@@H](C)O)[C@@H](C)CC JHPPUNFVXZAAKU-YNDCLQMTSA-N - - 6.6 6.6 Refs
B1 (Secretin) Glucagon receptor family GLR glucagon GCGR Human Glucagon (Human) Principal 1 Protein NCCCC[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)O)[C@H](O)C)CC(=O)N)CCSC)CC(C)C)Cc1c[nH]c2c1cccc2)CCC(=O)N)C(C)C)Cc1ccccc1)CC(=O)O)CCC(=O)N)C)CCCN=C(N)N)CCCN=C(N)N)CO)CC(=O)O)CC(C)C)Cc1ccc(cc1)O)NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)[C@@H](NC(=O)[C@H]([C@H](O)C)NC(=O)CNC(=O)[C@@H](NC(=O)[C@@H](NC(=O)[C@H](Cc1nc[nH]c1)N)CO)CCC(=O)N)Cc1ccccc1)CO)CC(=O)O)Cc1ccc(cc1)O)CO MASNOZXLGMXCHN-ZLPAWPGGSA-N - 9.0 9.0 Refs
B1 (Secretin) Glucagon receptor family SCTR secretin SCTR Human Vip (Human) 2 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)CC(=O)N)CC(C)C)C(CC)C)CO)CC(=O)N)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(C)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(Cc1nc[nH]c1)N)CO)CC(=O)O)C)Cc1ccccc1)CC(=O)O)CC(=O)N)Cc1ccc(cc1)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N VBUWHHLIZKOSMS-UHFFFAOYSA-N - Refs
B1 (Secretin) Glucagon receptor family SCTR secretin SCTR Human Secretin (Mouse) 2 Peptide - - -
B1 (Secretin) Glucagon receptor family SCTR secretin SCTR Human Secretin (Pig) 1 Peptide OCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)O)C(C)C)CC(C)C)CCC(=O)N)CC(C)C)CC(C)C)CCCNC(=N)N)CCC(=O)N)CC(C)C)CCCNC(=N)N)C)CO)CC(=O)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(O)C)NC(=O)CNC(=O)C(NC(=O)C(NC(=O)C(Cc1[nH]ccn1)N)CO)CC(=O)O)Cc1ccccc1)CO)CCC(=O)O)CC(C)C KKNIUBFRGPFELP-UHFFFAOYSA-N - 9.7 9.7 Refs
B1 (Secretin) Glucagon receptor family SCTR secretin Sctr Rat Vip (Human) 2 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)CC(=O)N)CC(C)C)C(CC)C)CO)CC(=O)N)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(C)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(Cc1nc[nH]c1)N)CO)CC(=O)O)C)Cc1ccccc1)CC(=O)O)CC(=O)N)Cc1ccc(cc1)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N VBUWHHLIZKOSMS-UHFFFAOYSA-N - - Refs
B1 (Secretin) Glucagon receptor family SCTR secretin Sctr Rat Secretin (Rat) 2 Peptide - - - - 8.0 8.5 9.0 Refs
B1 (Secretin) Parathyroid hormone PTH1R PTH1 PTH1R Human Pth (Human) 3 Peptide - - -
B1 (Secretin) Parathyroid hormone PTH1R PTH1 PTH1R Human Pth (Mouse) 3 Peptide - - -
B1 (Secretin) Parathyroid hormone PTH1R PTH1 PTH1R Human Pth (Rat) 3 Peptide - - -
B1 (Secretin) Parathyroid hormone PTH1R PTH1 PTH1R Human Pthrp (Human) 3 Peptide - - -
B1 (Secretin) Parathyroid hormone PTH1R PTH1 PTH1R Human Pthrp-(1-36) (Human) 2 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](C)N)C(C)C)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O)C(=O)O NNRMZXDHMCWWRV-RHBZDGMUSA-N - 8HAF Refs
B1 (Secretin) Parathyroid hormone PTH1R PTH1 PTH1R Human Tip39 (Human) 1 Peptide - - - Refs
B1 (Secretin) Parathyroid hormone PTH2R PTH2 PTH2R Human Pth (Human) 5 Peptide - - -
B1 (Secretin) Parathyroid hormone PTH2R PTH2 PTH2R Human Pth (Mouse) 5 Peptide - - -
B1 (Secretin) Parathyroid hormone PTH2R PTH2 PTH2R Human Pth (Rat) 5 Peptide - - -
B1 (Secretin) Parathyroid hormone PTH2R PTH2 PTH2R Human Pthrp (Human) 5 Peptide - - -
B1 (Secretin) Parathyroid hormone PTH2R PTH2 PTH2R Human Pthrp-(1-34) (Human) (Human) 3 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](C)N)C(C)C)[C@@H](C)CC)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@H](C(=O)N[C@@H](C)C(=O)O)[C@@H](C)O)[C@@H](C)CC ZOWOHMFPXMYFKJ-WBTWNKCNSA-N - Refs
B1 (Secretin) Parathyroid hormone PTH2R PTH2 PTH2R Human Pthrp-(1-36) (Human) 4 Peptide CC[C@H](C)[C@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H](NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CCCCN)NC(=O)CNC(=O)[C@H](CCCCN)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H](NC(=O)[C@H](C)N)C(C)C)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O)C(=O)O NNRMZXDHMCWWRV-RHBZDGMUSA-N - Refs
B1 (Secretin) Parathyroid hormone PTH2R PTH2 PTH2R Human Tip39 (Human) 1 Peptide - - - Refs
B1 (Secretin) Parathyroid hormone PTH2R PTH2 PTH2R Human Tip39 (Mouse) 2 Peptide - - - Refs
B1 (Secretin) Parathyroid hormone PTH2R PTH2 Pth2r Rat Tip39 (Mouse) 2 Peptide - - - - Refs
B1 (Secretin) VIP and PACAP PACR PAC1 ADCYAP1R1 Human Pacap-27 (Human) 1 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N)CC(C)C)C(C)C)C)C)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(CC)C)NC(=O)CNC(=O)C(NC(=O)C(NC(=O)C(Cc1[nH]cnc1)N)CO)CC(=O)O)Cc1ccccc1)CC(=O)O)CO)Cc1ccc(cc1)O)CO)CCCNC(=N)N)Cc1ccc(cc1)O)CCCNC(=N)N RZGBUJXSKLDAFE-UHFFFAOYSA-N - 8E3X 10.0 10.1 10.1 8.5 8.7 8.8 Refs
B1 (Secretin) VIP and PACAP PACR PAC1 ADCYAP1R1 Human Pacap-38 (Human) 2 Peptide - - - 9.5 9.8 10.0 8.4 8.6 8.8 Refs
B1 (Secretin) VIP and PACAP PACR PAC1 ADCYAP1R1 Human Phi (Mouse) 4 Peptide - - -
B1 (Secretin) VIP and PACAP PACR PAC1 ADCYAP1R1 Human Phm (Human) 4 Peptide - - -
B1 (Secretin) VIP and PACAP PACR PAC1 ADCYAP1R1 Human Phv (Human) 4 Peptide - - -
B1 (Secretin) VIP and PACAP PACR PAC1 ADCYAP1R1 Human Phv (Rat) 4 Peptide - - -
B1 (Secretin) VIP and PACAP PACR PAC1 ADCYAP1R1 Human Vip (Human) 3 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)CC(=O)N)CC(C)C)C(CC)C)CO)CC(=O)N)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(C)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(Cc1nc[nH]c1)N)CO)CC(=O)O)C)Cc1ccccc1)CC(=O)O)CC(=O)N)Cc1ccc(cc1)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N VBUWHHLIZKOSMS-UHFFFAOYSA-N - 7.1 7.1 7.1 5.5 5.7 5.8 Refs
B1 (Secretin) VIP and PACAP PACR PAC1 Adcyap1r1 Rat Pacap-27 (Human) 1 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N)CC(C)C)C(C)C)C)C)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(CC)C)NC(=O)CNC(=O)C(NC(=O)C(NC(=O)C(Cc1[nH]cnc1)N)CO)CC(=O)O)Cc1ccccc1)CC(=O)O)CO)Cc1ccc(cc1)O)CO)CCCNC(=N)N)Cc1ccc(cc1)O)CCCNC(=N)N RZGBUJXSKLDAFE-UHFFFAOYSA-N - - 10.0 10.1 10.1 8.5 8.7 8.8 Refs
B1 (Secretin) VIP and PACAP PACR PAC1 Adcyap1r1 Rat Pacap-38 (Human) 2 Peptide - - - - 9.5 9.8 10.0 8.4 8.6 8.8 Refs
B1 (Secretin) VIP and PACAP PACR PAC1 Adcyap1r1 Rat Vip (Human) 3 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)CC(=O)N)CC(C)C)C(CC)C)CO)CC(=O)N)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(C)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(Cc1nc[nH]c1)N)CO)CC(=O)O)C)Cc1ccccc1)CC(=O)O)CC(=O)N)Cc1ccc(cc1)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N VBUWHHLIZKOSMS-UHFFFAOYSA-N - - 7.1 7.1 7.1 5.5 5.7 5.8 Refs
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Ghrh (Human) 4 Peptide - - - 6.2 6.2 Refs
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Ghrh (Mouse) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Ghrh (Rat) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Pacap-27 (Human) 2 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N)CC(C)C)C(C)C)C)C)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(CC)C)NC(=O)CNC(=O)C(NC(=O)C(NC(=O)C(Cc1[nH]cnc1)N)CO)CC(=O)O)Cc1ccccc1)CC(=O)O)CO)Cc1ccc(cc1)O)CO)CCCNC(=N)N)Cc1ccc(cc1)O)CCCNC(=N)N RZGBUJXSKLDAFE-UHFFFAOYSA-N - 6VN7 7.6 8.6 9.9 8.9 8.9 Refs
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Pacap-38 (Human) 3 Peptide - - - 7.4 8.6 9.7 8.2 8.2 Refs
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Phi (Mouse) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Phm (Human) 4 Peptide - - - 5.7 5.7 Refs
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Vip (Human) 1 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)CC(=O)N)CC(C)C)C(CC)C)CO)CC(=O)N)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(C)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(Cc1nc[nH]c1)N)CO)CC(=O)O)C)Cc1ccccc1)CC(=O)O)CC(=O)N)Cc1ccc(cc1)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N VBUWHHLIZKOSMS-UHFFFAOYSA-N - 7.9 9.0 10.0 8.5 9.2 9.8 Refs
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Secretin (Mouse) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Secretin (Pig) 4 Peptide OCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)O)C(C)C)CC(C)C)CCC(=O)N)CC(C)C)CC(C)C)CCCNC(=N)N)CCC(=O)N)CC(C)C)CCCNC(=N)N)C)CO)CC(=O)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(O)C)NC(=O)CNC(=O)C(NC(=O)C(NC(=O)C(Cc1[nH]ccn1)N)CO)CC(=O)O)Cc1ccccc1)CO)CCC(=O)O)CC(C)C KKNIUBFRGPFELP-UHFFFAOYSA-N -
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 VIPR1 Human Secretin (Rat) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 Vipr1 Rat Pacap-27 (Human) 2 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N)CC(C)C)C(C)C)C)C)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(CC)C)NC(=O)CNC(=O)C(NC(=O)C(NC(=O)C(Cc1[nH]cnc1)N)CO)CC(=O)O)Cc1ccccc1)CC(=O)O)CO)Cc1ccc(cc1)O)CO)CCCNC(=N)N)Cc1ccc(cc1)O)CCCNC(=N)N RZGBUJXSKLDAFE-UHFFFAOYSA-N - - 7.6 8.6 9.9 8.9 8.9 Refs
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 Vipr1 Rat Phv (Rat) 4 Peptide - - - - Refs
B1 (Secretin) VIP and PACAP VIPR1 VPAC1 Vipr1 Rat Vip (Human) 1 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)CC(=O)N)CC(C)C)C(CC)C)CO)CC(=O)N)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(C)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(Cc1nc[nH]c1)N)CO)CC(=O)O)C)Cc1ccccc1)CC(=O)O)CC(=O)N)Cc1ccc(cc1)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N VBUWHHLIZKOSMS-UHFFFAOYSA-N - - 7.9 9.0 10.0 8.5 9.2 9.8 Refs
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Ghrh (Human) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Ghrh (Mouse) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Ghrh (Rat) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Pacap-27 (Human) 2 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N)CC(C)C)C(C)C)C)C)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(CC)C)NC(=O)CNC(=O)C(NC(=O)C(NC(=O)C(Cc1[nH]cnc1)N)CO)CC(=O)O)Cc1ccccc1)CC(=O)O)CO)Cc1ccc(cc1)O)CO)CCCNC(=N)N)Cc1ccc(cc1)O)CCCNC(=N)N RZGBUJXSKLDAFE-UHFFFAOYSA-N - 7WBJ 7.6 8.5 9.4 Refs
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Pacap-38 (Human) 1 Peptide - - - 7.7 8.5 9.3 Refs
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Phi (Mouse) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Vip (Human) 3 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)CC(=O)N)CC(C)C)C(CC)C)CO)CC(=O)N)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(C)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(Cc1nc[nH]c1)N)CO)CC(=O)O)C)Cc1ccccc1)CC(=O)O)CC(=O)N)Cc1ccc(cc1)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N VBUWHHLIZKOSMS-UHFFFAOYSA-N - 7.3 8.3 9.3 7.8 8.4 8.8 Refs
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Secretin (Mouse) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Secretin (Pig) 4 Peptide OCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NCC(=O)NC(C(=O)NC(C(=O)O)C(C)C)CC(C)C)CCC(=O)N)CC(C)C)CC(C)C)CCCNC(=N)N)CCC(=O)N)CC(C)C)CCCNC(=N)N)C)CO)CC(=O)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(O)C)NC(=O)CNC(=O)C(NC(=O)C(NC(=O)C(Cc1[nH]ccn1)N)CO)CC(=O)O)Cc1ccccc1)CO)CCC(=O)O)CC(C)C KKNIUBFRGPFELP-UHFFFAOYSA-N -
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 VIPR2 Human Secretin (Rat) 4 Peptide - - -
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 Vipr2 Rat Pacap-27 (Human) 2 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)N)CC(C)C)C(C)C)C)C)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(CC)C)NC(=O)CNC(=O)C(NC(=O)C(NC(=O)C(Cc1[nH]cnc1)N)CO)CC(=O)O)Cc1ccccc1)CC(=O)O)CO)Cc1ccc(cc1)O)CO)CCCNC(=N)N)Cc1ccc(cc1)O)CCCNC(=N)N RZGBUJXSKLDAFE-UHFFFAOYSA-N - - 7.6 8.5 9.4 Refs
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 Vipr2 Rat Phv (Rat) 4 Peptide - - - - Refs
B1 (Secretin) VIP and PACAP VIPR2 VPAC2 Vipr2 Rat Vip (Human) 3 Protein NCCCCC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)NC(C(=O)O)CC(=O)N)CC(C)C)C(CC)C)CO)CC(=O)N)CC(C)C)Cc1ccc(cc1)O)CCCCN)CCCCN)C(C)C)C)CCSC)CCC(=O)N)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(C(O)C)NC(=O)C(NC(=O)C(C(C)C)NC(=O)C(NC(=O)C(NC(=O)C(NC(=O)C(Cc1nc[nH]c1)N)CO)CC(=O)O)C)Cc1ccccc1)CC(=O)O)CC(=O)N)Cc1ccc(cc1)O)CCCNC(=N)N)CC(C)C)CCCNC(=N)N VBUWHHLIZKOSMS-UHFFFAOYSA-N - - 7.3 8.3 9.3 7.8 8.4 8.8 Refs
B2 (Adhesion) ADGRB AGRB1 ADGRB1 ADGRB1 Human Phosphatidylserine Principal 1 Small molecule CCCC(=O)O[C@@H](COP(=O)(OC[C@@H](C(=O)O)N)O)COC(=O)CC UNJJBGNPUUVVFQ-ZJUUUORDSA-N - - Refs
B2 (Adhesion) ADGRD AGRD1 ADGRD1 ADGRD1 Human Dihydrotestosterone Principal 1 Small molecule O=C1CC[C@]2([C@H](C1)CC[C@@H]1[C@@H]2CC[C@]2([C@H]1CC[C@@H]2O)C)C NVKAWKQGWWIWPM-ABEVXSGRSA-N - 9IV2
B2 (Adhesion) ADGRL AGRL1 ADGRL1 Adgrl1 Rat Lasso D (Rat) Principal 1 Peptide - - - - Refs
B2 (Adhesion) ADGRL AGRL3 ADGRL3 Adgrl3 Rat Flrt3 (Rat) Principal 1 Peptide - - - - Refs
C (Glutamate) Calcium-sensing CASR CaS CASR Human Ca2+ None 2 Small molecule - - - - Refs
C (Glutamate) Calcium-sensing CASR CaS CASR Human D-Tryptophan None 1 Small molecule OC(=O)[C@@H](Cc1c[nH]c2c1cccc2)N QIVBCDIJIAJPQS-SECBINFHSA-N - 9C1P Refs
C (Glutamate) Calcium-sensing CASR CaS CASR Human Mg2+ None 3 Small molecule - - - -
C (Glutamate) Calcium-sensing CASR CaS CASR Human Spermine None 1 Small molecule NCCCNCCCCNCCCN PFNFFQXMRSDOHW-UHFFFAOYSA-N - 8SZH Refs
C (Glutamate) Calcium-sensing CASR CaS Casr Mouse Ca2+ None 2 Small molecule - - - - Refs
C (Glutamate) Calcium-sensing CASR CaS Casr Rat Ca2+ None 2 Small molecule - - - - Refs
C (Glutamate) Calcium-sensing CASR CaS Casr Rat Mg2+ None 3 Small molecule - - - - Refs
C (Glutamate) GABAB GABR1 GABAB1 GABBR1 Human Gaba Principal 1 Small molecule NCCCC(=O)O BTCSSZJGUNDROE-UHFFFAOYSA-N - -
C (Glutamate) GABAB GABR1 GABAB1 Gabbr1 Rat Gaba Principal 1 Small molecule NCCCC(=O)O BTCSSZJGUNDROE-UHFFFAOYSA-N - - Refs
C (Glutamate) Metabotropic glutamate GRM1 mGlu1 GRM1 Human L-Glutamic Acid Principal 1 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - 9WQM 4.8 4.9 5.0 6.4 6.5 6.5 Refs
C (Glutamate) Metabotropic glutamate GRM1 mGlu1 Grm1 Rat L-Glutamic Acid Principal 1 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - - 4.8 4.9 5.0 6.4 6.5 6.5 Refs
C (Glutamate) Metabotropic glutamate GRM2 mGlu2 GRM2 Human L-Glutamic Acid Principal 1 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - 8JD3 4.7 5.1 5.4 5.4 5.7 5.9 Refs
C (Glutamate) Metabotropic glutamate GRM2 mGlu2 Grm2 Rat L-Glutamic Acid Principal 1 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - - 4.7 5.1 5.4 5.4 5.7 5.9 Refs
C (Glutamate) Metabotropic glutamate GRM3 mGlu3 GRM3 Human L-Glutamic Acid None 1 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - 9II3 5.3 5.4 5.4 6.4 6.4 Refs
C (Glutamate) Metabotropic glutamate GRM3 mGlu3 GRM3 Human Naag None 2 Small molecule OC(=O)CC[C@@H](C(=O)O)NC(=O)[C@@H](NC(=O)C)CC(=O)O OPVPGKGADVGKTG-BQBZGAKWSA-N - - 4.7 4.7 Refs
C (Glutamate) Metabotropic glutamate GRM3 mGlu3 Grm3 Rat L-Glutamic Acid None 1 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - - 5.3 5.4 5.4 6.4 6.4 Refs
C (Glutamate) Metabotropic glutamate GRM4 mGlu4 GRM4 Human L-Glutamic Acid None 2 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - 8WGB 4.7 5.1 5.5 4.9 5.2 5.5 Refs
C (Glutamate) Metabotropic glutamate GRM4 mGlu4 GRM4 Human L-Serine-O-Phosphate None 1 Small molecule OC(=O)[C@H](COP(=O)(O)O)N BZQFBWGGLXLEPQ-REOHCLBHSA-N - 7E9H 5.9 5.9 Refs
C (Glutamate) Metabotropic glutamate GRM4 mGlu4 Grm4 Rat L-Glutamic Acid None 2 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - - 4.7 5.1 5.5 4.9 5.2 5.5 Refs
C (Glutamate) Metabotropic glutamate GRM4 mGlu4 Grm4 Rat L-Serine-O-Phosphate None 1 Small molecule OC(=O)[C@H](COP(=O)(O)O)N BZQFBWGGLXLEPQ-REOHCLBHSA-N - - 5.9 5.9 Refs
C (Glutamate) Metabotropic glutamate GRM5 mGlu5 GRM5 Human L-Glutamic Acid Principal 1 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - 9WQL 5.0 5.3 5.5 Refs
C (Glutamate) Metabotropic glutamate GRM5 mGlu5 Grm5 Rat L-Glutamic Acid Principal 1 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - - 5.0 5.3 5.5 Refs
C (Glutamate) Metabotropic glutamate GRM6 mGlu6 GRM6 Human L-Glutamic Acid None 2 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - - 4.8 4.4 4.4 Refs
C (Glutamate) Metabotropic glutamate GRM6 mGlu6 GRM6 Human L-Serine-O-Phosphate None 1 Small molecule OC(=O)[C@H](COP(=O)(O)O)N BZQFBWGGLXLEPQ-REOHCLBHSA-N - 9LLZ 6.4 6.4 Refs
C (Glutamate) Metabotropic glutamate GRM6 mGlu6 Grm6 Rat L-Glutamic Acid None 2 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - - 4.8 4.4 4.4 Refs
C (Glutamate) Metabotropic glutamate GRM7 mGlu7 GRM7 Human L-Glutamic Acid None 2 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - - 3.0 3.0 3.1 3.1 Refs
C (Glutamate) Metabotropic glutamate GRM7 mGlu7 GRM7 Human L-Serine-O-Phosphate None 1 Small molecule OC(=O)[C@H](COP(=O)(O)O)N BZQFBWGGLXLEPQ-REOHCLBHSA-N - - 4.5 4.5 4.4 4.4 Refs
C (Glutamate) Metabotropic glutamate GRM8 mGlu8 GRM8 Human L-Glutamic Acid None 1 Small molecule OC(=O)CC[C@@H](C(=O)O)N WHUUTDBJXJRKMK-VKHMYHEASA-N - 9MBA 4.9 5.3 5.6 Refs
C (Glutamate) Metabotropic glutamate GRM8 mGlu8 GRM8 Human L-Serine-O-Phosphate None 2 Small molecule OC(=O)[C@H](COP(=O)(O)O)N BZQFBWGGLXLEPQ-REOHCLBHSA-N - - Refs
C (Glutamate) Orphan GPC6A GPRC6 GPRC6A Human L-Alanine None 3 Small molecule C[C@@H](C(=O)O)N QNAYBMKLOCPYGJ-REOHCLBHSA-N - - 3.8 3.8 Refs
C (Glutamate) Orphan GPC6A GPRC6 GPRC6A Human L-Arginine None 1 Small molecule OC(=O)[C@H](CCCN=C(N)N)N ODKSFYDXXFIFQN-BYPYZUCNSA-N - - 4.4 4.4 Refs
C (Glutamate) Orphan GPC6A GPRC6 GPRC6A Human L-Citrulline None 4 Small molecule NC(=O)NCCC[C@@H](C(=O)O)N RHGKLRLOHDJJDR-BYPYZUCNSA-N - - 3.6 3.6 Refs
C (Glutamate) Orphan GPC6A GPRC6 GPRC6A Human L-Glutamine None 5 Small molecule NC(=O)CC[C@@H](C(=O)O)N ZDXPYRJPNDTMRX-VKHMYHEASA-N - - 3.2 3.2 Refs
C (Glutamate) Orphan GPC6A GPRC6 GPRC6A Human L-Lysine None 3 Small molecule NCCCC[C@@H](C(=O)O)N KDXKERNSBIXSRK-YFKPBYRVSA-N - - 3.8 3.8 Refs
C (Glutamate) Orphan GPC6A GPRC6 GPRC6A Human L-Ornithine None 2 Small molecule N[C@H](C(=O)O)CCCN AHLPHDHHMVZTML-BYPYZUCNSA-N - - 4.0 4.0 Refs
C (Glutamate) Orphan GPC6A GPRC6 GPRC6A Human L-Serine None 5 Small molecule OC[C@@H](C(=O)O)N MTCFGRXMJLQNBG-REOHCLBHSA-N - - 3.2 3.2 Refs
C (Glutamate) Orphan GPC6A GPRC6 GPRC6A Human Glycine None 4 Small molecule NCC(=O)O DHMQDGOQFOQNFH-UHFFFAOYSA-N - - 3.6 3.6 Refs
F (Frizzled) WNT FZD1 FZD1 FZD1 Human Wnt-1 (Human) Peptide - - - -
F (Frizzled) WNT FZD1 FZD1 FZD1 Human Wnt-2 (Human) Peptide - - - -
F (Frizzled) WNT FZD1 FZD1 FZD1 Human Wnt-3a (Human) Peptide - - - -
F (Frizzled) WNT FZD1 FZD1 FZD1 Human Wnt-5a (Human) Peptide - - - -
F (Frizzled) WNT FZD1 FZD1 FZD1 Human Wnt-7b (Human) Peptide - - - -
F (Frizzled) WNT FZD2 FZD2 FZD2 Human Wnt-5a (Human) Principal 1 Peptide - - - -
F (Frizzled) WNT FZD4 FZD4 Fzd4 Mouse Norrin (Mouse) Principal 1 Peptide - - - - Refs
F (Frizzled) WNT FZD6 FZD6 FZD6 Human Wnt-3a (Human) Peptide - - - - Refs
F (Frizzled) WNT FZD6 FZD6 FZD6 Human Wnt-4 (Human) Peptide - - - Refs
F (Frizzled) WNT FZD6 FZD6 FZD6 Human Wnt-5a (Human) Peptide - - - Refs
Unclassified Orphan GP107 GPR107 GPR107 Human Neuronostatin (Human) Principal 1 Peptide CC(C)C[C@H](N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)N[C@@H](C)C(=O)O QMXYKUFZQPEQES-UZSBMYCGSA-N - -
Unclassified Orphan GP143 GPR143 GPR143 Human Levodopa Principal 1 Small molecule OC(=O)[C@H](Cc1ccc(c(c1)O)O)N WTDRDQBEARUVNC-LURJTMIESA-N - - Refs