abaloparatide |
Anti-osteoporotic |
pth1r_human |
primary |
Class B1 (Secretin) |
Parathyroid hormone receptors |
approved |
4 |
- |
2017 |
peptide |
agonist |
28389324
|
26562265
|
no |
abarelix |
Antineoplastic |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
2003 |
peptide |
antagonist |
16985933
|
no |
acamprosate |
Antineoplastic |
grm5_human |
secondary |
Class C (Glutamate) |
Metabotropic glutamate receptors |
approved |
4 |
- |
2004 |
small molecule |
antagonist |
15963001
|
yes |
acebutolol |
Antihypertensive |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
2453744
|
2568935
|
16268148
|
11752352
|
yes |
acepromazine, aceprometazine |
Antipsychotic |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
7918347
|
no |
acepromazine, aceprometazine |
Antipsychotic |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
10821438
|
8593484
|
no |
acepromazine, aceprometazine |
Antipsychotic |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
11103886
|
11873706
|
15694263
|
16867246
|
11752352
|
20643630
|
no |
acepromazine, aceprometazine |
Antipsychotic |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
11755134
|
9760039
|
no |
acepromazine, aceprometazine |
Hypnotics and Sedatives |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
17139284
|
17016423
|
4406367
|
11752352
|
no |
acetophenazine |
schizophrenia |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1961 |
small molecule |
antagonist |
17139284
|
17016423
|
no |
acetophenazine |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1961 |
small molecule |
antagonist |
17139284
|
17016423
|
11873706
|
6147851
|
11752352
|
no |
acetylcholine |
Antiglaucomic |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1973 |
small molecule |
agonist |
508313
|
yes |
acipimox |
lipid-lowering |
hcar2_human |
primary |
Class A (Rhodopsin) |
Hydroxycarboxylic acid receptors |
approved |
4 |
- |
2003 |
small molecule |
agonist |
22267479
|
yes |
agomelatine |
Anti-depressant |
5ht2c_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
15289999
|
yes |
agomelatine |
Anti-depressant |
mtr1a_human |
primary |
Class A (Rhodopsin) |
Melatonin |
approved |
4 |
- |
2009 |
small molecule |
agonist |
15289999
|
yes |
agomelatine |
Anti-depressant |
mtr1b_human |
primary |
Class A (Rhodopsin) |
Melatonin |
approved |
4 |
- |
2009 |
small molecule |
agonist |
15289999
|
yes |
aclidinium |
Bronchodilator |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2012 |
small molecule |
antagonist |
19710368
|
19478135
|
yes |
aclidinium |
Bronchodilator |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2012 |
small molecule |
antagonist |
19710368
|
19478135
|
yes |
aclidinium |
Bronchodilator |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2012 |
small molecule |
antagonist |
19710368
|
19478135
|
yes |
aclidinium |
Bronchodilator |
acm4_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2012 |
small molecule |
antagonist |
19710368
|
19478135
|
yes |
aclidinium |
Bronchodilator |
acm5_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2012 |
small molecule |
antagonist |
19710368
|
19478135
|
yes |
acrivastine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1994 |
small molecule |
antagonist |
1715267
|
yes |
adenosine |
Analgesics |
aa3r_human |
primary |
Class A (Rhodopsin) |
Adenosine receptors |
approved |
4 |
- |
1989 |
small molecule |
agonist |
11752352
|
20370662
|
20370661
|
17321471
|
16339914
|
20136829
|
17438146
|
17442976
|
yes |
adenosine |
Analgesics |
aa2ar_human |
primary |
Class A (Rhodopsin) |
Adenosine receptors |
approved |
4 |
- |
1989 |
small molecule |
agonist |
20370662
|
20370661
|
17321471
|
16339914
|
19749080
|
20136829
|
17438146
|
17442976
|
yes |
adenosine |
Analgesics |
aa2br_human |
primary |
Class A (Rhodopsin) |
Adenosine receptors |
approved |
4 |
- |
1989 |
small molecule |
agonist |
20370662
|
20370661
|
17321471
|
16339914
|
20136829
|
17438146
|
17442976
|
yes |
adenosine |
Analgesics |
aa1r_human |
primary |
Class A (Rhodopsin) |
Adenosine receptors |
approved |
4 |
- |
1989 |
small molecule |
agonist |
20370662
|
20370661
|
17321471
|
20136829
|
17438146
|
17442976
|
yes |
albiglutide |
Antidiabetic |
glp1r_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
2014 |
protein |
agonist |
25136065
|
yes |
albuterol |
chronic obstructive pulmonary disease (COPD) |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1981 |
small molecule |
agonist |
17996583
|
no |
alcaftadine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2010 |
small molecule |
antagonist |
22035879
|
no |
almotriptan |
Anti-migraine |
5ht1d_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
10193663
|
11134654
|
11642004
|
11752352
|
yes |
alfentanil |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1986 |
small molecule |
agonist |
10955836
|
15694871
|
16906017
|
11240090
|
11752352
|
yes |
alfuzosin |
benign prostatic hyperplasia |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2003 |
small molecule |
agonist |
11752352
|
8799556
|
12892027
|
9122046
|
15639685
|
9223558
|
8196478
|
9870119
|
16613526
|
16553574
|
11750253
|
yes |
alfuzosin |
benign prostatic hyperplasia |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2003 |
small molecule |
agonist |
11752352
|
8799556
|
9122046
|
15639685
|
8196478
|
16613526
|
16553574
|
11750253
|
yes |
alfuzosin |
benign prostatic hyperplasia |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2003 |
small molecule |
agonist |
11752352
|
8799556
|
9122046
|
15639685
|
8196478
|
9870119
|
16613526
|
16553574
|
11750253
|
yes |
almotriptan |
Anti-migraine |
5ht1b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
10193663
|
10824628
|
11050304
|
11069595
|
11134654
|
11752352
|
yes |
alprenolol |
Anti-Arrhythmia ; Antihypertensive |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1966 |
small molecule |
antagonist |
2439825
|
2859531
|
2871880
|
no |
alprenolol |
Anti-Arrhythmia ; Antihypertensive |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1966 |
small molecule |
antagonist |
7678677
|
7606348
|
10433496
|
12522078
|
2828119
|
11752352
|
no |
alprostadil |
sexual dysfunction |
pe2r2_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1981 |
small molecule |
agonist |
10509658
|
15840408
|
11752352
|
yes |
alprostadil |
sexual dysfunction |
pe2r1_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1981 |
small molecule |
agonist |
15560119
|
14561849
|
10670413
|
16516814
|
11524243
|
yes |
alverine |
Antispasmodics |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2014 |
small molecule |
antagonist |
11697552
|
yes |
alvimopan |
opioid-induced bowel dysfunction |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2008 |
small molecule |
antagonist |
17909271
|
19086236
|
16597533
|
11752352
|
15882122
|
11755894
|
no |
alvimopan |
Opiate Antagonists |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2008 |
small molecule |
antagonist |
17909271
|
19086236
|
16597533
|
11752352
|
15882122
|
11755894
|
no |
amantadine hcl |
dyskinesias |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1968 |
small molecule |
antagonist |
9195603
|
10443547
|
no |
ambrisentan |
Antihypertensive |
ednra_human |
primary |
Class A (Rhodopsin) |
Endothelin receptors |
approved |
4 |
- |
2007 |
small molecule |
antagonist |
20811346
|
19389876
|
19601701
|
19920913
|
yes |
amiodarone |
Anti-Arrhythmia |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1985 |
small molecule |
antagonist |
12083991
|
yes |
amitriptyline |
Analgesics |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1961 |
small molecule |
antagonist |
7855217
|
yes |
amoxapine |
unipolar depression |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1980 |
small molecule |
antagonist |
11180191
|
yes |
amoxapine |
unipolar depression |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1980 |
small molecule |
antagonist |
16135699
|
yes |
amoxapine |
unipolar depression |
drd4_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1980 |
small molecule |
antagonist |
16135699
|
yes |
amoxapine |
unipolar depression |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1980 |
small molecule |
antagonist |
1966571
|
11180191
|
yes |
amphetamine |
cognitive dysfunction; ADHD |
taar1_human |
secondary |
Class A (Rhodopsin) |
Trace amine receptors |
approved |
4 |
- |
1996 |
small molecule |
agonist |
17218486
|
17234900
|
17212650
|
17234899
|
15764732
|
no |
anileridine |
Analgesics; Narcotics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
17139284
|
17016423
|
11752352
|
no |
anisotropine methylbromide |
Antispasmodics; Anti-ulcer |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
4555460
|
no |
anisotropine methylbromide |
Antispasmodics; Anti-ulcer |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
4555460
|
no |
anisotropine methylbromide |
Antispasmodics; Anti-ulcer |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
4555460
|
6897316
|
20391952
|
no |
antazoline |
atrial fibrillation |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1994 |
small molecule |
antagonist |
16129921
|
yes |
apomorphine |
anti-parkisonian |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2004 |
small molecule |
agonist |
11752352
|
yes |
apomorphine |
anti-parkisonian |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2004 |
small molecule |
agonist |
11343576
|
11752352
|
11212866
|
18691132
|
10641988
|
11692072
|
11215397
|
10494453
|
yes |
apomorphine |
anti-parkisonian |
drd4_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2004 |
small molecule |
agonist |
15007532
|
11752352
|
18691132
|
9497025
|
17067298
|
9871530
|
17164075
|
yes |
asenapine |
schizophrenia |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
10592235
|
18308814
|
yes |
apraclonidine |
Antiglaucomic |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1987 |
small molecule |
agonist |
1676991
|
yes |
apraclonidine |
Antiglaucomic |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1987 |
small molecule |
agonist |
1676991
|
yes |
apraclonidine |
Antiglaucomic |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1987 |
small molecule |
agonist |
17139284
|
17016423
|
11481271
|
17824139
|
16921219
|
12630335
|
14575724
|
15748550
|
20399934
|
17572343
|
16935593
|
yes |
aprepitant |
Antiemetics |
nk1r_human |
primary |
Class A (Rhodopsin) |
Tachykinin receptors |
approved |
4 |
- |
2003 |
small molecule |
antagonist |
11752352
|
12590540
|
17643344
|
12784346
|
12227806
|
15121485
|
yes |
arbutamine |
Cardiotonic |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1997 |
small molecule |
agonist |
17139284
|
17016423
|
8723169
|
no |
arformoterol |
Bronchodilator |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2006 |
small molecule |
agonist |
14725487
|
17594727
|
17352511
|
20406080
|
16022567
|
18501650
|
17472819
|
11752352
|
no |
aripiprazole |
schizophrenia |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2002 |
small molecule |
partial agonist |
12063084
|
14647959
|
14709325
|
15257633
|
15862515
|
yes |
aripiprazole |
psychosis |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2015 |
small molecule |
partial agonist |
12063084
|
14647959
|
14709325
|
15257633
|
15862515
|
yes |
aripiprazole |
schizophrenia |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2002 |
small molecule |
partial agonist |
14642974
|
17242925
|
17265076
|
yes |
aripiprazole |
psychosis |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2015 |
small molecule |
partial agonist |
14642974
|
17242925
|
17265076
|
yes |
aripiprazole |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2002 |
small molecule |
partial agonist |
16366516
|
9083792
|
16925992
|
16981227
|
17501690
|
11752352
|
yes |
aripiprazole |
psychosis |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2015 |
small molecule |
partial agonist |
16366516
|
9083792
|
16925992
|
16981227
|
17501690
|
11752352
|
yes |
asenapine |
schizophrenia |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
10592235
|
21655346
|
18308814
|
yes |
asenapine |
schizophrenia |
5ht2c_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
10592235
|
21655346
|
18308814
|
yes |
asenapine |
schizophrenia |
5ht6r_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
10592235
|
21655346
|
18308814
|
yes |
atropine |
nerve antidote |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1973 |
small molecule |
antagonist |
7855217
|
17139284
|
17016423
|
yes |
atropine |
nerve antidote |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1973 |
small molecule |
antagonist |
7855217
|
17139284
|
17016423
|
yes |
atropine |
nerve antidote |
acm4_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1973 |
small molecule |
antagonist |
7855217
|
17139284
|
17016423
|
yes |
asenapine |
schizophrenia |
5ht1b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
21655346
|
18308814
|
yes |
asenapine |
schizophrenia |
5ht5a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
21655346
|
18308814
|
yes |
asenapine |
schizophrenia |
5ht7r_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
21655346
|
18308814
|
yes |
asenapine |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
21655346
|
21658377
|
18308814
|
yes |
asfotase alfa |
hypophosphatasia |
s1pr1_human |
primary |
Class A (Rhodopsin) |
Lysophospholipid (S1P) receptors |
approved |
4 |
- |
2015 |
enzyme |
agonist |
20446681
|
21345969
|
no |
astemizole |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1988 |
small molecule |
antagonist |
8001268
|
6146346
|
3147222
|
10597865
|
10597866
|
6204835
|
2892659
|
11752352
|
no |
atenolol |
Anti-Arrhythmia ; Antihypertensive |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1981 |
small molecule |
antagonist |
10913016
|
12065078
|
17628611
|
9300315
|
11752352
|
yes |
atosiban |
labor repressant |
oxyr_human |
primary |
Class A (Rhodopsin) |
Vasopressin and oxytocin receptors |
approved |
4 |
- |
2013 |
small molecule |
antagonist |
22069312
|
no |
atropine |
nerve antidote |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1973 |
small molecule |
antagonist |
16248990
|
17087737
|
15333678
|
17588565
|
16188951
|
7855217
|
yes |
atropine |
nerve antidote |
acm5_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1973 |
small molecule |
antagonist |
7855217
|
17139284
|
17016423
|
11752352
|
yes |
azatadine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1977 |
small molecule |
antagonist |
9638277
|
2568212
|
2523301
|
7528133
|
11752352
|
yes |
azilsartan medoxomil |
Antihypertensive |
agtr1_human |
primary |
Class A (Rhodopsin) |
Angiotensin receptors |
approved |
4 |
- |
2011 |
small molecule |
antagonist |
11752352
|
23563275
|
yes |
azelastine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1996 |
small molecule |
antagonist |
2540229
|
8829888
|
9585822
|
11752352
|
19209282
|
17723160
|
10478514
|
yes |
azelastine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2012 |
small molecule |
antagonist |
2540229
|
8829888
|
9585822
|
11752352
|
19209282
|
17723160
|
10478514
|
yes |
baclofen |
anti-spastic |
gabr2_human |
primary |
Class C (Glutamate) |
GABAB receptors |
approved |
4 |
- |
1977 |
small molecule |
agonist |
10658574
|
15235087
|
8388192
|
10751439
|
11008066
|
19303900
|
10328880
|
10545129
|
yes |
baclofen |
anti-spastic |
gabr1_human |
primary |
Class C (Glutamate) |
GABAB receptors |
approved |
4 |
- |
1977 |
small molecule |
agonist |
8388192
|
11752352
|
10386831
|
19303900
|
10444662
|
10482760
|
10494996
|
10545129
|
10094428
|
yes |
benperidol |
Antipsychotic |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2006 |
small molecule |
antagonist |
27241797
|
yes |
benzphetamine |
Central Nervous System Stimulants |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
17139284
|
17016423
|
no |
benzphetamine |
Central Nervous System Stimulants |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
17139284
|
17016423
|
no |
benztropine |
Antiparkinson |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1954 |
small molecule |
antagonist |
16460947
|
no |
bepotastine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
16914135
|
11752352
|
no |
betahistine |
vertigo |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1970 |
small molecule |
agonist |
18447604
|
11700150
|
yes |
betahistine |
vertigo |
hrh3_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1970 |
small molecule |
antagonist |
18447604
|
11700150
|
20530654
|
yes |
betanechol |
Antidiabetic |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1970 |
small molecule |
agonist |
11798291
|
17413603
|
no |
betaxolol |
Antihypertensive |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1985 |
small molecule |
antagonist |
12181453
|
17513029
|
2077180
|
2891463
|
11752352
|
yes |
betazole |
Diagnostic |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
2892392
|
3661710
|
2886642
|
2874214
|
7213132
|
11752352
|
no |
bethanechol |
eosinophilic esophagitis |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1948 |
small molecule |
agonist |
17139284
|
17016423
|
17413603
|
11798291
|
16953191
|
yes |
brimonidine |
Antiglaucomic |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1996 |
small molecule |
agonist |
14610637
|
8097565
|
yes |
bethanidine |
Antihypertensive |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
11752352
|
no |
bethanidine |
Antihypertensive |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
11752352
|
no |
bethanidine |
Antihypertensive |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
11752352
|
no |
bromocriptine |
Antidiabetic |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1978 |
small molecule |
agonist |
12010185
|
11752352
|
18691132
|
10641988
|
10626749
|
12753422
|
10721819
|
11444429
|
yes |
bethanidine |
Antihypertensive |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
11752352
|
2545383
|
no |
bethanidine |
Antihypertensive |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
11752352
|
2545383
|
no |
bethanidine |
Antihypertensive |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
11752352
|
2545383
|
no |
bilastine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2010 |
small molecule |
antagonist |
27110120
|
yes |
bimatoprost |
Antiglaucomic |
pf2r_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
11740958
|
12222762
|
14733708
|
18452763
|
689791
|
19697832
|
17724194
|
11752352
|
yes |
bimatoprost |
Antiglaucomic |
pe2r1_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
14733708
|
16877408
|
yes |
bimatoprost |
Antiglaucomic |
pe2r3_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
14733708
|
19232013
|
16877408
|
yes |
biperiden |
Antidyskinetics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1959 |
small molecule |
antagonist |
17139284
|
17016423
|
10907719
|
9798802
|
10370904
|
8081071
|
11752352
|
yes |
bisoprolol |
Antihypertensive |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1992 |
small molecule |
antagonist |
1280737
|
14757145
|
16325050
|
1676675
|
1691366
|
11752352
|
yes |
bitolterol |
obstructive lung disease |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
agonist |
17139284
|
17016423
|
10796631
|
3278878
|
no |
bopindolol |
Antihypertensive |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
- |
small molecule |
partial agonist |
11752352
|
14608456
|
1687398
|
2148726
|
8884690
|
2907348
|
no |
bosentan |
Antihypertensive |
ednra_human |
primary |
Class A (Rhodopsin) |
Endothelin receptors |
approved |
4 |
- |
2001 |
small molecule |
antagonist |
11728166
|
11752352
|
11447307
|
11704565
|
10961375
|
11849873
|
yes |
bosentan |
Antihypertensive |
ednrb_human |
primary |
Class A (Rhodopsin) |
Endothelin receptors |
approved |
4 |
- |
2001 |
small molecule |
antagonist |
11752352
|
7921608
|
16335785
|
9806221
|
7858879
|
15629255
|
yes |
bromocriptine |
Antidiabetic |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1978 |
small molecule |
agonist |
18691132
|
10641988
|
yes |
brexpiprazole |
Anti-depressant |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2015 |
small molecule |
partial agonist |
24947465
|
no |
brexpiprazole |
Anti-depressant |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2015 |
small molecule |
partial agonist |
24947465
|
no |
brexpiprazole |
Anti-depressant |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2015 |
small molecule |
partial agonist |
24947465
|
no |
bromodiphenhydramine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1954 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
no |
brimonidine |
Antiglaucomic |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1996 |
small molecule |
agonist |
10799649
|
11481271
|
1373179
|
11752352
|
yes |
brimonidine |
Antiglaucomic |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1996 |
small molecule |
agonist |
14610637
|
11606316
|
12670699
|
16757535
|
yes |
bromopride |
Antiemetics |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
14871277
|
no |
brompheniramine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1957 |
small molecule |
antagonist |
1680053
|
1970615
|
7714410
|
7855217
|
10212017
|
11752352
|
yes |
buclizine |
Antiemetics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
no |
buclizine |
Antiemetics |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
no |
bupranolol |
Antihypertensive |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
19439807
|
no |
buserelin |
LHRH analogue |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
- |
peptide |
not available |
20053189
|
yes |
buprenorphine |
Anti-depressant; Analgesics; opioid addiction |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1981 |
small molecule |
agonist |
10729371
|
10942856
|
11275413
|
12435410
|
15100703
|
11752352
|
yes |
buprenorphine |
Anti-depressant; Analgesics; opioid addiction |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2016 |
small molecule |
agonist |
10729371
|
10942856
|
11275413
|
12435410
|
15100703
|
11752352
|
yes |
buspirone |
Anti-anxiety |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1986 |
small molecule |
partial agonist |
10027850
|
10064829
|
10215901
|
10221756
|
10428422
|
11752352
|
14769835
|
yes |
buprenorphine |
Anti-depressant; Analgesics; opioid addiction |
oprk_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2016 |
small molecule |
agonist |
17244875
|
16953647
|
yes |
buspirone |
Anti-anxiety |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1986 |
small molecule |
partial agonist |
12781354
|
11421254
|
11224194
|
14522358
|
16214127
|
yes |
butorphanol |
Analgesics |
oprk_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1978 |
small molecule |
partial agonist |
10381785
|
10779697
|
12127012
|
12470863
|
15942128
|
8968334
|
8746803
|
7705457
|
2555580
|
17909753
|
no |
buprenorphine |
Anti-depressant; Analgesics; opioid addiction |
oprk_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1981 |
small molecule |
agonist |
17244875
|
16953647
|
yes |
butorphanol |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1978 |
small molecule |
partial agonist |
10381785
|
12127012
|
12470863
|
15942128
|
8968334
|
8746803
|
9399970
|
7705457
|
17909753
|
no |
butorphanol |
Analgesics |
oprd_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1978 |
small molecule |
partial agonist |
12127012
|
12470863
|
15942128
|
8968334
|
8746803
|
7705457
|
17909753
|
11752352
|
no |
cabergoline |
Antiparkinson |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1996 |
small molecule |
agonist |
11752352
|
12464354
|
12008749
|
12721865
|
15341508
|
8951172
|
11436517
|
18303487
|
yes |
butriptyline |
Anti-depressant |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1974 |
small molecule |
antagonist |
6086881
|
3816971
|
9537821
|
no |
butriptyline |
Anti-depressant |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1974 |
small molecule |
antagonist |
6086881
|
3816971
|
9537821
|
no |
caffeine |
Central Nervous System Stimulants |
aa1r_human |
primary |
Class A (Rhodopsin) |
Adenosine receptors |
approved |
4 |
- |
1999 |
small molecule |
antagonist |
16702031
|
17372967
|
17126319
|
17162470
|
17085856
|
11752352
|
yes |
caffeine |
Central Nervous System Stimulants |
aa2ar_human |
primary |
Class A (Rhodopsin) |
Adenosine receptors |
approved |
4 |
- |
1999 |
small molecule |
antagonist |
17558310
|
17577101
|
17616786
|
11752352
|
yes |
calcitonin human |
parathyroid disease |
calcr_human |
primary |
Class B1 (Secretin) |
Calcitonin receptors |
approved |
4 |
- |
1986 |
peptide |
agonist |
22461211
|
no |
calcitonin salmon recombinant |
Paget's disease |
calcr_human |
primary |
Class B1 (Secretin) |
Calcitonin receptors |
approved |
4 |
- |
2005 |
peptide |
agonist |
7610922
|
no |
calcitonin salmon recombinant |
osteitis deformans |
calcr_human |
primary |
Class B1 (Secretin) |
Calcitonin receptors |
approved |
4 |
- |
2005 |
peptide |
agonist |
7610922
|
no |
calcitonin salmon recombinant |
postmenopausal osteoporosis |
calcr_human |
primary |
Class B1 (Secretin) |
Calcitonin receptors |
approved |
4 |
- |
1978 |
peptide |
agonist |
7610922
|
no |
candesartan cilexetil |
Antihypertensive |
agtr1_human |
primary |
Class A (Rhodopsin) |
Angiotensin receptors |
approved |
4 |
- |
1998 |
small molecule |
antagonist |
19436650
|
17588300
|
yes |
cangrelor |
antithrombotic |
p2y12_human |
primary |
Class A (Rhodopsin) |
P2Y receptors |
approved |
4 |
- |
2015 |
small molecule |
antagonist |
26402735
|
no |
captodiame |
anxiolytic |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
- |
small molecule |
agonist |
23863923
|
no |
captodiame |
anxiolytic |
5ht2c_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
23863923
|
no |
carbachol |
Antiglaucomic |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1972 |
small molecule |
agonist |
15059034
|
no |
carbachol |
Antiglaucomic |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1972 |
small molecule |
agonist |
15485827
|
15333678
|
12948933
|
12505062
|
16181410
|
no |
carbinoxamine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2003 |
small molecule |
antagonist |
7513381
|
16574052
|
1143714
|
19761204
|
11752352
|
no |
carboprost tromethamine |
Abortifacient |
pe2r1_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1965 |
small molecule |
agonist |
17016423
|
20519365
|
11338376
|
9462300
|
no |
cevimeline |
Parasympathomimetics |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2000 |
small molecule |
agonist |
17139284
|
17016423
|
18450949
|
11752352
|
no |
cariprazine |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2015 |
small molecule |
partial agonist |
23320989
|
no |
cariprazine |
schizophrenia |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2015 |
small molecule |
partial agonist |
23320989
|
no |
carphenazine |
schizophrenia |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
4889058
|
4887393
|
4861216
|
no |
carphenazine |
schizophrenia |
drd5_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
4889058
|
4887393
|
4861216
|
no |
carphenazine |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
4889058
|
4887393
|
4861216
|
11752352
|
no |
carteolol |
Antiglaucomic |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1988 |
small molecule |
antagonist |
11752352
|
15526107
|
10864881
|
16160085
|
yes |
carteolol |
cardiovascular disease |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1988 |
small molecule |
antagonist |
1349493
|
15526107
|
11752352
|
yes |
carvedilol |
cardiovascular disease |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1995 |
small molecule |
antagonist |
1712335
|
2575762
|
2577144
|
7908256
|
yes |
carvedilol |
congestive heart failure |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1995 |
small molecule |
antagonist |
17139284
|
17016423
|
yes |
celiprolol |
Antihypertensive |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
- |
small molecule |
agonist |
17141277
|
yes |
celiprolol |
Antihypertensive |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
17384462
|
17141277
|
18636069
|
yes |
ceruletide, caerulein |
Diagnostic |
cckar_human |
primary |
Class A (Rhodopsin) |
Cholecystokinin receptors |
withdrawn |
4 |
- |
1982 |
small molecule |
agonist |
2087492
|
1620654
|
8182534
|
1356589
|
2587420
|
3440035
|
no |
cetirizine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2007 |
small molecule |
antagonist |
11752352
|
12787835
|
15286093
|
14505791
|
10597865
|
15942272
|
yes |
cetrorelix |
Antineoplastic |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
2000 |
peptide |
antagonist |
11854630
|
12606421
|
14561652
|
14605254
|
16809153
|
11752352
|
yes |
cevimeline |
Parasympathomimetics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2000 |
small molecule |
agonist |
17139284
|
17016423
|
8624083
|
no |
chlophedianol |
Antitussive |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1987 |
small molecule |
antagonist |
2905706
|
no |
chlorcyclizine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
21058326
|
no |
chloropyramine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
19610651
|
no |
chlorpheniramine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1950 |
small molecule |
antagonist |
11736858
|
no |
chlorpromazine |
psychosis |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1957 |
small molecule |
antagonist |
10821438
|
8593484
|
yes |
chlorpromazine |
psychosis |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1957 |
small molecule |
antagonist |
11103886
|
11873706
|
15694263
|
16867246
|
11752352
|
20643630
|
7908055
|
8524985
|
yes |
chlorprothixene |
schizophrenia |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
3774629
|
2891550
|
yes |
chlorprothixene |
schizophrenia |
5ht2b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
17139284
|
17016423
|
yes |
chlorprothixene |
schizophrenia |
5ht2c_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
17139284
|
17016423
|
yes |
chlorprothixene |
schizophrenia |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
17139284
|
17016423
|
1830565
|
yes |
chlorprothixene |
schizophrenia |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
17139284
|
17016423
|
1830565
|
yes |
chlorprothixene |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
8101879
|
1830565
|
19091563
|
11752352
|
yes |
chorionic gonadotropin |
Antineoplastic |
lshr_human |
primary |
Class A (Rhodopsin) |
Glycoprotein hormone receptors |
approved |
4 |
- |
1973 |
protein |
agonist |
20836886
|
no |
chorionic gonadotropin |
stroke |
lshr_human |
primary |
Class A (Rhodopsin) |
Glycoprotein hormone receptors |
approved |
4 |
- |
1973 |
protein |
agonist |
20836886
|
no |
chorionic gonadotropin |
Fertility |
lshr_human |
primary |
Class A (Rhodopsin) |
Glycoprotein hormone receptors |
approved |
4 |
- |
1973 |
protein |
agonist |
20836886
|
no |
cimetidine |
Antihistamines |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1977 |
small molecule |
antagonist |
11752352
|
10950107
|
8863950
|
16723495
|
yes |
cimetidine |
GI Anti-Ulcer ; antihistamines |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1977 |
small molecule |
antagonist |
11752352
|
10950107
|
8863950
|
16723495
|
yes |
cinacalcet |
hyperparathyroidism |
casr_human |
primary |
Class C (Glutamate) |
Calcium-sensing receptors |
approved |
4 |
- |
2004 |
small molecule |
PAM |
15794735
|
15864123
|
15884662
|
16030053
|
16109140
|
19461861
|
19261825
|
19181759
|
19056615
|
11752352
|
yes |
cinacalcet |
Calcimimetics |
casr_human |
primary |
Class C (Glutamate) |
Calcium-sensing receptors |
approved |
4 |
- |
2004 |
small molecule |
PAM |
15794735
|
15864123
|
15884662
|
16030053
|
16109140
|
19461861
|
19261825
|
19181759
|
19056615
|
11752352
|
yes |
cinitapride |
gastrointestinal disorders |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
9211565
|
9562338
|
no |
cinitapride |
gastrointestinal disorders |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
- |
small molecule |
agonist |
9211565
|
9562338
|
no |
cinnarizine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1989 |
small molecule |
antagonist |
11752352
|
2866055
|
yes |
cisapride |
Parasympathomimetics |
5ht4r_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1993 |
small molecule |
agonist |
10027842
|
10328995
|
10556228
|
11034583
|
11218067
|
11752352
|
no |
clemastine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1977 |
small molecule |
antagonist |
11752352
|
2890562
|
6701456
|
6387510
|
1678430
|
7513381
|
4074605
|
6449094
|
1266718
|
8930778
|
yes |
glucagon |
for prevention of hypoglycemia |
glr_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
1960 |
peptide |
agonist |
17623014
|
17620721
|
yes |
clenbuterol |
Bronchodilator |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
- |
small molecule |
agonist |
11720783
|
12388476
|
1322047
|
1685013
|
17449161
|
11752352
|
no |
clidinium |
GI Anti-Ulcer ; anticholinergic; Antispasmodics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2013 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
no |
clofedanol |
antitussive |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1987 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
2905706
|
no |
cyclobenzaprine |
Muscle Relaxants |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1977 |
small molecule |
antagonist |
12498911
|
8884233
|
no |
clonidine |
diabetic neuropathy; ADHD; antimucositic |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1974 |
small molecule |
agonist |
28715875
|
yes |
clonidine |
diabetic neuropathy; ADHD; antimucositic |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1974 |
small molecule |
agonist |
28715875
|
yes |
clonidine |
diabetic neuropathy; ADHD; antimucositic |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1974 |
small molecule |
agonist |
11752127
|
12357167
|
15306201
|
14757140
|
12098614
|
yes |
clopidogrel |
antiplatelet |
p2y12_human |
primary |
Class A (Rhodopsin) |
P2Y receptors |
approved |
4 |
- |
1997 |
small molecule |
antagonist |
14668029
|
15199474
|
15269827
|
15291969
|
15308557
|
11752352
|
19463375
|
16835302
|
12615691
|
yes |
clopidogrel |
antithrombotic |
p2y12_human |
primary |
Class A (Rhodopsin) |
P2Y receptors |
approved |
4 |
- |
1997 |
small molecule |
antagonist |
14668029
|
15199474
|
15269827
|
15291969
|
15308557
|
11752352
|
19463375
|
16835302
|
12615691
|
yes |
clozapine |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1989 |
small molecule |
antagonist |
12769622
|
14575800
|
15286066
|
15781964
|
16040180
|
11752352
|
yes |
clozapine |
schizophrenia |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1989 |
small molecule |
antagonist |
12973385
|
14530903
|
14687870
|
14751426
|
15037867
|
7520908
|
yes |
cocaine |
local anesthetic |
drd3_human |
secondary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
15351386
|
yes |
cocaine |
local anesthetic |
oprk_human |
secondary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
15351386
|
2840298
|
yes |
codeine |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2009 |
small molecule |
agonist |
15509185
|
17620111
|
8306082
|
11752352
|
yes |
codeine |
Analgesics |
oprd_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2009 |
small molecule |
agonist |
16386786
|
7885194
|
12067475
|
8119316
|
2156065
|
11752352
|
yes |
codeine |
Analgesics |
oprk_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2009 |
small molecule |
agonist |
17139284
|
17016423
|
17620111
|
7885194
|
yes |
conivaptan |
hyponatremia |
v2r_human |
primary |
Class A (Rhodopsin) |
Vasopressin and oxytocin receptors |
approved |
4 |
- |
2005 |
small molecule |
antagonist |
11752352
|
15659304
|
16843091
|
17919259
|
17202666
|
17592003
|
19695403
|
16522696
|
19057376
|
20054444
|
17428103
|
19663609
|
no |
conivaptan |
hyponatremia |
v1ar_human |
primary |
Class A (Rhodopsin) |
Vasopressin and oxytocin receptors |
approved |
4 |
- |
2005 |
small molecule |
antagonist |
11752352
|
17919259
|
17202666
|
17592003
|
19695403
|
16522696
|
19057376
|
20054444
|
17428103
|
19663609
|
no |
corticorelin ovine triflutate |
Diagnostic |
crfr1_human |
primary |
Class B1 (Secretin) |
Corticotropin-releasing factor receptors |
approved |
4 |
- |
1996 |
small molecule |
agonist |
20809121
|
no |
cosyntropin |
Diagnostic |
acthr_human |
primary |
Class A (Rhodopsin) |
Melanocortin receptors |
approved |
4 |
- |
1970 |
peptide |
agonist |
15710205
|
2156274
|
20562554
|
11752352
|
no |
cromolyn sodium, chromoglycate |
anti-allergenic |
gpr35_human |
primary |
Class A (Rhodopsin) |
Class A orphans |
approved |
4 |
- |
2000 |
small molecule |
agonist |
20559017
|
no |
cyclizine |
Antiemetics |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
11752352
|
1983158
|
yes |
cyclobenzaprine |
Anti-depressant |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1977 |
small molecule |
antagonist |
12498911
|
8884233
|
no |
cyclopentolate |
Mydriatics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1974 |
small molecule |
antagonist |
17139284
|
17016423
|
yes |
cycrimine |
Antiparkinson |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
1267542
|
11752352
|
no |
cyproheptadine |
Anti-Allergic ; Appetite Stimulant |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1961 |
small molecule |
antagonist |
11752352
|
yes |
cyproheptadine |
Anti-Allergic ; Appetite Stimulant |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1961 |
small molecule |
antagonist |
12233819
|
12498911
|
1358088
|
1403790
|
16418149
|
yes |
danazol |
diabetic macular edema |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1976 |
small molecule |
agonist |
14571621
|
3004220
|
14605254
|
2404115
|
yes |
danazol |
Antiendometriosis ; Antineoplastic |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1976 |
small molecule |
agonist |
14571621
|
3004220
|
14605254
|
2404115
|
yes |
darifenacin |
overactive bladder |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2004 |
small molecule |
antagonist |
20395537
|
19416629
|
18046909
|
11752352
|
yes |
dapiprazole |
opthalmological |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1990 |
small molecule |
antagonist |
17139284
|
17016423
|
no |
dapiprazole |
opthalmological |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1990 |
small molecule |
antagonist |
17139284
|
17016423
|
no |
dapiprazole |
opthalmological |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1990 |
small molecule |
antagonist |
17139284
|
17016423
|
9401944
|
no |
degarelix |
Antineoplastic |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
2008 |
small molecule |
antagonist |
20110043
|
20053189
|
19450172
|
15705170
|
yes |
desipramine |
Anti-depressant |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1964 |
small molecule |
antagonist |
10467920
|
7855217
|
no |
desloratadine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2001 |
small molecule |
antagonist |
15564772
|
7581058
|
8174605
|
11752352
|
18336052
|
17902729
|
12642846
|
18797058
|
yes |
desmopressin |
Antidiuretic |
v1ar_human |
primary |
Class A (Rhodopsin) |
Vasopressin and oxytocin receptors |
approved |
4 |
- |
1978 |
peptide |
not available |
10731046
|
10594321
|
8957254
|
15613460
|
yes |
desmopressin |
Antidiuretic |
v1br_human |
primary |
Class A (Rhodopsin) |
Vasopressin and oxytocin receptors |
approved |
4 |
- |
1978 |
peptide |
not available |
15613460
|
14971638
|
18655906
|
yes |
desmopressin |
Antidiuretic |
v2r_human |
primary |
Class A (Rhodopsin) |
Vasopressin and oxytocin receptors |
approved |
4 |
- |
1978 |
peptide |
agonist |
18761325
|
16333859
|
11752352
|
yes |
dexbrompheniramine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1963 |
small molecule |
antagonist |
9691225
|
1680053
|
1970615
|
7714410
|
19085565
|
11752352
|
no |
dexchlorpheniramine |
sunburn |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1981 |
small molecule |
antagonist |
374215
|
no |
dexmedetomidine |
Analgesics |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1999 |
small molecule |
agonist |
15306201
|
no |
dexmedetomidine |
Antineoplastic |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1999 |
small molecule |
agonist |
15306201
|
no |
dexmedetomidine |
Analgesics; Hypnotics and Sedatives |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1999 |
small molecule |
agonist |
11752127
|
11834617
|
14583739
|
15087625
|
15306201
|
17692748
|
no |
dezocine |
Analgesics |
oprk_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1989 |
small molecule |
partial agonist |
17139284
|
17016423
|
16433932
|
11752352
|
no |
glucagon |
hypoglycemia |
glr_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
1998 |
peptide |
agonist |
17623014
|
17620721
|
yes |
glycopyrrolate |
Antineoplastic |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1961 |
small molecule |
antagonist |
8249551
|
no |
dezocine |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1989 |
small molecule |
partial agonist |
9399970
|
11702089
|
10958085
|
12513698
|
9972766
|
1361946
|
no |
dicyclomine |
Antispasmodics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1950 |
small molecule |
antagonist |
17139284
|
17016423
|
19533734
|
11752352
|
no |
difenoxin |
recurrent infection of the gastrointestinal tract |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1978 |
small molecule |
agonist |
8386327
|
no |
dihydrocodeine |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1958 |
small molecule |
agonist |
12665158
|
yes |
dihydroergotamine |
Anti-migraine |
5ht1b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1997 |
small molecule |
agonist |
10455274
|
14744615
|
1660351
|
8622623
|
9650800
|
no |
dipivefrin |
Antiglaucomic |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1980 |
small molecule |
agonist |
11752352
|
17622774
|
17417877
|
17597612
|
yes |
dihydroergotamine |
Anti-migraine |
5ht1d_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1997 |
small molecule |
agonist |
11752352
|
9605573
|
1379707
|
1324091
|
12558771
|
1407010
|
14744615
|
no |
dimenhydrinate |
Antiemetics |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1972 |
small molecule |
antagonist |
11752352
|
11835984
|
yes |
dimetindene |
Anti-Allergic |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
- |
small molecule |
antagonist |
8608784
|
no |
dimetindene |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
20800486
|
8608784
|
no |
dinoprost tromethamine |
Abortifacient |
pi2r_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1981 |
small molecule |
agonist |
17139284
|
17016423
|
11752352
|
no |
dinoprostone |
Abortifacient |
pe2r4_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1977 |
small molecule |
agonist |
16545798
|
18715952
|
20599704
|
19788928
|
17329241
|
yes |
dinoprostone |
Abortifacient |
pe2r1_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1977 |
small molecule |
agonist |
18715952
|
20599704
|
19788928
|
17329241
|
yes |
dinoprostone |
Abortifacient |
pe2r3_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1977 |
small molecule |
agonist |
18715952
|
20599704
|
19788928
|
17329241
|
yes |
dinoprostone |
Abortifacient |
pe2r2_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1977 |
small molecule |
agonist |
18715952
|
20599704
|
19788928
|
17329241
|
11752352
|
yes |
diphemanil |
Bronchodilator |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1976 |
small molecule |
antagonist |
6450282
|
no |
diphenhydramine |
Anti-Allergic ; Hypnotics and sedatives; Antiemetics; Antipruritics; Antitussives |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1946 |
small molecule |
antagonist |
11752352
|
17169617
|
16702624
|
17390763
|
17196194
|
17329841
|
2878016
|
yes |
diphenidol |
Antiemetics |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
10497897
|
9851542
|
9454790
|
9059856
|
8050463
|
12185001
|
10530931
|
1863523
|
no |
diphenidol |
Antiemetics |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
17139284
|
17016423
|
12185001
|
10530931
|
1863523
|
no |
diphenidol |
Antiemetics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
17139284
|
17016423
|
1863523
|
no |
diphenoxylate |
Antidiuretic |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
11752352
|
18192961
|
10202212
|
8583364
|
8386327
|
no |
diphenylpyraline |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
1912125
|
1678430
|
18977145
|
15627433
|
11752352
|
no |
dipivefrin |
opthalmological |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1980 |
small molecule |
agonist |
17139284
|
17016423
|
yes |
dipivefrin |
Antiglaucomic |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1980 |
small molecule |
agonist |
17603545
|
17658513
|
yes |
dobutamine |
Cardiotonic |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1978 |
small molecule |
agonist |
12098582
|
15564877
|
16325050
|
16627864
|
11752352
|
no |
dopamine |
hypotension |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1974 |
small molecule |
agonist |
23241039
|
no |
doxepin |
Hypnotics and Sedatives |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
2897127
|
2141000
|
yes |
doxacurium |
Muscle Relaxants |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1991 |
small molecule |
antagonist |
9523819
|
no |
doxazosin |
Anticholesteremic ; Antihypertensive ; Vasodilator |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1990 |
small molecule |
antagonist |
15573147
|
8736427
|
14767264
|
9205965
|
16225542
|
19002123
|
17070143
|
10393471
|
11752352
|
yes |
doxazosin |
Anticholesteremic ; Antihypertensive ; Vasodilator |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1990 |
small molecule |
antagonist |
18231614
|
19002123
|
17070143
|
10393471
|
yes |
doxazosin |
Anticholesteremic ; Antihypertensive ; Vasodilator |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1990 |
small molecule |
antagonist |
18231614
|
19002123
|
17070143
|
10393471
|
yes |
doxepin |
Hypnotics and Sedatives |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
15286093
|
7238574
|
15255990
|
3011460
|
6086881
|
7855217
|
19179941
|
17685877
|
2141000
|
11752352
|
yes |
doxepin |
Hypnotics and Sedatives |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
7855217
|
19179941
|
2329499
|
2141000
|
yes |
doxepin |
Hypnotics and Sedatives |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
7855217
|
309138
|
19179941
|
yes |
doxepin |
Hypnotics and Sedatives |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
7855217
|
2329499
|
2141000
|
yes |
doxepin |
Hypnotics and Sedatives |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
7855217
|
2329499
|
2141000
|
yes |
doxepin |
Hypnotics and Sedatives |
acm4_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
7855217
|
2329499
|
2141000
|
yes |
doxepin |
Hypnotics and Sedatives |
acm5_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
7855217
|
2329499
|
2141000
|
yes |
doxylamine |
Antihistamine; for nausea and vomiting of pregnancy |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1948 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
no |
doxepin |
Hypnotics and Sedatives |
5ht2b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
7855217
|
309138
|
yes |
doxepin |
Hypnotics and Sedatives |
5ht2c_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1969 |
small molecule |
antagonist |
7855217
|
309138
|
yes |
doxylamine |
Anti-Allergic ; Antiemetics; Antitussive ; Hypnotics and Sedatives |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1948 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
no |
dronabinol |
Analgesics |
cnr1_human |
primary |
Class A (Rhodopsin) |
Cannabinoid receptors |
approved |
4 |
- |
1985 |
small molecule |
agonist |
17139284
|
17016423
|
12686391
|
11204352
|
11752352
|
no |
dronabinol |
Appetite stimulant |
cnr1_human |
primary |
Class A (Rhodopsin) |
Cannabinoid receptors |
approved |
4 |
- |
1985 |
small molecule |
agonist |
17139284
|
17016423
|
12686391
|
11204352
|
11752352
|
no |
droperidol |
psychosis |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1970 |
small molecule |
antagonist |
2527092
|
no |
dronedarone |
Anti-Arrhythmia |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
17389667
|
yes |
dronedarone |
Anti-Arrhythmia |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
17389667
|
yes |
droperidol |
Adjuvants; Anesthesia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1970 |
small molecule |
antagonist |
1549935
|
2527092
|
14633536
|
20358234
|
no |
droxidopa |
orthostatic hypotension |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2014 |
small molecule |
agonist |
11482743
|
17266602
|
20412040
|
9138687
|
8825367
|
no |
droxidopa |
orthostatic hypotension |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2014 |
small molecule |
agonist |
17266602
|
20412040
|
7582530
|
7674815
|
no |
droxidopa |
orthostatic hypotension |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2014 |
small molecule |
agonist |
17266602
|
20412040
|
7773533
|
8166240
|
no |
droxidopa |
orthostatic hypotension |
adrb3_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2014 |
small molecule |
agonist |
19434307
|
9464897
|
19110970
|
18064417
|
no |
droxidopa |
orthostatic hypotension |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2014 |
small molecule |
agonist |
21173850
|
18680204
|
11306720
|
no |
droxidopa |
orthostatic hypotension |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2014 |
small molecule |
agonist |
21173850
|
18680204
|
18064417
|
no |
droxidopa |
orthostatic hypotension |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2014 |
small molecule |
agonist |
21173850
|
18680204
|
8590979
|
no |
droxidopa |
orthostatic hypotension |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2014 |
small molecule |
agonist |
9464897
|
19110970
|
18064417
|
no |
droxidopa |
orthostatic hypotension |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2014 |
small molecule |
agonist |
9464897
|
9666280
|
7969507
|
19110970
|
18064417
|
no |
dulaglutide |
Antidiabetic |
glp1r_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
2014 |
protein |
agonist |
25367716
|
yes |
eletriptan |
Anti-migraine |
5ht1b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2002 |
small molecule |
agonist |
10193663
|
11050304
|
11069595
|
11513839
|
12384251
|
11752352
|
yes |
eletriptan |
Anti-migraine |
5ht1f_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2002 |
small molecule |
agonist |
10193663
|
11834243
|
15185063
|
yes |
eletriptan |
Anti-migraine |
5ht1d_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2002 |
small molecule |
agonist |
11752352
|
10193663
|
15821444
|
11513839
|
12498013
|
11152011
|
yes |
eluxadoline |
irritable bowel syndrome |
oprd_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2015 |
small molecule |
agonist |
25261794
|
no |
eluxadoline |
irritable bowel syndrome |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2015 |
small molecule |
agonist |
25261794
|
23583433
|
no |
emedastine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1997 |
small molecule |
antagonist |
7714409
|
7714410
|
9747899
|
19558341
|
15553105
|
18714531
|
11752352
|
yes |
ephedrine |
Central Nervous System Stimulants |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1963 |
small molecule |
not available |
17405867
|
12557268
|
10592235
|
yes |
epinastine |
Anti-Allergic |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2003 |
small molecule |
antagonist |
16131920
|
yes |
epinastine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2003 |
small molecule |
antagonist |
17534605
|
1972625
|
11752352
|
yes |
epinephrine, adrenaline |
Anesthetics |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1976 |
small molecule |
agonist |
11306720
|
10742288
|
9836297
|
1980236
|
18680204
|
18064417
|
no |
epinephrine, adrenaline |
Anesthetics |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1976 |
small molecule |
agonist |
11752352
|
17622774
|
17417877
|
17597612
|
no |
epinephrine, adrenaline |
Anesthetics |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1976 |
small molecule |
agonist |
11752352
|
17622774
|
17541557
|
no |
epinephrine, adrenaline |
Anesthetics |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1976 |
small molecule |
agonist |
17603545
|
17658513
|
20412040
|
20857090
|
no |
epinephrine, adrenaline |
Anesthetics |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1976 |
small molecule |
agonist |
1979424
|
11728431
|
11053214
|
1980236
|
18064417
|
no |
epinephrine, adrenaline |
Anesthetics |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1976 |
small molecule |
agonist |
20954794
|
19730427
|
20412040
|
20857090
|
no |
epoprostenol |
Antihypertensive ; Platelet Aggregation Inhibitors |
pi2r_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1995 |
small molecule |
agonist |
19302827
|
12297509
|
20522800
|
11752352
|
yes |
eprosartan |
Antihypertensive |
agtr1_human |
primary |
Class A (Rhodopsin) |
Angiotensin receptors |
approved |
4 |
- |
1997 |
small molecule |
antagonist |
11752352
|
12927226
|
10856732
|
12540520
|
9602957
|
12782193
|
12184062
|
12766389
|
12517247
|
18093407
|
11320369
|
yes |
ergoloid, co-dergocrine mesilate |
cardiovascular disease |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1953 |
small molecule |
agonist |
8786706
|
2869188
|
no |
ergoloid, co-dergocrine mesilate |
cardiovascular disease |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1953 |
small molecule |
agonist |
8786706
|
2869188
|
no |
ergoloid |
cardiovascular disease |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1953 |
small molecule |
agonist |
8786706
|
2869188
|
yes |
ergoloid |
cardiovascular disease |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1953 |
small molecule |
agonist |
8786706
|
2869188
|
yes |
esmolol |
Anti-Arrhythmia |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1986 |
small molecule |
antagonist |
11752352
|
7612051
|
7957532
|
2568748
|
2894187
|
1975995
|
no |
ergoloid |
Nootropic ; Vasodilator |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1953 |
small molecule |
agonist |
8786706
|
2869188
|
yes |
ergoloid |
Nootropic ; Vasodilator |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1953 |
small molecule |
agonist |
8786706
|
2869188
|
yes |
ergonovine, ergometrine |
antihaemorrhagic |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1946 |
small molecule |
agonist |
2897449
|
19933260
|
no |
ergotamine |
Anti-migraine |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
18066532
|
yes |
ergotamine |
Anti-migraine |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
18066532
|
yes |
ergotamine |
Anti-migraine |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
18066532
|
yes |
ergotamine |
Anti-migraine |
5ht1b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
10188968
|
10455274
|
11015308
|
15224175
|
yes |
ergotamine |
Anti-migraine |
5ht1d_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
12558771
|
8384716
|
1407010
|
14504136
|
1646776
|
yes |
ergotamine |
Anti-migraine |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
17139284
|
17016423
|
yes |
ergotamine |
Anti-migraine |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
17139284
|
17016423
|
18066532
|
yes |
ergotamine |
Anti-migraine |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
17139284
|
17016423
|
18066532
|
yes |
etelcalcetide, amg 416, velcalcetide, kai-4169, ono-5163 |
parathyroid disorders |
casr_human |
primary |
Class C (Glutamate) |
Calcium-sensing receptors |
approved |
4 |
- |
2017 |
peptide |
agonist |
24235081
|
no |
ethopropazine |
Antidyskinetics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17016423
|
2904117
|
2236897
|
11752352
|
no |
ethylmorphine |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
- |
small molecule |
agonist |
16530171
|
16580639
|
16580848
|
16682505
|
11752352
|
no |
etomidate |
Anesthetics; Intravenous |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
PAM |
20496522
|
14508322
|
yes |
exenatide |
Antidiabetic |
glp1r_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
2005 |
peptide |
agonist |
16722815
|
17292977
|
17353295
|
16534527
|
17379930
|
20649595
|
15331551
|
15495988
|
15700891
|
16341288
|
16627399
|
11752352
|
yes |
exendin-4 |
Antidiabetic |
glp1r_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
2005 |
peptide |
agonist |
16374859
|
no |
famotidine |
acid reducer |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1986 |
small molecule |
antagonist |
11752352
|
17273750
|
16723495
|
16702624
|
16513821
|
12832840
|
12509588
|
2067140
|
1646056
|
19578661
|
18310651
|
yes |
famotidine |
gastric ulcer and gastroesophageal reflux |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1986 |
small molecule |
antagonist |
11752352
|
17273750
|
16723495
|
16702624
|
16513821
|
12832840
|
12509588
|
2067140
|
1646056
|
19578661
|
18310651
|
yes |
fenoldopam |
Antihypertensive |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1997 |
small molecule |
agonist |
11752352
|
19293728
|
8103596
|
no |
fenoldopam |
Antihypertensive |
drd5_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1997 |
small molecule |
agonist |
17139284
|
17016423
|
19293728
|
8103596
|
no |
fenoterol |
Bronchodilator ; Tocolytic |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
withdrawn |
- |
small molecule |
agonist |
11730729
|
16324695
|
6203844
|
8777955
|
8911881
|
11752352
|
yes |
fentanyl |
adjuvant to anesthesia |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1968 |
small molecule |
agonist |
15589524
|
16114980
|
16332149
|
16376082
|
16797997
|
11752352
|
19403616
|
yes |
fingolimod |
Multiple Sclerosis |
s1pr1_human |
primary |
Class A (Rhodopsin) |
Lysophospholipid (S1P) receptors |
approved |
4 |
- |
2010 |
small molecule |
agonist |
16374859
|
yes |
fingolimod |
Multiple Sclerosis |
s1pr5_human |
primary |
Class A (Rhodopsin) |
Lysophospholipid (S1P) receptors |
approved |
4 |
- |
2010 |
small molecule |
agonist |
23579459
|
23579456
|
yes |
flavoxate |
Antispasmodics |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1970 |
small molecule |
antagonist |
17139284
|
17016423
|
19002123
|
10858873
|
3247311
|
yes |
flavoxate |
Antispasmodics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1970 |
small molecule |
antagonist |
17139284
|
17016423
|
3247311
|
yes |
fentanyl |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1968 |
small molecule |
agonist |
15589524
|
16114980
|
16332149
|
16376082
|
16797997
|
11752352
|
19403616
|
yes |
flibanserin |
sexual dysfunction |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2015 |
small molecule |
agonist |
12890707
|
12177684
|
26412054
|
no |
fentanyl |
adjuvant to anesthesia |
oprd_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1968 |
small molecule |
agonist |
15665994
|
15828941
|
15868528
|
16372825
|
16861092
|
19403616
|
yes |
flunarizine |
Anticonvulsants; Vasodilator |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1968 |
small molecule |
antagonist |
17139284
|
17016423
|
20493137
|
yes |
flupentixol |
Antipsychotic |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1965 |
small molecule |
antagonist |
7052344
|
yes |
flupentixol |
Antipsychotic |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1965 |
small molecule |
antagonist |
17111172
|
yes |
flupentixol |
Antipsychotic |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1965 |
small molecule |
antagonist |
11752352
|
11873706
|
6149133
|
7498321
|
1674528
|
8797192
|
17111172
|
yes |
fentanyl |
Analgesics |
oprd_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1968 |
small molecule |
agonist |
15665994
|
15828941
|
15868528
|
16372825
|
16861092
|
19403616
|
yes |
fesoterodine |
prostate adenocarcinoma |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2007 |
small molecule |
antagonist |
19029429
|
yes |
fesoterodine |
overactive bladder syndrome |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
2007 |
small molecule |
antagonist |
11752352
|
12076307
|
yes |
fexofenadine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1996 |
small molecule |
antagonist |
11752352
|
10864400
|
15352500
|
12712828
|
15286093
|
10597865
|
18336052
|
18797058
|
19545214
|
9506246
|
yes |
flupentixol |
Antipsychotic |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1965 |
small molecule |
antagonist |
17139284
|
17016423
|
10531405
|
17111172
|
yes |
fluphenazine |
schizophrenia |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1959 |
small molecule |
antagonist |
11752352
|
11113312
|
10531405
|
11873706
|
yes |
fluphenazine |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1959 |
small molecule |
antagonist |
11873706
|
7508675
|
7828655
|
11752352
|
yes |
fluphenazine decanoate |
psychosis |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1972 |
small molecule |
antagonist |
7828655
|
yes |
fluphenazine enanthate |
psychosis |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
7828655
|
no |
fluspirilene |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1977 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
11842444
|
8935801
|
no |
formoterol |
Anti-Asthmatic |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2010 |
small molecule |
agonist |
12090787
|
14662724
|
16432501
|
2544117
|
7675115
|
11752352
|
9506248
|
14720051
|
18686730
|
1718682
|
17594727
|
yes |
follitropin |
Fertility |
fshr_human |
primary |
Class A (Rhodopsin) |
Glycoprotein hormone receptors |
approved |
4 |
- |
1997 |
protein |
agonist |
11299519
|
7755615
|
2108722
|
8319832
|
8070368
|
18020563
|
11752352
|
yes |
forasartan |
Antihypertensive |
agtr1_human |
primary |
Class A (Rhodopsin) |
Angiotensin receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
11569611
|
8981065
|
9156352
|
11752352
|
no |
formoterol |
Anti-Asthmatic |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
12090787
|
14662724
|
16432501
|
2544117
|
7675115
|
11752352
|
9506248
|
14720051
|
18686730
|
1718682
|
17594727
|
yes |
formoterol |
chronic obstructive pulmonary disease (COPD) |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2016 |
small molecule |
agonist |
12090787
|
14662724
|
16432501
|
2544117
|
7675115
|
11752352
|
9506248
|
14720051
|
18686730
|
1718682
|
17594727
|
yes |
formoterol |
chronic obstructive pulmonary disease (COPD) |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
12090787
|
14662724
|
16432501
|
2544117
|
7675115
|
11752352
|
9506248
|
14720051
|
18686730
|
1718682
|
17594727
|
yes |
formoterol |
Bronchodilator |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
12090787
|
14662724
|
16432501
|
2544117
|
7675115
|
11752352
|
9506248
|
14720051
|
18686730
|
1718682
|
17594727
|
yes |
formoterol |
Anti-Asthmatic ; COPD |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
12090787
|
14662724
|
16432501
|
2544117
|
7675115
|
11752352
|
9506248
|
14720051
|
18686730
|
1718682
|
17594727
|
yes |
frovatriptan |
Anti-migraine |
5ht1d_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
11752352
|
11735616
|
12028320
|
11152011
|
10883409
|
15185063
|
15311727
|
9700983
|
18360605
|
15342617
|
12028322
|
yes |
frovatriptan |
Anti-migraine |
5ht1b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2001 |
small molecule |
agonist |
11752352
|
15311727
|
12028320
|
9700983
|
11735616
|
17190530
|
11152011
|
10883409
|
18001261
|
18360605
|
15342617
|
12028322
|
yes |
ganirelix acetate |
for prevention of premature ovulation in fertility treatment |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1999 |
small molecule |
antagonist |
15932933
|
no |
gamma hydroxybutyric acid |
Hypnotics and Sedatives |
gabr1_human |
primary |
Class C (Glutamate) |
GABAB receptors |
approved |
4 |
- |
2002 |
small molecule |
agonist |
15745703
|
no |
gamma hydroxybutyric acid |
Hypnotics and Sedatives |
gabr2_human |
primary |
Class C (Glutamate) |
GABAB receptors |
approved |
4 |
- |
2002 |
small molecule |
agonist |
15745703
|
no |
ganirelix acetate |
Fertility |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1999 |
small molecule |
antagonist |
15932933
|
no |
glucagon |
Antidiabetic |
glr_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
1960 |
peptide |
agonist |
17623014
|
17620721
|
yes |
glucagon |
Antihypoglycemic |
glr_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
1960 |
peptide |
agonist |
17623014
|
17620721
|
yes |
icatibant |
hereditary angioedema |
bkrb2_human |
primary |
Class A (Rhodopsin) |
Bradykinin receptors |
approved |
4 |
- |
2008 |
small molecule |
antagonist |
14514033
|
11752352
|
yes |
glycopyrrolate |
chronic obstructive pulmonary disease (COPD) |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1961 |
small molecule |
antagonist |
8249551
|
no |
glycopyrronium |
chronic obstructive pulmonary disease (COPD) |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1961 |
small molecule |
antagonist |
28767773
|
yes |
gonadorelin |
Fertility |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
15967801
|
16962597
|
16973761
|
17002488
|
17068198
|
11752352
|
yes |
goserelin |
Antineoplastic |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1989 |
peptide |
agonist |
20053189
|
yes |
goserelin |
Antineoplastic s; Hormonal |
lshr_human |
primary |
Class A (Rhodopsin) |
Glycoprotein hormone receptors |
approved |
4 |
- |
1989 |
peptide |
agonist |
17139284
|
17016423
|
20053189
|
yes |
guanabenz |
Antihypertensive |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
8263811
|
7903385
|
8819507
|
15265636
|
9050980
|
no |
guanfacine |
ADHD |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1986 |
small molecule |
agonist |
10942848
|
17173664
|
15928018
|
11164065
|
1356794
|
20331927
|
yes |
haloperidol |
psychosis |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1986 |
small molecule |
antagonist |
27578530
|
yes |
haloperidol |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1967 |
small molecule |
antagonist |
15894081
|
16132064
|
17134027
|
11752352
|
16730699
|
17316700
|
7520908
|
20643630
|
yes |
hexocyclium |
digestive system disease |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
8075869
|
no |
hexocyclium |
digestive system disease |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
8075869
|
no |
histamine |
Anti-migraine |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1939 |
small molecule |
agonist |
16648669
|
17114052
|
17222324
|
17336292
|
17478759
|
no |
histamine |
for diagnosis of gastric acid secretory function |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1939 |
small molecule |
agonist |
17334413
|
17359382
|
11752352
|
no |
histrelin |
Antineoplastic |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1991 |
small molecule |
agonist |
10969915
|
9177416
|
yes |
homatropine methylbromide |
GI Anti-Ulcer ; Antimuscarinics |
acm5_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
no |
homatropine methylbromide |
GI Anti-Ulcer ; Antimuscarinics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
20085574
|
11124384
|
no |
homatropine methylbromide |
GI Anti-Ulcer ; Antimuscarinics |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
2612581
|
20085574
|
11124384
|
no |
homatropine methylbromide |
GI Anti-Ulcer ; Antimuscarinics |
acm4_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
6893558
|
no |
homatropine methylbromide |
GI Anti-Ulcer ; Antimuscarinics |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
6893558
|
11124384
|
no |
icosapent |
hypertriglyceridemia |
ffar1_human |
secondary |
Class A (Rhodopsin) |
Free fatty acid receptors |
approved |
4 |
- |
- |
small molecule |
agonist |
16214394
|
no |
hydrocodone |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1943 |
small molecule |
agonist |
11752352
|
10640321
|
16291875
|
2849950
|
14600248
|
20665209
|
18606504
|
no |
irbesartan |
Antihypertensive |
agtr1_human |
primary |
Class A (Rhodopsin) |
Angiotensin receptors |
approved |
4 |
- |
1997 |
small molecule |
antagonist |
11752352
|
17408613
|
15030294
|
11486244
|
14716205
|
7843749
|
10069682
|
10075381
|
10082498
|
10373224
|
10822210
|
18627212
|
15101793
|
yes |
iloperidone |
Antipsychotic ; atypical |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
8997630
|
12861482
|
no |
iloperidone |
Antipsychotic ; atypical |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2009 |
small molecule |
antagonist |
8997630
|
12861482
|
no |
hydrocodone |
Analgesics |
oprd_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1943 |
small molecule |
agonist |
16291875
|
14600248
|
11752352
|
no |
hydromorphone |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1984 |
small molecule |
agonist |
11869661
|
12479250
|
11305075
|
18789923
|
yes |
hydromorphone |
Analgesics |
oprk_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1984 |
small molecule |
agonist |
17139284
|
17016423
|
16433932
|
yes |
hydromorphone |
Analgesics |
oprd_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1984 |
small molecule |
agonist |
9301669
|
2849950
|
7511163
|
17658959
|
2478994
|
11752352
|
yes |
hydroxyzine |
Antipruritics; Anxiolytics sedatives and hypnotics |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1956 |
small molecule |
antagonist |
11752352
|
17222324
|
19057127
|
18781943
|
1979798
|
yes |
hyoscyamine |
Antispasmodics |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
- |
small molecule |
antagonist |
17139284
|
17016423
|
11495349
|
no |
hyoscyamine |
Antispasmodics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
- |
small molecule |
antagonist |
17139284
|
17016423
|
9732369
|
no |
iloprost |
Antihypertensive |
pd2r2_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
2004 |
small molecule |
agonist |
9579725
|
yes |
iloprost |
Antihypertensive |
pi2r_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
2004 |
small molecule |
agonist |
11792366
|
1375507
|
17257398
|
17273558
|
2456096
|
15163595
|
20395700
|
19683911
|
19475782
|
yes |
iloprost |
Antihypertensive |
pe2r1_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
2004 |
small molecule |
agonist |
11999132
|
11739243
|
yes |
indacaterol |
Bronchodilator |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2009 |
small molecule |
agonist |
16022567
|
yes |
indoramin |
Antihypertensive |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1993 |
small molecule |
not available |
7536677
|
yes |
indoramin |
Antihypertensive |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1993 |
small molecule |
not available |
7536677
|
yes |
indoramin |
Antihypertensive |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1993 |
small molecule |
not available |
7536677
|
yes |
isoetharine |
Anti-Asthmatic |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1979 |
small molecule |
antagonist |
6125600
|
no |
ipratropium |
chronic obstructive pulmonary disease (COPD) |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1986 |
small molecule |
antagonist |
15987237
|
yes |
ipratropium |
chronic obstructive pulmonary disease (COPD) |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1986 |
small molecule |
antagonist |
15987237
|
yes |
ipratropium |
chronic obstructive pulmonary disease (COPD) |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1986 |
small molecule |
antagonist |
15987237
|
yes |
isoetharine |
Bronchodilator |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1979 |
small molecule |
agonist |
6125600
|
no |
isometheptene |
migraines |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
- |
small molecule |
agonist |
15094323
|
3129549
|
yes |
isometheptene |
Anti-migraine |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1962 |
small molecule |
agonist |
15094323
|
3129549
|
yes |
isopropamide |
digestive system disease |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1957 |
small molecule |
antagonist |
3580704
|
29133
|
no |
isopropamide |
digestive system disease |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1957 |
small molecule |
antagonist |
3580704
|
29133
|
no |
isoproterenol |
cardiovascular ; Anti-Asthmatic |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1956 |
small molecule |
agonist |
10988267
|
no |
isoproterenol |
Bronchodilator ; Cardiotonic |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1956 |
small molecule |
agonist |
10988267
|
no |
isoproterenol |
cardiovascular ; Anti-Asthmatic |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1956 |
small molecule |
agonist |
11791000
|
no |
isoproterenol |
Bronchodilator ; Cardiotonic |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1956 |
small molecule |
agonist |
11791000
|
no |
isothipendyl |
antipruritic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
8546983
|
no |
itraconazole |
Antineoplastic |
smo_human |
primary |
Class F (Frizzled) |
Frizzled |
approved |
4 |
- |
1992 |
small molecule |
antagonist |
20385363
|
yes |
ketobemidone |
Analgesics |
oprd_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
- |
small molecule |
agonist |
8153059
|
no |
ketobemidone |
Analgesics |
oprk_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
- |
small molecule |
agonist |
8153059
|
no |
ketobemidone |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
- |
small molecule |
agonist |
8878254
|
8153059
|
no |
ketotifen |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1999 |
small molecule |
antagonist |
7893266
|
1434122
|
16404130
|
8836617
|
8101246
|
18490184
|
11752352
|
yes |
levobunolol |
Antiglaucomic |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1985 |
small molecule |
antagonist |
11752352
|
6147147
|
11572462
|
7928182
|
1351412
|
2892662
|
2891463
|
yes |
labetalol |
cardiovascular disease |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
6355664
|
yes |
labetalol |
cardiovascular disease |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
6355664
|
yes |
labetalol |
cardiovascular disease |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
6355664
|
yes |
labetalol |
Antihypertensive |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
1361547
|
2907566
|
11752352
|
6355664
|
19879818
|
8104240
|
7684671
|
yes |
labetalol |
Antihypertensive |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
1687367
|
6151824
|
6355664
|
7286847
|
11752352
|
19879818
|
8104240
|
7684671
|
yes |
levobunolol |
Antiglaucomic |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1985 |
small molecule |
antagonist |
2891463
|
7928182
|
10864881
|
11572462
|
1351412
|
2892662
|
yes |
labetalol |
cardiovascular disease |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
2696507
|
10529655
|
yes |
labetalol |
cardiovascular disease |
adrb3_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
2696507
|
10529655
|
yes |
labetalol |
Antihypertensive |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
2696507
|
10529655
|
yes |
labetalol |
Antihypertensive |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1984 |
small molecule |
antagonist |
2696507
|
10529655
|
yes |
lanreotide |
acromegaly |
ssr1_human |
primary |
Class A (Rhodopsin) |
Somatostatin receptors |
approved |
4 |
- |
2007 |
peptide |
agonist |
15103227
|
yes |
lanreotide |
acromegaly |
ssr5_human |
primary |
Class A (Rhodopsin) |
Somatostatin receptors |
approved |
4 |
- |
2007 |
peptide |
agonist |
26416534
|
yes |
lanreotide |
Antineoplastic |
ssr2_human |
primary |
Class A (Rhodopsin) |
Somatostatin receptors |
approved |
4 |
- |
2007 |
peptide |
agonist |
26416534
|
yes |
levocabastine |
Anti-Allergic |
ntr2_human |
primary |
Class A (Rhodopsin) |
Neurotensin receptors |
approved |
4 |
- |
1993 |
small molecule |
antagonist |
11723247
|
8647296
|
9080465
|
yes |
levocabastine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1993 |
small molecule |
antagonist |
11752352
|
10631382
|
8647296
|
9627096
|
9551716
|
11915520
|
yes |
latanoprost |
Antiglaucomic |
pf2r_human |
primary |
Class A (Rhodopsin) |
Prostanoid receptors |
approved |
4 |
- |
1996 |
small molecule |
agonist |
16249494
|
14646172
|
15037111
|
9733584
|
12204699
|
11752352
|
yes |
leuprolide |
Antineoplastic |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1985 |
peptide |
agonist |
16809153
|
10687850
|
9625809
|
15758569
|
10394541
|
no |
levocetirizine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
2007 |
small molecule |
antagonist |
21639816
|
18336052
|
yes |
leuprolide |
Antineoplastic ; endometriosis |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1985 |
peptide |
agonist |
16809153
|
10687850
|
9625809
|
15758569
|
10394541
|
no |
leuprolide |
Alzheimer's disease |
gnrhr_human |
primary |
Class A (Rhodopsin) |
Gonadotrophin-releasing hormone receptors |
approved |
4 |
- |
1985 |
peptide |
agonist |
16809153
|
10687850
|
9625809
|
15758569
|
10394541
|
no |
levallorphan |
Opiate Antagonists |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
8968334
|
7723747
|
9016350
|
8819494
|
9862398
|
no |
levodopa |
Antiparkinson |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1993 |
small molecule |
agonist |
17553470
|
15710490
|
15824260
|
15728856
|
18549347
|
11978145
|
9633680
|
yes |
levodopa |
Antiparkinson |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2015 |
small molecule |
agonist |
17553470
|
15710490
|
15824260
|
15728856
|
18549347
|
11978145
|
9633680
|
yes |
levomepromazine |
psychosis |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
2870716
|
yes |
levomepromazine |
psychosis |
drd4_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
2870716
|
yes |
levomepromazine |
psychosis |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
10741754
|
yes |
levodopa |
Antiparkinson |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1993 |
small molecule |
agonist |
18549347
|
11978145
|
9633680
|
yes |
levodopa |
Antiparkinson |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1993 |
small molecule |
agonist |
18549347
|
11978145
|
9633680
|
yes |
levodopa |
Antiparkinson |
drd4_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1993 |
small molecule |
agonist |
18549347
|
11978145
|
9633680
|
yes |
levodopa |
Antiparkinson |
drd5_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1993 |
small molecule |
agonist |
18549347
|
11978145
|
9633680
|
yes |
levomepromazine |
schizophrenia |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
10741754
|
yes |
levodopa |
Antiparkinson |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2015 |
small molecule |
agonist |
18549347
|
11978145
|
9633680
|
yes |
levodopa |
Antiparkinson |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2015 |
small molecule |
agonist |
18549347
|
11978145
|
9633680
|
yes |
levodopa |
Antiparkinson |
drd4_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2015 |
small molecule |
agonist |
18549347
|
11978145
|
9633680
|
yes |
levodopa |
Antiparkinson |
drd5_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2015 |
small molecule |
agonist |
18549347
|
11978145
|
9633680
|
yes |
levomepromazine |
schizophrenia |
5ht2b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
15701205
|
yes |
levomethadyl acetate |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1993 |
small molecule |
agonist |
9360954
|
2471291
|
10911931
|
11561100
|
11752352
|
no |
levonordefrin |
decongestant |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
19326476
|
no |
levonordefrin |
nasal decongestant |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1960 |
small molecule |
agonist |
19326476
|
no |
levorphanol |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1953 |
small molecule |
agonist |
12975489
|
17039381
|
no |
levosalbutamol |
Anti-Asthmatic |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1999 |
small molecule |
agonist |
21453221
|
no |
liraglutide |
Antidiabetic |
glp1r_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
2009 |
protein |
agonist |
14678021
|
18333889
|
yes |
liraglutide |
Antidiabetic |
glp1r_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
2010 |
protein |
agonist |
14678021
|
18333889
|
yes |
lisuride |
Antiparkinson |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2011 |
small molecule |
agonist |
11224054
|
18691132
|
12373423
|
1678728
|
1783326
|
2887435
|
no |
lisdexamfetamine |
Central Nervous System Stimulants |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2007 |
small molecule |
antagonist |
17016423
|
11752352
|
yes |
lisdexamfetamine |
Central Nervous System Stimulants |
taar1_human |
primary |
Class A (Rhodopsin) |
Trace amine receptors |
approved |
4 |
- |
2007 |
small molecule |
antagonist |
17016423
|
11752352
|
yes |
lisuride |
Antiparkinson |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2011 |
small molecule |
agonist |
11752352
|
18691132
|
no |
lisuride |
Antiparkinson |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2011 |
small molecule |
agonist |
17139284
|
17016423
|
18691132
|
no |
lixisenatide |
Antidiabetic |
glp1r_human |
primary |
Class B1 (Secretin) |
Glucagon receptor family |
approved |
4 |
- |
2016 |
small molecule |
agonist |
25119443
|
yes |
lofexidine |
opiate withdrawal |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2006 |
small molecule |
agonist |
1357064
|
10598217
|
yes |
lofexidine |
opiate withdrawal |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2006 |
small molecule |
agonist |
1357064
|
10598217
|
yes |
lofexidine |
opiate withdrawal |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
2006 |
small molecule |
agonist |
1357064
|
10598217
|
10882840
|
yes |
loperamide |
Antidiuretic |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1976 |
small molecule |
agonist |
10087042
|
14592702
|
8488368
|
11752352
|
6319884
|
18284554
|
yes |
morphine |
Analgesics |
oprk_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2002 |
small molecule |
agonist |
17139284
|
17016423
|
9808678
|
7959748
|
16753266
|
yes |
loratadine |
Anti-Asthmatic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1993 |
small molecule |
antagonist |
11752352
|
1303772
|
7581058
|
8174605
|
10597865
|
15942272
|
1303773
|
9444440
|
1977506
|
11291777
|
yes |
lorcaserin |
Anti-obesity |
5ht2c_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2012 |
small molecule |
agonist |
16625817
|
16259227
|
no |
losartan |
Antihypertensive ; for Diabetic neuropathy |
agtr1_human |
primary |
Class A (Rhodopsin) |
Angiotensin receptors |
approved |
4 |
- |
1995 |
small molecule |
antagonist |
11752352
|
15026875
|
15991937
|
12710529
|
12719755
|
15573751
|
yes |
losartan |
Antihypertensive |
agtr1_human |
primary |
Class A (Rhodopsin) |
Angiotensin receptors |
approved |
4 |
- |
1995 |
small molecule |
antagonist |
11752352
|
15026875
|
15991937
|
12710529
|
12719755
|
15573751
|
yes |
loxapine |
schizophrenia |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1975 |
small molecule |
antagonist |
12664192
|
yes |
loxapine |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1975 |
small molecule |
antagonist |
6239298
|
15694653
|
9570468
|
8101879
|
9342550
|
8665533
|
11752352
|
yes |
mepenzolate |
digestive system disease |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1956 |
small molecule |
antagonist |
7623487
|
2791613
|
7122991
|
yes |
mepenzolate |
digestive system disease |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1956 |
small molecule |
antagonist |
7623487
|
2791613
|
7122991
|
yes |
meperidine, pethidine |
Analgesics |
oprk_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1942 |
small molecule |
agonist |
28625303
|
26732307
|
no |
lurasidone |
schizophrenia |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
2010 |
small molecule |
antagonist |
23545936
|
yes |
lurasidone |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2010 |
small molecule |
antagonist |
23545936
|
yes |
lutropin alfa |
Fertility |
lshr_human |
primary |
Class A (Rhodopsin) |
Glycoprotein hormone receptors |
approved |
4 |
- |
2004 |
peptide |
agonist |
17139284
|
17016423
|
20161981
|
11752352
|
yes |
macitentan |
cardiovascular disease |
ednra_human |
primary |
Class A (Rhodopsin) |
Endothelin receptors |
approved |
4 |
- |
2013 |
small molecule |
antagonist |
22862294
|
22458347
|
24261583
|
yes |
macitentan |
cardiovascular disease |
ednrb_human |
primary |
Class A (Rhodopsin) |
Endothelin receptors |
approved |
4 |
- |
2013 |
small molecule |
antagonist |
22862294
|
22458347
|
24261583
|
yes |
maraviroc |
antiviral ; HIV |
ccr5_human |
primary |
Class A (Rhodopsin) |
Chemokine receptors |
approved |
4 |
- |
2007 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
19098484
|
19692476
|
16298345
|
yes |
marinol |
Antiemetics |
cnr1_human |
primary |
Class A (Rhodopsin) |
Cannabinoid receptors |
approved |
4 |
- |
1985 |
small molecule |
agonist |
17828291
|
no |
meclizine |
Antiemetics |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1957 |
small molecule |
antagonist |
7513381
|
1350745
|
1362160
|
1678430
|
no |
melatonin |
Hypnotics and Sedatives |
mtr1a_human |
primary |
Class A (Rhodopsin) |
Melatonin |
approved |
4 |
- |
2005 |
small molecule |
agonist |
19463840
|
11752352
|
15992934
|
19449447
|
20827520
|
20674373
|
19966183
|
yes |
melatonin |
Hypnotics and Sedatives |
mtr1b_human |
primary |
Class A (Rhodopsin) |
Melatonin |
approved |
4 |
- |
2005 |
small molecule |
agonist |
19463840
|
15992934
|
19449447
|
20827520
|
20674373
|
19966183
|
yes |
methacholine |
Anti-Asthmatic |
acm3_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1986 |
small molecule |
agonist |
20888332
|
20347047
|
19951374
|
19460789
|
no |
methadone |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1947 |
small molecule |
agonist |
17139284
|
17016423
|
11933204
|
17850768
|
14991152
|
yes |
melevodopa |
Antiparkinson |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2000 |
small molecule |
agonist |
20302892
|
no |
melevodopa |
Antiparkinson |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2000 |
small molecule |
agonist |
20302892
|
no |
melevodopa |
Antiparkinson |
drd3_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2000 |
small molecule |
agonist |
20302892
|
no |
melevodopa |
Antiparkinson |
drd4_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2000 |
small molecule |
agonist |
20302892
|
no |
melevodopa |
Antiparkinson |
drd5_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
2000 |
small molecule |
agonist |
20302892
|
no |
menotropins, menotrophin |
Fertility |
lshr_human |
primary |
Class A (Rhodopsin) |
Glycoprotein hormone receptors |
approved |
4 |
- |
1975 |
protein |
agonist |
17139284
|
17016423
|
14680547
|
7872378
|
no |
menotropins, menotrophin |
Fertility |
fshr_human |
primary |
Class A (Rhodopsin) |
Glycoprotein hormone receptors |
approved |
4 |
- |
1975 |
protein |
agonist |
17139284
|
17016423
|
14680547
|
7872378
|
11752352
|
no |
methadyl acetate |
Analgesics |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
1993 |
small molecule |
agonist |
20163389
|
6268422
|
19153939
|
11752352
|
no |
methamphetamine |
neuroprotectant |
taar1_human |
secondary |
Class A (Rhodopsin) |
Trace amine receptors |
approved |
4 |
- |
1943 |
small molecule |
agonist |
17888514
|
11459929
|
17218486
|
17234900
|
17212650
|
17234899
|
15764732
|
no |
mephentermine |
cardiovascular disease |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1951 |
small molecule |
agonist |
21182601
|
5334234
|
no |
mephentermine |
cardiovascular disease |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1951 |
small molecule |
agonist |
21182601
|
5334234
|
no |
mephentermine |
cardiovascular disease |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1951 |
small molecule |
agonist |
21182601
|
5334234
|
no |
mephentermine |
cardiovascular disease |
ada2b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1951 |
small molecule |
agonist |
21182601
|
5334234
|
no |
mephentermine |
cardiovascular disease |
ada2c_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1951 |
small molecule |
agonist |
21182601
|
5334234
|
no |
mephentermine |
cardiovascular disease |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1951 |
small molecule |
agonist |
21182601
|
5334234
|
no |
mephentermine |
cardiovascular disease |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1951 |
small molecule |
agonist |
21182601
|
5334234
|
no |
mephentermine |
cardiovascular disease |
adrb3_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1951 |
small molecule |
agonist |
21182601
|
5334234
|
no |
mephentermine |
Antihypotensive ; Vasoconstrictor |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1951 |
small molecule |
agonist |
21182601
|
5334234
|
no |
mequitazine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
9454781
|
7650688
|
8808167
|
7511558
|
12244568
|
6418550
|
11752352
|
no |
mesoridazine |
schizophrenia |
drd2_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1970 |
small molecule |
antagonist |
11752352
|
16135699
|
15357957
|
no |
mesoridazine |
schizophrenia |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1970 |
small molecule |
antagonist |
15357957
|
11561066
|
10991983
|
no |
metaproterenol, orciprenaline |
Anti-Asthmatic |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1973 |
small molecule |
agonist |
10490901
|
3168573
|
2870555
|
8760245
|
10973730
|
11752352
|
no |
metaraminol |
Antihypotensive ; Vasoconstrictor |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1954 |
small molecule |
agonist |
17139284
|
17016423
|
9663612
|
no |
methantheline |
GI Anti-Ulcer ; anticholinergic; Antispasmodics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1951 |
small molecule |
antagonist |
17139284
|
17016423
|
no |
methamphetamine |
neuroprotectant |
ada2b_human |
secondary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1943 |
small molecule |
agonist |
9551769
|
15955613
|
no |
methamphetamine |
neuroprotectant |
ada2c_human |
secondary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1943 |
small molecule |
agonist |
9551769
|
15955613
|
no |
methamphetamine |
neuroprotectant |
ada2a_human |
secondary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1943 |
small molecule |
agonist |
9551769
|
15955613
|
12453616
|
no |
methantheline |
digestive system disease |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1951 |
small molecule |
antagonist |
6116801
|
no |
methdilazine |
Anti-Allergic |
hrh1_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
1982 |
small molecule |
antagonist |
17139284
|
17016423
|
11752352
|
9700532
|
20012879
|
no |
methoxamine |
cardiovascular disease |
ada1d_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
19493707
|
no |
methoxamine |
Antihypotensive ; Vasoconstrictor |
ada1b_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
2546049
|
2988814
|
8635240
|
11752352
|
11331292
|
no |
methoxamine |
Antihypotensive ; Vasoconstrictor |
ada1a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1982 |
small molecule |
agonist |
7875228
|
1978244
|
1680715
|
7511752
|
8986981
|
no |
methyldopa |
Antihypertensive |
ada2a_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1962 |
small molecule |
agonist |
17139284
|
17016423
|
17485976
|
9284427
|
10415926
|
8743022
|
1363322
|
14557373
|
yes |
methylergonovine |
Abortifacient |
drd1_human |
primary |
Class A (Rhodopsin) |
Dopamine receptors |
approved |
4 |
- |
1946 |
small molecule |
partial agonist |
15930499
|
no |
methylnaltrexone |
opioid-induced constipation |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2008 |
small molecule |
antagonist |
17504835
|
yes |
methylnaltrexone |
OIC treatment |
oprm_human |
primary |
Class A (Rhodopsin) |
Opioid receptors |
approved |
4 |
- |
2008 |
small molecule |
antagonist |
17504835
|
yes |
methylscopolamine, methscopolamine |
Anti-ulcer |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1953 |
small molecule |
antagonist |
17139284
|
17016423
|
20590642
|
no |
methylscopolamine, methscopolamine |
Antispasmodics |
acm1_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1953 |
small molecule |
antagonist |
17139284
|
17016423
|
20590642
|
no |
methylscopolamine |
Anti-ulcer |
acm2_human |
primary |
Class A (Rhodopsin) |
Acetylcholine receptors (muscarinic) |
approved |
4 |
- |
1953 |
small molecule |
antagonist |
19565307
|
11752352
|
no |
methysergide |
Anti-migraine |
5ht2b_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1962 |
small molecule |
antagonist |
8743744
|
yes |
methysergide |
Anti-migraine s; Vasoconstrictor |
5ht7r_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1962 |
small molecule |
antagonist |
14501155
|
yes |
methysergide |
Anti-migraine s; Vasoconstrictor |
5ht2a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1962 |
small molecule |
antagonist |
10080233
|
10455282
|
11061982
|
11704657
|
11720080
|
yes |
methysergide |
Anti-migraine s; Vasoconstrictor |
5ht1a_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1962 |
small molecule |
antagonist |
11049861
|
14501155
|
14517765
|
14581123
|
1838579
|
yes |
methysergide |
Anti-migraine s; Vasoconstrictor |
5ht2c_human |
primary |
Class A (Rhodopsin) |
5-Hydroxytryptamine receptors |
approved |
4 |
- |
1962 |
small molecule |
antagonist |
11752352
|
12555241
|
yes |
metiamide |
acid reducer |
hrh2_human |
primary |
Class A (Rhodopsin) |
Histamine receptors |
approved |
4 |
- |
- |
small molecule |
antagonist |
7725982
|
no |
metipranolol |
Anti-Arrhythmia ; Antihypertensive ; Anti-glaucoma |
adrb1_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1989 |
small molecule |
antagonist |
17139284
|
17016423
|
2895037
|
12967722
|
2885244
|
yes |
metipranolol |
Anti-Arrhythmia ; Antihypertensive ; Anti-glaucoma |
adrb2_human |
primary |
Class A (Rhodopsin) |
Adrenoceptors |
approved |
4 |
- |
1989 |
small molecule |
antagonist |