GPCRdb

Ligand source activities (1 row/activity)

Potency
Affinity

Get vendors

Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Potency)	# tested GPCRs (Potency)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	11337	2883	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Measuring β-arrestin recruitment using the PathHunter assay system.Measuring β-arrestin recruitment using the PathHunter assay system.	Guide to Pharmacology	440	4	0	4	3.9	O=c1c2CN(CCc2n2c(=NCC2)n1Cc1ccc(cc1)C(F)(F)F)Cc1ccccc1	31127149
	124085867	2883	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Measuring β-arrestin recruitment using the PathHunter assay system.Measuring β-arrestin recruitment using the PathHunter assay system.	Guide to Pharmacology	440	4	0	4	3.9	O=c1c2CN(CCc2n2c(=NCC2)n1Cc1ccc(cc1)C(F)(F)F)Cc1ccccc1	31127149
	5312830	187	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology	296	14	2	2	4.9	CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O	16236715
	5567	187	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology	296	14	2	2	4.9	CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O	16236715
	CHEMBL1230670	187	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology	296	14	2	2	4.9	CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O	16236715
	DB07302	187	0	None	-	1	Human	5.7	pEC50	=	5.7	Functional	UnclassifiedUnclassified	Guide to Pharmacology	296	14	2	2	4.9	CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O	16236715
	12945	2825	0	None	-	1	Human	7.3	pEC50	=	7.3	Functional	UnclassifiedUnclassified	Guide to Pharmacology	351	6	2	4	4.0	CC1=C(OC2=C1C=C(NC(=O)CCC(=O)C3=CC=CC=C3)C=C2)C(O)=O	37770763
	12944	2824	0	None	-	1	Human	7.8	pIC50	=	7.8	Functional	Efficacy 90%Efficacy 90%	Guide to Pharmacology	359	6	2	4	3.0	CC1=C(OC2=C1C=C(C=C2)S(=O)(=O)NCCC3=CC=CC=C3)C(O)=O	37770763
	4319354	2824	0	None	-	1	Human	7.8	pIC50	=	7.8	Functional	Efficacy 90%Efficacy 90%	Guide to Pharmacology	359	6	2	4	3.0	CC1=C(OC2=C1C=C(C=C2)S(=O)(=O)NCCC3=CC=CC=C3)C(O)=O	37770763

Get vendors

Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Affinity)	# tested GPCRs (Affinity)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI