GPCRdb

Ligand source activities (1 row/activity)

Potency
Affinity

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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Potency)	# tested GPCRs (Potency)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	10321	1675	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	In a TCF/LEF reporter assay with WRE-GFP constructs.In a TCF/LEF reporter assay with WRE-GFP constructs.	Guide to Pharmacology	322	3	4	3	3.9	O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O	29293331
	137553171	1675	0	None	-	1	Human	6.4	pEC50	=	6.4	Functional	In a TCF/LEF reporter assay with WRE-GFP constructs.In a TCF/LEF reporter assay with WRE-GFP constructs.	Guide to Pharmacology	322	3	4	3	3.9	O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O	29293331
	10321	1675	0	None	-	1	Human	6.7	pIC50	=	6.7	Functional	In TCF/LEF reporter assays with WRE-GFP constructsIn TCF/LEF reporter assays with WRE-GFP constructs	Guide to Pharmacology	322	3	4	3	3.9	O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O	25751279
	137553171	1675	0	None	-	1	Human	6.7	pIC50	=	6.7	Functional	In TCF/LEF reporter assays with WRE-GFP constructsIn TCF/LEF reporter assays with WRE-GFP constructs	Guide to Pharmacology	322	3	4	3	3.9	O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O	25751279
	10322	1674	0	None	-	1	Human	6.2	pIC50	=	6.2	Functional	In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs.	Guide to Pharmacology	360	3	3	3	5.9	O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1	25751279
	10322	1674	0	None	-	1	Human	6.2	pIC50	=	6.2	Functional	In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs.	Guide to Pharmacology	360	3	3	3	5.9	O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1	29293331
	90478321	1674	0	None	-	1	Human	6.2	pIC50	=	6.2	Functional	In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs.	Guide to Pharmacology	360	3	3	3	5.9	O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1	25751279
	90478321	1674	0	None	-	1	Human	6.2	pIC50	=	6.2	Functional	In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs.	Guide to Pharmacology	360	3	3	3	5.9	O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1	29293331

Get vendors

Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Affinity)	# tested GPCRs (Affinity)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	2947	2822	0	None	-	1	Mouse	8.4	pKd	None	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	15035989