PDB
Resolution
3.3 Å
Released
Aug. 27, 2025
Receptor
Class
A
Species
Homo sapiens
Ligand
I-BOP
Function
Agonist
Reference
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Ligand Amino Acid Generic Number Segment Interaction Type
I-BOP A31 1.39x39 TM1 hydrophobic
I-BOP L78 2.54x54 TM2 hydrophobic
I-BOP V85 2.61x61 TM2 hydrophobic
I-BOP H89 2.65x65 TM2 polar (hydrogen bond)
I-BOP H89 2.65x65 TM2 Van der Waals
I-BOP M112 3.32x32 TM3 Van der Waals
I-BOP G116 3.36x36 TM3 Van der Waals
I-BOP S181 ECL2 Van der Waals
I-BOP W182 ECL2 hydrophobic
I-BOP W182 ECL2 Van der Waals
I-BOP F184 45.51x51 ECL2 Van der Waals
I-BOP W258 6.48x48 TM6 hydrophobic
I-BOP W258 6.48x48 TM6 Van der Waals
I-BOP L291 7.36x35 TM7 Van der Waals
I-BOP L294 7.39x38 TM7 hydrophobic
I-BOP L294 7.39x38 TM7 Van der Waals
I-BOP R295 7.40x39 TM7 Van der Waals
I-BOP T298 7.43x42 TM7 Van der Waals
I-BOP Q301 7.46x46 TM7 Van der Waals

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Snake plot — Download: PNG | SVG
ICL1 G G S H T R ICL1ECL1 L F E W H A V D P G ECL1ICL2 P F S R P A V A ICL2ECL2 V G R Y T V Q Y P G S W C F L T L G A ECL2ICL3 E A A Q ICL3ECL3 N P P A M S P A G Q L ECL3N-term M W P N G S S L G P C F R P T N I T L E E R R L I A N-termC-term L Q P Q L T Q R S G L Q C-term S P W F A A S F C V V G L A S N L L A L S V L A G A R Q S S F L T F L C G L V L T D F L G L L V T G T I V V S Q H A A C R L C R F M G V V M I F F G L S P L L L G A A M A S E R Y L G I T R S Q R R A W A T V G L V W A A A L A L G L L P L L G E S G D V A F G L L F S M L G G L S V G L S F L L N T V S V A T L C H V Y H G Q Q R P R D S E V E M M A Q L L G I M V V A S V C W L P L L V F I A Q T V L R S R T T E K E L L I Y L R V A T W N Q I L D P W V Y I L F R R A L Q P R P R V L R R R L S T S L S
Helix box plot — Download: PNG | SVG L N S A L G V V C F S A A F W P S 1 C G L V L T D F L G L L V T G T I V V S 2 A A G L L L P S L G F F I M V V G M F R 3 A W A T V G L V W A A A L A L G L L P L 4 N L L F S L G V S L G G L M S F L L G F 5 L G I M V V A S V C W L P L L V F I A Q 6 W P D L I Q N W T A V R L Y I L L E K 7

GPCRdb(A)
GPCRdb(A)
TP receptor
TM1
1x39 1.39x39 A31
TM2
2x54 2.54x54 L78
2x61 2.61x61 V85
2x65 2.65x65 H89
TM3
3x32 3.32x32 M112
3x36 3.36x36 G116
ECL2
45x51 45.51x51 F184
TM6
6x48 6.48x48 W258
TM7
7x35 7.36x35 L291
7x38 7.39x38 L294
7x39 7.40x39 R295
7x42 7.43x42 T298
7x46 7.46x46 Q301