PDB
Resolution
2.9 Å
Released
March 4, 2026
Receptor
Class
A
Species
Homo sapiens
Ligand
Function
oridonin
Agonist
Reference
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Ligand Amino Acid Generic Number Segment Interaction Type
oridonin R127 3.32x32 TM3 hydrophobic
oridonin V131 3.36x36 TM3 Van der Waals
oridonin E182 4.60x61 TM4 Van der Waals
oridonin C221 5.42x43 TM5 hydrophobic
oridonin F222 5.43x44 TM5 Van der Waals
oridonin F225 5.46x461 TM5 hydrophobic
oridonin N287 6.51x51 TM6 polar (hydrogen bond)
oridonin H288 6.52x52 TM6 Van der Waals
oridonin Y291 6.55x55 TM6 hydrophobic
oridonin R316 7.39x38 TM7 Van der Waals

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Snake plot — Download: PNG | SVG
ICL1 K S M Q ICL1ECL1 E G W L F ECL1ICL2 P L E R Q P S N ICL2ECL2 N V Y T F R D P N K N M T F E S C T S Y P V S ECL2ICL3 P T E E Q S ICL3ECL3 Q T Y V D P ECL3N-term M A Q R Q P H S P N Q T L I S I T N D T E S S S S V V S N D N T N K G W S G D N S P G N-termC-term C C K A E R P E P P V A D T S L T T L A V M G T V P G T G S I Q M S E I S V T S F T G C S V K Q A E D R F C-term I E A L C A I Y I T Y A V I I S V G I L G N A I L I K V F F K T T V P N I F I T S L A F G D L L L L L T C V P V D A T H Y L A G R I G C K V L S F I R L T S V G V S V F T L T I L S A D R Y K A V V K A I L K T C V K A G C V W I V S M I F A L P E A I F S K K L L Q E I H S L L C F L V F Y I I P L S I I S V Y Y S L I A R T L Y K S T L N I H A R K Q I E S R K R I A R T V L V L V A L F A L C W L P N H L L Y L Y H S F T S S A M H F I F T I F S R V L A F S N S C V N P F A L Y W L S K S F K A F Q K H Q L F
Helix box plot — Download: PNG | SVG A N G L I G V S I I V A Y T I Y I A C L 1 T S L A F G D L L L L T L C V P V D A T H 2 I T L T F V S V G V S T L R I F S L V K 3 T C V K A G C V W I V S M I F A L P E 4 Y Y V S I I S L P I I Y F V L F C L L S H 5 L V L V A L F A L C W L P N H L L Y L Y 6 F P N V C S N S F A L V R S F I T F I 7

GPCRdb(A)
GPCRdb(A)
BB3 receptor
TM3
3x32 3.32x32 R127
3x36 3.36x36 V131
TM4
4x61 4.60x61 E182
TM5
5x43 5.42x43 C221
5x44 5.43x44 F222
5x461 5.46x461 F225
TM6
6x51 6.51x51 N287
6x52 6.52x52 H288
6x55 6.55x55 Y291
TM7
7x38 7.39x38 R316