PDB
Resolution
2.7 Å
Released
March 4, 2026
Receptor
Class
A
Species
Danio rerio
Ligands
Function
Agmatine (R:402)
Agonist
Agmatine (R:401)
Unknown
Reference
—
Agmatine (R:402) Agmatine (R:401)

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Ligand Amino Acid Generic Number Segment Interaction Type
Agmatine (R:402) D112 3.32x32 TM3 polar (hydrogen bond)
Agmatine (R:402) D112 3.32x32 TM3 polar (charge-charge)
Agmatine (R:402) L113 3.33x33 TM3 hydrophobic
Agmatine (R:402) T116 3.36x36 TM3 polar (hydrogen bond)
Agmatine (R:402) S117 3.37x37 TM3 polar (hydrogen bond)
Agmatine (R:402) Y163 4.56x56 TM4 Van der Waals
Agmatine (R:401) Y180 ECL2 Van der Waals
Agmatine (R:401) T191 45.51x51 ECL2 Van der Waals
Agmatine (R:401) L192 45.52x52 ECL2 polar (hydrogen bond with backbone)
Agmatine (R:401) Y193 ECL2 polar (hydrogen bond)
Agmatine (R:401) Y193 ECL2 hydrophobic
Agmatine (R:402) D202 5.42x43 TM5 polar (charge-charge)
Agmatine (R:402) D202 5.42x43 TM5 polar (hydrogen bond)
Agmatine (R:402) T206 5.46x461 TM5 Van der Waals
Agmatine (R:402) W269 6.48x48 TM6 hydrophobic
Agmatine (R:402) W269 6.48x48 TM6 aromatic (pi-cation)
Agmatine (R:402) F272 6.51x51 TM6 hydrophobic
Agmatine (R:402) F273 6.52x52 TM6 Van der Waals
Agmatine (R:401) D279 6.58x58 TM6 polar (charge-charge)
Agmatine (R:401) F284 ECL3 Van der Waals
Agmatine (R:401) V288 7.32x31 TM7 Van der Waals
Agmatine (R:401) F291 7.35x34 TM7 aromatic (pi-cation)
Agmatine (R:402) V295 7.39x38 TM7 Van der Waals

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Snake plot — Download: PNG | SVG
ICL1 K Q L Q ICL1ECL1 C W Y ECL1ICL2 P L Q Y P T M I ICL2ECL2 G L D E Y I Q S M Y C V G G C T L Y F ECL2ICL3 N Q N E I ICL3ECL3 F S T ECL3N-term M D L S S Q E Y D P S Q F C F P A V N N S C L K G T H N-termC-term R R I F E P N S S D I N I F T L C-term H V S T Q T V V Y L I L A S A M T V T I L G N S V V I I S I A H F T T T N I L V M S L A L A D L L L G L V V M P F S M I R S V D G Y G E T F C M L H S S F D L F L T S V S I F H L I F I A V D R H Q A V C F T I P V A W V M V M I S W S M A A L Y S Y G L V Y S K A N M E N A L W S V L D T L I T F F L P C S V M I G L Y A R I F V V A K K H A R I I N E A D G T F K S S R R S E Q K A A K T L G I V V G A F I M C W L P F F I N S L M D P Y I N P V A L F E A F V W L G Y I N S T M N P I I Y G F F Y P W F Y L I R K T L I T
Helix box plot — Download: PNG | SVG S N G L I T V T M A S A L I L Y V V T Q 1 M S L A L A D L L L G V L V M P F S M I R 2 F I L H F I S V S T L F L D F S S H L M 3 A W V M V M I S W S M A A L Y S Y G L V 4 Y L G I M V S C P L F F T I L T D L V S W 5 G I V V G A F I M C W L P F F I N S L M 6 I P N M T S N I Y G L W V F A E F L A 7

GPCRdb(A)
GPCRdb(A)
taar13d
TM3
3x32 3.32x32 D112
3x33 3.33x33 L113
3x36 3.36x36 T116
3x37 3.37x37 S117
TM4
4x56 4.56x56 Y163
ECL2
45x51 45.51x51 T191
45x52 45.52x52 L192
TM5
5x43 5.42x43 D202
5x461 5.46x461 T206
TM6
6x48 6.48x48 W269
6x51 6.51x51 F272
6x52 6.52x52 F273
6x58 6.58x58 D279
TM7
7x31 7.32x31 V288
7x34 7.35x34 F291
7x38 7.39x38 V295