PDB
Resolution
2.4 Å
Released
March 4, 2026
Receptor
Class
A
Species
Mus musculus
Ligand
DAMGO
Function
Agonist
Reference
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Ligand Amino Acid Generic Number Segment Interaction Type
DAMGO V143 3.28x28 TM3 hydrophobic
DAMGO I144 3.29x29 TM3 hydrophobic
DAMGO D147 3.32x32 TM3 polar (charge-assisted hydrogen bond)
DAMGO C217 45.50x50 ECL2 Van der Waals
DAMGO V236 5.42x43 TM5 hydrophobic
DAMGO V236 5.42x43 TM5 Van der Waals
DAMGO I296 6.51x51 TM6 hydrophobic
DAMGO H297 6.52x52 TM6 Van der Waals
DAMGO V300 6.55x55 TM6 hydrophobic
DAMGO V300 6.55x55 TM6 Van der Waals
DAMGO W318 7.35x34 TM7 hydrophobic
DAMGO W318 7.35x34 TM7 Van der Waals
DAMGO Y326 7.43x42 TM7 Van der Waals

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Snake plot — Download: PNG | SVG
ICL1 T K M K ICL1ECL1 T W P F ECL1ICL2 P V K A L D F R ICL2ECL2 T T K Y R Q G S I D C T L T F S H ECL2ICL3 R M L S G ICL3ECL3 T I P E ECL3N-term M D S S A G P G N I S D C S D P L A P A S C S P A P G S W L N L S H V D G N Q S D P C G P N R T G L G G S H S L C P Q T G S P S N-termC-term P T S S T I E Q Q N S A R I R Q N T R E H P S T A N T V D R T N H Q L E N L E A E T A P L P C-term M V T A I T I M A L Y S I V C V V G L F G N F L V M Y V I V R Y T A T N I Y I F N L A L A D A L A T S T L P F Q S V N Y L M G G N I L C K I V I S I D Y Y N M F T S I F T L C T M S V D R Y I A V C H T P R N A K I V N V C N W I L S S A I G L P V M F M A P T W Y W E N L L K I C V F I F A F I M P V L I I T V C Y G L M I L R L K S V S K E K D R N L R R I T R M V L V V V A V F I V C W T P I H I Y V I I K A L I T T F Q T V S W H F C I A L G Y T N S C L N P V L Y A F L D E N F R E F K R C F C I
Helix box plot — Download: PNG | SVG F N G F L G V V C V I S Y L A M I T I A 1 F N L A L A D A L A T S T L P F Q S V N 2 T C L T F I S T F M N Y Y D I S I V I K 3 A K I V N V C N W I L S S A I G L P V M 4 Y C V T I I L V P M I F A F I F V C I K L 5 L V V V A V F I V C W T P I H I Y V I I 6 V P N L C S N T Y G L A I C F H W S V 7

GPCRdb(A)
GPCRdb(A)
μ receptor
TM3
3x28 3.28x28 V143
3x29 3.29x29 I144
3x32 3.32x32 D147
ECL2
45x50 45.50x50 C217
TM5
5x43 5.42x43 V236
TM6
6x51 6.51x51 I296
6x52 6.52x52 H297
6x55 6.55x55 V300
TM7
7x34 7.35x34 W318
7x42 7.43x42 Y326