PDB
Resolution
3.1 Å
Released
May 20, 2026
Receptor
Class
A
Species
Homo sapiens
Ligand
AR234958
Function
Agonist
Reference
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Ligand Amino Acid Generic Number Segment Interaction Type
AR234958 I84 2.57x57 TM2 hydrophobic
AR234958 L87 2.60x60 TM2 hydrophobic
AR234958 Y91 2.64x64 TM2 hydrophobic
AR234958 Y95 ECL1 polar (hydrogen bond)
AR234958 Y95 ECL1 Van der Waals
AR234958 H262 7.35x34 TM7 Van der Waals
AR234958 H263 7.36x35 TM7 Van der Waals
AR234958 L266 7.39x38 TM7 Van der Waals
AR234958 L266 7.39x38 TM7 hydrophobic

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Snake plot — Download: PNG | SVG
ICL1 R R ICL1ECL1 Y E L ECL1ICL2 P I W Y R C H R ICL2ECL2 I D R E E E S H S R N ECL2ICL3 A S H ICL3ECL3 W S T F ECL3N-term M D G S N V T S F V V E E P T N I S T G R N A S V G N A H R Q N-termC-term L T R A F K D E M Q P R R Q K D N C N T V T V E T V V C-term I P I V H W V I M S I S P V G F V E N G I L L W F L C F R M N P F T V Y I T H L S I A D I S L L F C I F I L S I D Y A L D S S G H Y Y T I V T L S V T F L F G Y N T G L Y L L T A I S V E R C L S V L Y P K Y Q S A L V C A L L W A L S C L V T T M E Y V M C D C R A V I I F I A I L S F L V F T P L M L V S S T I L V V K I R K N T W S S K L Y I V I M V T I I I F L I F A M P M R L L Y L L Y Y E Y G N L H H I S L L F S T I N S S A N P F I Y F F V G S S F K E V K K K R S L K V
Helix box plot — Download: PNG | SVG G N E V F G V P S I S M I V W H V I P I 1 T H L S I A D I S L L F C I F I L S I D 2 A T L L Y L G T N Y G F L F T V S L T V 3 S A L V C A L L W A L S C L V T T M E Y 4 I T S S V L M L P T F V L F S L I A I F I 5 M V T I I I F L I F A M P M R L L Y L L 6 F P N A S S N I T S F L L S I H H L N 7

GPCRdb(A)
GPCRdb(A)
MAS1
TM2
2x57 2.57x57 I84
2x60 2.60x60 L87
2x64 2.64x64 Y91
TM7
7x34 7.35x34 H262
7x35 7.36x35 H263
7x38 7.39x38 L266