PDB
Resolution
2.8 Å
Released
July 8, 2026
Receptor
Class
A
Species
Homo sapiens
Ligand
BMS-986187
Function
Ago-PAM
Reference
—

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Ligand Amino Acid Generic Number Segment Interaction Type
BMS-986187 A123 3.27x27 TM3 hydrophobic
BMS-986187 I127 3.31x31 TM3 hydrophobic
BMS-986187 Y130 3.34x34 TM3 hydrophobic
BMS-986187 N131 3.35x35 TM3 polar (hydrogen bond)
BMS-986187 N131 3.35x35 TM3 Van der Waals
BMS-986187 S177 4.54x54 TM4 Van der Waals
BMS-986187 V181 4.58x58 TM4 hydrophobic
BMS-986187 V181 4.58x58 TM4 Van der Waals
BMS-986187 M184 4.61x61 TM4 Van der Waals
BMS-986187 M184 4.61x61 TM4 hydrophobic

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Snake plot — Download: PNG | SVG
ICL1 T K M K ICL1ECL1 T W P F ECL1ICL2 P V K A L D F R ICL2ECL2 V T R P R D G A V V C M L Q F P S ECL2ICL3 R L L S G ICL3ECL3 D I D R R ECL3N-term M E P A P S A G A E L Q P P L F A N A S D A Y P S A C P S A G A N A S G P P N-termC-term P C G R P D P S S F S R A R E A T A R E R V T A C T P S D G P G G G A A A C-term G A R S A S S L A L A I A I T A L Y S A V C A V G L L G N V L V M F G I V R Y T A T N I Y I F N L A L A D A L A T S T L P F Q S A K Y L M E G E L L C K A V L S I D Y Y N M F T S I F T L T M M S V D R Y I A V C H T P A K A K L I N I C I W V L A S G V G V P I M V M A P S W Y W D T V T K I C V F L F A F V V P I L I I T V C Y G L M L L R L R S V S K E K D R S L R R I T R M V L V V V G A F V V C W A P I H I F V I V W T L V D P L V V A A L H L C I A L G Y A N S S L N P V L Y A F L D E N F R Q F K R C L C R K
Helix box plot — Download: PNG | SVG V N G L L G V A C V A S Y L A T I A I A 1 F N L A L A D A L A T S T L P F Q S A K 2 M T L T F I S T F M N Y Y D I S L V A K 3 A K L I N I C I W V L A S G V G V P I M 4 Y C V T I I L I P V V F A F L F V C I K T 5 L V V V G A F V V C W A P I H I F V I V 6 V P N L S S N A Y G L A I C L H L A A 7

GPCRdb(A)
GPCRdb(A)
δ receptor
TM3
3x27 3.27x27 A123
3x31 3.31x31 I127
3x34 3.34x34 Y130
3x35 3.35x35 N131
TM4
4x54 4.54x54 S177
4x58 4.58x58 V181
4x61 4.61x61 M184