BIM 23056


SMILES None
InChIKey None
Sequence FFYWKVFA

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
H3 HRH3 Human Histamine A pKi 8.4 8.8 9.2 Guide to Pharmacology
H3 HRH3 Human Histamine A pKd 9.2 9.2 9.2 Guide to Pharmacology
H4 HRH4 Mouse Histamine A pKi 6.4 6.4 6.4 Guide to Pharmacology
H4 HRH4 Rat Histamine A pKi 6.2 6.2 6.2 Guide to Pharmacology
H3 HRH3 Rat Histamine A pKi 8.0 8.35 8.7 Guide to Pharmacology
H3 HRH3 Mouse Histamine A pKi 8.4 8.4 8.4 Guide to Pharmacology
H4 HRH4 Human Histamine A pKd 7.2 7.2 7.2 Guide to Pharmacology
H4 HRH4 Human Histamine A pKi 6.5 6.7 6.9 Guide to Pharmacology
H3 HRH3 Guinea pig Histamine A pKi 8.82 9.38 10.07 ChEMBL
H3 HRH3 Guinea pig Histamine A pKd 7.8 7.8 7.8 ChEMBL
H4 HRH4 Human Histamine A pKi 6.6 6.73 6.84 ChEMBL
H3 HRH3 Human Histamine A pKi 7.2 8.61 9.26 ChEMBL
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
H3 HRH3 Rat Histamine A pIC50 8.82 8.82 8.82 ChEMBL
H4 HRH4 Human Histamine A pEC50 5.95 6.08 6.2 ChEMBL
H3 HRH3 Human Histamine A pEC50 7.4 8.65 9.5 ChEMBL
H3 HRH3 Human Histamine A pIC50 8.64 8.64 8.64 ChEMBL