[Leu8,des-Arg9]bradykinin
SMILES | None |
InChIKey | BGAPYBBQGHUQNM-YYGRSCHNSA-N |
Sequence | RPPGFSPL |
Chemical properties
Hydrogen bond acceptors | None |
Hydrogen bond donors | None |
Rotatable bonds | None |
Molecular weight (Da) |
Drug properties
Molecular type | Peptide |
Physiological/Surrogate | Surrogate |
Approved drug | No |
Database connections
Bioactivities
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
B1 | BKRB1 | Mouse | Bradykinin | A | pKi | 8.4 | 8.4 | 8.4 | Guide to Pharmacology |
B1 | BKRB1 | Rat | Bradykinin | A | pKi | 7.4 | 7.55 | 7.7 | Guide to Pharmacology |
B1 | BKRB1 | Human | Bradykinin | A | pKi | 6.42 | 6.42 | 6.42 | ChEMBL |
B1 | BKRB1 | Human | Bradykinin | A | pKi | 5.8 | 6.5 | 7.2 | Guide to Pharmacology |
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
B1 | BKRB1 | Mouse | Bradykinin | A | pA2 | 6.9 | 6.9 | 6.9 | Guide to Pharmacology |
B1 | BKRB1 | Mouse | Bradykinin | A | pEC50 | 7.3 | 7.3 | 7.3 | Guide to Pharmacology |