GPCRdb

procainamide

Agent/drug
Bioactivity

procainamide

SMILES	CCN(CC)CCNC(=O)c1ccc(N)cc1
InChIKey	REQCZEXYDRLIBE-UHFFFAOYSA-N

Chemical Properties

Hydrogen bond acceptors	3
Hydrogen bond donors	2
Rotatable bonds	6
Molecular weight (Da)	235.2

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids DrugBank Drug Central GPCRdb

Bioactivities

Affinity
Potency

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

M₂	ACM2	Human	Acetylcholine (muscarinic)	A	pKi	7.81	7.81	7.81	PDSP Ki database
M₂	ACM2	Human	Acetylcholine (muscarinic)	A	pKi	8.11	8.11	8.11	Drug Central

Showing 1 to 2 of 2 entries

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

M₁	ACM1	Rat	Acetylcholine (muscarinic)	A	Potency	5.20	5.20	5.20	ChEMBL
TAS2R9	TA2R9	Human	Taste 2	T2	pEC50	2.55	2.55	2.55	Guide to Pharmacology
TSH	TSHR	Human	Glycoprotein hormone	A	Potency	4.80	4.80	4.80	ChEMBL

Showing 1 to 3 of 3 entries

procainamide

Drug properties

Molecular type	Small molecule
Physiological/Surrogate	Surrogate
Approved drug	Yes

Clinical Trials

Phase I 0

Phase II 0

Phase III 0

Approved No

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids DrugBank Drug Central GPCRdb

Compound is not listed as a drug.