gastrin-17


SMILES None
InChIKey None
Sequence XGPWLEEEEEAYGWMDF

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Endogenous
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
D1 DRD1 Human Dopamine A pKi 7.82 7.99 8.15 ChEMBL
5-HT1A 5HT1A Human 5-Hydroxytryptamine A pKi 5.26 5.26 5.26 PDSP Ki database
D1 DRD1 Human Dopamine A pKi 6.95 6.95 6.95 PDSP Ki database
D2 DRD2 Human Dopamine A pKi 5.0 5.0 5.0 PDSP Ki database
D2 DRD2 Human Dopamine A pKi 5.1 5.8 6.51 ChEMBL
D3 DRD3 Human Dopamine A pKi 5.0 5.55 6.1 PDSP Ki database
5-HT2C 5HT2C Rat 5-Hydroxytryptamine A pKi 5.82 5.82 5.82 PDSP Ki database
D1 DRD1 Rat Dopamine A pKi 8.72 8.72 8.72 PDSP Ki database
D1 DRD1 Rat Dopamine A pKi 8.7 8.7 8.7 Guide to Pharmacology
D2 DRD2 Rat Dopamine A pKi 5.9 5.9 5.9 PDSP Ki database
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
D5 DRD5 Human Dopamine A pEC50 8.85 8.85 8.85 ChEMBL
D1 DRD1 Human Dopamine A pEC50 5.02 6.6 8.33 ChEMBL
TA1 TAAR1 Human Trace amine A pEC50 5.18 5.18 5.18 ChEMBL
GAL3 GALR3 Human Galanin A pIC50 5.42 5.42 5.42 ChEMBL