4-fluorobenzoyl-FGLRW-NH2


SMILES None
InChIKey None
Sequence FGLRW

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
α2A ADA2A Rat Adrenoceptors A pKd 6.59 6.59 6.59 ChEMBL
α2A ADA2A Rat Adrenoceptors A pKi 7.34 7.34 7.34 ChEMBL
α1D ADA1D Rat Adrenoceptors A pKd 8.6 8.7 8.8 ChEMBL
α1D ADA1D Rat Adrenoceptors A pKi 8.2 8.56 8.92 ChEMBL
α1B ADA1B Rat Adrenoceptors A pKd 8.16 8.2 8.21 ChEMBL
α1B ADA1B Rat Adrenoceptors A pKi 7.59 7.84 8.1 ChEMBL
α1A ADA1A Human Adrenoceptors A pKi 9.37 9.45 9.8 ChEMBL
α1D ADA1D Human Adrenoceptors A pKi 9.1 9.3 9.6 ChEMBL
5-HT1A 5HT1A Rat 5-Hydroxytryptamine A pKi 8.14 8.36 8.57 ChEMBL
5-HT1A 5HT1A Human 5-Hydroxytryptamine A pKi 8.68 8.68 8.68 ChEMBL
α1A ADA1A Human Adrenoceptors A pKi 9.7 9.75 9.8 Guide to Pharmacology
α1B ADA1B Human Adrenoceptors A pKi 7.24 8.14 10.42 ChEMBL
α1B ADA1B Human Adrenoceptors A pKi 8.5 8.75 9.0 Guide to Pharmacology
α1D ADA1D Human Adrenoceptors A pKi 9.6 9.6 9.6 Guide to Pharmacology
α2A ADA2A Human Adrenoceptors A pKi 8.46 8.46 8.46 ChEMBL
α2A ADA2A Human Adrenoceptors A pKi 7.6 8.25 8.9 Guide to Pharmacology
α2B ADA2B Human Adrenoceptors A pKi 7.55 7.55 7.55 ChEMBL
α2B ADA2B Human Adrenoceptors A pKi 7.0 7.7 8.4 Guide to Pharmacology
α2C ADA2C Human Adrenoceptors A pKi 9.1 9.1 9.1 ChEMBL
α2C ADA2C Human Adrenoceptors A pKi 8.2 8.8 9.4 Guide to Pharmacology
D3 DRD3 Rat Dopamine A pKi 6.97 6.97 6.97 ChEMBL
α1A ADA1A Rat Adrenoceptors A pKd 9.18 9.37 9.51 ChEMBL
α1A ADA1A Rat Adrenoceptors A pKi 8.89 9.5 10.1 ChEMBL
α1A ADA1A Rat Adrenoceptors A pKi 10.2 10.2 10.2 Guide to Pharmacology
D2 DRD2 Rat Dopamine A pKi 6.91 6.91 6.91 ChEMBL
α1A ADA1A Bovine Adrenoceptors A pKi 9.21 9.3 9.46 ChEMBL
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
α1A ADA1A Human Adrenoceptors A pIC50 9.0 9.0 9.0 ChEMBL