icatibant


SMILES None
InChIKey QURWXBZNHXJZBE-MCDGZUPGSA-N
Sequence RRPXGXSXXR

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug Yes

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
δ OPRD Mouse Opioid A pKi 9.2 9.2 9.2 Guide to Pharmacology
κ OPRK Human Opioid A pKi 8.4 8.4 8.4 Guide to Pharmacology
μ OPRM Human Opioid A pKi 8.8 8.8 8.8 Guide to Pharmacology
δ OPRD Human Opioid A pKi 8.43 8.59 8.74 ChEMBL
δ OPRD Human Opioid A pKi 8.43 8.7 9.18 PDSP Ki database
κ OPRK Human Opioid A pKi 7.26 7.84 8.43 PDSP Ki database
κ OPRK Guinea pig Opioid A pKi 8.15 8.15 8.15 PDSP Ki database
δ A0A286XTF2 Guinea pig Opioid A pKi 8.38 8.38 8.38 PDSP Ki database
μ OPRM Human Opioid A pKi 7.74 8.25 8.77 PDSP Ki database
δ OPRD Human Opioid A pKi 8.4 8.4 8.4 Guide to Pharmacology
μ OPRM Human Opioid A pKi 8.72 8.72 8.72 ChEMBL
κ OPRK Guinea pig Opioid A pKi 7.18 7.32 7.47 ChEMBL
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database