[D-Phe6,β-Ala11,Phe13,Nle14]bombesin-(6-14)
| SMILES | None |
| InChIKey | None |
| Sequence | FQWAVAHFX |
Chemical properties
| Hydrogen bond acceptors | None |
| Hydrogen bond donors | None |
| Rotatable bonds | None |
| Molecular weight (Da) |
Drug properties
| Molecular type | Peptide |
| Physiological/Surrogate | Surrogate |
| Approved drug | No |
Database connections
Bioactivities
| Receptor | Activity | Source | |||||||
|---|---|---|---|---|---|---|---|---|---|
| GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
| BB1 | NMBR | Human | Bombesin | A | pKi | 7.8 | 8.75 | 9.7 | Guide to Pharmacology |
| BB2 | GRPR | Human | Bombesin | A | pKi | 7.82 | 7.91 | 8.0 | Guide to Pharmacology |
| BB3 | BRS3 | Human | Bombesin | A | pKi | 8.05 | 8.21 | 8.38 | Guide to Pharmacology |
| BB3 | BRS3 | Mouse | Bombesin | A | pKi | 8.82 | 8.82 | 8.82 | Guide to Pharmacology |
| BB3 | BRS3 | Rat | Bombesin | A | pKi | 9.0 | 9.0 | 9.0 | Guide to Pharmacology |
| Receptor | Activity | Source | |||||||
|---|---|---|---|---|---|---|---|---|---|
| GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
| BB1 | NMBR | Human | Bombesin | A | pIC50 | 9.49 | 9.59 | 9.68 | Guide to Pharmacology |
| BB2 | GRPR | Human | Bombesin | A | pIC50 | 10.07 | 10.2 | 10.32 | Guide to Pharmacology |