gastrin-releasing peptide
SMILES | None |
InChIKey | BNEIPTFKHBHJBM-XKNFJVFFSA-N |
Sequence | VPLPAGGGTVLTKMYPRGNHWAVGHLM |
Chemical properties
Hydrogen bond acceptors | None |
Hydrogen bond donors | None |
Rotatable bonds | None |
Molecular weight (Da) |
Drug properties
Molecular type | Peptide |
Physiological/Surrogate | Endogenous |
Approved drug | No |
Database connections
Bioactivities
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
BB2 | GRPR | Human | Bombesin | A | pKi | 6.34 | 7.28 | 8.21 | Guide to Pharmacology |
BB2 | GRPR | Rat | Bombesin | A | pKi | 7.74 | 7.74 | 7.74 | Guide to Pharmacology |
BB1 | NMBR | Rat | Bombesin | A | pKi | 6.36 | 6.38 | 6.39 | Guide to Pharmacology |
BB2 | GRPR | Mouse | Bombesin | A | pKi | 8.6 | 8.75 | 8.91 | Guide to Pharmacology |
BB1 | NMBR | Human | Bombesin | A | pKi | 8.04 | 8.04 | 8.04 | ChEMBL |
BB2 | GRPR | Human | Bombesin | A | pKi | 10.4 | 10.4 | 10.4 | ChEMBL |
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
BB2 | GRPR | Human | Bombesin | A | pIC50 | 9.92 | 9.94 | 9.96 | Guide to Pharmacology |