probe 2.1 [PMID: 24187130]



probe 2.1 [PMID: 24187130]


SMILES Cc1ccc(NC(=O)[C@H]2CC=C[C@H]3CCN(c4ccccc4F)C(=O)[C@@H]23)cc1C(F)(F)F
InChIKey LRJGJDKBKCTWKM-HZUJVAHNSA-N

Chemical Properties

Hydrogen bond acceptors 2
Hydrogen bond donors 1
Rotatable bonds 3
Molecular weight (Da) 446.2

Database connections



No bioactivity data available.

probe 2.1 [PMID: 24187130]


Drug properties

Molecular type Small molecule
Physiological/Surrogate Surrogate
Approved drug No

Distribution across phases (no. indications)

Phase I
Phase II
Phase III
Phase IV

Database connections



Compound is not listed as a drug.