Ligand source activities (1 row/activity)





Ligands Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb ID #Vendors Reference
ligand
Fold selectivity
(Potency)
# tested GPCRs
(Potency)
Species p-value
(-log)
Type Activity
Relation
Activity
Value
Assay Type Assay Description Source Mol
weight
Rot
Bonds
H don H acc LogP Smiles DOI
3647 4040 0 None - 1 Human 7.3 pEC50 ~ 7.3 Functional
Measuring Ca<sup>2+</sup> fluxMeasuring Ca<sup>2+</sup> flux
Guide to Pharmacology None None None None 25497737
4370 4041 0 None - 1 Human 7.3 pEC50 ~ 7.3 Functional
Measuring Ca<sup>2+</sup> fluxMeasuring Ca<sup>2+</sup> flux
Guide to Pharmacology None None None None 25497737




Ligands Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb ID #Vendors Reference
ligand
Fold selectivity
(Affinity)
# tested GPCRs
(Affinity)
Species p-value
(-log)
Type Activity
Relation
Activity
Value
Assay Type Assay Description Source Mol
weight
Rot
Bonds
H don H acc LogP Smiles DOI