Ligand source activities (1 row/activity)
Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Potency) |
# tested GPCRs (Potency) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |
1001 | 617 | 95 | None | -11 | 4 | Mouse | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | 121 | 2 | 1 | 1 | 1.2 | NCCc1ccccc1 | 16878137 | ||
2144 | 617 | 95 | None | -11 | 4 | Mouse | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | 121 | 2 | 1 | 1 | 1.2 | NCCc1ccccc1 | 16878137 | ||
CHEMBL610 | 617 | 95 | None | -11 | 4 | Mouse | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | 121 | 2 | 1 | 1 | 1.2 | NCCc1ccccc1 | 16878137 | ||
DB04325 | 617 | 95 | None | -11 | 4 | Mouse | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | 121 | 2 | 1 | 1 | 1.2 | NCCc1ccccc1 | 16878137 |
Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Affinity) |
# tested GPCRs (Affinity) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |