Ligand source activities (1 row/activity)
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
|
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Activity
| Chemical information
| |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
5572 | 1928 | None | 0 | Rat | Functional | pA2 | = | 7.6 | 7.6 | - | 1 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | None | ||||
129631922 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
132274287 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
132451761 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
155817470 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
16132393 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
16133850 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
16133850.0 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
4448 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
4514 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
91933454 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
CHEMBL525610 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
DB06285 | 3781 | None | 9 | Rat | Functional | pIC50 | = | 8.2 | 8.2 | -34 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
129631922 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
132274287 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
132451761 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
155817470 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
16132393 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
16133850 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
16133850.0 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
4448 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
4514 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
91933454 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
CHEMBL525610 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
DB06285 | 3781 | None | 9 | Human | Functional | pIC50 | = | 8.1 | 8.1 | -7 | 4 | NoneNone |
Drug Central | None | None | None | None | None | ||||
155817427 | 3232 | None | 0 | Rat | Functional | pIC50 | = | 5.5 | 5.5 | -158 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
1788 | 3232 | None | 0 | Rat | Functional | pIC50 | = | 5.5 | 5.5 | -158 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
129316189 | 3229 | None | 0 | Rat | Functional | pIC50 | = | 6.8 | 6.8 | -35 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
155817471 | 3229 | None | 0 | Rat | Functional | pIC50 | = | 6.8 | 6.8 | -35 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
16201228 | 3229 | None | 0 | Rat | Functional | pIC50 | = | 6.8 | 6.8 | -35 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
4449 | 3229 | None | 0 | Rat | Functional | pIC50 | = | 6.8 | 6.8 | -35 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
1824 | 2003 | None | 0 | Human | Functional | pIC50 | = | 7 | 7.0 | - | 1 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 10537121 | ||||
155817427 | 3232 | None | 0 | Human | Functional | pIC50 | = | 7.5 | 7.5 | -1 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
155817427 | 3232 | None | 0 | Human | Functional | pIC50 | = | 7.5 | 7.5 | -1 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | ||||
1788 | 3232 | None | 0 | Human | Functional | pIC50 | = | 7.5 | 7.5 | -1 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
1788 | 3232 | None | 0 | Human | Functional | pIC50 | = | 7.5 | 7.5 | -1 | 3 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | ||||
129631922 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
129631922 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | ||||
132274287 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
132274287 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | ||||
132451761 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
132451761 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | ||||
155817470 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
155817470 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | ||||
16132393 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
16132393 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | ||||
16133850 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
16133850 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 | ||||
16133850.0 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 11602681 | ||||
16133850.0 | 3781 | None | 9 | Human | Functional | pIC50 | = | 7.8 | 7.8 | -7 | 4 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 8702701 |
Showing 1 to 50 of 127 entries
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
|
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Activity
| Chemical information
| |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
No data available in table |
Showing 0 to 0 of 0 entries