Ligand source activities (1 row/activity)





Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
AssayType

Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI

5572 1928 0 None - 1 Rat 7.6 pA2 = 7.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None None
129631922 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
132274287 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
132451761 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
155817470 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
16132393 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
16133850 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
4448 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
4514 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
91933454 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
CHEMBL525610 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
DB06285 3781 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
129631922 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
132274287 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
132451761 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
155817470 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
16132393 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
16133850 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
4448 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
4514 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
91933454 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
CHEMBL525610 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
DB06285 3781 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
155817427 3232 0 None -158 3 Rat 5.5 pIC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1788 3232 0 None -158 3 Rat 5.5 pIC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
129316189 3229 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817471 3229 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16201228 3229 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4449 3229 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1824 2003 0 None - 1 Human 7.0 pIC50 = 7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
155817427 3232 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817427 3232 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1788 3232 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1788 3232 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
129631922 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
129631922 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
132274287 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132274287 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
132451761 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132451761 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
155817470 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817470 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
16132393 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16132393 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
16133850 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16133850 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
4448 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4448 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
4514 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4514 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
91933454 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
91933454 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
CHEMBL525610 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
CHEMBL525610 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
DB06285 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
DB06285 3781 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
3624 3826 0 None -5 2 Rat 8.1 pIC50 = 8.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1815 3825 0 None 25 3 Human 8.4 pIC50 = 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
1815 3825 0 None 25 3 Human 8.4 pIC50 = 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
3624 3826 0 None 5 2 Human 8.8 pIC50 = 8.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817432 3233 0 None -446 3 Rat 5.3 pIC50 None 5.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16144017 3233 0 None -446 3 Rat 5.3 pIC50 None 5.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1822 3233 0 None -446 3 Rat 5.3 pIC50 None 5.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817428 3234 0 None -6 2 Human 5.7 pIC50 None 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1790 3234 0 None -6 2 Human 5.7 pIC50 None 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
155817432 3233 0 None -70 3 Human 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16144017 3233 0 None -70 3 Human 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1822 3233 0 None -70 3 Human 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817433 3828 0 None -125 3 Rat 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16134968 3828 0 None -125 3 Rat 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1827 3828 0 None -125 3 Rat 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1825 1996 0 None - 1 Human 6.2 pIC50 None 6.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1820 1497 0 None -10 2 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1807 3104 0 None -5 2 Human 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
129631922 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132274287 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132451761 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817470 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16132393 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16133850 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4448 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4514 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
91933454 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
CHEMBL525610 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
DB06285 3781 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817434 3829 0 None -50 2 Rat 6.5 pIC50 None 6.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1828 3829 0 None -50 2 Rat 6.5 pIC50 None 6.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1794 1930 0 None 19 3 Human 6.6 pIC50 None 6.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
155817429 3235 0 None -3 2 Human 6.7 pIC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1814 3235 0 None -3 2 Human 6.7 pIC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1801 2001 0 None -3 2 Human 6.8 pIC50 None 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1819 1498 0 None -3 2 Human 6.9 pIC50 None 6.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1821 2002 0 None -1 2 Human 7.0 pIC50 None 7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1815 3825 0 None -25 3 Rat 7.0 pIC50 None 7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817433 3828 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
155817433 3828 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16134968 3828 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
16134968 3828 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1827 3828 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1827 3828 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1800 2000 0 None -3 2 Human 7.2 pIC50 None 7.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1820 1497 0 None 10 2 Human 7.3 pIC50 None 7.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1799 1999 0 None -1 2 Human 7.3 pIC50 None 7.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1808 3872 0 None 2 2 Human 7.4 pIC50 None 7.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9360953
1809 3871 0 None 1 2 Human 7.5 pIC50 None 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1798 1998 0 None -1 2 Human 7.6 pIC50 None 7.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1798 1998 0 None -1 2 Human 7.6 pIC50 None 7.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1797 2004 0 None 1 2 Human 7.7 pIC50 None 7.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9360953
155817434 3829 0 None 50 2 Human 8.2 pIC50 None 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1828 3829 0 None 50 2 Human 8.2 pIC50 None 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
129316189 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
129316189 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
129316189 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817471 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
155817471 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
155817471 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16201228 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
16201228 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
16201228 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4449 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
4449 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
4449 3229 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681




Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Similar-
ity
Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
Assay
Type
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI