CCR5

PROTEIN CLASS

Class A (Rhodopsin)

RECEPTOR

PDB CODE

SPECIES

Homo sapiens

RESOLUTION

2.800

PREFERRED CHAIN

B

REFERENCE

PUBLICATION DATE

Oct. 24, 2018

RECEPTOR PDB

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INTERACTING RESIDUES

LIGANDS

N-[(1S)-3-{(3-exo)-3-[3-methyl-5-(propan-2-yl)-4H-1,2,4-triazol-4-yl]-8-azabicyclo[3.2.1]octan-8-yl}-1-(thiophen-2-yl)propyl]cyclopentanecarboxamide - Antagonist pubchem

ENDOGENOUS LIGANDS

CCL14, CCL5, CCL2, CCL4, CCL3, CCL13, CCL8, CCL7, CCL16, CCL11