CRF1 receptor

GPCR CLASS (FAMILY)

Class B1 (Secretin)

PDB CODE

SPECIES

Homo sapiens

RESOLUTION

2.6 Å

PREFERRED CHAIN

A

REFERENCE

PUBLICATION DATE

Sept. 13, 2023

3D VIEW

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LIGAND INTERACTIONS

LIGANDS

7-(4-bromanyl-2,6-dimethoxy-phenyl)-4,8-dimethyl-~{N},~{N}-bis[4,4,4-tris(fluoranyl)butyl]-1$l^{4},3,5,9-tetrazabicyclo[4.3.0]nona-1(6),2,4,8-tetraen-2-amine - Antagonist

ENDOGENOUS LIGANDS

urocortin 1, corticotrophin-releasing hormone, urocortin 2