GPCR CLASS (FAMILY)
Class B1 (Secretin)
PDB CODE
SPECIES
Homo sapiens
RESOLUTION
2.6 Å
PREFERRED CHAIN
A
REFERENCE
PUBLICATION DATE
Sept. 13, 2023
LIGAND INTERACTIONS
LIGANDS
7-(4-bromanyl-2,6-dimethoxy-phenyl)-4,8-dimethyl-~{N},~{N}-bis[4,4,4-tris(fluoranyl)butyl]-1$l^{4},3,5,9-tetrazabicyclo[4.3.0]nona-1(6),2,4,8-tetraen-2-amine - Antagonist
ENDOGENOUS LIGANDS
urocortin 1, corticotrophin-releasing hormone, urocortin 2