GPCR CLASS (FAMILY)
Class A (Rhodopsin)
GPCR SPECIES
Homo sapiens
GPCR PREFERRED CHAIN
r
G PROTEIN (FAMILY)
Gi/o
G PROTEIN SPECIES
Homo sapiens
PDB CODE
RESOLUTION
3.6 Å
PUBLICATION DATE
May 27, 2026
LIGAND INTERACTIONS
LIGANDS
salvinorin A - Agonist pubchem gtoplig chembl_ligand chembl_ligand pubchem chembl_ligand pubchem chembl_ligand pubchem drugbank
PHYSIOLOGICAL LIGANDS
[Met]enkephalin (Human), β-neoendorphin (Human), dynorphin A (Human), dynorphin A-(1-8) (Human), dynorphin A-(1-13) (Human), big dynorphin (Human), β-endorphin (Mouse), β-endorphin (Rat), dynorphin B (Human), β-endorphin (Human), α-neoendorphin (Human), [Leu]enkephalin (Human)