PDB
Resolution
3.2 Å
Released
Jan. 15, 2025
Receptor
Class
A
Species
Homo sapiens
Ligand
Function
CXCL6
Agonist

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Ligand Amino Acid Generic Number Segment Interaction Type
CXCL6 D35 N-term polar (charge-charge)
CXCL6 D35 N-term polar (hydrogen bond)
CXCL6 A36 N-term hydrophobic
CXCL6 A37 N-term Van der Waals
CXCL6 P38 N-term hydrophobic
CXCL6 C39 N-term hydrophobic
CXCL6 C39 N-term polar (hydrogen bond with backbone)
CXCL6 P41 N-term hydrophobic
CXCL6 S43 N-term Van der Waals
CXCL6 K108 2.64x64 TM2 Van der Waals
CXCL6 V187 ECL2 hydrophobic
CXCL6 S189 ECL2 Van der Waals
CXCL6 N191 ECL2 Van der Waals
CXCL6 V192 ECL2 hydrophobic
CXCL6 S193 ECL2 polar (hydrogen bond)
CXCL6 A195 ECL2 Van der Waals
CXCL6 Y197 45.51x51 ECL2 hydrophobic
CXCL6 E198 45.52x52 ECL2 Van der Waals
CXCL6 D199 ECL2 Van der Waals
CXCL6 G201 ECL2 Van der Waals
CXCL6 N202 ECL2 Van der Waals
CXCL6 N203 ECL2 Van der Waals
CXCL6 T204 5.31x32 TM5 Van der Waals
CXCL6 R208 5.35x36 TM5 polar (hydrogen bond)
CXCL6 R208 5.35x36 TM5 polar (charge-charge)
CXCL6 R212 5.39x40 TM5 polar (charge-charge)
CXCL6 D274 6.58x58 TM6 polar (charge-charge)
CXCL6 R278 6.62x62 TM6 polar (hydrogen bond)
CXCL6 R278 6.62x62 TM6 polar (charge-charge)
CXCL6 E284 ECL3 hydrophobic
CXCL6 R289 7.28x27 TM7 polar (hydrogen bond)
CXCL6 D293 7.32x31 TM7 polar (hydrogen bond)
CXCL6 D293 7.32x31 TM7 polar (charge-charge)
CXCL6 L296 7.35x34 TM7 hydrophobic

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Snake plot — Download: PNG | SVG
ICL1 R V G R ICL1ECL1 G W I F ECL1ICL2 A T R T L T Q K R Y ICL2ECL2 R T V Y S S N V S P A C Y E D M G N ECL2ICL3 H M G ICL3ECL3 V I Q E ECL3N-term M E D F N M E S D S F E D F W K G E D L S N Y S Y S S T L P P F L L D A A P C E P E S L N-termC-term G L I S K D S L P K D S R P S F V G S S S G H T S T T L C-term E I N K Y F V V I I Y A L V F L L S L L G N S L V M L V I L Y S S V T D V Y L L N L A L A D L L F A L T L P I W A A S K V N G T F L C K V V S L L K E V N F Y S G I L L L A C I S V D R Y L A I V H L V K F I C L S I W G L S L L L A L P V L L F R N T A N W R M L L R I L P Q S F G F I V P L L I M L F C Y G F T L R T L F K A Q K H R A M R V I F A V V L I F L L C W L P Y N L V L L A D T L M R T Q T C E R R N H I D R A L D A T E I L G I L H S C L N P L I Y A F I G Q K L L K H F R H G I L A I
Helix box plot — Download: PNG | SVG S N G L L S L L F V L A Y I I V V F Y K 1 L N L A L A D L L F A L T L P I W A A S 2 C A L L L I G S Y F N V E K L L S V V K 3 V K F I C L S I W G L S L L L A L P V 4 Y C F L M I L L P V I F G F S Q P L I R L 5 F A V V L I F L L C W L P Y N L V L L A 6 L P N L C S H L I G L I E T A D L A R 7

GPCRdb(A)
GPCRdb(A)
CXCR2
TM2
2x64 2.64x64 K108
ECL2
45x51 45.51x51 Y197
45x52 45.52x52 E198
TM5
5x32 5.31x32 T204
5x36 5.35x36 R208
5x40 5.39x40 R212
TM6
6x58 6.58x58 D274
6x62 6.62x62 R278
TM7
7x27 7.28x27 R289
7x31 7.32x31 D293
7x34 7.35x34 L296