PDB
Resolution
2.9 Å
Released
July 1, 2026
Receptor
Class
A
Species
Homo sapiens
Ligand
PHENCYCLIDINE
Function
Agonist (partial)

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Ligand Amino Acid Generic Number Segment Interaction Type
PHENCYCLIDINE Y150 3.33x33 TM3 hydrophobic
PHENCYCLIDINE M153 3.36x36 TM3 hydrophobic
PHENCYCLIDINE I298 6.51x51 TM6 hydrophobic
PHENCYCLIDINE W320 7.35x34 TM7 hydrophobic
PHENCYCLIDINE I324 7.39x38 TM7 hydrophobic
PHENCYCLIDINE Y328 7.43x42 TM7 hydrophobic

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Snake plot — Download: PNG | SVG
ICL1 T K M K ICL1ECL1 T W P F ECL1ICL2 P V K A L D F R ICL2ECL2 T T K Y R Q G S I D C T L T F S H ECL2ICL3 R M L S G ICL3ECL3 T I P E ECL3N-term M D S S A A P T N A S N C T D A L A Y S S C S P A P S P G S W V N L S H L D G N L S D P C G P N R T D L G G R D S L C P P T G S P S N-termC-term P T S S N I E Q Q N S T R I R Q N T R D H P S T A N T V D R T N H Q L E N L E A E T A P L P C-term M I T A I T I M A L Y S I V C V V G L F G N F L V M Y V I V R Y T A T N I Y I F N L A L A D A L A T S T L P F Q S V N Y L M G G T I L C K I V I S I D Y Y N M F T S I F T L C T M S V D R Y I A V C H T P R N A K I I N V C N W I L S S A I G L P V M F M A P T W Y W E N L L K I C V F I F A F I M P V L I I T V C Y G L M I L R L K S V S K E K D R N L R R I T R M V L V V V A V F I V C W T P I H I Y V I I K A L V T T F Q T V S W H F C I A L G Y T N S C L N P V L Y A F L D E N F R E F K R C F C I
Helix box plot — Download: PNG | SVG F N G F L G V V C V I S Y L A M I T I A 1 F N L A L A D A L A T S T L P F Q S V N 2 T C L T F I S T F M N Y Y D I S I V I K 3 A K I I N V C N W I L S S A I G L P V M 4 Y C V T I I L V P M I F A F I F V C I K L 5 L V V V A V F I V C W T P I H I Y V I I 6 V P N L C S N T Y G L A I C F H W S V 7

GPCRdb(A)
GPCRdb(A)
μ receptor
TM3
3x33 3.33x33 Y150
3x36 3.36x36 M153
TM6
6x51 6.51x51 I298
TM7
7x34 7.35x34 W320
7x38 7.39x38 I324
7x42 7.43x42 Y328