GSK256073


SMILES CCCCCn1c(=O)[nH]c(=O)c2c1nc([nH]2)Cl
InChIKey CGAMDQCXAAOFSR-UHFFFAOYSA-N

Chemical properties

Hydrogen bond acceptors 4
Hydrogen bond donors 2
Rotatable bonds 4
Molecular weight (Da) 256.1

Drug properties

Molecular type Small molecule
Endogenous/Surrogate Surrogate
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
β2 ADRB2 Human Adrenoceptors A pKi 6.28 6.28 6.28 ChEMBL
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
β2 ADRB2 Guinea pig Adrenoceptors A pIC50 7.32 7.32 7.32 ChEMBL
β2 ADRB2 Human Adrenoceptors A pEC50 7.41 7.41 7.41 ChEMBL