Ligand source activities (1 row/activity)



Get vendors


Ligands (move mouse cursor over ligand name to see structure) Receptor Activity Chemical information
Sel. page Common
name		 GPCRdb
ID		 Reference
ligand		 Vendors

 Species

 Assay
Type

 Activity
Type		 Activity
Relation		 Activity
Value		 p-value
(-log)		 Fold
selectivity		 Tested
GPCRs		 Assay
Description		 Source

 Mol
weight		 Rot
Bonds		 H don

 H acc

 LogP

 Smiles

 DOI
44314644 13515 None 0 Rat Functional pEC50 = 9.1 9.1 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1193573 13515 None 0 Rat Functional pEC50 = 9.1 9.1 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL545002 13515 None 0 Rat Functional pEC50 = 9.1 9.1 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314965 12919 None 0 Rat Functional pEC50 = 9 9.0 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1189070 12919 None 0 Rat Functional pEC50 = 9 9.0 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL538008 12919 None 0 Rat Functional pEC50 = 9 9.0 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 533 10 2 5 4.2 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
9937590 108082 None 0 Rat Functional pEC50 = 9 9.0 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL319460 108082 None 0 Rat Functional pEC50 = 9 9.0 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL545465 108082 None 0 Rat Functional pEC50 = 9 9.0 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314574 12918 None 0 Rat Functional pEC50 = 8.9 8.9 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 547 11 2 5 4.6 CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1189066 12918 None 0 Rat Functional pEC50 = 8.9 8.9 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 547 11 2 5 4.6 CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL538004 12918 None 0 Rat Functional pEC50 = 8.9 8.9 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 547 11 2 5 4.6 CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
178024 1971 None 27 Rat Functional pEC50 = 8.8 8.8 -1 3
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 528 8 2 6 1.8 O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C 10.1016/S0960-894X(97)00421-6
5867 1971 None 27 Rat Functional pEC50 = 8.8 8.8 -1 3
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 528 8 2 6 1.8 O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C 10.1016/S0960-894X(97)00421-6
CHEMBL13817 1971 None 27 Rat Functional pEC50 = 8.8 8.8 -1 3
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 528 8 2 6 1.8 O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C 10.1016/S0960-894X(97)00421-6
22867267 13703 None 0 Rat Functional pEC50 = 8.7 8.7 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1194874 13703 None 0 Rat Functional pEC50 = 8.7 8.7 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL553478 13703 None 0 Rat Functional pEC50 = 8.7 8.7 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
44293557 101142 None 0 Rat Functional pEC50 = 8 8.0 -1 2
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 447 7 2 3 3.7 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL294923 101142 None 0 Rat Functional pEC50 = 8 8.0 -1 2
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 447 7 2 3 3.7 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL540001 101142 None 0 Rat Functional pEC50 = 8 8.0 -1 2
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 447 7 2 3 3.7 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
9890375 98323 None 0 Rat Functional pEC50 = 7.9 7.9 -1 3
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 458 5 3 3 3.4 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL274599 98323 None 0 Rat Functional pEC50 = 7.9 7.9 -1 3
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 458 5 3 3 3.4 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL558802 98323 None 0 Rat Functional pEC50 = 7.9 7.9 -1 3
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 458 5 3 3 3.4 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
10026738 162864 None 0 Rat Functional pEC50 = 7.8 7.8 -1 2
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 449 7 2 4 2.9 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL417182 162864 None 0 Rat Functional pEC50 = 7.8 7.8 -1 2
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 449 7 2 4 2.9 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
CHEMBL557206 162864 None 0 Rat Functional pEC50 = 7.8 7.8 -1 2
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 449 7 2 4 2.9 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1 10.1016/S0960-894X(97)00421-6
44315065 13496 None 0 Rat Functional pEC50 = 8.7 8.7 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1193375 13496 None 0 Rat Functional pEC50 = 8.7 8.7 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL544769 13496 None 0 Rat Functional pEC50 = 8.7 8.7 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 9 2 5 3.8 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314651 13609 None 0 Rat Functional pEC50 = 8.7 8.7 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1194179 13609 None 0 Rat Functional pEC50 = 8.7 8.7 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL545704 13609 None 0 Rat Functional pEC50 = 8.7 8.7 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
22867284 13114 None 0 Rat Functional pEC50 = 8.6 8.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1190399 13114 None 0 Rat Functional pEC50 = 8.6 8.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL540805 13114 None 0 Rat Functional pEC50 = 8.6 8.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 505 9 3 4 3.8 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
22867266 13113 None 0 Rat Functional pEC50 = 8.6 8.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 10 3 4 4.1 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1190394 13113 None 0 Rat Functional pEC50 = 8.6 8.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 10 3 4 4.1 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL540800 13113 None 0 Rat Functional pEC50 = 8.6 8.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 519 10 3 4 4.1 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
44314888 13689 None 0 Rat Functional pEC50 = 8.6 8.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1194776 13689 None 0 Rat Functional pEC50 = 8.6 8.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL553290 13689 None 0 Rat Functional pEC50 = 8.6 8.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 491 8 3 4 3.4 CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
44314948 13468 None 0 Rat Functional pEC50 = 8.5 8.5 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1193173 13468 None 0 Rat Functional pEC50 = 8.5 8.5 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL544536 13468 None 0 Rat Functional pEC50 = 8.5 8.5 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314963 13799 None 0 Rat Functional pEC50 = 7.6 7.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1195548 13799 None 0 Rat Functional pEC50 = 7.6 7.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL554852 13799 None 0 Rat Functional pEC50 = 7.6 7.6 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
9872740 26473 None 26 Rat Functional pEC50 = 8.5 8.5 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 567 10 4 7 3.6 C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc2ccc(-c3ccccc3-c3nn[nH]n3)cc2)C1=O 10.1016/S0960-894X(97)00421-6
CHEMBL13600 26473 None 26 Rat Functional pEC50 = 8.5 8.5 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 567 10 4 7 3.6 C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc2ccc(-c3ccccc3-c3nn[nH]n3)cc2)C1=O 10.1016/S0960-894X(97)00421-6
44314653 13516 None 0 Rat Functional pEC50 = 8.4 8.4 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 493 8 3 5 2.6 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1193574 13516 None 0 Rat Functional pEC50 = 8.4 8.4 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 493 8 3 5 2.6 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL545003 13516 None 0 Rat Functional pEC50 = 8.4 8.4 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 493 8 3 5 2.6 CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
22867262 13983 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 516 7 4 4 3.5 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL1196866 13983 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 516 7 4 4 3.5 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
CHEMBL558422 13983 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 516 7 4 4 3.5 CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12 10.1016/S0960-894X(97)00421-6
44314767 13705 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1194891 13705 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL553507 13705 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44314881 13663 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1194592 13663 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL552911 13663 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 521 9 2 6 3.0 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
121879 2234 None 25 Rat Functional pEC50 = 7.2 7.2 -1 5
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 509 7 3 6 3.6 O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2 10.1016/S0960-894X(97)00421-6
5868 2234 None 25 Rat Functional pEC50 = 7.2 7.2 -1 5
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 509 7 3 6 3.6 O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2 10.1016/S0960-894X(97)00421-6
CHEMBL308716 2234 None 25 Rat Functional pEC50 = 7.2 7.2 -1 5
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 509 7 3 6 3.6 O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2 10.1016/S0960-894X(97)00421-6
44314642 13643 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1194442 13643 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL552657 13643 None 0 Rat Functional pEC50 = 8.2 8.2 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 544 8 3 5 3.9 CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
44315063 13878 None 0 Rat Functional pEC50 = 8.1 8.1 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL1196053 13878 None 0 Rat Functional pEC50 = 8.1 8.1 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
CHEMBL555821 13878 None 0 Rat Functional pEC50 = 8.1 8.1 - 1
Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay
ChEMBL 530 7 3 5 3.5 CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21 10.1016/S0960-894X(97)00421-6
1104 1792 None 0 Rat Functional pIC50 = 9.1 9.1 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 1534126
1122 2701 None 0 Rat Functional pIC50 None 10.2 10.2 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431
1123 2702 None 0 Rat Functional pIC50 None 10.2 10.2 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431
1105 1793 None 0 Rat Functional pIC50 None 8 8.0 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 1534126
1103 1791 None 0 Rat Functional pIC50 None 8.2 8.2 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 1534126
CHEMBL440262 1791 None 0 Rat Functional pIC50 None 8.2 8.2 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 1534126


Get vendors


Ligands (move mouse cursor over ligand name to see structure) Receptor Activity Chemical information
Sel. page Common
name		 GPCRdb
ID		 Reference
ligand		 Vendors

 Species

 Assay
Type		 Activity
Type		 Activity
Relation		 Activity
Value		 p-value
(-log)		 Fold
selectivity		 Tested
GPCRs		 Assay
Description		 Source

 Mol
weight		 Rot
Bonds		 H don

 H acc

 LogP

 Smiles

 DOI
148124 209557 None 54 Human Binding pIC50 = 9.9 9.9 - 1
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
ChEMBL 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C 10.1073/pnas.0610860104
CHEMBL3545252 209557 None 54 Human Binding pIC50 = 9.9 9.9 - 1
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
ChEMBL 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C 10.1073/pnas.0610860104
CHEMBL92 209557 None 54 Human Binding pIC50 = 9.9 9.9 - 1
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
ChEMBL 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C 10.1073/pnas.0610860104
44387407 141913 None 0 Rat Binding pIC50 = 9.1 9.1 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3354 116 47 46 -12.4 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928715 141913 None 0 Rat Binding pIC50 = 9.1 9.1 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3354 116 47 46 -12.4 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL386366 141913 None 0 Rat Binding pIC50 = 9.1 9.1 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3354 116 47 46 -12.4 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
1103 1791 None 0 Rat Binding pIC50 = 9.1 9.1 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None None 10.1021/jm00088a023
CHEMBL440262 1791 None 0 Rat Binding pIC50 = 9.1 9.1 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None None 10.1021/jm00088a023
CHEMBL385308 214808 None 0 Rat Binding pIC50 = 8.7 8.7 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O 10.1021/jm00088a023
CHEMBL412221 215437 None 0 Rat Binding pIC50 = 6 6.0 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL269263 213242 None 0 Rat Binding pIC50 = 6 6.0 - 0
Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]GRF in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL264522 213083 None 0 Rat Binding pIC50 = 6.9 6.9 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
44387431 96574 None 0 Rat Binding pIC50 = 7.9 7.9 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3441 119 50 48 -15.1 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928702 96574 None 0 Rat Binding pIC50 = 7.9 7.9 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3441 119 50 48 -15.1 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL262750 96574 None 0 Rat Binding pIC50 = 7.9 7.9 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3441 119 50 48 -15.1 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
44387406 161337 None 0 Rat Binding pIC50 = 6.9 6.9 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3136 108 44 42 -11.2 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928713 161337 None 0 Rat Binding pIC50 = 6.9 6.9 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3136 108 44 42 -11.2 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL411913 161337 None 0 Rat Binding pIC50 = 6.9 6.9 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3136 108 44 42 -11.2 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL427794 215845 None 0 Rat Binding pIC50 = 7.8 7.8 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL413014 215504 None 0 Rat Binding pIC50 = 7.8 7.8 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL414943 215623 None 0 Rat Binding pIC50 = 7.7 7.7 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL437461 216182 None 0 Rat Binding pIC50 = 7.7 7.7 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)C(C)C)[C@@H](C)O 10.1021/jm00088a023
44387434 169089 None 0 Rat Binding pIC50 = 7.7 7.7 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3497 123 50 48 -13.5 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928693 169089 None 0 Rat Binding pIC50 = 7.7 7.7 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3497 123 50 48 -13.5 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL439108 169089 None 0 Rat Binding pIC50 = 7.7 7.7 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3497 123 50 48 -13.5 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL269041 213235 None 0 Rat Binding pIC50 = 6.7 6.7 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None None 10.1021/jm00088a023
CHEMBL428284 215894 None 0 Rat Binding pIC50 = 6.5 6.5 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](N)CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL439306 216296 None 0 Rat Binding pIC50 = 6.4 6.4 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL427665 215824 None 0 Rat Binding pIC50 = 7.4 7.4 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O 10.1021/jm00088a023
CHEMBL262536 212999 None 0 Rat Binding pIC50 = 7.3 7.3 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL428135 215879 None 11 Rat Binding pIC50 = 8.3 8.3 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
44387430 81926 None 0 Rat Binding pIC50 = 8.2 8.2 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3469 121 50 48 -14.3 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
91928698 81926 None 0 Rat Binding pIC50 = 8.2 8.2 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3469 121 50 48 -14.3 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL216479 81926 None 0 Rat Binding pIC50 = 8.2 8.2 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL 3469 121 50 48 -14.3 CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL438545 216236 None 0 Rat Binding pIC50 = 8.1 8.1 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL415373 215646 None 0 Rat Binding pIC50 = 6.1 6.1 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL266658 213150 None 0 Rat Binding pIC50 = 8.0 8.0 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
CHEMBL265167 213099 None 15 Rat Binding pIC50 = 8.0 8.0 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1c[nH]cn1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O 10.1021/jm00088a023
CHEMBL412558 215463 None 0 Rat Binding pIC50 = 7.0 7.0 - 0
Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates
ChEMBL None None None CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O 10.1021/jm00088a023
148124 209557 None 54 Human Binding pIC50 = 8.0 8.0 - 1
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
Drug Central 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C None
CHEMBL3545252 209557 None 54 Human Binding pIC50 = 8.0 8.0 - 1
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
Drug Central 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C None
CHEMBL92 209557 None 54 Human Binding pIC50 = 8.0 8.0 - 1
Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells
Drug Central 807 8 5 14 3.3 CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C None
9114 2118 None 0 Human Binding pIC50 = 9.9 9.9 - 0
Measuring displacement of [<sup>12</sup>5I]JV-1-42 in a radioligand binding assay.Measuring displacement of [<sup>12</sup>5I]JV-1-42 in a radioligand binding assay.
Guide to Pharmacology None None None None 17261802
1109 2159 None 0 Rat Binding pKi = 10.1 10.1 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10542394
1109 2159 None 0 Rat Binding pKi = 10.1 10.1 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1109 2159 None 0 Rat Binding pKi = 10.1 10.1 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1107 2157 None 0 Rat Binding pKi = 10.3 10.3 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10542394
1107 2157 None 0 Rat Binding pKi = 10.3 10.3 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1107 2157 None 0 Rat Binding pKi = 10.3 10.3 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1110 2160 None 0 Rat Binding pKi None 10.1 10.1 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1115 2165 None 0 Rat Binding pKi None 10.2 10.2 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1116 2166 None 0 Rat Binding pKi None 10.2 10.2 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1121 2700 None 0 Rat Binding pKi None 10.2 10.2 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431
1124 2703 None 0 Rat Binding pKi None 10.2 10.2 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1106 2156 None 0 Rat Binding pKi None 10.3 10.3 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1118 2696 None 0 Rat Binding pKi None 10.3 10.3 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1108 2158 None 0 Rat Binding pKi None 10.4 10.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1111 2161 None 0 Rat Binding pKi None 10.4 10.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1112 2162 None 0 Rat Binding pKi None 10.4 10.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1113 2163 None 0 Rat Binding pKi None 10.4 10.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1114 2164 None 0 Rat Binding pKi None 10.4 10.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1117 2695 None 0 Rat Binding pKi None 10.4 10.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1119 2697 None 0 Rat Binding pKi None 10.4 10.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1125 281 None 0 Rat Binding pKi None 8.4 8.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 14755056
1125 281 None 0 Rat Binding pKi None 8.4 8.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1125 281 None 0 Rat Binding pKi None 8.4 8.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431
1125 281 None 0 Rat Binding pKi None 8.4 8.4 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9892695
1120 2699 None 0 Rat Binding pKi None 9.9 9.9 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 7991622
1120 2699 None 0 Rat Binding pKi None 9.9 9.9 - 1
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9145431