GPCR CLASS (FAMILY)
Class A (Rhodopsin)
PDB CODE
SPECIES
Homo sapiens
RESOLUTION
3.4 Å
PREFERRED CHAIN
R
PUBLICATION DATE
Nov. 12, 2025
LIGAND INTERACTIONS
LIGANDS
naloxone - Agonist (partial) pubchem gtoplig chembl_ligand drugbank drug_central chembl_ligand pubchem pubchem
PHYSIOLOGICAL LIGANDS
[Met]enkephalin (Human), dynorphin A-(1-8) (Human), dynorphin A (Human), dynorphin A-(1-13) (Human), β-endorphin (Mouse), endomorphin-1 (Human), β-endorphin (Rat), dynorphin B (Human), β-endorphin (Human), [Leu]enkephalin (Human), endomorphin-2 (Human)