BIM 23058


SMILES None
InChIKey None
Sequence FFYWKVFT

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
A1 AA1R Human Adenosine A pKi 6.08 6.08 6.08 Guide to Pharmacology
A2A AA2AR Human Adenosine A pKi 7.04 7.48 7.92 Guide to Pharmacology
A2B AA2BR Human Adenosine A pKi 5.0 5.0 5.0 Guide to Pharmacology
A3 AA3R Human Adenosine A pKi 5.35 5.35 5.35 Guide to Pharmacology
A1 AA1R Rat Adenosine A pKi 6.64 6.64 6.64 Guide to Pharmacology
A2A AA2AR Rat Adenosine A pKi 8.35 8.5 8.66 Guide to Pharmacology
A2A AA2AR Rat Adenosine A pKi 7.89 8.41 8.7 ChEMBL
A1 AA1R Rat Adenosine A pKi 6.24 6.62 6.82 ChEMBL
A2B AA2BR Human Adenosine A pKi 5.75 5.75 5.75 ChEMBL
A3 AA3R Human Adenosine A pKi 5.35 5.35 5.35 ChEMBL
A2A AA2AR Human Adenosine A pKi 6.7 7.56 8.66 ChEMBL
A2A AA2AR Human Adenosine A pKd 5.9 5.9 5.9 ChEMBL
A1 AA1R Human Adenosine A pKi 5.52 5.77 6.08 ChEMBL
A1 AA1R Human Adenosine A pKi 8.22 8.22 8.22 Drug Central
A2A AA2AR Human Adenosine A pKi 8.06 8.06 8.06 Drug Central
A2B AA2BR Human Adenosine A pKi 8.24 8.24 8.24 Drug Central
A3 AA3R Human Adenosine A pKi 8.27 8.27 8.27 Drug Central
A1 AA1R Rat Adenosine A pKi 8.17 8.17 8.17 Drug Central
A2A AA2AR Rat Adenosine A pKi 8.06 8.06 8.06 Drug Central
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
A2A AA2AR Rat Adenosine A pIC50 6.64 6.64 6.64 ChEMBL
A2A AA2AR Human Adenosine A pIC50 5.28 5.28 5.28 ChEMBL