substance P-OMe


SMILES None
InChIKey None
Sequence RPKPQQFFGLM

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug No

Database connections


Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
H4 HRH4 Human Histamine A pKi 7.1 7.44 7.7 ChEMBL
H4 HRH4 Human Histamine A pKd 7.7 7.7 7.7 ChEMBL
H3 HRH3 Human Histamine A pKi 4.7 4.98 5.4 ChEMBL
H4 HRH4 Human Histamine A pKi 7.1 7.1 7.1 Guide to Pharmacology
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
H4 HRH4 Human Histamine A pIC50 6.28 6.57 6.86 ChEMBL
H3 HRH3 Human Histamine A pEC50 5.5 5.5 5.5 ChEMBL