d(CH2)5[Tyr(Et)2,Val4,des-Gly9]AVP


SMILES None
InChIKey DRLYXDZRLDZVIS-XXNQTUAPSA-N
Sequence CYFVNCPR

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
β1 ADRB1 Human Adrenoceptors A pKi 6.24 6.24 6.24 ChEMBL
β2 ADRB2 Human Adrenoceptors A pKi 6.8 6.8 6.8 ChEMBL
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
β3 ADRB3 Human Adrenoceptors A pEC50 10.1 10.1 10.1 Guide to Pharmacology
β1 ADRB1 Human Adrenoceptors A pIC50 6.7 6.7 6.7 ChEMBL
β1 ADRB1 Human Adrenoceptors A pEC50 6.48 6.48 6.48 ChEMBL
β3 ADRB3 Human Adrenoceptors A pEC50 9.0 9.3 9.37 ChEMBL
β2 ADRB2 Human Adrenoceptors A pIC50 5.52 6.12 6.72 ChEMBL
β2 ADRB2 Human Adrenoceptors A pEC50 7.7 7.7 7.7 ChEMBL
TSH TSHR Human Glycoprotein hormone A Potency 4.7 4.7 4.7 ChEMBL