d(CH2)5[Tyr(Me)2,Thr4]OVT


SMILES None
InChIKey None
Sequence CYITNCPXG

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug No

Database connections


Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
5-HT1D 5HT1D Human 5-Hydroxytryptamine A pKi 9.05 9.05 9.05 ChEMBL
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
5-HT1B 5HT1B Human 5-Hydroxytryptamine A pIC50 6.8 6.8 6.8 Guide to Pharmacology
5-HT1D 5HT1D Human 5-Hydroxytryptamine A pIC50 9.0 9.0 9.0 Guide to Pharmacology
5-HT1B 5HT1B Human 5-Hydroxytryptamine A pIC50 6.73 6.78 6.82 ChEMBL
5-HT1D 5HT1D Human 5-Hydroxytryptamine A pEC50 8.96 9.01 9.1 ChEMBL
5-HT1D 5HT1D Human 5-Hydroxytryptamine A pIC50 9.05 9.05 9.05 ChEMBL
5-HT1A 5HT1A Human 5-Hydroxytryptamine A pIC50 7.18 7.18 7.18 ChEMBL
5-HT2A 5HT2A Human 5-Hydroxytryptamine A pIC50 5.96 5.96 5.96 ChEMBL
5-HT1A 5HT1A Human 5-Hydroxytryptamine A pIC50 7.2 7.2 7.2 Guide to Pharmacology
5-HT7 5HT7R Rat 5-Hydroxytryptamine A pIC50 6.27 6.27 6.27 ChEMBL