d(CH2)5[Tyr(Me)2,Arg8]VP


SMILES None
InChIKey None
Sequence YFQNCPRG

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
NOP OPRX Human Opioid A pKi 10.55 10.55 10.55 ChEMBL
δ OPRD Human Opioid A pKi 6.37 6.37 6.37 ChEMBL
μ OPRM Human Opioid A pKi 7.13 7.13 7.13 ChEMBL
κ OPRK Human Opioid A pKi 8.36 8.36 8.36 ChEMBL
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
NOP OPRX Guinea pig Opioid A pEC50 9.17 9.17 9.17 ChEMBL
NOP OPRX Mouse Opioid A pEC50 9.24 9.24 9.24 ChEMBL
NOP OPRX Rat Opioid A pEC50 8.34 8.34 8.34 ChEMBL
NOP OPRX Human Opioid A pEC50 10.55 10.55 10.55 ChEMBL
NOP OPRX Human Opioid A pEC50 8.39 9.05 9.71 Guide to Pharmacology