CGP42112


SMILES None
InChIKey UXGNARZDONUMMK-LRMQDCNJSA-N
Sequence YKHPI

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
PAR1 PAR1 Human Proteinase-activated A pKi 7.89 8.22 8.96 ChEMBL
PAR1 PAR1 Human Proteinase-activated A pKi 8.09 8.09 8.09 Drug Central
PAR1 PAR1 Human Proteinase-activated A pKi 8.09 8.09 8.09 Guide to Pharmacology
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
PAR1 PAR1 Human Proteinase-activated A pIC50 6.6 7.56 8.96 ChEMBL