labradimil
| SMILES | None |
| InChIKey | IDXCXSCCZNCXCL-XMADEQCMSA-N |
| Sequence | RPXGXSPYR |
Chemical properties
| Hydrogen bond acceptors | None |
| Hydrogen bond donors | None |
| Rotatable bonds | None |
| Molecular weight (Da) |
Drug properties
| Molecular type | Peptide |
| Endogenous/Surrogate | Surrogate |
| Approved drug | Yes |
Database connections
Bioactivities
| Receptor | Activity | Source | |||||||
|---|---|---|---|---|---|---|---|---|---|
| GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
| PAR4 | PAR4 | Human | Proteinase-activated | A | pKd | 10.01 | 10.08 | 10.15 | ChEMBL |
| Receptor | Activity | Source | |||||||
|---|---|---|---|---|---|---|---|---|---|
| GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
| PAR4 | PAR4 | Human | Proteinase-activated | A | pIC50 | 9.3 | 9.3 | 9.3 | Guide to Pharmacology |
| PAR4 | PAR4 | Human | Proteinase-activated | A | pIC50 | 8.01 | 8.58 | 9.4 | ChEMBL |
| PAR4 | PAR4 | Human | Proteinase-activated | A | pEC50 | 9.37 | 9.37 | 9.37 | ChEMBL |