CCK-58


SMILES None
InChIKey None
Sequence AVQKVDGEPRAHLGALLARYIQQARKAPSGRMSVIKNLQNLDPSHRISDRDYMGWMDF

Chemical properties

Hydrogen bond acceptors None
Hydrogen bond donors None
Rotatable bonds None
Molecular weight (Da)

Drug properties

Molecular type Peptide
Endogenous/Surrogate Surrogate
Approved drug No

Database connections

Bioactivities

Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
mGlu5 GRM5 Rat Metabotropic glutamate C pKi 5.42 5.42 5.42 ChEMBL
mGlu5 GRM5 Human Metabotropic glutamate C pKi 6.6 6.6 6.6 ChEMBL
Receptor Activity Source
GTP Uniprot Species Family Class Type Min Avg Max Database
mGlu5 GRM5 Human Metabotropic glutamate C pEC50 7.6 7.8 8.0 Guide to Pharmacology
mGlu5 GRM5 Rat Metabotropic glutamate C pEC50 7.7 7.7 7.7 Guide to Pharmacology
mGlu5 GRM5 Rat Metabotropic glutamate C pEC50 7.01 7.27 7.7 ChEMBL
mGlu5 GRM5 Human Metabotropic glutamate C pEC50 6.75 7.27 8.0 ChEMBL