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Ligand source activities (1 row/activity)

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Ligands (move mouse cursor over ligand name to see structure)					Receptor		Activity									Chemical information
Sel. page	Common name No matches found	GPCRdb ID No matches found	Reference ligand No matches found	Vendors	Species No matches found		Assay Type No matches found	Activity Type No matches found	Activity Relation No matches found	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description No matches found	Source No matches found	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles No matches found	DOI No matches found

Ligands (move mouse cursor over ligand name to see structure)					Receptor	Activity									Chemical information
Sel. page	Common name No matches found	GPCRdb ID No matches found	Reference ligand No matches found	Vendors	Species No matches found	Assay Type No matches found	Activity Type No matches found	Activity Relation No matches found	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description No matches found	Source No matches found	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles No matches found	DOI No matches found
	90656213	110966	None	0	Human	Functional	pEC50	=	7	7.0	1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation countingAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation counting	ChEMBL	635	13	7	13	-0.3	O=c1[nH]/c(=N\OCCCc2cccc(F)c2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	CHEMBL3261362	110966	None	0	Human	Functional	pEC50	=	7	7.0	1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation countingAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation counting	ChEMBL	635	13	7	13	-0.3	O=c1[nH]/c(=N\OCCCc2cccc(F)c2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	1734	3966	None	29	Human	Functional	pEC50	=	7	7.0	-1	7	Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptorAgonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptor	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/s0960-894x(00)00612-0
	3639	3966	None	29	Human	Functional	pEC50	=	7	7.0	-1	7	Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptorAgonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptor	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/s0960-894x(00)00612-0
	6133	3966	None	29	Human	Functional	pEC50	=	7	7.0	-1	7	Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptorAgonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptor	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/s0960-894x(00)00612-0
	CHEMBL336296	3966	None	29	Human	Functional	pEC50	=	7	7.0	-1	7	Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptorAgonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptor	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/s0960-894x(00)00612-0
	DB04005	3966	None	29	Human	Functional	pEC50	=	7	7.0	-1	7	Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptorAgonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 receptor	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/s0960-894x(00)00612-0
	1731	130	None	8	Human	Functional	pEC50	=	5	5.0	-10	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as calcium elevation by fura2/AM assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as calcium elevation by fura2/AM assay	ChEMBL	562	8	7	12	-1.7	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cc(Br)c(=O)[nH]c1=O	10.1021/jm901450d
	9872620	130	None	8	Human	Functional	pEC50	=	5	5.0	-10	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as calcium elevation by fura2/AM assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as calcium elevation by fura2/AM assay	ChEMBL	562	8	7	12	-1.7	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cc(Br)c(=O)[nH]c1=O	10.1021/jm901450d
	CHEMBL384527	130	None	8	Human	Functional	pEC50	=	5	5.0	-10	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as calcium elevation by fura2/AM assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as calcium elevation by fura2/AM assay	ChEMBL	562	8	7	12	-1.7	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cc(Br)c(=O)[nH]c1=O	10.1021/jm901450d
	90656214	110967	None	0	Human	Functional	pEC50	=	7.0	7.0	5	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation countingAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation counting	ChEMBL	635	13	7	13	-0.3	O=c1[nH]/c(=N\OCCCc2ccc(F)cc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	CHEMBL3261363	110967	None	0	Human	Functional	pEC50	=	7.0	7.0	5	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation countingAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation counting	ChEMBL	635	13	7	13	-0.3	O=c1[nH]/c(=N\OCCCc2ccc(F)cc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	54584406	62940	None	0	Human	Functional	pEC50	=	6.0	6.0	4	2	Agonist activity at human P2Y4Agonist activity at human P2Y4	ChEMBL	509	9	6	12	-1.2	[N-]=[N+]=N[C@@H]1[C@H](O)[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O[C@H]1n1ccc(=O)[nH]c1=O	10.1021/jm101591j
	CHEMBL1784888	62940	None	0	Human	Functional	pEC50	=	6.0	6.0	4	2	Agonist activity at human P2Y4Agonist activity at human P2Y4	ChEMBL	509	9	6	12	-1.2	[N-]=[N+]=N[C@@H]1[C@H](O)[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O[C@H]1n1ccc(=O)[nH]c1=O	10.1021/jm101591j
	44586045	184254	None	0	Human	Functional	pEC50	=	6.0	6.0	1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	638	14	9	17	-3.0	O=c1ccn([C@@H]2O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)OP(=O)(O)OCC(O)CO)[C@@H](O)[C@H]2O)c(=O)[nH]1	10.1016/j.bmc.2008.05.013
	CHEMBL482895	184254	None	0	Human	Functional	pEC50	=	6.0	6.0	1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	638	14	9	17	-3.0	O=c1ccn([C@@H]2O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)OP(=O)(O)OCC(O)CO)[C@@H](O)[C@H]2O)c(=O)[nH]1	10.1016/j.bmc.2008.05.013
	90656216	110969	None	0	Human	Functional	pEC50	=	6.9	6.9	2	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation countingAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation counting	ChEMBL	743	13	7	13	0.2	O=c1[nH]/c(=N\OCCCc2cccc(I)c2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	CHEMBL3261365	110969	None	0	Human	Functional	pEC50	=	6.9	6.9	2	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation countingAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation counting	ChEMBL	743	13	7	13	0.2	O=c1[nH]/c(=N\OCCCc2cccc(I)c2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	46831686	14206	None	0	Human	Functional	pEC50	=	5.9	5.9	-3	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assayAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assay	ChEMBL	509	9	6	11	-0.9	O=c1[nH]/c(=N\OCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm100287t
	CHEMBL1084612	14206	None	0	Human	Functional	pEC50	=	5.9	5.9	-3	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assayAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assay	ChEMBL	509	9	6	11	-0.9	O=c1[nH]/c(=N\OCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm100287t
	CHEMBL1198872	14206	None	0	Human	Functional	pEC50	=	5.9	5.9	-3	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assayAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assay	ChEMBL	509	9	6	11	-0.9	O=c1[nH]/c(=N\OCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm100287t
	CHEMBL4866937	14206	None	0	Human	Functional	pEC50	=	5.9	5.9	-3	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assayAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation proximity assay	ChEMBL	509	9	6	11	-0.9	O=c1[nH]/c(=N\OCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm100287t
	46831686	14206	None	0	Human	Functional	pEC50	=	5.9	5.9	-3	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysisAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysis	ChEMBL	509	9	6	11	-0.9	O=c1[nH]/c(=N\OCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1039/c3md00132f
	CHEMBL1084612	14206	None	0	Human	Functional	pEC50	=	5.9	5.9	-3	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysisAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysis	ChEMBL	509	9	6	11	-0.9	O=c1[nH]/c(=N\OCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1039/c3md00132f
	CHEMBL1198872	14206	None	0	Human	Functional	pEC50	=	5.9	5.9	-3	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysisAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysis	ChEMBL	509	9	6	11	-0.9	O=c1[nH]/c(=N\OCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1039/c3md00132f
	CHEMBL4866937	14206	None	0	Human	Functional	pEC50	=	5.9	5.9	-3	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysisAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells using [3H]inositol as substrate assessed as [3H]inositol phosphate formation after 30 mins by liquid scintillation counting analysis	ChEMBL	509	9	6	11	-0.9	O=c1[nH]/c(=N\OCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1039/c3md00132f
	11525909	141692	None	6	Human	Functional	pEC50	=	5.9	5.9	-19	2	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	483	8	7	12	-2.5	N[C@@H]1[C@H](O)[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O[C@H]1n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	CHEMBL385098	141692	None	6	Human	Functional	pEC50	=	5.9	5.9	-19	2	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	483	8	7	12	-2.5	N[C@@H]1[C@H](O)[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O[C@H]1n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	11525909	141692	None	6	Human	Functional	pEC50	=	5.9	5.9	-19	2	Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CAgonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase C	ChEMBL	483	8	7	12	-2.5	N[C@@H]1[C@H](O)[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O[C@H]1n1ccc(=O)[nH]c1=O	10.1021/jm060903o
	CHEMBL385098	141692	None	6	Human	Functional	pEC50	=	5.9	5.9	-19	2	Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CAgonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase C	ChEMBL	483	8	7	12	-2.5	N[C@@H]1[C@H](O)[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O[C@H]1n1ccc(=O)[nH]c1=O	10.1021/jm060903o
	44586007	192704	None	1	Human	Functional	pEC50	=	5.9	5.9	1	2	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	498	8	7	12	-2.1	C[C@@]1(O)[C@H](O)[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O[C@H]1n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	CHEMBL521487	192704	None	1	Human	Functional	pEC50	=	5.9	5.9	1	2	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	498	8	7	12	-2.1	C[C@@]1(O)[C@H](O)[C@@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)O[C@H]1n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	90656225	110978	None	0	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation countingAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation counting	ChEMBL	667	13	7	13	0.8	O=c1[nH]/c(=N\OCCCc2ccc3ccccc3c2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	CHEMBL3261374	110978	None	0	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation countingAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as stimulation of [3H]inositol phosphate accumulation by liquid scintillation counting	ChEMBL	667	13	7	13	0.8	O=c1[nH]/c(=N\OCCCc2ccc3ccccc3c2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	148197	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	148197.0	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	1736	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	4900	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	CHEMBL221326	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	DB15919	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1016/j.bmc.2008.05.013
	148197	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CAgonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase C	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm060903o
	148197.0	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CAgonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase C	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm060903o
	1736	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CAgonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase C	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm060903o
	4900	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CAgonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase C	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm060903o
	CHEMBL221326	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CAgonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase C	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm060903o
	DB15919	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CAgonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase C	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm060903o
	148197	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by scintillation proximity assayAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm101591j
	148197.0	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by scintillation proximity assayAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm101591j
	1736	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by scintillation proximity assayAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm101591j
	4900	1438	None	20	Human	Functional	pEC50	=	6.9	6.9	-1	3	Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by scintillation proximity assayAgonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by scintillation proximity assay	ChEMBL	790	14	10	21	-4.2	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(OP(=O)(OC[C@H]2O[C@H]([C@@H]([C@@H]2O)O)n2ccc(=O)[nH]c2=O)O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/jm101591j

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Ligands (move mouse cursor over ligand name to see structure)					Receptor		Activity									Chemical information
Sel. page	Common name No matches found	GPCRdb ID No matches found	Reference ligand No matches found	Vendors	Species No matches found		Assay Type No matches found	Activity Type No matches found	Activity Relation No matches found	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description No matches found	Source No matches found	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles No matches found	DOI No matches found

Ligands (move mouse cursor over ligand name to see structure)					Receptor	Activity									Chemical information
Sel. page	Common name No matches found	GPCRdb ID No matches found	Reference ligand No matches found	Vendors	Species No matches found	Assay Type No matches found	Activity Type No matches found	Activity Relation No matches found	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description No matches found	Source No matches found	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles No matches found	DOI No matches found
	1713	520	None	42	Rat	Binding	pEC50	=	5.9	5.9	-	2	Antagonist activity at rat P2Y4Antagonist activity at rat P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	5957	520	None	42	Rat	Binding	pEC50	=	5.9	5.9	-	2	Antagonist activity at rat P2Y4Antagonist activity at rat P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	91	520	None	42	Rat	Binding	pEC50	=	5.9	5.9	-	2	Antagonist activity at rat P2Y4Antagonist activity at rat P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	CHEMBL14249	520	None	42	Rat	Binding	pEC50	=	5.9	5.9	-	2	Antagonist activity at rat P2Y4Antagonist activity at rat P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	DB00171	520	None	42	Rat	Binding	pEC50	=	5.9	5.9	-	2	Antagonist activity at rat P2Y4Antagonist activity at rat P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	90656232	110982	None	0	Human	Binding	pEC50	=	5.9	5.9	-	0	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells by functional assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells by functional assay	ChEMBL	1056	24	10	23	0.0	O=c1[nH]/c(=N\OCCCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)OP(=O)(O)OC[C@H]2O[C@@H](n3cc/c(=N/OCCCc4ccccc4)[nH]c3=O)[C@H](O)[C@@H]2O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	CHEMBL3261380	110982	None	0	Human	Binding	pEC50	=	5.9	5.9	-	0	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells by functional assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells by functional assay	ChEMBL	1056	24	10	23	0.0	O=c1[nH]/c(=N\OCCCc2ccccc2)ccn1[C@@H]1O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)OP(=O)(O)OC[C@H]2O[C@@H](n3cc/c(=N/OCCCc4ccccc4)[nH]c3=O)[C@H](O)[C@@H]2O)[C@@H](O)[C@H]1O	10.1021/jm500367e
	1734	3966	None	29	Human	Binding	pEC50	=	6.3	6.3	-	2	Agonist activity at human P2Y4 transfected in human 1321N1 cellsAgonist activity at human P2Y4 transfected in human 1321N1 cells	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/acs.jmedchem.5b01972
	3639	3966	None	29	Human	Binding	pEC50	=	6.3	6.3	-	2	Agonist activity at human P2Y4 transfected in human 1321N1 cellsAgonist activity at human P2Y4 transfected in human 1321N1 cells	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/acs.jmedchem.5b01972
	6133	3966	None	29	Human	Binding	pEC50	=	6.3	6.3	-	2	Agonist activity at human P2Y4 transfected in human 1321N1 cellsAgonist activity at human P2Y4 transfected in human 1321N1 cells	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/acs.jmedchem.5b01972
	CHEMBL336296	3966	None	29	Human	Binding	pEC50	=	6.3	6.3	-	2	Agonist activity at human P2Y4 transfected in human 1321N1 cellsAgonist activity at human P2Y4 transfected in human 1321N1 cells	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/acs.jmedchem.5b01972
	DB04005	3966	None	29	Human	Binding	pEC50	=	6.3	6.3	-	2	Agonist activity at human P2Y4 transfected in human 1321N1 cellsAgonist activity at human P2Y4 transfected in human 1321N1 cells	ChEMBL	484	8	7	12	-2.5	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1ccc(=O)[nH]c1=O	10.1021/acs.jmedchem.5b01972
	1713	520	None	42	Human	Binding	pEC50	=	5.2	5.2	257	2	Antagonist activity at human P2Y4Antagonist activity at human P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	5957	520	None	42	Human	Binding	pEC50	=	5.2	5.2	257	2	Antagonist activity at human P2Y4Antagonist activity at human P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	91	520	None	42	Human	Binding	pEC50	=	5.2	5.2	257	2	Antagonist activity at human P2Y4Antagonist activity at human P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	CHEMBL14249	520	None	42	Human	Binding	pEC50	=	5.2	5.2	257	2	Antagonist activity at human P2Y4Antagonist activity at human P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	DB00171	520	None	42	Human	Binding	pEC50	=	5.2	5.2	257	2	Antagonist activity at human P2Y4Antagonist activity at human P2Y4	ChEMBL	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10.1021/acs.jmedchem.5b01972
	136677322	3296	None	17	Rat	Binding	pEC50	=	5.2	5.2	-	1	Antagonist activity at rat P2Y4 transfected in xenopus oocyte cellAntagonist activity at rat P2Y4 transfected in xenopus oocyte cell	ChEMBL	773	9	7	15	3.9	OS(=O)(=O)c1cc(Nc2ccc(c(c2)S(=O)(=O)O)Nc2nc(Cl)nc(n2)Nc2cccc(c2)S(=O)(=O)O)c2c(c1N)C(=O)c1c(C2=O)cccc1	10.1021/acs.jmedchem.5b01972
	1739	3296	None	17	Rat	Binding	pEC50	=	5.2	5.2	-	1	Antagonist activity at rat P2Y4 transfected in xenopus oocyte cellAntagonist activity at rat P2Y4 transfected in xenopus oocyte cell	ChEMBL	773	9	7	15	3.9	OS(=O)(=O)c1cc(Nc2ccc(c(c2)S(=O)(=O)O)Nc2nc(Cl)nc(n2)Nc2cccc(c2)S(=O)(=O)O)c2c(c1N)C(=O)c1c(C2=O)cccc1	10.1021/acs.jmedchem.5b01972
	656725	3296	None	17	Rat	Binding	pEC50	=	5.2	5.2	-	1	Antagonist activity at rat P2Y4 transfected in xenopus oocyte cellAntagonist activity at rat P2Y4 transfected in xenopus oocyte cell	ChEMBL	773	9	7	15	3.9	OS(=O)(=O)c1cc(Nc2ccc(c(c2)S(=O)(=O)O)Nc2nc(Cl)nc(n2)Nc2cccc(c2)S(=O)(=O)O)c2c(c1N)C(=O)c1c(C2=O)cccc1	10.1021/acs.jmedchem.5b01972
	CHEMBL1160031	3296	None	17	Rat	Binding	pEC50	=	5.2	5.2	-	1	Antagonist activity at rat P2Y4 transfected in xenopus oocyte cellAntagonist activity at rat P2Y4 transfected in xenopus oocyte cell	ChEMBL	773	9	7	15	3.9	OS(=O)(=O)c1cc(Nc2ccc(c(c2)S(=O)(=O)O)Nc2nc(Cl)nc(n2)Nc2cccc(c2)S(=O)(=O)O)c2c(c1N)C(=O)c1c(C2=O)cccc1	10.1021/acs.jmedchem.5b01972
	90656231	110981	None	0	Human	Binding	pEC50	=	7.0	7.0	-	0	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells by functional assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells by functional assay	ChEMBL	923	19	10	22	-2.1	O=c1ccn([C@@H]2O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)OP(=O)(O)OC[C@H]3O[C@@H](n4cc/c(=N/OCCCc5ccccc5)[nH]c4=O)[C@H](O)[C@@H]3O)[C@@H](O)[C@H]2O)c(=O)[nH]1	10.1021/jm500367e
	CHEMBL3261379	110981	None	0	Human	Binding	pEC50	=	7.0	7.0	-	0	Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells by functional assayAgonist activity at human P2Y4 receptor expressed in human 1321N1 cells by functional assay	ChEMBL	923	19	10	22	-2.1	O=c1ccn([C@@H]2O[C@H](COP(=O)(O)OP(=O)(O)OP(=O)(O)OP(=O)(O)OC[C@H]3O[C@@H](n4cc/c(=N/OCCCc5ccccc5)[nH]c4=O)[C@H](O)[C@@H]3O)[C@@H](O)[C@H]2O)c(=O)[nH]1	10.1021/jm500367e
	1713	520	None	42	Human	Binding	pKd	=	6.2	6.2	257	2	UnclassifiedUnclassified	Guide to Pharmacology	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10779375
	5957	520	None	42	Human	Binding	pKd	=	6.2	6.2	257	2	UnclassifiedUnclassified	Guide to Pharmacology	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10779375
	91	520	None	42	Human	Binding	pKd	=	6.2	6.2	257	2	UnclassifiedUnclassified	Guide to Pharmacology	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10779375
	CHEMBL14249	520	None	42	Human	Binding	pKd	=	6.2	6.2	257	2	UnclassifiedUnclassified	Guide to Pharmacology	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10779375
	DB00171	520	None	42	Human	Binding	pKd	=	6.2	6.2	257	2	UnclassifiedUnclassified	Guide to Pharmacology	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	10779375
	1713	520	None	42	Human	Binding	pKi	=	8.2	8.2	257	2	GRAC: human P2Y4 selective antagonistGRAC: human P2Y4 selective antagonist	Drug Central	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	None
	5957	520	None	42	Human	Binding	pKi	=	8.2	8.2	257	2	GRAC: human P2Y4 selective antagonistGRAC: human P2Y4 selective antagonist	Drug Central	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	None
	91	520	None	42	Human	Binding	pKi	=	8.2	8.2	257	2	GRAC: human P2Y4 selective antagonistGRAC: human P2Y4 selective antagonist	Drug Central	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	None
	CHEMBL14249	520	None	42	Human	Binding	pKi	=	8.2	8.2	257	2	GRAC: human P2Y4 selective antagonistGRAC: human P2Y4 selective antagonist	Drug Central	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	None
	DB00171	520	None	42	Human	Binding	pKi	=	8.2	8.2	257	2	GRAC: human P2Y4 selective antagonistGRAC: human P2Y4 selective antagonist	Drug Central	507	8	7	14	-1.6	O[C@@H]1[C@@H](COP(=O)(OP(=O)(OP(=O)(O)O)O)O)O[C@H]([C@@H]1O)n1cnc2c1ncnc2N	None

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