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Ligand source activities (1 row/activity)

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Ligands (move mouse cursor over ligand name to see structure)					Receptor		Activity									Chemical information
Sel. page	Common name No matches found	GPCRdb ID No matches found	Reference ligand No matches found	Vendors	Species No matches found		Assay Type No matches found	Activity Type No matches found	Activity Relation No matches found	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description No matches found	Source No matches found	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles No matches found	DOI No matches found

Ligands (move mouse cursor over ligand name to see structure)					Receptor	Activity									Chemical information
Sel. page	Common name No matches found	GPCRdb ID No matches found	Reference ligand No matches found	Vendors	Species No matches found	Assay Type No matches found	Activity Type No matches found	Activity Relation No matches found	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description No matches found	Source No matches found	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles No matches found	DOI No matches found
	71460332	80964	None	5	Human	Functional	pIC50	=	5.7	5.7	-181	3	Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assayAntagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assay	ChEMBL	429	7	1	3	6.2	C[C@H](NC(=O)CCCc1ccc2cccnc2n1)c1ccc(-c2cccc(Cl)c2)cc1	10.1016/j.bmcl.2011.04.091
	CHEMBL2153446	80964	None	5	Human	Functional	pIC50	=	5.7	5.7	-181	3	Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assayAntagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assay	ChEMBL	429	7	1	3	6.2	C[C@H](NC(=O)CCCc1ccc2cccnc2n1)c1ccc(-c2cccc(Cl)c2)cc1	10.1016/j.bmcl.2011.04.091
	71456641	80991	None	0	Human	Functional	pIC50	=	5.3	5.3	-125	3	Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assayAntagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assay	ChEMBL	426	6	0	5	6.2	Clc1cccc(-c2ccc(-c3nnc(CCCc4ccc5cccnc5n4)o3)cc2)c1	10.1016/j.bmcl.2011.04.091
	CHEMBL2153586	80991	None	0	Human	Functional	pIC50	=	5.3	5.3	-125	3	Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assayAntagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assay	ChEMBL	426	6	0	5	6.2	Clc1cccc(-c2ccc(-c3nnc(CCCc4ccc5cccnc5n4)o3)cc2)c1	10.1016/j.bmcl.2011.04.091
	71462027	80958	None	0	Human	Functional	pIC50	=	5.2	5.2	-173	3	Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assayAntagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assay	ChEMBL	415	7	1	3	5.6	O=C(CCCc1ccc2cccnc2n1)NCc1ccc(-c2cccc(Cl)c2)cc1	10.1016/j.bmcl.2011.04.091
	CHEMBL2153440	80958	None	0	Human	Functional	pIC50	=	5.2	5.2	-173	3	Antagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assayAntagonist activity at human GPR99 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induced increase in intracellular calcium level at by FLIPR assay	ChEMBL	415	7	1	3	5.6	O=C(CCCc1ccc2cccnc2n1)NCc1ccc(-c2cccc(Cl)c2)cc1	10.1016/j.bmcl.2011.04.091
	3636	361	None	69	Human	Functional	pEC50	=	3.9	3.9	-22908	2	UnclassifiedUnclassified	Guide to Pharmacology	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	15141213
	3636	361	None	69	Human	Functional	pEC50	=	3.9	3.9	-22908	2	UnclassifiedUnclassified	Guide to Pharmacology	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	23396314
	51	361	None	69	Human	Functional	pEC50	=	3.9	3.9	-22908	2	UnclassifiedUnclassified	Guide to Pharmacology	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	15141213
	51	361	None	69	Human	Functional	pEC50	=	3.9	3.9	-22908	2	UnclassifiedUnclassified	Guide to Pharmacology	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	23396314
	CHEMBL1686	361	None	69	Human	Functional	pEC50	=	3.9	3.9	-22908	2	UnclassifiedUnclassified	Guide to Pharmacology	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	15141213
	CHEMBL1686	361	None	69	Human	Functional	pEC50	=	3.9	3.9	-22908	2	UnclassifiedUnclassified	Guide to Pharmacology	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	23396314
	DB08845	361	None	69	Human	Functional	pEC50	=	3.9	3.9	-22908	2	UnclassifiedUnclassified	Guide to Pharmacology	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	15141213
	DB08845	361	None	69	Human	Functional	pEC50	=	3.9	3.9	-22908	2	UnclassifiedUnclassified	Guide to Pharmacology	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	23396314

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Ligands (move mouse cursor over ligand name to see structure)					Receptor		Activity									Chemical information
Sel. page	Common name No matches found	GPCRdb ID No matches found	Reference ligand No matches found	Vendors	Species No matches found		Assay Type No matches found	Activity Type No matches found	Activity Relation No matches found	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description No matches found	Source No matches found	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles No matches found	DOI No matches found

Ligands (move mouse cursor over ligand name to see structure)					Receptor	Activity									Chemical information
Sel. page	Common name No matches found	GPCRdb ID No matches found	Reference ligand No matches found	Vendors	Species No matches found	Assay Type No matches found	Activity Type No matches found	Activity Relation No matches found	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description No matches found	Source No matches found	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles No matches found	DOI No matches found
	46875342	204633	None	0	Rat	Binding	pKi	=	8	8.0	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	449	11	5	10	-0.4	CC(=O)NCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL609487	204633	None	0	Rat	Binding	pKi	=	8	8.0	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	449	11	5	10	-0.4	CC(=O)NCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	46875317	204431	None	0	Rat	Binding	pKi	=	6.0	6.0	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	414	3	4	9	0.1	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NC23CC4CC(CC(C4)C2)C3)[C@@H](O)[C@H]1O	10.1021/jm000150k
	CHEMBL608000	204431	None	0	Rat	Binding	pKi	=	6.0	6.0	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	414	3	4	9	0.1	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NC23CC4CC(CC(C4)C2)C3)[C@@H](O)[C@H]1O	10.1021/jm000150k
	10089226	79321	None	0	Rat	Binding	pKi	=	7.9	7.9	50	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	350	6	4	9	-0.7	CCCCCNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL2113492	79321	None	0	Rat	Binding	pKi	=	7.9	7.9	50	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	350	6	4	9	-0.7	CCCCCNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	10738295	77849	None	0	Rat	Binding	pKi	=	7.9	7.9	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	376	3	4	9	-0.3	C[C@H]1CC[C@H](NC(=O)[C@H]2O[C@@H](n3cnc4c(N)ncnc43)[C@H](O)[C@@H]2O)CC1	10.1021/jm000150k
	CHEMBL2092859	77849	None	0	Rat	Binding	pKi	=	7.9	7.9	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	376	3	4	9	-0.3	C[C@H]1CC[C@H](NC(=O)[C@H]2O[C@@H](n3cnc4c(N)ncnc43)[C@H](O)[C@@H]2O)CC1	10.1021/jm000150k
	46875267	204676	None	0	Rat	Binding	pKi	=	6.9	6.9	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	434	12	4	9	1.7	CCCCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL609768	204676	None	0	Rat	Binding	pKi	=	6.9	6.9	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	434	12	4	9	1.7	CCCCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	46875320	204432	None	0	Rat	Binding	pKi	=	6.9	6.9	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	430	6	4	11	-0.6	COc1ccc(CNC(=O)[C@H]2OC(n3cnc4c(N)ncnc43)[C@H](O)[C@@H]2O)cc1OC	10.1021/jm000150k
	CHEMBL608003	204432	None	0	Rat	Binding	pKi	=	6.9	6.9	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	430	6	4	11	-0.6	COc1ccc(CNC(=O)[C@H]2OC(n3cnc4c(N)ncnc43)[C@H](O)[C@@H]2O)cc1OC	10.1021/jm000150k
	46875266	204632	None	0	Rat	Binding	pKi	=	6.8	6.8	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	448	13	4	9	2.1	CCCCCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL609485	204632	None	0	Rat	Binding	pKi	=	6.8	6.8	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	448	13	4	9	2.1	CCCCCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	9996282	19496	None	0	Rat	Binding	pKi	=	6.8	6.8	-3	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	323	4	5	10	-2.9	NCCNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL129903	19496	None	0	Rat	Binding	pKi	=	6.8	6.8	-3	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	323	4	5	10	-2.9	NCCNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	49797674	204604	None	0	Rat	Binding	pKi	=	7.8	7.8	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	336	5	4	9	-1.1	CCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL609186	204604	None	0	Rat	Binding	pKi	=	7.8	7.8	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	336	5	4	9	-1.1	CCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	10316575	79318	None	0	Rat	Binding	pKi	=	7.8	7.8	141	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	362	3	4	9	-0.5	Nc1ncnc2c1ncn2[C@@H]1O[C@H](C(=O)NC2CCCCC2)[C@@H](O)[C@H]1O	10.1021/jm000150k
	CHEMBL2113489	79318	None	0	Rat	Binding	pKi	=	7.8	7.8	141	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	362	3	4	9	-0.5	Nc1ncnc2c1ncn2[C@@H]1O[C@H](C(=O)NC2CCCCC2)[C@@H](O)[C@H]1O	10.1021/jm000150k
	21152082	204395	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	364	7	4	9	-0.3	CCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL607719	204395	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	364	7	4	9	-0.3	CCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	46875402	204561	None	0	Rat	Binding	pKi	=	6.7	6.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	336	4	4	9	-1.1	CCC(C)NC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL608895	204561	None	0	Rat	Binding	pKi	=	6.7	6.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	336	4	4	9	-1.1	CCC(C)NC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	56668023	63282	None	0	Rat	Binding	pKi	=	7.7	7.7	44	3	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	291	2	4	9	-2.0	C#CC(O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL1791423	63282	None	0	Rat	Binding	pKi	=	7.7	7.7	44	3	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	291	2	4	9	-2.0	C#CC(O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	46875323	204471	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	352	5	4	10	-1.3	CC(C)CONC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL608293	204471	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	352	5	4	10	-1.3	CC(C)CONC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	46875257	204559	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	378	8	4	9	0.1	CCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL608888	204559	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	378	8	4	9	0.1	CCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	46875347	204679	None	0	Rat	Binding	pKi	=	5.7	5.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	414	3	4	9	-0.0	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NC2C3CC4CC(C3)CC2C4)[C@@H](O)[C@H]1O	10.1021/jm000150k
	CHEMBL609774	204679	None	0	Rat	Binding	pKi	=	5.7	5.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	414	3	4	9	-0.0	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NC2C3CC4CC(C3)CC2C4)[C@@H](O)[C@H]1O	10.1021/jm000150k
	46875326	204472	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	392	9	4	9	0.5	CCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL608296	204472	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	392	9	4	9	0.5	CCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	46875346	204678	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	376	3	4	9	-0.1	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NC2CCCCCC2)[C@@H](O)[C@H]1O	10.1021/jm000150k
	CHEMBL609773	204678	None	0	Rat	Binding	pKi	=	7.7	7.7	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	376	3	4	9	-0.1	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NC2CCCCCC2)[C@@H](O)[C@H]1O	10.1021/jm000150k
	46875336	204560	None	0	Rat	Binding	pKi	=	7.6	7.6	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	390	3	4	9	0.3	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NC2CCCCCCC2)[C@@H](O)[C@H]1O	10.1021/jm000150k
	CHEMBL608893	204560	None	0	Rat	Binding	pKi	=	7.6	7.6	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	390	3	4	9	0.3	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NC2CCCCCCC2)[C@@H](O)[C@H]1O	10.1021/jm000150k
	377	2758	None	42	Rat	Binding	pKi	=	7.6	7.6	-70	15	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	10.1021/jm000150k
	425	2758	None	42	Rat	Binding	pKi	=	7.6	7.6	-70	15	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	10.1021/jm000150k
	448222	2758	None	42	Rat	Binding	pKi	=	7.6	7.6	-70	15	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	10.1021/jm000150k
	CHEMBL464859	2758	None	42	Rat	Binding	pKi	=	7.6	7.6	-70	15	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	308	3	4	9	-1.8	CCNC(=O)[C@H]1O[C@H]([C@@H]([C@@H]1O)O)n1cnc2c1ncnc2N	10.1021/jm000150k
	46875307	205072	None	0	Rat	Binding	pKi	=	7.6	7.6	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	420	11	4	9	1.3	CCCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL612154	205072	None	0	Rat	Binding	pKi	=	7.6	7.6	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	420	11	4	9	1.3	CCCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	46875349	204681	None	0	Rat	Binding	pKi	=	7.5	7.5	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	407	10	5	10	-0.6	NCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL609776	204681	None	0	Rat	Binding	pKi	=	7.5	7.5	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	407	10	5	10	-0.6	NCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	3044933	16490	None	4	Rat	Binding	pKi	=	7.5	7.5	-2	6	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	322	4	4	9	-1.4	CCCNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL1235128	16490	None	4	Rat	Binding	pKi	=	7.5	7.5	-2	6	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	322	4	4	9	-1.4	CCCNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	46875268	204677	None	0	Rat	Binding	pKi	=	7.5	7.5	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	406	10	4	9	0.9	CCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k
	CHEMBL609769	204677	None	0	Rat	Binding	pKi	=	7.5	7.5	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranesBinding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	406	10	4	9	0.9	CCCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	10.1021/jm000150k

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Ligand source activities (1 row/activity)